Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.715 prodotti)
- Apoptosi(6.164 prodotti)
- Ciclo cellulare/Checkpoint(4.727 prodotti)
- Cromatina/Epigenetica(2.400 prodotti)
- Segnalazione citoscheletrica(1.492 prodotti)
- Danno al DNA/Riparazione del DNA(2.928 prodotti)
- Endocrinologia/Ormoni(3.653 prodotti)
- Enzima(3.661 prodotti)
- Proteina G/GPCR(8.861 prodotti)
- Immunologia e infiammazione(3.801 prodotti)
- Virus dell'influenza(299 prodotti)
- Segnalazione JAK/STAT(412 prodotti)
- Segnalazione MAPK(1.239 prodotti)
- Trasportatore di membrana/canale ionico(2.979 prodotti)
- Metabolismo(10.029 prodotti)
- Microbiologia/Virologia(7.445 prodotti)
- Neuroscienza(10.281 prodotti)
- Altri inibitori(36.478 prodotti)
- Ossidazione-riduzione(44 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.443 prodotti)
- Proteasi/Proteasoma(1.695 prodotti)
- Cellule staminali e Derivati(829 prodotti)
- Adattatori Tirosin-chinasi(2.035 prodotti)
- Ubiquitinazione(1.693 prodotti)
Mostrare 16 più sottocategorie
Trovati 66676 prodotti di "Inibitori"
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BMS-986163
CAS:BMS-986163, a prodrug, quickly becomes BMS-986169, a GluN2B inhibitor (Ki=4 nM, IC50=24 nM).Formula:C23H28FN2O5PPurezza:98%Colore e forma:SolidPeso molecolare:462.45PF-06380101
CAS:PF-06380101, a potent auristatin analog and Dolastatin 10 derivative, shows strong anti-tumor activity and unique ADME attributes.Formula:C39H62N6O6SPurezza:98%Colore e forma:SolidPeso molecolare:743.01Samuraciclib
CAS:Samuraciclib (CT7001) is an oral CDK7 inhibitor with 41 nM IC50, notable for its high selectivity and potency against breast cancer cells.Formula:C22H30N6OColore e forma:SolidPeso molecolare:394.51Idraparinux Na
CAS:Idraparinux Na is an Antithrombotic, Indirect, Selective, Synthetic Factor Xa InhibitorFormula:C38H55Na9O49S7Colore e forma:SolidPeso molecolare:1727.14KUSC-5037
KUSC-5037 inhibits HIF-1 (IC50 = 1.2 μM) and mitochondrial complex V/FoF1ATP synthase.Formula:C18H17F3N6O2Colore e forma:SolidPeso molecolare:406.13651TLR7/8 agonist 7
CAS:<p>TLR7/8 agonist 7 activates immune cells, useful in ISAC synthesis and immunity research.</p>Formula:C26H37N7O2Colore e forma:SolidPeso molecolare:479.62AMG-315
CAS:AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.Formula:C24H41NO2Colore e forma:SolidPeso molecolare:375.59KMH-233
CAS:KMH-233 effectively blocks LAT1, inhibiting L-leucine uptake and cell growth, boosting betastatin and cisplatin efficacy at 25 μM.Formula:C32H25N7O5Colore e forma:SolidPeso molecolare:587.58PqsR-IN-1
PqsR-IN-1, potent PqsR inhibitor, curbs pyocyanin in Pseudomonas aeruginosa with low cytotoxicity.Formula:C17H18ClN3OSColore e forma:SolidPeso molecolare:347.86IRAK4-IN-15
CAS:IRAK4-IN-15: selective IRAK4 inhibitor, IC50 0.002 μM, good PK, low clearance, synergizes with Acalabrutinib in MyD88/CD79 mutant ABC-DLBCL.Formula:C25H29FN10Colore e forma:SolidPeso molecolare:488.562R,4R-Sacubitril
CAS:2R,4R-Sacubitril is the impurity of Sacubitril. Sacubitril is used in combination with valsartan for the treatment of patients with heart failure.Formula:C24H29NO5Purezza:98%Colore e forma:SolidPeso molecolare:411.49EGFR/BRAF-IN-1
