Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.811 prodotti)
- Apoptosi(6.295 prodotti)
- Ciclo cellulare/Checkpoint(4.842 prodotti)
- Cromatina/Epigenetica(2.526 prodotti)
- Segnalazione citoscheletrica(1.550 prodotti)
- Danno al DNA/Riparazione del DNA(2.917 prodotti)
- Endocrinologia/Ormoni(3.708 prodotti)
- Enzima(3.671 prodotti)
- Proteina G/GPCR(9.024 prodotti)
- Immunologia e infiammazione(3.896 prodotti)
- Virus dell'influenza(302 prodotti)
- Segnalazione JAK/STAT(418 prodotti)
- Segnalazione MAPK(1.248 prodotti)
- Trasportatore di membrana/canale ionico(3.094 prodotti)
- Metabolismo(10.157 prodotti)
- Microbiologia/Virologia(7.623 prodotti)
- Neuroscienza(10.360 prodotti)
- Altri inibitori(35.913 prodotti)
- Ossidazione-riduzione(40 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.440 prodotti)
- Proteasi/Proteasoma(1.711 prodotti)
- Cellule staminali e Derivati(792 prodotti)
- Adattatori Tirosin-chinasi(2.013 prodotti)
- Ubiquitinazione(1.722 prodotti)
Mostrare 16 più sottocategorie
Trovati 66619 prodotti di "Inibitori"
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Purine phosphoribosyltransferase-IN-2
Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.Formula:C11H15N5Na4O10P2Colore e forma:SolidPeso molecolare:531.17Antitubercular agent-13
Compound 3d: antitubercular, MIC 0.007 μg/mL vs MTB H37Rv, 1.851 μg/mL vs MDR-MTB 16833, metabolically unstable.Formula:C18H18N4O5Colore e forma:SolidPeso molecolare:370.36Marizomib
CAS:Marizomib is a novel irreversible brain-permeable proteasome inhibitor that inhibits CT-L, CT-T-laspase-like, and trypsin-like 20S proteasomes.Cost-effective and quality-assured.Formula:C15H20ClNO4Purezza:98.03% - 99.41%Colore e forma:SolidPeso molecolare:313.78ONO-5334
CAS:ONO-5334: selective cathepsin K inhibitor, potential for osteoporosis study; Ki: 0.10 nM (human), 0.049 nM (rabbit), 0.85 nM (rat).Formula:C21H34N4O4SPurezza:98.22% - 99.60%Colore e forma:SolidPeso molecolare:438.58Alentemol hydrobromide
CAS:Alentemol hydrobromide is a Dopamine agonist.Formula:C19H26BrNOPurezza:98%Colore e forma:SolidPeso molecolare:364.32YM158 free base
CAS:YM158 free base is a potent and selective antagonist of TXA2 and LTD4 receptor (pA2s: about 8.81 and 8.87).Formula:C32H33ClN6O5S2Purezza:98%Colore e forma:SolidPeso molecolare:681.22JTZ-951 HCl
CAS:JTZ-951 is a potent and orally active inhibitor of hypoxia inducible factor prolyl hydroxylase (PHD).Formula:C17H17ClN4O4Purezza:98%Colore e forma:SolidPeso molecolare:376.79(1R,3S)-THCCA-Asn
(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.Formula:C24H24N4O6Colore e forma:SolidPeso molecolare:464.47L 691816
CAS:L 691816 is an effective inhibitor of the 5-LO reaction.Formula:C36H35ClN6OSPurezza:98%Colore e forma:SolidPeso molecolare:635.22Sekikaic Acid
CAS:Sekikaic acid, a phenolic lichen metabolite in H. obscurata, has antioxidant and antiviral properties, inhibiting MLL1-CBP.Formula:C22H26O8Colore e forma:SolidPeso molecolare:418.44Antitumor agent-78
Antitumor agent-78 blocks GPx-4, raises COX2, triggers apoptosis, halts EMT, and stifles cancer cell growth and migration.Colore e forma:SoildLp-PLA2-IN-6
CAS:Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.Formula:C25H21F5N4O3Colore e forma:SolidPeso molecolare:520.45BILA 1906 BS
CAS:BILA 1906 BS is an inhibitor of substrate analog protease.Formula:C41H52N6O4SPurezza:98%Colore e forma:SolidPeso molecolare:724.95Cilengitide hydrochloride
CAS:Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.Formula:C27H41ClN8O7Colore e forma:SolidPeso molecolare:625.12Hit 1
Hit 1 is an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 μM) and reduces glucose-stimulated insulin secretion.Formula:C22H24N4O3S2Colore e forma:SolidPeso molecolare:456.58WF-47-JS03
WF-47-JS03: RET kinase inhibitor, crosses blood-brain barrier, 500x more selective for KDR, IC50: 1.7 nM in Ba/F3 cells, 5.3 nM in LC-2/ad lung cancer cells.
