
Recettore degli oppioidi
I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.
Trovati 326 prodotti di "Recettore degli oppioidi"
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MCOPPB triHydrochloride
CAS:MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.Formula:C26H43Cl3N4Purezza:99.89% - 99.91%Colore e forma:SolidPeso molecolare:518.01Ref: TM-T2071
2mg34,00€5mg50,00€10mg87,00€25mg163,00€50mg255,00€100mg375,00€200mg535,00€1mL*10mM (DMSO)58,00€Deltorphin I
CAS:Deltorphin I is an agonist of δ-opioid receptor.Formula:C37H52N8O10Purezza:>99.99%Colore e forma:SolidPeso molecolare:768.86Tyr-Gly-Gly-Phe-Met-OH
CAS:<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formula:C27H35N5O7SPurezza:≥95%Colore e forma:White Lyophilised SolidPeso molecolare:573.66Endomorphin 2
CAS:EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.Formula:C32H37N5O5Purezza:99.64%Colore e forma:SolidPeso molecolare:571.67EST73502 HCl
CAS:EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.Formula:C19H27ClF2N2O2Purezza:99.96%Colore e forma:SolidPeso molecolare:388.88Ref: TM-T39284
1mg92,00€5mg180,00€10mg258,00€25mg424,00€50mg598,00€100mg792,00€200mg1.074,00€1mL*10mM (DMSO)197,00€JTC-801
CAS:JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.Formula:C26H25N3O2·HClPurezza:99.27% - 99.59%Colore e forma:SolidPeso molecolare:447.96BMS-986122
CAS:BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1Formula:C16H15BrClNO3S2Purezza:98.42%Colore e forma:SolidPeso molecolare:448.78Ref: TM-T26869
1mg48,00€5mg96,00€10mg160,00€25mg311,00€50mg472,00€100mg658,00€200mg929,00€1mL*10mM (DMSO)96,00€Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Formula:C19H23NO4Purezza:99.02% - 99.73%Colore e forma:White PowderPeso molecolare:329.39ADL-5747 (HCl)
CAS:ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.Formula:C24H29ClN2O3Colore e forma:SolidPeso molecolare:428.95PZM21
CAS:<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Formula:C19H27N3O2SPurezza:99.93% - >99.99%Colore e forma:SolidPeso molecolare:361.5BMS986187
CAS:BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.Formula:C31H34O4Purezza:99.09%Colore e forma:SolidPeso molecolare:470.6GR103545
CAS:GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.Formula:C23H29Cl2N3O7Purezza:99.75%Colore e forma:SolidPeso molecolare:530.4Ref: TM-T9459
1mg87,00€2mg143,00€5mg188,00€10mg283,00€25mg509,00€50mg727,00€100mg1.017,00€1mL*10mM (DMSO)250,00€LY2795050
CAS:LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).Formula:C23H22ClN3O2Purezza:97.77%Colore e forma:SolidPeso molecolare:407.89Ref: TM-TQ0091
1mg52,00€2mg74,00€5mg116,00€10mg180,00€25mg298,00€50mgPrezzo su richiesta1mL*10mM (DMSO)127,00€DAMGO
CAS:DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.Formula:C26H35N5O6Purezza:98.83% - 99.92%Colore e forma:SolidPeso molecolare:513.59Ref: TM-T4351
1mg50,00€2mg60,00€5mg87,00€10mg140,00€25mg283,00€50mg423,00€100mg623,00€1mL*10mM (DMSO)88,00€Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).Formula:C50H72N15O15SPurezza:>99.99%Colore e forma:SolidPeso molecolare:1326.26Ref: TM-T7567L
1mg48,00€5mg125,00€10mg180,00€25mg325,00€50mg467,00€100mg645,00€200mg868,00€1mL*10mM (DMSO)187,00€[D-Ala2]leucine-enkephalin
CAS:[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.Formula:C29H39N5O7Purezza:98.06%Colore e forma:SolidPeso molecolare:569.65Difelikefalin acetate
CAS:Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.Formula:C38H57N7O8Purezza:99.55%Colore e forma:SolidPeso molecolare:739.9BAM 22P acetate
BAM 22P acetate is a potent opioid agonist.Formula:C132H188N38O33S2Purezza:99.87%Colore e forma:SoildPeso molecolare:2899.27Ref: TM-TP1211L
1mg105,00€5mg398,00€10mg595,00€25mg1.064,00€50mg1.434,00€100mg1.948,00€200mg2.622,00€Dynorphin A acetate(80448-90-4 free base)
Dynorphin A acetate is an Endogenous kappa receptor agonist.Formula:C101H159N31O25Purezza:99.69%Colore e forma:SolidPeso molecolare:2207.58(D-Ser2)-Leu-Enkephalin-Thr
(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.Formula:C33H46N6O10Purezza:94.17%Colore e forma:SoildPeso molecolare:686.75
