AChR
Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.
Trovati 617 prodotti di "AChR"
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Valethamate bromide
CAS:<p>Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.</p>Formula:C19H32BrNO2Purezza:>99.99%Colore e forma:SolidPeso molecolare:386.37Fipexide
CAS:Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.Formula:C20H21ClN2O4Purezza:97.6% - 99.95%Colore e forma:SolidPeso molecolare:388.849-Cyclopentyladenine
CAS:9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signalingFormula:C10H13N5Purezza:99.98%Colore e forma:SolidPeso molecolare:203.24Zelminemab
CAS:Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].Purezza:98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)Colore e forma:LiquidOrphenadrine Citrate
CAS:<p>Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.</p>Formula:C18H23NO·C6H8O7Purezza:98% - 99.58%Colore e forma:White SolidPeso molecolare:461.52',5'-Dideoxyadenosine
CAS:2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).Formula:C10H13N5O2Purezza:99.55%Colore e forma:White SolidPeso molecolare:235.24Dequalinium chloride
CAS:<p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>Formula:C30H40Cl2N4Purezza:99.79% - 99.9%Colore e forma:SolidPeso molecolare:527.59Ipratropium bromide monohydrate
CAS:<p>Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.</p>Formula:C20H32BrNO4Purezza:97.85%Colore e forma:SolidPeso molecolare:430.38Pancuronium dibromide
CAS:Pancuronium dibromide (Pavulon), a competitive AChR antagonist, acts as a skeletal muscle relaxant. Pancuronium dibromide blocks neuromuscular transmission.Formula:C35H60Br2N2O4Purezza:99.86%Colore e forma:solidPeso molecolare:732.67Carbetapentane citrate
CAS:Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Formula:C20H31NO3·C6H8O7Purezza:99.46%Colore e forma:White To Off-White SolidPeso molecolare:525.59Tiotropium bromide
CAS:<p>Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).</p>Formula:C19H22BrNO4S2Purezza:96.82% - 99.97%Colore e forma:White SolidPeso molecolare:472.42Ribavirin
CAS:Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.Formula:C8H12N4O5Purezza:99.09% - 99.83%Colore e forma:Less Solid Colourless SolidPeso molecolare:244.20Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formula:C21H25NO·CH4SO3Purezza:98.41% - 99.96%Colore e forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecolare:403.53Nicardipine hydrochloride
CAS:<p>Nicardipine hydrochloride is a potent calcium channel blocker used to dilate cerebral and coronary vessels.</p>Formula:C26H30ClN3O6Purezza:99.58% - 99.89%Colore e forma:Yellow SolidPeso molecolare:515.99Adiphenine hydrochloride
CAS:Adiphenine hydrochloride (Patrovina), a nicotinic receptor inhibitor, can be used as an antispasmodic drug.Formula:C20H25NO2·HClPurezza:97.76% - 99.53%Colore e forma:White Or Almost White PowderPeso molecolare:347.88Pyrantel pamoate
CAS:<p>Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent.</p>Formula:C34H30N2O6SPurezza:99.71%Peso molecolare:594.69Deschloroclozapine
CAS:Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist.Formula:C18H20N4Purezza:99.61% - 99.98%Colore e forma:SolidPeso molecolare:292.38(Rac)-Sabcomeline HCl
CAS:<p>Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.</p>Formula:C10H16ClN3OPurezza:99.58%Colore e forma:SoildPeso molecolare:229.71Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formula:C17H20N2S·HClPurezza:99.85%Colore e forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecolare:320.88Lysipressin acetate(50-57-7(fb_acetate))
CAS:<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Formula:C48H69N13O14S2Purezza:98.08%Colore e forma:SolidPeso molecolare:1116.28Fesoterodine fumarate
CAS:<p>Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.</p>Formula:C26H37NO3·C4H4O4Purezza:99.16%Colore e forma:White SolidPeso molecolare:527.65Atropine methyl bromide
CAS:<p>Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.</p>Formula:C18H26BrNO3Purezza:99.7%Colore e forma:SolidPeso molecolare:384.308Primidone
CAS:Primidone (NCI-C56360) is a potent anticonvulsant agent.Formula:C12H14N2O2Purezza:99.91%Colore e forma:Crystals (Ntp 1992)Peso molecolare:218.25Methscopolamine