Formula:C30H38N6O2Colore e forma:SolidPeso molecolare:514.66AM9405
AM9405: peripheral CB1/5-HT3 agonist, suppresses gut motility, relieves GI disorder symptoms in mice.Formula:C24H33BrN2O2Purezza:98%Colore e forma:SolidPeso molecolare:461.44(Rac)-Plevitrexed
CAS:(Rac)-Plevitrexed is a racemate of Plevitrexed. Plevitrexed is an orally active and potent inhibitor of thymidylate synthase (TS).Formula:C26H25FN8O4Purezza:98%Colore e forma:SolidPeso molecolare:532.53NITD-688
CAS:NITD-688 is a pan-serotype inhibitor targeting the dengue virus NS4B protein, effective through oral administration.Formula:C25H32N4O3S2Colore e forma:SolidPeso molecolare:500.68BMS-901715
CAS:BMS-901715 is an effective and selective inhibitor of adapter protein-2 associated kinase 1 (AAK1; IC50: 3.3 nM).Formula:C22H28N10OPurezza:98%Colore e forma:SolidPeso molecolare:448.52Cdc7-IN-19
CAS:Cdc7-IN-19 (compound 1-1) is a potent CDC7 inhibitor with an IC 50 of 1.49 nM [1].Formula:C19H21N5O2Colore e forma:SolidPeso molecolare:351.40GGTI298
CAS:GGTI298 is a potent GGTase I inhibitor; IC50 3μM for Rap1A, >20μM for Ha-Ras.Formula:C27H33N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:479.63Antitumor agent-47
Antitumor agent-47, a silibinin derivative, shows cytotoxicity in NCI-H1299 (IC50: 8.07µM) and HT29 (IC50: 6.27µM) cells.Formula:C30H27NO11Colore e forma:SolidPeso molecolare:577.54Anticancer agent 12
Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.Formula:C16H17BrN4O2SColore e forma:SolidPeso molecolare:409.34-Bromo A23187
CAS:4-Bromo A23187 is a halogenated analog of the calcium ionophore A-23187. 4-Bromo A23187 is a calcium modulator and induces apoptosis in different cells.Formula:C29H36BrN3O6Purezza:98%Colore e forma:SolidPeso molecolare:602.52Ro-51
CAS:dual P2X3 and P2X2/3 antagonistFormula:C17H23IN4O4Purezza:98%Colore e forma:SolidPeso molecolare:474.29METTL3-IN-2
CAS:METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.Formula:C25H26N8OColore e forma:SolidPeso molecolare:454.53GDC-0927 Racemate
CAS:GDC-0927 Racemate is a degrader of estrogen receptor, is used in the research of ER-related diseases, potently inhibits ER-α activity, with an IC50 of 0.2 nM.Formula:C28H28FNO4Purezza:98%Colore e forma:SolidPeso molecolare:461.52DNA-PK-IN-2
CAS:DNA-PK-IN-2 is an inhibitor of the DNA-PK enzyme complex, useful in cancer research.Formula:C20H23N5O3Colore e forma:SolidPeso molecolare:381.43Anticancer agent 36
Compound 11: Sulfonylurea derivative, antimicrobial, anticancer; MIC 0.039-0.156 mg/mL; A549 IC50: 19.7 μg/mL, PC3 IC50: 11.9 μg/mL.Formula:C21H17N3O3S2Colore e forma:SolidPeso molecolare:423.51Esorubicin
CAS:Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.Formula:C27H29NO10Colore e forma:SolidPeso molecolare:527.52Mu opioid receptor antagonist 2
Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.Formula:C25H28N2O4SColore e forma:SolidPeso molecolare:452.57Asimicin