<p>EGFR/BRAF-IN-1 inhibits EGFR/BRAF (BRAFV600E IC50: 45 nM, GI50: 35 nM) and has antioxidant properties.</p>Formula:C26H28ClN3O4Colore e forma:SolidPeso molecolare:481.97Leualacin
CAS:Leualacin is a novel calcium blocker from Hapsidospora irregularis.Formula:C31H47N3O7Purezza:98%Colore e forma:SolidPeso molecolare:573.72LY 215890
CAS:LY 215890 is a compound that exhibits potent Gram-negative and Gram-positive antibacterial activity.Formula:C13H12ClN5O5SPurezza:98%Colore e forma:SolidPeso molecolare:385.78PTP1B-IN-21
PTP1B-IN-21 inhibits PTP1B (IC50=1.56μM) selectively over TCPTP, a type 2 diabetes target.Formula:C22H22O11Colore e forma:SolidPeso molecolare:462.4Elacestrant S enantiomer dihydrochloride
Elacestrant (RAD1901) dihydrochloride, an oral ERR degrader, has IC50 of 48 nM (ERα) and 870 nM (ERβ). Its S enantiomer has low activity.Formula:C30H40Cl2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:531.56Alkyne-probe 1
Alkyne-probe 1 is usually used as an Alkyne-labeled fluorescent or chemical probe.Formula:C14H23N5O2Purezza:98%Colore e forma:SolidPeso molecolare:293.36Glycyl H-1152 hydrochloride
CAS:<p>Glycyl-H-1152 is a potent ROCK-II inhibitor (IC50=11.8 nM) with high selectivity over CaMKII, PKG, Aurora A, PKA, and PKC. Better than Y-27632 and HA-1077.</p>Formula:C18H26Cl2N4O3SColore e forma:SolidPeso molecolare:449.39PqsR-IN-2
PqsR-IN-2, potent PqsR inhibitor, curbs Pseudomonas aeruginosa communication, reduces pyocyanin, with low toxicity.Formula:C18H20ClN3OSColore e forma:SolidPeso molecolare:361.89Monoamine oxidase/Aromatase-IN-1
Compound 2q: Dual MAO/aromatase inhibitor; IC50: 39 nM (MAO-B), 31 nM (aromatase). Useful in neurological/breast cancer research.Formula:C19H19N3O3SColore e forma:SolidPeso molecolare:369.44L 689065
CAS:L 689065 is a 5-lipoxygenase inhibitor.Formula:C35H33ClN2O3SPurezza:98%Colore e forma:SolidPeso molecolare:597.17HER2-IN-6
CAS:<p>HER2-IN-6, a potent HER2 inhibitor, may target wild/mutant EGFR and HER2-mediated tumors. (Patent WO2021164697A1, compound 11)</p>Formula:C26H32N8O3Colore e forma:SolidPeso molecolare:504.58Mifepristone methochloride
CAS:<p>Mifepristone methochloride is a glucocorticoid antagonist. This product will be sold for research use only.</p>Formula:C30H38ClNO2Colore e forma:SolidPeso molecolare:480.08264W94
CAS:264W94 robustly inhibits IBAT, induces CYP7A1, and significantly reduces cholesterol.Formula:C23H31NO4SPurezza:98%Colore e forma:SolidPeso molecolare:417.56Plm IV inhibitor-2
CAS:"Plm IV inhibitor-2: Potent for Plm IV (IC50=24nM), affects Plm II/Plm I; malaria research compound."Formula:C39H54N4O4Colore e forma:SolidPeso molecolare:642.87P7170
CAS:<p>P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.</p>Formula:C21H16F3N9Colore e forma:SolidPeso molecolare:451.42Dersimelagon phosphate
CAS:Dersimelagon phosphate: MC1R agonist, boosts melanin, enhances light tolerance in EPP/XLP without sun.Formula:C36H48F4N3O9PColore e forma:SolidPeso molecolare:773.75ATR-IN-17
CAS:ATR-IN-17 is a potent inhibitor of ATR kinase with good anti-cancer effects in LoVo cells (IC50: 1 nM).Formula:C22H28N6O2SColore e forma:SolidPeso molecolare:440.56FXIa-IN-9
CAS:FXIa-IN-9, a potent FXIa inhibitor (K i : human 0.17 nM, rabbit 0.5 nM), forms hydrogen bonds and has anticoagulant properties.Formula:C23H18Cl2F3N9O2Colore e forma:SolidPeso molecolare:580.35Azotomycin
