Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.542 prodotti)
- Apoptosi(5.816 prodotti)
- Ciclo cellulare/Checkpoint(4.466 prodotti)
- Cromatina/Epigenetica(2.252 prodotti)
- Segnalazione citoscheletrica(1.381 prodotti)
- Danno al DNA/Riparazione del DNA(2.830 prodotti)
- Endocrinologia/Ormoni(3.518 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.362 prodotti)
- Immunologia e infiammazione(3.540 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(405 prodotti)
- Segnalazione MAPK(1.201 prodotti)
- Trasportatore di membrana/canale ionico(2.809 prodotti)
- Metabolismo(9.462 prodotti)
- Microbiologia/Virologia(7.003 prodotti)
- Neuroscienza(9.942 prodotti)
- Altri inibitori(37.827 prodotti)
- Ossidazione-riduzione(40 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.399 prodotti)
- Proteasi/Proteasoma(1.598 prodotti)
- Cellule staminali e Derivati(830 prodotti)
- Adattatori Tirosin-chinasi(2.012 prodotti)
- Ubiquitinazione(1.651 prodotti)
Mostrare 16 più sottocategorie
Trovati 66618 prodotti di "Inibitori"
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EGFR/HER2-IN-4
<p>EGFR/HER2-IN-4: oral, irreversible dual EGFR inhibitor (IC50: 0.6 nM), targets L858R/T790M mutations, potent anti-lung cancer effects in vivo.</p>Colore e forma:SolidPqsR-IN-1
<p>PqsR-IN-1, potent PqsR inhibitor, curbs pyocyanin in Pseudomonas aeruginosa with low cytotoxicity.</p>Formula:C17H18ClN3OSColore e forma:SolidPeso molecolare:347.86TNP-470
CAS:<p>TNP-470 is a methionine aminopeptidase-2 inhibitor. TNP-470 is also an angiogenesis inhibitor.</p>Formula:C19H28ClNO6Purezza:98%Colore e forma:SolidPeso molecolare:401.88Cortistatin A
CAS:<p>Cortistatin A is a potent and selective mediator-associated kinase CDK8 and its paralogue CDK19 inhibitor.</p>Formula:C30H36N2O3Purezza:98%Colore e forma:SolidPeso molecolare:472.62MSK-195
CAS:<p>MSK-195 is an effective TRPV1 agonist.</p>Formula:C28H40N2O5Purezza:98%Colore e forma:SolidPeso molecolare:484.6320S Proteasome-IN-4
CAS:<p>20S Proteasome-IN-4: brain-penetrant, parasite-specific, oral, inhibits T.b. brucei proteasome (IC50: 6.3nM), for HAT research.</p>Formula:C20H18ClF2N3O3Colore e forma:SolidPeso molecolare:421.83HIV-1 inhibitor-41
<p>HIV-1 inhibitor-41 (B23): Oral non-nucleoside reverse transcriptase blocker, EC50 of 50 nM (E138K), 20.8 nM (WT), low hERG/CYP impact, non-toxic.</p>Formula:C16H15F2N3OSColore e forma:SolidPeso molecolare:335.37D-473
CAS:<p>D-473 is a novel orally active triple reuptake inhibitor targeting dopamine, serotonin and norepinephrine transporters.</p>Formula:C26H27F2NO3Colore e forma:SolidPeso molecolare:439.49Carbonic anhydrase inhibitor 10
<p>CA inhibitor 10 targets MCF-7 cells, IC50: 11.9 μM; potent h CA IX inhibitor, Ki: 6.2 nM. Anti-cancer research.</p>Formula:C14H17N5O3SColore e forma:SolidPeso molecolare:335.38LolCDE-IN-2
CAS:<p>LolCDE-IN-2 is a potent Lol protein (LolCDE) inhibitor. LolCDE-IN-2 shows antibacterial activity with a MIC of 2 μg/ml against E. coli MG1655 [1].</p>Formula:C22H17N5OPurezza:98%Colore e forma:SolidPeso molecolare:367.40GNE-203
