AChR
Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.
Trovati 617 prodotti di "AChR"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Tolterodine tartrate
CAS:Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.Formula:C22H31NO·C4H6O6Purezza:99.95%Colore e forma:White-To-Off-White Crystalline PowderPeso molecolare:475.58Dequalinium chloride
CAS:<p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>Formula:C30H40Cl2N4Purezza:99.79% - 99.9%Colore e forma:SolidPeso molecolare:527.59Bambuterol hydrochloride
CAS:Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.Formula:C18H30ClN3O5Purezza:99.53% - 99.61%Colore e forma:White SolidPeso molecolare:403.91Vecuronium bromide
CAS:Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking agent, with muscleFormula:C34H57BrN2O4Purezza:99.63% - 99.92%Colore e forma:White PowderPeso molecolare:637.73Ribavirin
CAS:Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.Formula:C8H12N4O5Purezza:99.09% - 99.83%Colore e forma:Less Solid Colourless SolidPeso molecolare:244.20Benzethonium chloride
CAS:Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.Formula:C27H42ClNO2Purezza:99.91%Colore e forma:White To Off-White Solid Solid Particulate/PowderPeso molecolare:448.09Atropine methyl bromide
CAS:<p>Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.</p>Formula:C18H26BrNO3Purezza:99.7%Colore e forma:SolidPeso molecolare:384.308Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formula:C21H25NO·CH4SO3Purezza:98.41% - 99.96%Colore e forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecolare:403.53Oxybutynin
CAS:Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.Formula:C22H31NO3Purezza:97.81% - 99.57%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:357.49V-11-0711 HCl
V-11-0711 HCl is a selective and highly effective choline kinase α (ChoKα) inhibitor that inhibits the catalytic activity of Chk.Formula:C27H36ClNO3Purezza:99.87%Colore e forma:SolidPeso molecolare:458.03Solifenacin succinate
CAS:<p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>Formula:C23H26N2O2·C4H6O4Purezza:99.85% - 99.98%Colore e forma:SolidPeso molecolare:480.56Bethanechol chloride
CAS:Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.Formula:C7H17N2O2·ClPurezza:95% - 99.73%Colore e forma:White CrystallinePeso molecolare:196.68Carbetapentane citrate
CAS:Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Formula:C20H31NO3·C6H8O7Purezza:99.46%Colore e forma:White To Off-White SolidPeso molecolare:525.59Dicyclomine hydrochloride
CAS:<p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>Formula:C19H36ClNO2Purezza:99.81%Colore e forma:SolidPeso molecolare:345.95Pancuronium dibromide
CAS:Pancuronium dibromide (Pavulon), a competitive AChR antagonist, acts as a skeletal muscle relaxant. Pancuronium dibromide blocks neuromuscular transmission.Formula:C35H60Br2N2O4Purezza:99.86%Colore e forma:solidPeso molecolare:732.67Temephos
CAS:<p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>Formula:C16H20O6P2S3Purezza:≥95%Colore e forma:White Crystalline Solid Or LiquidPeso molecolare:466.47Methscopolamine
CAS:Methscopolamine (Hyoscine methyl bromide) (Pamine), as a natural plant alkaloid, is a muscarinic acetylcholine receptor blocker.Formula:C18H24BrNO4Purezza:99.12% - ≥98%Colore e forma:SolidPeso molecolare:398.29PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Formula:C36H51Cl3N4O7SPurezza:99.85%Colore e forma:SolidPeso molecolare:790.24Hexamethonium Bromide
CAS:Hexamethonium Bromide blocks neural nicotinic AChR, poorly absorbed in the gut, doesn't pass the blood-brain barrier.Formula:C12H30Br2N2Purezza:99.76%Colore e forma:White Crystalline Powder And AgglomeratesPeso molecolare:362.19Flavoxate hydrochloride
