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Recettore degli oppioidi

Recettore degli oppioidi

I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.

Trovati 327 prodotti di "Recettore degli oppioidi"

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  • N-Desmethyl Loperamide
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    N-Desmethyl Loperamide

    CAS:
    N-Desmethyl Loperamide is the major metabolite of loperamide. It is also used as the precusor for radiolabelled loperamide.
    Formula:C28H31ClN2O2
    Colore e forma:Solid
    Peso molecolare:463.01

    Ref: TM-T33615

  • (Rac)-SNC80
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    (Rac)-SNC80

    CAS:
    (Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.
    Formula:C28H39N3O2
    Colore e forma:Solid
    Peso molecolare:449.63

    Ref: TM-T73631

  • Nocistatin
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    Nocistatin

    CAS:
    Nocistatin, a neuropeptide, blocks Nociceptin effects and inhibits 5-HT release, acting on an opioid-related receptor.
    Formula:C32H56N10O12
    Colore e forma:Solid
    Peso molecolare:772.85

    Ref: TM-T76420

  • β-Naltrexamine dihydrochloride
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    β-Naltrexamine dihydrochloride

    CAS:
    β-Naltrexamine dihydrochloride is an orally administered, irreversible opioid receptor antagonist. Its derivatives exhibit optimised subtype selectivity and can be used for pain research.
    Formula:C20H28Cl2N2O3
    Purezza:95.98%
    Colore e forma:Soild
    Peso molecolare:415.35

    Ref: TM-T204075L

  • BAM-22P
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    BAM-22P

    CAS:
    Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.
    Formula:C130H184N38O31S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:2839.22

    Ref: TM-TP1211

  • β-Endorphin, equine
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    β-Endorphin, equine

    CAS:
    Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.
    Formula:C154H248N42O44S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3423.94

    Ref: TM-TP1647

  • SNC 80
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    SNC 80

    CAS:
    SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.
    Formula:C28H39N3O2
    Purezza:99.65%
    Colore e forma:Solid
    Peso molecolare:449.63

    Ref: TM-T8414

  • [Nphe1]Nociceptin(1-13)NH2
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    [Nphe1]Nociceptin(1-13)NH2

    CAS:
    <p>Competitive nociceptin receptor antagonist with pKi=8.4; no agonist activity; blocks nociceptin effects in vitro/in vivo.</p>
    Formula:C61H100N22O15
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1381.6

    Ref: TM-TP1987

  • Clocinnamox mesylate
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    Clocinnamox mesylate

    CAS:
    Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).
    Formula:C30H33ClN2O7S
    Colore e forma:Solid
    Peso molecolare:601.11

    Ref: TM-T41184

  • U-54494A hydrochloride
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    U-54494A hydrochloride

    CAS:
    U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.
    Formula:C18H25Cl3N2O
    Colore e forma:Solid
    Peso molecolare:391.76

    Ref: TM-T36372

  • ICI 174,864
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    ICI 174,864

    CAS:
    <p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>
    Formula:C38H53N5O7
    Purezza:98%
    Colore e forma:White Solid
    Peso molecolare:691.87

    Ref: TM-TP2013

  • Gluten Exorphin B5
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    Gluten Exorphin B5

    CAS:
    Gluten exorphin B5 (GE-B5) is a food-derived opioid peptide identified in digests of wheat gluten.
    Formula:C30H38N6O7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:594.66

    Ref: TM-TP1815

  • Herkinorin
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    Herkinorin

    CAS:
    Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.
    Formula:C28H30O8
    Colore e forma:Solid
    Peso molecolare:494.53

    Ref: TM-T27534

  • Dermorphin
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    Dermorphin

    CAS:
    <p>Dermorphin is agonist of μ-opioid receptor (MOR) agonist.</p>
    Formula:C40H50N8O10
    Purezza:98.82%
    Colore e forma:Solid
    Peso molecolare:802.87

    Ref: TM-T7404

  • Orphanin FQ(1-11)
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    Orphanin FQ(1-11)

    CAS:
    <p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>
    Formula:C49H75N15O14
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1098.2

    Ref: TM-TP1882

  • Dynorphin B (1-13)
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    Dynorphin B (1-13)

    CAS:
    Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.
    Formula:C74H115N21O17
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1570.84

    Ref: TM-TP1826

  • Ro 64-6198
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    Ro 64-6198

    CAS:
    Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.
    Formula:C26H31N3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:401.54

    Ref: TM-T16772

  • CTAP
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    CTAP

    CAS:
    Potent μ opioid antagonist, IC50 3.5 nM, 1200x selectivity over δ and somatostatin, brain-penetrant, active in vivo.
    Formula:C51H69N13O11S2
    Purezza:98%
    Colore e forma:White Solid/Powder
    Peso molecolare:1104.32

    Ref: TM-TP2050

  • UFP-101
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    UFP-101

    CAS:
    <p>Strong, selective NOP receptor antagonist with pKi=10.24; &gt;3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>
    Formula:C82H138N32O21
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1908.19

    Ref: TM-TP2105

  • Logo CymitQuimica
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    Helianorphin-19

    <p>Helianorphin-19: Potent KOR agonist (Ki=25 nM; EC50=45 nM), 200x selective over μ/δ receptors, effective in mouse pain model, non-sedative.</p>
    Colore e forma:Liquid

    Ref: TM-T41183