CAS:Azotomycin is an antagonist of L-glutamine and may be used as an immunosuppressant.Formula:C17H23N7O8Purezza:98%Colore e forma:SolidPeso molecolare:453.41SIK1 activator 1
CAS:SIK1 activator 1 boosts SIK1 phosphorylation, reduces type 2 diabetes hyperglycemia, and inhibits liver gluconeogenesis.Formula:C23H32O6Colore e forma:SolidPeso molecolare:404.50PD 135158
CAS:PD 135158 is a CCK2 receptor antagonist.Formula:C42H61N5O11Purezza:98%Colore e forma:SolidPeso molecolare:811.9613(R)-HODE
CAS:13(R)-HODE, produced from linoleic acid, inhibits platelet aggregation (IC50=2.7μM) and is found in bovine endothelial cells.Formula:C18H32O3Colore e forma:SolidPeso molecolare:296.44CDK7-IN-18
CAS:<p>CDK7-IN-18: potent, pyrimidine-based CDK7 inhibitor with cancer research potential.</p>Formula:C22H24F3N7OSColore e forma:SolidPeso molecolare:491.53UNC7467
CAS:UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.Formula:C20H13NO3Purezza:98.28% - 98.64%Colore e forma:SoildPeso molecolare:315.32Cacospongionolide B
CAS:<p>Cacospongionolide B from Fasciospongia cavernosa inhibits secretory phospholipase A2, curbing inflammation.</p>Formula:C25H36O4Colore e forma:SolidPeso molecolare:400.55Transthyretin-IN-1
Transthyretin-IN-1 inhibits TTR fibril formation, aiding Alzheimer’s research.Formula:C10H9Br2NO4Colore e forma:SolidPeso molecolare:366.99Triphen diol
CAS:Triphen diol, a phenol diol, fights pancreatic cancer & cholangiocarcinoma, inducing apoptosis via caspase-dependent & -independent paths.Formula:C22H20O4Colore e forma:SolidPeso molecolare:348.39Homopteroic Acid
CAS:Homopteroic Acid, a precursor to Homofolic Acid, inhibits L1210 mouse leukemia growth by targeting folate uptake.Formula:C15H14N6O3Colore e forma:SolidPeso molecolare:326.31FK-906 HCl
CAS:FK-906 HCl is a human renin inhibitor used for the long-term treatment of patients with essential hypertension.Formula:C40H64ClN7O7Colore e forma:SolidPeso molecolare:790.44Carumonam Sodium
CAS:Carumonam Sodium is a monobactam, penicillin-binding protein inhibitor. It is used as antibacterials.Formula:C12H12N6Na2O10S2Purezza:98%Colore e forma:SolidPeso molecolare:510.37JTP-117968
CAS:JTP-117968: Non-steroidal SGRM, glucocorticoid receptor modulator, IC50 = 6.8 nM, offers better inhibitory/activatory balance.Formula:C31H31F3N2O2Colore e forma:SolidPeso molecolare:520.59P-gp modulator 1
CAS:P-gp modulator 1 is a high affinity and orally available P-glycoprotein (Pgp) modulatorFormula:C41H72N2O6Purezza:98%Colore e forma:SolidPeso molecolare:689.02Urease-IN-2
Urease-IN-2 is a non-competitive inhibitor of urease (IC50: 0.94 μM, Ki: 1.6 μM) that non-competitively inhibits Jack bean urease (JBU).Formula:C26H25N5O5S3Colore e forma:SolidPeso molecolare:583.7ddCTP trisodium
ddCTP trisodium, an HIV reverse transcriptase target, aids AIDS research and DNA sequencing as a ddNTP.Formula:C9H13N3Na3O12P3Colore e forma:SolidPeso molecolare:517.1Topoisomerase II inhibitor 6
Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.Formula:C19H18N4O2Colore e forma:SolidPeso molecolare:334.37hCAIX/XII-IN-5
<p>Coumarin 9a: Selective inhibitor of hCA IX/XII (Ki 93.3/85.7 nM), blocks cancer cell growth, and induces apoptosis.</p>Formula:C18H13NO3Colore e forma:SolidPeso molecolare:291.3BMS-248360