CAS:Asimicin is a effective complex I inhibitor.Formula:C37H66O7Purezza:98%Colore e forma:SolidPeso molecolare:622.92Mibefradil
CAS:Mibefradil is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels (IC50s: 2.7 μM and 18.6 μM for T-type and L-type currents).Formula:C29H38FN3O3Purezza:98%Colore e forma:SolidPeso molecolare:495.63FXIa-IN-8
FXIa-IN-8: potent FXIa blocker (IC50: 14.2 nM), anti-thrombotic, low bleeding/toxicity risk.Colore e forma:SolidFuraprevir
CAS:Furaprevir is an HCV NS3/4A InhibitorFormula:C47H56N6O10SColore e forma:SolidPeso molecolare:897.05TRPV1 antagonist 3
TRPV1 antagonist 3 (7q) strongly blocks TRPV1 at 2.66 nM IC50, is selective, 60% bioavailable, and crosses the blood-brain barrier.Formula:C23H25N3OSColore e forma:SolidPeso molecolare:391.53SCO-792
SCO-792: potent, reversible oral enteropeptidase inhibitor, with slow in vitro dissociation and in vivo protein digestion blocking.Formula:C22H22N4O8·xH2OColore e forma:SolidJAK3/BTK-IN-3
CAS:JAK3/BTK-IN-3: strong dual JAK3/BTK suppressor, promising for autoimmune disease research.Formula:C22H28N8OColore e forma:SolidPeso molecolare:420.51α-Amylase-IN-1
CAS:α-Amylase-IN-1 is an α-Amylase inhibitor (IC50: 0.5509 μM).Formula:C18H18N2O3Purezza:99.92%Colore e forma:SoildPeso molecolare:310.35c-Myc inhibitor 4
Potent oral c-Myc inhibitor 4 reduces the proto-oncogene linked to tumor development.Formula:C26H33FN6O3Colore e forma:SolidPeso molecolare:496.58MM-589 TFA
CAS:MM-589 TFA is a potent WD repeat domain 5 (WDR5)inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.Formula:C30H45F3N8O7Purezza:98%Colore e forma:SolidPeso molecolare:686.72BACE1-IN-2
CAS:BACE1-IN-2 is a BACE1 inhibitor (IC50: 22 nM).Formula:C19H15F4N5O2Purezza:98%Colore e forma:SolidPeso molecolare:421.35TRβ agonist 1
CAS:TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.Formula:C29H25FN2O8Colore e forma:SolidPeso molecolare:548.52Methysergide maleate
CAS:Methysergide prevents migraines/cluster headaches; treats serotonin syndrome, carcinoid-induced diarrhea; risk of fibrosis limits use.Formula:C25H31N3O6Purezza:98%Colore e forma:White To Off-WhitePeso molecolare:469.54Asukamycin
CAS:Asukamycin, from S. nodosus asukaensis, is a polyketide antibiotic inhibiting tumor cells by activating caspases 8 and 3.Formula:C31H34N2O7Colore e forma:SolidPeso molecolare:546.61AFM-30a hydrochloride
AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.Formula:C24H28ClFN6O3Colore e forma:SolidPeso molecolare:502.97EGFR-IN-38
CAS:EGFR-IN-38: low-toxic acrylamide-derived EGFR inhibitor, targets NSCLC, patented for research on EGFR mutation-related diseases.Formula:C25H24ClN7O2Colore e forma:SolidPeso molecolare:489.96EGFR-IN-58
EGFR-IN-58 is a potent, selective, ATP-competitive inhibitor of EGFR. EGFR-IN-58 exhibits significant cytotoxicity against melanoma, colon and blood cancers.Formula:C31H30FN7OColore e forma:SolidPeso molecolare:535.61Human carbonic anhydrase II-IN-1