CAS:<p>Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.</p>Formula:C24H26ClNO4Purezza:99.78%Colore e forma:White SolidPeso molecolare:427.92Homatropine Methylbromide
CAS:<p>Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.</p>Formula:C17H24BrNO3Purezza:98.97%Colore e forma:SolidPeso molecolare:370.29SSR 180
CAS:<p>SSR 180 is a potent and subtype-selective α7 agonist with applications in the study of Alzheimer;s disease and schizophrenia.</p>Formula:C14H17BrN2O2Purezza:98.82%Colore e forma:SoildPeso molecolare:325.20Pirenzepine dihydrochloride
CAS:Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.Formula:C19H21N5O2·2HClPurezza:99.48% - 99.62%Colore e forma:White PowderPeso molecolare:424.32Diphenmanil methylsulfate
CAS:Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.Formula:C20H24N·CH3O4SPurezza:98% - 99.27%Colore e forma:SolidPeso molecolare:389.51Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formula:C17H20N2S·HClPurezza:99.85%Colore e forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecolare:320.88Procainamide hydrochloride
CAS:Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analogFormula:C13H21N3O·HClPurezza:99.83% - 99.97%Colore e forma:White To Slightly Yellow PowderPeso molecolare:271.79Tiotropium bromide
CAS:<p>Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).</p>Formula:C19H22BrNO4S2Purezza:96.82% - 99.97%Colore e forma:White SolidPeso molecolare:472.42Valethamate bromide
CAS:<p>Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.</p>Formula:C19H32BrNO2Purezza:>99.99%Colore e forma:SolidPeso molecolare:386.37VU 0365114
CAS:VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).Formula:C22H14F3NO3Purezza:99.86%Colore e forma:SolidPeso molecolare:397.35Fesoterodine fumarate
CAS:<p>Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.</p>Formula:C26H37NO3·C4H4O4Purezza:99.16%Colore e forma:White SolidPeso molecolare:527.65Adiphenine hydrochloride
CAS:Adiphenine hydrochloride (Patrovina), a nicotinic receptor inhibitor, can be used as an antispasmodic drug.Formula:C20H25NO2·HClPurezza:97.76% - 99.53%Colore e forma:White Or Almost White PowderPeso molecolare:347.889-Cyclopentyladenine
CAS:9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signalingFormula:C10H13N5Purezza:99.98%Colore e forma:SolidPeso molecolare:203.24Nefiracetam
CAS:<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Formula:C14H18N2O2Purezza:97.37%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:246.3Gallamine triethiodide
CAS:Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.Formula:C30H60I3N3O3Purezza:98.90%Colore e forma:White Amorphous Powder SolidPeso molecolare:891.53Zelminemab
CAS:Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].Purezza:98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)Colore e forma:LiquidDroperidol
CAS:<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Formula:C22H22FN3O2Purezza:97.16% - 98%Colore e forma:SolidPeso molecolare:379.43Cotinine
CAS:Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.Formula:C10H12N2OPurezza:98% - 99.89%Colore e forma:Viscous Oil SolidPeso molecolare:176.22Orphenadrine Citrate
CAS:<p>Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.</p>Formula:C18H23NO·C6H8O7Purezza:98% - 99.58%Colore e forma:White SolidPeso molecolare:461.5Nicardipine hydrochloride
CAS:<p>Nicardipine hydrochloride is a potent calcium channel blocker used to dilate cerebral and coronary vessels.</p>Formula:C26H30ClN3O6Purezza:99.58% - 99.89%Colore e forma:Yellow SolidPeso molecolare:515.99Dipivefrin hydrochloride