CAS:BMS-248360: Oral dual hAT1/hETA antagonist with Kis of 10nM & 1.9nM, respectively; treats hypertension.Formula:C36H45N5O5SPurezza:98%Colore e forma:SolidPeso molecolare:659.84GID4 Ligand 1
<p>GID4 Ligand 1: cell-permeable, selective binder, IC50 5.4 μM, Kd 5.6 μM, binds in cells with EC50 558 nM, useful for PROTAC synthesis.</p>Formula:C28H34N4O5SColore e forma:SolidPeso molecolare:538.66AAK1-IN-3 TFA
AAK1-IN-3 TFA, an AAK1 inhibitor with IC50 of 11 nM, crosses the blood-brain barrier, is a quinoline analogue, and may aid neuropathic pain research.Formula:C24H22F6N4O4Colore e forma:SolidPeso molecolare:544.45BSc5367
CAS:<p>BSc5367 inhibits Nek1 kinase (IC50: 11.5 nM), key in cell cycle, DNA repair, impacting ALS, PKD, cancer.</p>Formula:C20H15N3O2Colore e forma:SoildPeso molecolare:329.35TMX-4113
<p>TMX-4113 has potential to be used in cancer that is a phosphodiesterase 6D(PDE6D) and casein kinase 1α(CK1α) degrader [1].</p>Formula:C12H12N4O2S2Colore e forma:SolidPeso molecolare:308.38SGLT1/2-IN-1
CAS:SGLT1/2-IN-1 is a dual SGLT1/SGLT2 inhibitor.Formula:C25H28O8Colore e forma:SolidPeso molecolare:456.48LY 190388
CAS:<p>LY 190388 is a penicillamine-containing enkephalin analog used as an mu receptor agonist with analgesia activity.</p>Formula:C30H41N5O7SPurezza:98%Colore e forma:SolidPeso molecolare:615.74MI-1851
CAS:<p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>Formula:C34H53N15O6Colore e forma:SolidPeso molecolare:767.88IDO2-IN-1
CAS:<p>IDO2-IN-1: potent oral IDO2 inhibitor, IC50 = 112 nM, for inflammatory autoimmunity research.</p>Formula:C21H21BrN10O3Colore e forma:SolidPeso molecolare:541.36HSP90-IN-11
HSP90-IN-11: potent HSP90 inhibitor, akin to AUY-922; hinders CRC/NSCLC cell proliferation; degrades EGFR, Akt proteins.Formula:C27H30FN3O6Colore e forma:SolidPeso molecolare:511.54JBJ-09-063
CAS:JBJ-09-063: EGFR inhibitor, IC50s 0.147-0.396 nM for various mutants; hinders EGFR/Akt/ERK1/2 phosphorylation; targets TKI-sensitive/resistant lung cancer.Formula:C31H29FN4O3SColore e forma:SolidPeso molecolare:556.65Antidepressant agent 2
<p>Antidepressant agent 2 showed significant antidepressant effects with a MED value of 0.1 mg/kg.</p>Formula:C21H22ClFN2O3SColore e forma:SolidPeso molecolare:436.93LY 254155
CAS:LY 254155, an antifolate,binds to mFBP and inhibits hGARFT with Kis of 1.7±0.1 and 2.1±0.2 nM, respectively.Formula:C19H23N5O6SPurezza:98%Colore e forma:SolidPeso molecolare:449.48Integrase-LEDGF/p75 allosteric inhibitor 1
CAS:Oral HIV-1 allosteric integrase inhibitor, blocks DNA integration, antiviral, potent against NL432 (EC50: 3.9 nM).Formula:C33H41NO6SColore e forma:SolidPeso molecolare:579.75Atiratecan
CAS:Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.Formula:C31H34N6O6Purezza:98%Colore e forma:SolidPeso molecolare:586.64KRAS inhibitor-21
CAS:KRAS inhibitor-21 (22b) is a KRAS G12C inhibitor (IC50<0.01 μM) that can be used in cancer research.Formula:C33H41N5O3Colore e forma:SolidPeso molecolare:555.71L-Afegostat
CAS:<p>L-Afegostat (5-epi-Isofagomine), an iminosugar, inhibits glycosidase and β-Glucosidase (K i 30 μM), aids in carbohydrate synthesis.</p>Formula:C6H13NO3Colore e forma:SolidPeso molecolare:147.17HDAC-IN-37