CAS:Methscopolamine (Hyoscine methyl bromide) (Pamine), as a natural plant alkaloid, is a muscarinic acetylcholine receptor blocker.Formula:C18H24BrNO4Purezza:99.12% - ≥98%Colore e forma:SolidPeso molecolare:398.29MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Formula:C25H25N3O2Purezza:99.77% - 99.8%Colore e forma:SolidPeso molecolare:399.48Cotinine
CAS:Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.Formula:C10H12N2OPurezza:98% - 99.89%Colore e forma:Viscous Oil SolidPeso molecolare:176.22PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Formula:C36H51Cl3N4O7SPurezza:99.85%Colore e forma:SolidPeso molecolare:790.24(Rac)-ABT-202 dihydrochloride
CAS:(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.Formula:C9H15Cl2N3Purezza:97.4%Colore e forma:SolidPeso molecolare:236.142Bambuterol hydrochloride
CAS:Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.Formula:C18H30ClN3O5Purezza:99.53% - 99.61%Colore e forma:White SolidPeso molecolare:403.91Procainamide hydrochloride
CAS:Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analogFormula:C13H21N3O·HClPurezza:99.83% - 99.97%Colore e forma:White To Slightly Yellow PowderPeso molecolare:271.79Acetamiprid
CAS:Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.Formula:C10H11ClN4Purezza:99.66%Colore e forma:White PowderPeso molecolare:222.67Rocuronium bromide
CAS:<p>Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.</p>Formula:C32H53BrN2O4Purezza:99.77% - >99.99%Colore e forma:White Or Off-White PowderPeso molecolare:609.68TAK-071
CAS:<p>TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).</p>Formula:C24H24FN3O3Purezza:98.02%Colore e forma:SolidPeso molecolare:421.46Carbachol
CAS:<p>Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.</p>Formula:C6H15ClN2O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:182.65Benzethonium chloride
CAS:Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.Formula:C27H42ClNO2Purezza:99.91%Colore e forma:White To Off-White Solid Solid Particulate/PowderPeso molecolare:448.09DL-trihexyphenidyl hydrochloride
CAS:DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.Formula:C20H32ClNOPurezza:99.63% - 99.71%Colore e forma:SolidPeso molecolare:337.93Dicyclomine hydrochloride
CAS:<p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>Formula:C19H36ClNO2Purezza:99.81%Colore e forma:SolidPeso molecolare:345.95VU 0365114
CAS:VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).Formula:C22H14F3NO3Purezza:99.86%Colore e forma:SolidPeso molecolare:397.35Bethanechol chloride
CAS:Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.Formula:C7H17N2O2·ClPurezza:95% - 99.73%Colore e forma:White CrystallinePeso molecolare:196.68Benactyzine hydrochloride
CAS:<p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>Formula:C20H26ClNO3Purezza:99.03% - 99.94%Colore e forma:SolidPeso molecolare:363.88Solifenacin succinate
CAS:<p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>Formula:C23H26N2O2·C4H6O4Purezza:99.85% - 99.98%Colore e forma:SolidPeso molecolare:480.56Diphenmanil methylsulfate
CAS:Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.Formula:C20H24N·CH3O4SPurezza:98% - 99.27%Colore e forma:SolidPeso molecolare:389.51Pirenzepine dihydrochloride
CAS:Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.Formula:C19H21N5O2·2HClPurezza:99.48% - 99.62%Colore e forma:White PowderPeso molecolare:424.32Nefiracetam
CAS:<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Formula:C14H18N2O2Purezza:97.37%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:246.3Gallamine triethiodide
CAS:Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.Formula:C30H60I3N3O3Purezza:98.90%Colore e forma:White Amorphous Powder SolidPeso molecolare:891.53Temephos
CAS:<p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>Formula:C16H20O6P2S3Purezza:≥95%Colore e forma:White Crystalline Solid Or LiquidPeso molecolare:466.47Nebracetam hydrochloride
CAS:Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.Formula:C12H17ClN2OPurezza:99.23%Colore e forma:SolidPeso molecolare:240.729Pyrantel tartrate
CAS:Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.Formula:C15H20N2O6SPurezza:99.96%Colore e forma:White CrystalsPeso molecolare:356.39Droperidol
CAS:<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Formula:C22H22FN3O2Purezza:97.16% - 98%Colore e forma:SolidPeso molecolare:379.43Dipivefrin hydrochloride
CAS:<p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>Formula:C19H27NO5·HClPurezza:99.22% - 99.92%Colore e forma:Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorPeso molecolare:387.9