CAS:<p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>Formula:C19H27NO5·HClPurezza:99.22% - 99.92%Colore e forma:Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorPeso molecolare:387.9Clidinium bromide
CAS:Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.Formula:C22H26BrNO3Purezza:98.89% - 99.86%Colore e forma:White Crystalline SolidPeso molecolare:432.35Trospium chloride
CAS:<p>Trospium chloride treats urinary incontinence without causing liver damage.</p>Formula:C25H30ClNO3Purezza:99.84% - >99.99%Colore e forma:White To Off-White PowderPeso molecolare:427.964Propantheline bromide
CAS:Propantheline bromide (Pro-Banthine) competitively antagonizes acetylcholine activity mediated by muscarinic receptors at neuroeffector sites on smooth muscleFormula:C23H30BrNO3Purezza:98% - ≥98%Peso molecolare:448.4Darifenacin hydrobromide
CAS:<p>Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome.</p>Formula:C28H31BrN2O2Purezza:99.75% - >99.99%Colore e forma:SolidPeso molecolare:505.45Tazomeline
CAS:Tazomeline is a muscarinic M1 receptor agonist with neuroprotective activity.Formula:C14H23N3S2Purezza:99.63%Colore e forma:SolidPeso molecolare:297.48Lysipressin acetate(50-57-7(fb_acetate))
CAS:<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Formula:C48H69N13O14S2Purezza:98.08%Colore e forma:SolidPeso molecolare:1116.28nAChR agonist 1
CAS:<p>nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine receptor (α7 nAChR)modulator.</p>Formula:C20H18ClNO3S2Purezza:97.59%Colore e forma:SolidPeso molecolare:419.94Methacholine Chloride
CAS:<p>Methacholine Chloride (Acetyl-β-methylcholine chloride) is a quaternary ammonium parasympathomimetic agent with the muscarinic actions of acetylcholine.</p>Formula:C8H18ClNO2Purezza:99.37% - 99.74%Colore e forma:White Hygroscopic Crystals With Slight Odor Of Dead FishPeso molecolare:195.69Ipratropium bromide monohydrate
CAS:<p>Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.</p>Formula:C20H32BrNO4Purezza:97.85%Colore e forma:SolidPeso molecolare:430.38MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Formula:C25H25N3O2Purezza:99.77% - 99.8%Colore e forma:SolidPeso molecolare:399.48Deschloroclozapine
CAS:Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist.Formula:C18H20N4Purezza:99.61% - 99.98%Colore e forma:SolidPeso molecolare:292.38Benactyzine hydrochloride
CAS:<p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>Formula:C20H26ClNO3Purezza:99.03% - 99.94%Colore e forma:SolidPeso molecolare:363.88Fipexide
CAS:Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.Formula:C20H21ClN2O4Purezza:97.6% - 99.95%Colore e forma:SolidPeso molecolare:388.842',5'-Dideoxyadenosine
CAS:2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).Formula:C10H13N5O2Purezza:99.55%Colore e forma:White SolidPeso molecolare:235.24DL-trihexyphenidyl hydrochloride
CAS:DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.Formula:C20H32ClNOPurezza:99.63% - 99.71%Colore e forma:SolidPeso molecolare:337.93Pyrantel pamoate
CAS:<p>Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent.</p>Formula:C34H30N2O6SPurezza:99.71%Peso molecolare:594.69(Rac)-ABT-202 dihydrochloride
CAS:(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.Formula:C9H15Cl2N3Purezza:97.4%Colore e forma:SolidPeso molecolare:236.142Primidone
CAS:Primidone (NCI-C56360) is a potent anticonvulsant agent.Formula:C12H14N2O2Purezza:99.91%Colore e forma:Crystals (Ntp 1992)Peso molecolare:218.25Nebracetam hydrochloride
CAS:Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.Formula:C12H17ClN2OPurezza:99.23%Colore e forma:SolidPeso molecolare:240.729Pyrantel tartrate