HDAC-IN-37 inhibits HDACs 1, 3, 8, & 6, induces histone acetylation, halts G1 to S phase, and triggers early apoptosis.Formula:C23H24ClN7OColore e forma:SolidPeso molecolare:449.94p38 MAPK-IN-3
<p>Compound 2c is a potent p38α MAPK inhibitor with antitumor effects, enhancing apoptosis and ROS.</p>Formula:C22H17BrO2Colore e forma:SolidPeso molecolare:393.27PAT-347
CAS:PAT-347 is a potent inhibitor of Autotaxin, an enzyme linked to cell survival and diseases like cancer and fibrosis.Formula:C28H21ClF2N2O3SColore e forma:SolidPeso molecolare:538.99CM-352
CAS:CM-352 is a metalloproteinase inhibitor that reduces brain damage and improves functional recovery in rat models of cerebral hemorrhage.Formula:C24H29N3O6SPurezza:97.24%Colore e forma:SolidPeso molecolare:487.57Antimalarial agent 2
Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.Formula:C27H25N3O5Colore e forma:SolidPeso molecolare:471.5Pyripyropene A
CAS:Pyripyropene A is a potent and selective inhibitor of sterol O-acyltransferase 2 (SOAT2)/acyl-coenzyme A:cholesterol acyltransferase 2 (ACAT2)(IC50 of 0.07 μM).Formula:C31H37NO10Purezza:98%Colore e forma:SolidPeso molecolare:583.63Carnostatine
<p>Carnostatine (SAN9812), a potent CN1 inhibitor with 11 nM K i, may boost renal carnosine to treat DN.</p>Formula:C10H16N4O4Purezza:98%Colore e forma:SolidPeso molecolare:256.26L-Sepiapterin
CAS:L-Sepiapterin aids in making BH4, a coenzyme essential for eNOS, enhancing artery function and angiogenesis, while suppressing ovarian cancer cell growth.Formula:C9H11N5O3Colore e forma:SolidPeso molecolare:237.22MtTMPK-IN-9
MtTMPK-IN-9 moderately inhibits MtbTMPK (IC50: 48 μM), has submicromolar Mycobacterium activity, and is non-toxic, aiding tuberculosis research.Formula:C25H26N6O7Colore e forma:SolidPeso molecolare:522.51FLT3/TrKA-IN-1
FLT3/TrKA-IN-1: Potent dual kinase inhibitor for FLT3 & TrKA, promising for AML research.Formula:C28H30N4O2Colore e forma:SolidPeso molecolare:454.56ent-8-iso-15(S)-Prostaglandin F2α
CAS:Isoprostanes are produced by the non-enzymatic, free radical peroxidation of phospholipid-esterified arachidonic acid.Formula:C20H34O5Colore e forma:SolidPeso molecolare:354.48TRPC4/5-IN-1
TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.Formula:C21H21N3OColore e forma:SolidPeso molecolare:331.41LasR-IN-2
LasR-IN-2 blocks LasR via H-bond with TRY-56, useful in bacterial infection and CF research.Formula:C21H16ClN3O2Colore e forma:SolidPeso molecolare:377.82GDC-6036-NH
CAS:GDC-6036-NH is a precursor of compound 17a /b, which is a RAS inhibitor that can be used in cancer research.Formula:C26H30ClF4N7OPurezza:99.84%Colore e forma:SolidPeso molecolare:568.01SOS1-IN-10
SOS1-IN-10 is a potent inhibitor of SOS1 that acts on KRAS G12C-SOS1 (IC50: 13 nM).Formula:C22H19F5N4OColore e forma:SolidPeso molecolare:450.4Enantiomer of Sofosbuvir
Inactive enantiomer of Sofosbuvir, used for chronic hepatitis C; lacks reported biological activity.Formula:C22H29FN3O9PPurezza:98%Colore e forma:SolidPeso molecolare:529.45Moxaverine hydrochloride
CAS:<p>Moxaverine HCL, a papaverine derivative, is in Phase III trials for treating ocular blood flow in macular degeneration and glaucoma.</p>Formula:C20H22ClNO2Colore e forma:SolidPeso molecolare:343.85Tubulin polymerization-IN-35
