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AChR

AChR

Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.

Trovati 620 prodotti di "AChR"

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  • Thiochrome
    Targetmol
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    Thiochrome

    CAS:
    Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.
    Formula:C12H14N4OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:262.33

    Ref: TM-T13924

  • VU0090157
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    VU0090157

    CAS:
    VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.
    Formula:C19H21N3O7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:403.39

    Ref: TM-T29122

  • GAT107
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    GAT107

    CAS:
    GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.
    Formula:C18H17BrN2O2S
    Purezza:99.33%
    Colore e forma:Solid
    Peso molecolare:405.31

    Ref: TM-T27404

  • S-(+)-Mecamylamine hydrochloride
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    S-(+)-Mecamylamine hydrochloride

    CAS:
    Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.
    Formula:C11H22ClN
    Colore e forma:Solid
    Peso molecolare:203.75

    Ref: TM-T31401

  • T761-0184
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    T761-0184

    CAS:
    T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].
    Formula:C16H20FN3O
    Colore e forma:Solid
    Peso molecolare:289.35

    Ref: TM-T60588

  • Revatropate
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    Revatropate

    CAS:
    Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.
    Formula:C19H27NO4S
    Colore e forma:Solid
    Peso molecolare:365.49

    Ref: TM-T28523

  • Rispenzepine
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    Rispenzepine

    CAS:
    Rispenzepine, a novel mAChRs M1/M3 antagonist, treats immune, infections, and respiratory issues.
    Formula:C19H20N4O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:336.39

    Ref: TM-T16758

  • SCH 57790
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    SCH 57790

    CAS:
    SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.
    Formula:C25H31N3O2S
    Purezza:99.12% - 99.69%
    Colore e forma:Solid
    Peso molecolare:437.6

    Ref: TM-T28722

  • Milameline
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    Milameline

    CAS:
    Milameline is a muscarinic receptor agonist that improves cognition.
    Formula:C8H14N2O
    Colore e forma:Solid
    Peso molecolare:154.21

    Ref: TM-T70772

  • Biricodar dicitrate
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    Biricodar dicitrate

    CAS:
    Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.
    Formula:C46H57N3O21
    Purezza:97.78% - 99.78%
    Colore e forma:Solid
    Peso molecolare:987.95

    Ref: TM-T67790

  • Tarafenacin
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    Tarafenacin

    CAS:
    Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.
    Formula:C21H20F4N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:408.39

    Ref: TM-T16990

  • Sofiniclin
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    Sofiniclin

    CAS:
    Sofiniclin (ABT 894) is an agonist of nicotinic acetylcholine receptor (nAChR). It is used for the research for attention-deficit/hyperactivity disorder (ADHD).
    Formula:C10H11Cl2N3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:244.12

    Ref: TM-T10226

  • Bibn 99
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    Bibn 99

    CAS:
    <p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>
    Formula:C31H42ClN5O3
    Colore e forma:Solid
    Peso molecolare:568.15

    Ref: TM-T26799

  • SR 16584
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    SR 16584

    CAS:
    α3β4 nAChR antagonist
    Formula:C17H22N2O
    Purezza:99.84%
    Colore e forma:Solid
    Peso molecolare:270.37

    Ref: TM-T23388

  • VU 6008667
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    VU 6008667

    CAS:
    VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).
    Formula:C24H17ClF2N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:438.85

    Ref: TM-T13315

  • Rivanicline
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    Rivanicline

    CAS:
    Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.
    Formula:C10H14N2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:162.23

    Ref: TM-T12738L

  • Rapacuronium bromide
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    Rapacuronium bromide

    CAS:
    Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.
    Formula:C37H61BrN2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:677.8

    Ref: TM-T12690

  • ML375
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    ML375

    CAS:
    ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).
    Formula:C23H15ClF2N2O2
    Colore e forma:Solid
    Peso molecolare:424.83

    Ref: TM-T28068

  • CP-601927
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    CP-601927

    CAS:
    CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.
    Formula:C12H12F3N
    Colore e forma:Solid
    Peso molecolare:227.23

    Ref: TM-T31066

  • Arecaidine propargyl ester tosylate
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    Arecaidine propargyl ester tosylate

    CAS:
    Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.
    Formula:C17H21NO5S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:351.42

    Ref: TM-T22585