Compound S-13: Potent hCA II inhibitor, Kis 4.4, 9.2, 480.2, 14.7 nM for hCA II, I, IV, IX. Used in glaucoma research.Formula:C20H25N3O4SColore e forma:SolidPeso molecolare:403.5MtTMPK-IN-1
MtTMPK-IN-1 inhibits MtTMPK with 2.5 μM IC50, shows moderate anti-tuberculosis activity, and is low in cytotoxicity.Formula:C22H24N4O3Colore e forma:SolidPeso molecolare:392.45Rodatristat
CAS:Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).Formula:C27H27ClF3N5O3Purezza:98%Colore e forma:SolidPeso molecolare:561.98PF-03715455
CAS:PF-03715455 is a potent p38 MAPK inhibitor, reducing TNFα in blood (IC50=1.7 nM) with selectivity for p38α, and may treat COPD.Formula:C35H34ClN7O3S2Purezza:98%Colore e forma:SolidPeso molecolare:700.27Agosterol A
CAS:Agosterol A is isolated from marine sponge Spongia.Formula:C33H52O8Colore e forma:SolidPeso molecolare:576.76TDI-11861
CAS:TDI-11861 is a second-gen sAC (ADCY10) inhibitor with an IC50 of 5.5 nM and slow dissociation.Formula:C22H25ClF2N6O3Colore e forma:SolidPeso molecolare:494.92HDAC6-IN-13
HDAC6-IN-13: potent, selective HDAC6 inhibitor; oral; IC50=0.019μM; targets HDAC1/2/3; crosses blood-brain barrier; anti-inflammatory.Formula:C23H22N4OColore e forma:SolidPeso molecolare:370.45U91356
CAS:U91356 is an agonist of the dopamine receptors.Formula:C13H17N3OPurezza:98%Colore e forma:SolidPeso molecolare:231.29ADP-2341
ADP-2341 is a soluble analog of FiVe1.Formula:C24H29Cl2N5O3Colore e forma:SolidPeso molecolare:506.43J-113397
CAS:J-113397 is a potent and selective NOP receptor antagonist (IC50 = 2.3 nM).Formula:C24H37N3O2Purezza:98%Colore e forma:SolidPeso molecolare:399.57CDK9-IN-13
CDK9-IN-13 is a potent and selective CDK inhibitor (IC50<3 nM). CDK9-IN-13 has a very short half-life in rodents.Formula:C27H35N5O2Colore e forma:SolidPeso molecolare:461.6Gabaculine HCl
CAS:Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.Formula:C7H10ClNO2Colore e forma:SolidPeso molecolare:175.61VDR agonist 1
CAS:Compound 28 is a nonsteroidal VDR agonist with 690 nM potency, inducing cell cycle arrest and apoptosis in MCF-7 cells.Formula:C32H51N3O2Purezza:98%Colore e forma:SolidPeso molecolare:509.77JAK3-IN-11
CAS:JAK3-IN-11: potent oral JAK3 inhibitor (IC50=1.7 nM), noncytotoxic, >588-fold selectivity, blocks T-cell growth; useful in autoimmune research.Formula:C23H23N5O2Colore e forma:SolidPeso molecolare:401.46Sesamodil
CAS:Sesamodil (SD 3211) is a novel calcium antagonist that can be used to study hypertension.Formula:C29H32N2O6SPurezza:98.87% - 99.87%Colore e forma:SolidPeso molecolare:536.64Tubulin polymerization-IN-4
CAS:Tubulin polymerization-IN-4: inhibits tubulin (IC50=4.6 μM), blocks G2/M phase, induces apoptosis, hinders cell cloning/migration, damages vasculature.Formula:C21H21ClN2O4Colore e forma:SolidPeso molecolare:400.86ATX inhibitor 12
Oral ATX inhibitor 12 (IC50: 1.72 nM) at 60 mg/kg prevents lung damage in C57Bl/6J mice.
