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Cellule staminali e Derivati

Cellule staminali e Derivati

Gli inibitori delle cellule staminali sono composti che bersagliano specificamente le vie di segnalazione e le proteine coinvolte nel mantenimento, nella differenziazione e nella proliferazione delle cellule staminali. Questi inibitori sono cruciali per comprendere la biologia delle cellule staminali e per sviluppare strategie per manipolare le cellule staminali a fini terapeutici, come la medicina rigenerativa e il trattamento del cancro. Controllando il destino delle cellule staminali, questi inibitori possono aiutare a guidare la differenziazione delle cellule staminali in tipi cellulari specifici o a prevenire una crescita cellulare indesiderata. Presso CymitQuimica, offriamo una selezione di inibitori delle cellule staminali di alta qualità per supportare la tua ricerca in biologia delle cellule staminali, biologia dello sviluppo e medicina rigenerativa.

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Trovati 693 prodotti di "Cellule staminali e Derivati"

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  • YAP-TEAD-IN-2

    CAS:
    <p>YAP-TEAD-IN-2 (compound 6) serves as a potent inhibitor of the YAP-TEAD protein-protein interaction (PPI), demonstrating an inhibitory concentration 50 (IC50)</p>
    Formula:C25H24ClFN2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:470.92
  • Tubulin/JAK2-IN-1

    CAS:
    <p>Tubulin/JAK2-IN-1 (compound 7g) serves as a potent dual inhibitor targeting both Janus kinase 2 (JAK2) and microtubules, demonstrating significant</p>
    Formula:C22H20N6O3
    Colore e forma:Solid
    Peso molecolare:416.43
  • QL-1200186

    CAS:
    <p>QL-1200186 is an orally active, selective TYK2 inhibitor that, upon dose-dependent oral administration, suppresses interferon-γ (IFNγ) production following</p>
    Formula:C26H27N7O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:485.54
  • JAK kinase-IN-1

    CAS:
    <p>JAK kinase-IN-1 (Example 1) functions as a potent inhibitor targeting the JAK family, which includes TYK2, JAK1, JAK2, and JAK3, with IC50 values of 4.2 nM, 32</p>
    Formula:C17H19F2N7OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:407.44
  • Yhhu-3792 hydrochloride

    CAS:
    <p>Yhhu-3792 hydrochloride is a compound that bolsters the self-renewal capacity of neural stem cells (NSCs), catalyzes the Notch signaling pathway, and upregulates expression of Hes3 and Hes5. It augments the NSC pool, stimulates endogenous neurogenesis in the mouse hippocampal dentate gyrus (DG), and enhances mice's spatial and episodic memory skills. This compound shows promise for researching learning and memory impairments linked to DG dysfunction [1].</p>
    Formula:C24H25ClN4O2
    Colore e forma:Solid
    Peso molecolare:436.93
  • Casein kinase 1δ-IN-4

    CAS:
    <p>"Casein kinase 1δ-IN-4 (compound 567) is a potent inhibitor of casein kinase 1δ with potential application in Alzheimer's disease research [1]."</p>
    Formula:C16H12N6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:320.37
  • STAT3-IN-B9

    CAS:
    <p>STAT3-IN-B9 (B9) is an inhibitor of abnormal STAT3 activation and inhibits the proliferation of tumor cells including MDA-MB-468, MDA-MB-231, and DU145.</p>
    Formula:C20H13NO5S
    Purezza:98.19%
    Colore e forma:Solid
    Peso molecolare:379.39
  • LX7101

    CAS:
    LX7101 is an effective inhibitor of LIMK and ROCK2 (IC50: 24, 1.6, and 10 nM for LIMK1, LIMK2, and ROCK2, respectively). It also inhibits PKA (IC50 <1 nM).
    Formula:C23H29N7O3
    Purezza:99.08%
    Colore e forma:Solid
    Peso molecolare:451.52
  • Myristoyl tetrapeptide-12

    CAS:
    <p>Myristoyl Tetrapeptide-12 activates SMAD2 and facilitates the association of SMAD3 with DNA, promoting eyelash hair growth [1] [2].</p>
    Formula:C32H63N7O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:625.89
  • ROCK-IN-7

    CAS:
    <p>ROCK-IN-7 (compound 9) serves as a ROCK kinase inhibitor and is utilized in the investigation of ocular conditions, including glaucoma and retinal diseases [1].</p>
    Formula:C17H17N3O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:327.4
  • BRD5648

    CAS:
    <p>BRD5648 ((R)-BRD0705) is an inactive (R)-enantiomer of BRD0705.</p>
    Formula:C20H23N3O
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:321.42
  • JAK-IN-26

    CAS:
    <p>JAK-IN-26 (compound 2) is an orally active inhibitor of the Janus kinase (JAK) enzyme with favorable pharmacokinetic properties, exhibiting potency in</p>
    Formula:C22H24N6O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:420.46
  • inS3-54A18

    CAS:
    <p>inS3-54A18 is an effective inhibitor of STAT3. inS3-54A18 has anticancer effects.</p>
    Formula:C23H16ClNO2
    Purezza:99.68%
    Colore e forma:Solid
    Peso molecolare:373.83
  • FM-479

    CAS:
    <p>FM-479, a structural analog of FM-381, lacks inhibition of JAK3/kinases within 100-300 nM, serving as FM-381's negative control.</p>
    Formula:C25H26N6O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:442.523
  • Casein kinase 1δ-IN-5

    CAS:
    <p>Casein kinase 1δ-IN-5 is a potent and selective CK-1δ inhibitor, exhibiting an IC50 of 47 nM, and demonstrates neuroprotective and anti-inflammatory effects in</p>
    Formula:C16H11F3N2OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:336.33
  • JW 67

    CAS:
    <p>JW 67 is an inhibitor of canonical Wnt pathway signaling.</p>
    Formula:C21H18N2O6
    Purezza:99.02%
    Colore e forma:Solid
    Peso molecolare:394.38
  • A 1070722

    CAS:
    <p>A 1070722: potent GSK-3 inhibitor, Ki = 0.6 nM for both α/β isoforms, crosses BBB, potential brain GSK-3 PET radiotracer.</p>
    Formula:C17H13F3N4O2
    Purezza:99.9%
    Colore e forma:Solid
    Peso molecolare:362.31
  • JAK-IN-31

    CAS:
    <p>JAK-IN-31 (Example 75), a JAK inhibitor, demonstrates IC50 values of ≤0.01 µM for JAK1, ≤0.01 µM for JAK2, 0.01-0.1 µM for JAK3, and ≤0.01 µM for Tyk2,</p>
    Formula:C21H19N7O2S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:465.55
  • 3,7-DMF

    CAS:
    3,7-Dimethylfumarate (3,7-DMF) serves as an oral inhibitor of transforming growth factor-beta 1 (TGF-β1)-mediated hepatic stellate cell (HSC) activation.
    Formula:C17H14O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:282.29
  • ROCK2-IN-2

    CAS:
    <p>ROCK2-IN-2 is a selective inhibitor of ROCK2 (IC50 of &lt;1 μM).</p>
    Formula:C18H12N6OS
    Purezza:99.65%
    Colore e forma:Solid
    Peso molecolare:360.39