Recettore degli oppioidi
I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.
Trovati 325 prodotti di "Recettore degli oppioidi"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Dynorphin B (1-13) acetate(83335-41-5 free base)
Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.Formula:C76H119N21O19Purezza:99.72%Colore e forma:SolidPeso molecolare:1630.89CTAP(TFA) (103429-32-9 free base)
CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.Formula:C53H70F3N13O13S2Purezza:99.62%Colore e forma:SolidPeso molecolare:1218.33Nociceptin (1-13) amide TFA
Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).Formula:C63H101F3N22O17Purezza:97.64%Colore e forma:SolidPeso molecolare:1495.61Ac-RYYRIK-NH2 acetate
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.Formula:C46H74N14O11Purezza:99.84%Colore e forma:SolidPeso molecolare:999.17[Met5]-Enkephalin, amide TFA
[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.Formula:C29H37F3N6O8SPurezza:99.81%Colore e forma:SolidPeso molecolare:686.7Leuphasyl TFA
CAS:Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.Formula:C31H40F3N5O9Purezza:98.79%Colore e forma:SolidPeso molecolare:683.67Ref: TM-T20435L
1mg81,00€2mg105,00€5mg168,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€Orphanin FQ(1-11) acetate(178249-41-7 free base)
Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.Formula:C51H79N15O16Purezza:95.54%Colore e forma:SolidPeso molecolare:1158.26N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.Formula:C30H39N5O8Purezza:>99.99%Colore e forma:SolidPeso molecolare:597.66b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.Formula:C25H31N3O7Purezza:98.99%Colore e forma:SolidPeso molecolare:485.53Ref: TM-T21660L
5mg42,00€10mg57,00€25mg87,00€50mg131,00€100mg190,00€200mg285,00€1mL*10mM (DMSO)55,00€Ac-RYYRWK-NH2 acetate
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.Formula:C51H73N15O11Purezza:98.59%Colore e forma:SolidPeso molecolare:1072.22Hemorphin-7 acetate(152685-85-3 free base)
Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.Formula:C51H68N12O13Purezza:99.66%Colore e forma:SolidPeso molecolare:1057.16Dynorphin A 1-10 acetate(79994-24-4 free base)
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.Formula:C59H95N19O14Purezza:99.88%Colore e forma:SolidPeso molecolare:1294.53[Leu5]-Enkephalin, amide acetate
[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.Formula:C30H42N6O8Purezza:99.36%Colore e forma:SolidPeso molecolare:614.69Nociceptin (1-7) acetate
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.Formula:C31H41N7O9Purezza:98.92%Colore e forma:SoildPeso molecolare:655.7Ref: TM-T23076L
1mg294,00€2mg439,00€5mg660,00€10mg999,00€25mg1.468,00€50mg1.998,00€100mg2.692,00€1mL*10mM (DMSO)897,00€AR-M 1000390 hydrochloride
CAS:ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.Formula:C23H29ClN2OPurezza:98.66%Colore e forma:SolidPeso molecolare:384.94Bisacodyl
CAS:Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.Formula:C22H19NO4Purezza:99.45% - 99.78%Colore e forma:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecolare:361.39BRL 52537 hydrochloride
CAS:BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.Formula:C18H25Cl3N2OPurezza:99.04%Colore e forma:SolidPeso molecolare:391.76Aticaprant
CAS:Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.Formula:C26H27FN2O2Purezza:99.9% - 99.97%Colore e forma:SolidPeso molecolare:418.5Ref: TM-TQ0082
1mg40,00€2mg52,00€5mg88,00€10mg126,00€25mg259,00€50mg406,00€100mg607,00€1mL*10mM (DMSO)87,00€BMS986188
CAS:BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.Formula:C30H31BrO4Purezza:98.76%Colore e forma:SolidPeso molecolare:535.47BW-180C
CAS:BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.Formula:C29H39N5O7Purezza:>99.99%Colore e forma:SolidPeso molecolare:569.65Ref: TM-TP1905
2mg39,00€5mg58,00€10mg93,00€25mg145,00€50mg260,00€100mg462,00€200mg655,00€1mL*10mM (DMSO)73,00€
![[Met5]-Enkephalin, amide TFA](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1254.webp&w=3840&q=75)
![[Leu5]-Enkephalin, amide acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1113L.webp&w=3840&q=75)