CAS:Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.Formula:C15H20N2O6SPurezza:99.96%Colore e forma:White CrystalsPeso molecolare:356.39(Rac)-Sabcomeline HCl
CAS:<p>Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.</p>Formula:C10H16ClN3OPurezza:99.58%Colore e forma:SoildPeso molecolare:229.71Carbachol
CAS:<p>Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.</p>Formula:C6H15ClN2O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:182.65TAK-071
CAS:<p>TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).</p>Formula:C24H24FN3O3Purezza:98.02%Colore e forma:SolidPeso molecolare:421.46Acetamiprid
CAS:Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.Formula:C10H11ClN4Purezza:99.66%Colore e forma:White PowderPeso molecolare:222.67Rocuronium bromide
CAS:<p>Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.</p>Formula:C32H53BrN2O4Purezza:99.77% - >99.99%Colore e forma:White Or Off-White PowderPeso molecolare:609.68β2AR/M-receptor agonist-1
CAS:β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor andFormula:C43H56BrN3O7Colore e forma:SolidPeso molecolare:806.82Methylatropine (nitrate)
CAS:Methylatropine: Muscarinic antagonist, <0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.Formula:C18H26N2O6Colore e forma:SolidPeso molecolare:366.414Lupanine hydrochloride
CAS:Lupanine hydrochloride, a Sparteine derivative, binds to nAChR with a Ki of 500 nM and has ganglioplegic properties.Formula:C15H25ClN2OColore e forma:SolidPeso molecolare:284.83nAChR modulator-1
CAS:nAChR modulator-1, a insecticide, is a insect nAChR orthosteric modulator [1] .Formula:C12H8ClN3O2Colore e forma:SolidPeso molecolare:261.66Navafenterol saccharinate
CAS:AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).Formula:C45H47N7O9S3Colore e forma:SolidPeso molecolare:926.09Epiboxidine
CAS:Epiboxidine: Potent, selective nAChR agonist; Ki 0.46/1.2 nM for rat/human α4β2; analogous to Epibatidine and ABT 418.Formula:C10H14N2OColore e forma:SolidPeso molecolare:178.23Lobeline sulfate
CAS:Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.Formula:C22H29NO6SPurezza:98%Colore e forma:White PowderPeso molecolare:435.54trans-Cevimeline hydrochloride
CAS:<p>AF 102A hydrochloride is a biochemical.</p>Formula:C10H18ClNOSColore e forma:SolidPeso molecolare:235.77TC-2559 difumarate
CAS:TC-2559 difumarate: Oral α4β2 nAChR partial agonist, CNS-selective, EC50 0.18 μM, prefers α4β2 over α2β4/α4β4/α3β4, antinociceptive.Formula:C20H26N2O9Colore e forma:SolidPeso molecolare:438.43Perindoprilat
CAS:Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.Formula:C17H28N2O5Purezza:99.48%Colore e forma:SolidPeso molecolare:340.41Dicloromezotiaz
CAS:Dicloromezotiaz: Potent insecticide targeting nAChRs, controls various lepidoptera.Formula:C19H12Cl3N3O2SColore e forma:SolidPeso molecolare:452.74Muscarine
CAS:Muscarine is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.Formula:C9H20NO2Purezza:98%Colore e forma:SolidPeso molecolare:174.26(R)-Dinotefuran
CAS:(R)-Dinotefuran, a neonicotinoid, is 1.7-2.4x more effective against pests like Aphis gossypii and safer for bees.Formula:C7H14N4O3Colore e forma:SolidPeso molecolare:202.21(Rac)-5-Hydroxymethyl Tolterodine hydrochloride
CAS:<p>(Rac)-5-Hydroxymethyl Tolterodine HCl, or (Rac)-Desfesoterodine HCl, is a potent mAChR blocker researched for overactive bladder.</p>Formula:C22H32ClNO2Colore e forma:SolidPeso molecolare:377.95(rel)-Asperparaline A
CAS:<p>Aspergillimide, from A. japonicus, inhibits silkworm neuron nAChRs (IC50s: 20.2/39.6 nM), not affecting chicken nAChRs, and paralyzes silkworm larvae.</p>Formula:C20H29N3O3Colore e forma:SolidPeso molecolare:359.47DSPE-PEG1000-RVG29