Formula:C30H34FN5O2Colore e forma:SolidPeso molecolare:515.62AAK1-IN-2 TFA
AAK1-IN-2 TFA (compound (S)-31) is a selective and potent AAK1 inhibitor (IC50: 5.8 nM) that can cross the blood-brain barrier.Formula:C24H22F6N4O4Colore e forma:SolidPeso molecolare:544.45ErSO-DFP
ErSO-DFP activates a-UPR, targets ERα+ cancer cells with high selectivity, and effectively reduces MCF-7 tumours.Formula:C20H17F5N2O2Colore e forma:SolidPeso molecolare:412.35PSB 36
CAS:A1 adenosine receptor antagonistFormula:C21H30N4O3Purezza:98%Colore e forma:SolidPeso molecolare:386.49CYP1B1-IN-2
CYP1B1-IN-2 (compound 9j) is a highly potent and selective inhibitor of CYP1B1, a cytochrome P450 enzyme. It exhibits an IC50 value of 0.52 nM [1].Formula:C20H11F3O2Colore e forma:SolidPeso molecolare:340.3DSM705 hydrochloride
DSM705 hydrochloride: potent antimalarial, pyrrole-based DHODH inhibitor effective against Plasmodium, non-toxic to mammalian DHODH.Formula:C19H20ClF3N6OColore e forma:SolidPeso molecolare:440.85Antiallergic agent-1
Antiallergic agent-1, an Src family kinase inhibitor, is a new and valuable lead compound with potential as an anti-allergic agent.Formula:C27H19F6N5OColore e forma:SolidPeso molecolare:543.46RdRP-IN-4
RdRP-IN-4, an oral arylbenzohydrazide, inhibits influenza A/B by targeting PB1 of RdRP, with EC50s of 53 nM (H1N1) and 20 nM (Flu B), and aids infected mice.Formula:C17H17Br2N3O2Colore e forma:SolidPeso molecolare:455.14hCAIX/XII-IN-5
Coumarin 9a: Selective inhibitor of hCA IX/XII (Ki 93.3/85.7 nM), blocks cancer cell growth, and induces apoptosis.Formula:C18H13NO3Colore e forma:SolidPeso molecolare:291.3ND-2158
CAS:ND-2158 is a potent and selective inhibitor of IRAK4.Formula:C22H30N4O4SPurezza:98%Colore e forma:SolidPeso molecolare:446.56L 689065
CAS:L 689065 is a 5-lipoxygenase inhibitor.Formula:C35H33ClN2O3SPurezza:98%Colore e forma:SolidPeso molecolare:597.17Cav 3.2 inhibitor 3
Cav 3.2 inhibitor 3 is a potent inhibitor of the Cav3.2 T-type Ca2+channel (IC50: 0.1534 μM) and has a low binding affinity for D2 receptors.Formula:C32H37N3O2Colore e forma:SolidPeso molecolare:495.66MMAF sodium
CAS:MMAF sodium, a potent tubulin inhibitor in ADCs like Vorsetuzumab mafodotin and SGN-CD19A, acts as an antitumor agent.Formula:C39H64N5NaO8Purezza:98%Colore e forma:SolidPeso molecolare:753.94TRK-IN-19
TRK-IN-19 (I-10) inhibits TRKA (1.1 nM IC50) & TRKAG595R (5.3 nM), promising for cancer research.Formula:C22H26FN5O2Colore e forma:SolidPeso molecolare:411.47MK-8876
CAS:MK-8876 is an Inhibitor of HCV NS5B Site D.Formula:C32H24F2N4O5SPurezza:98%Colore e forma:SolidPeso molecolare:614.62HIF-1/2α-IN-1
HIF-1/2α-IN-1, an orally active compound, functions as an inhibitor of HIF-2α.Formula:C17H16N6O4Colore e forma:SolidPeso molecolare:368.35Monoamine oxidase/Aromatase-IN-1
Compound 2q: Dual MAO/aromatase inhibitor; IC50: 39 nM (MAO-B), 31 nM (aromatase). Useful in neurological/breast cancer research.Formula:C19H19N3O3SColore e forma:SolidPeso molecolare:369.44MDL-43291
CAS:MDL-43291 is a leukotriene receptor antagonist.Formula:C25H42O4SColore e forma:SolidPeso molecolare:438.66BNTX maleate