Tubulin-IN-35 inhibits oxazolylisoindole microtubule formation, targeting VL51 marginal zone lymphoma.Formula:C31H35N3O5Colore e forma:SolidPeso molecolare:529.63KF 20274
CAS:KF 20274 is an adenosine A1 antagonist; purinergic receptor antagonist.Formula:C21H29N5OColore e forma:SolidPeso molecolare:367.49Anti-inflammatory agent 23
Anti-inflammatory agent 23 blocks LPS-induced NO (IC50: 0.449 μM) and binds p65 well.Formula:C34H49NO6Colore e forma:SolidPeso molecolare:567.76YM158 free base
CAS:YM158 free base is a potent and selective antagonist of TXA2 and LTD4 receptor (pA2s: about 8.81 and 8.87).Formula:C32H33ClN6O5S2Purezza:98%Colore e forma:SolidPeso molecolare:681.22Myxothiazol
CAS:Myxothiazol blocks mitochondrial complex III and triggers SESN2, a gene important for stress response.Formula:C25H33N3O3S2Colore e forma:SolidPeso molecolare:487.68LY210073
CAS:<p>LY210073 is an antagonist of the Leukotriene B4 (LTB4) receptor (IC50: 6.2 nM).</p>Formula:C30H28O8Purezza:98%Colore e forma:SolidPeso molecolare:516.54IRAK4-IN-12
IRAK4-IN-12 (compound 37) is a potent inhibitor of IRAK4 (IC50: 0.015 μM) with cellular pIRAK4 potency (IC50: 0.5 μM).Formula:C24H31FN8OColore e forma:SolidPeso molecolare:466.55Deltasonamide 2 hydrochloride
Deltasonamide 2 hydrochloride is a competitive high-affinity PDEδ inhibitor with a Kd of approximately 385 pM.Formula:C30H40Cl2N6O4S2Purezza:98%Colore e forma:SolidPeso molecolare:683.71PARP10/15-IN-1
PARP10/15-IN-1 (compound 8l) is a dual PARP10 and PARP15 inhibitor with IC50s of 160 nM and 370 nM, respectively. It can be used in cancer research[1].Formula:C13H10N2O3SColore e forma:SolidPeso molecolare:274.3Metocurine chloride
CAS:Metocurine: a muscle relaxant, not for kidney failure patients as it's kidney-excreted.Formula:C40H48Cl2N2O6Colore e forma:SolidPeso molecolare:723.72AChE/BChE-IN-1
<p>AChE/BChE-IN-1: dual AChE/BChE inhibitor, IC50 of 1.06 nM/7.3 nM, crosses blood-brain barrier, with antioxidant properties for Alzheimer's research.</p>Formula:C32H35ClN6O3Colore e forma:SolidPeso molecolare:587.11S100A2-p53-IN-1
CAS:<p>S100A2-p53-IN-1 inhibits S100A2-p53 in pancreatic cancer, stunting MiaPaCa-2 cell growth at 1.2-3.4 μM.</p>Formula:C20H20F6N2O4SColore e forma:SolidPeso molecolare:498.44Sunobinop
CAS:Sunobinop (S 117957) is an opioid receptor-like orphan receptor (ORL1) modulator.Formula:C26H33N3O3Colore e forma:SolidPeso molecolare:435.56SG3199
CAS:<p>SG3199, a PBD dimer, binds DNA's minor groove, forms covalent cross-links, and is cytotoxic to various human cancer cells.</p>Formula:C33H36N4O6Colore e forma:SolidPeso molecolare:584.66α-Glucosidase-IN-12
α-Glucosidase-IN-12 is a potent inhibitor of α-glucosidase (IC50: 10.20 μM).Formula:C25H30N4O4S2Colore e forma:SolidPeso molecolare:514.66RET-IN-14
CAS:RET-IN-14 inhibits RET (IC50: <0.51-9.3 nM) & BTK (C481S) (IC50: 9.2-15 nM), promising for tumor research.Formula:C24H23FN8O4Colore e forma:SolidPeso molecolare:506.49PDHK-IN-3
PDHK-IN-3 (compound 7) is a potent inhibitor of pyruvate dehydrogenase kinase(PDHK) with IC50s of 0.21 and 1.54 μM for PDHK2 and PDHK4, respectively [1].Formula:C17H16N2O2Colore e forma:SolidPeso molecolare:280.32Avorelin acetate
CAS:Avorelin acetate is a luteinizing hormone releasing hormone (LH-RH) agonist.Formula:C67H89N17O14Colore e forma:SolidPeso molecolare:1356.55