DSPE-PEG1000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 can specifically bind to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and cross the BBB.Colore e forma:Odour SolidTMPH
CAS:TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.Formula:C16H31NO2Purezza:99.78%Colore e forma:SoildPeso molecolare:269.428-Aminoadenine
CAS:<p>8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.</p>Formula:C5H6N6Purezza:99.82%Colore e forma:SolidPeso molecolare:150.14M3/PDE4 modulator-1
M3/PDE4 Modulator-1 (compound 10f) serves as a bifunctional entity functioning both as an M3 mAChR antagonist and a PDE4 inhibitor.Formula:C38H41Cl2N3O8SColore e forma:SolidPeso molecolare:770.72Doxacurium Chloride
CAS:Doxacurium Chloride is a muscarinic acetylcholine receptor M2 antagonist.Formula:C56H78ClN2O16Purezza:98%Colore e forma:SolidPeso molecolare:1070.69nAChR modulator-2
CAS:nAChR modulator-2, a insecticide, is a insect nAChR orthosteric modulator [1] .Formula:C12H8ClN3O2Colore e forma:SolidPeso molecolare:261.66nAChR agonist CMPI hydrochloride
CAS:CMPI hydrochloride: Potent α4:α4 nAChR PAM; EC50 0.26 μM for (α4)3(β2)2 response to ACh; may aid nicotine dependence, neuropsychiatric research.Formula:C18H20Cl2N4OColore e forma:SolidPeso molecolare:379.29MK-0969
CAS:MK-0969 (J-104135) is a possible M3 antagonist for the treatment of chronic obstructive pulmonary disease.Formula:C24H30F2N4O2Colore e forma:SolidPeso molecolare:444.52Atracurium
CAS:Atracurium (BW-33A) is a competitive AChR antagonist and non-depolarizing muscle relaxant that may cause bronchoconstriction.Formula:C53H72N2O122Colore e forma:SolidPeso molecolare:929.14α-Conotoxin PIA
CAS:Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nMFormula:C79H125N27O25S4Purezza:98%Colore e forma:SolidPeso molecolare:1981.3α-Conotoxin PIA TFA
α-Conotoxin PIA TFA, targeting nicotinic acetylcholine receptor (nAChR) subtypes with α6 and α3 subunits, acts as an antagonist.Formula:C81H126F3N27O27S4Purezza:98.81%Colore e forma:SolidPeso molecolare:2095.3Epiboxidine hydrochloride
CAS:Epiboxidine HCl: potent α4β2 nAChR agonist; Ki 0.46 nM (rat), 1.2 nM (human); Epibatidine analog.Formula:C10H15ClN2OColore e forma:SolidPeso molecolare:214.69Navafenterol
CAS:AZD-8871, a potential COPD and asthma treatment, may work well with ICS.Formula:C38H42N6O6S2Colore e forma:SolidPeso molecolare:742.91α-Conotoxin AuIB
CAS:Selective antagonist of α3β4 nicotinic acetylcholine receptors.Formula:C65H89N17O21S4Purezza:98%Colore e forma:SolidPeso molecolare:1572.76α-Conotoxin imi
CAS:alpha-Conotoxin imi is a nicotinic acetylcholine receptor ligand.Formula:C52H78N20O15S4Purezza:98%Colore e forma:SolidPeso molecolare:1351.56AC1-IN-1
CAS:<p>AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 µM).</p>Formula:C18H18FN5O2Purezza:99.89%Colore e forma:SolidPeso molecolare:355.37Heliosupine N-oxide
Heliosupine N-oxide is a useful organic compound for research related to life sciences and the catalog number is T125058.Formula:C20H31NO8Colore e forma:SolidPeso molecolare:413.467rac-Desethyl Oxybutynin (hydrochloride)
CAS:<p>rac-Desethyl oxybutynin, active oxybutynin metabolite, binds to mAChRs; K_i values 3.12-16 nM; lowers rat micturition pressure.</p>Formula:C20H28ClNO3Colore e forma:SolidPeso molecolare:365.89α-Bungarotoxin
CAS:<p>Neurotoxin that blocks neuromuscular transmission via irreversible inhibition of nicotinic ACh receptors (nAChRs).</p>Formula:C338H529N97O105S11Purezza:98%Colore e forma:SolidPeso molecolare:7984.14DSPE-PEG5000-RVG29
DSPE-PEG5000-RVG29 is a PEG compound comprised of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and facilitates passage through the BBB.Colore e forma:Odour Solid