CAS:δ1 opioid receptor antagonistFormula:C31H31NO8Purezza:98%Colore e forma:SolidPeso molecolare:545.58TrxR-IN-2
TrxR-IN-2 is a potential thioredoxin reductase (TrxR) inhibitor. TrxR-IN-2 has research value in the chemotherapy of drug-resistant hepatocellular carcinoma.Formula:C22H22N4O4Colore e forma:SolidPeso molecolare:406.43Topo I-IN-1
Topo I-IN-1 (14d) is a powerful Topo I inhibitor with antitumor effects and DNA intercalation, inducing apoptosis.Formula:C20H14BrN3O2Colore e forma:SolidPeso molecolare:408.25Antitumor agent-37
Antitumor agent-37: strong anti-growth, anti-spread, induces DNA damage, apoptosis via Bcl-2/Bax/caspase3, boosts immune response.Formula:C16H18Cl2N2O4PtColore e forma:SolidPeso molecolare:568.32Butaprost
CAS:Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.Formula:C24H40O5Purezza:98%Colore e forma:SolidPeso molecolare:408.57MRTX849 ethoxypropanoic acid
CAS:MRTX849 is a KRAS G12C ligand and PROTAC linker for creating potent LC-2, degrading KRAS G12C with DC50 of 0.25-0.76 μM.Formula:C37H43ClFN7O5Colore e forma:SolidPeso molecolare:720.24Laulimalide
CAS:Microtubule stabilizer; halts cancer cell growth (IC50: 3-30 nM); arrests cells in prometaphase; prevents bipolar spindle formation.Formula:C30H42O7Colore e forma:SolidPeso molecolare:514.65BTK-IN-10
CAS:BTK-IN-10 is a potent inhibitor of BTK, acting on wild-type BTK (IC50<5 nM) or mutant BTK (C481S) (IC50<5 nM).Formula:C25H24F2N4O2Colore e forma:SolidPeso molecolare:450.48KP 10614
CAS:KP 10614 is a new prostacyclin analog that inhibits platelet-polymorphonuclear leukocyte interaction.Formula:C23H32O4Colore e forma:SolidPeso molecolare:372.50SB-612111
CAS:SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.Formula:C24H29Cl2NOColore e forma:SolidPeso molecolare:418.40Antioxidant agent-8
Antioxidant agent-8, an oral Aβ 1-42 inhibitor, reduces fibril aggregation & promotes disaggregation; it's neuroprotective & BBB permeable.Formula:C13H12O5Colore e forma:SolidPeso molecolare:248.23Bim-IN-1
Bim-IN-1 is a potent inhibitor of Bim expression with low toxicity, Bim-IN-1 reduces Bim expression levels with little inhibition of protein kinase A.Formula:C19H20Cl2FNO2SColore e forma:SolidPeso molecolare:416.34PSMA-1007
CAS:PSMA-1007 is a novel Glu-Ureido-type prostate-specific membrane antigen (PSMA) inhibitor.Formula:C49H55FN8O16Colore e forma:SolidPeso molecolare:1030.01Glutaminyl Cyclase Inhibitor 3
CAS:Designed anti-Alzheimer’s compound; potent Glutaminyl Cyclase inhibitor; IC50 at 4.5 nM; reduces brain Aβ; improves cognition.Formula:C24H32N6O2SPurezza:98%Colore e forma:SolidPeso molecolare:468.61Antitumor agent-58
Antitumor agent-58 suppresses tumor growth, colony formation, cell migration, and induces mitochondrial dysfunction in MGC-803 cells.Formula:C27H28F3N9SColore e forma:SolidPeso molecolare:567.63Elocalcitol
CAS:Elocalcitol is a calcitriol analog for inhibition of prostate cell growth.Formula:C29H43FO2Colore e forma:SolidPeso molecolare:442.65Antibacterial synergist 1
Compound 20P is a potent antibacterial, inhibits biofilms with IC50 4.5 μM, and reduces pyocyanin at IC50 8.6 μM.Formula:C19H24N2O4Colore e forma:SolidPeso molecolare:344.4