CAS:<p>GNE-203 is a Met inhibitor.</p>Formula:C30H29Cl2F3N8O3Colore e forma:SolidPeso molecolare:677.50SHP2-IN-9
<p>SHP2-IN-9: Potent SHP2 inhibitor, IC50=1.174 μM, 85x SHP1 selectivity, crosses blood-brain barrier, hampers cancer growth.</p>Formula:C20H20FN3O2SColore e forma:SolidPeso molecolare:385.46MK-6913
CAS:<p>MK-6913 is a potent and selective agonist of estrogen receptor β.</p>Formula:C25H27N3O2Purezza:98%Colore e forma:SolidPeso molecolare:401.5Antibacterial agent 78
<p>Antibacterial agent 78 (compound 30) is an antibacterial agent with improved cytotoxicity profile[1].</p>Formula:C16H23N3S2Colore e forma:SolidPeso molecolare:321.5LRRK2-IN-4
CAS:<p>LRRK2-IN-4: Potent, selective LRRK2 inhibitor, oral, BBB-penetrating, IC50=2.6 nM, potential for Parkinson's.</p>Formula:C25H29ClF2N6O2Colore e forma:SolidPeso molecolare:518.99Trichostatin A S-isomer
CAS:<p>Trichostatin A S-isomer, a HDAC 1, 3, 4, 6, 10 inhibitor with IC50 ~20 nM, has wide-ranging epigenetic effects.</p>Formula:C17H22N2O3Purezza:98%Colore e forma:SolidPeso molecolare:302.37nNOS-IN-25
CAS:nNOS-IN-25 is an effective, selective, and cell-permeable inhibitor of neuronal nitric oxide synthase.Formula:C21H22N4Purezza:98%Colore e forma:SolidPeso molecolare:330.43Hetrombopag olamine
CAS:<p>Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.</p>Formula:C29H36N6O7Purezza:98%Colore e forma:SolidPeso molecolare:580.63Cap-dependent endonuclease-IN-14
CAS:<p>Cap-dependent endonuclease-IN-14 hinders CEN and could treat influenza virus infections. (Patent CN113620948A, compound 1-c).</p>Formula:C30H23FN2O6SColore e forma:SolidPeso molecolare:558.58Antitubercular agent-22
<p>Antitubercular agent-22 combats Candida albicans (MIC: 2.34 μg/ml) and M. tuberculosis (MIC: 2 μg/ml).</p>Formula:C24H28FN5O8Colore e forma:SolidPeso molecolare:533.51Efrapeptin F
CAS:<p>Efrapeptin F, from Tolypocladium fungi, inhibits mitochondrial complex V and targets nutrient-deprived tumor cells.</p>Formula:C82H141N18O16Colore e forma:SolidPeso molecolare:1635.11Anticancer agent 26
<p>Anticancer agent 26 is a promising candidate for cancer therapy and deserves further development.</p>Formula:C28H33NO5Colore e forma:SolidPeso molecolare:463.57Aeruginosin 98-B
CAS:<p>Aeruginosin 98-B, a protease inhibitor, effectively inhibits trypsin, plasmin, and thrombin with IC50 values of 0.6, 7.0, and 10.0 μg/mL, respectively.</p>Formula:C29H46N6O9SColore e forma:SolidPeso molecolare:654.78PARL-IN-1
<p>PARL-IN-1: Strong PARL blocker, IC50 28 nM, boosts PINK1/Parkin mitophagy.</p>Formula:C40H58N6O7Colore e forma:SolidPeso molecolare:734.92P-gp modulator 1
CAS:<p>P-gp modulator 1 is a high affinity and orally available P-glycoprotein (Pgp) modulator</p>Formula:C41H72N2O6Purezza:98%Colore e forma:SolidPeso molecolare:689.02AA 497 (Free Base)
CAS:<p>AA 497, a beta-2 agonist, causes relaxation and suppresses Ca spike frequency.</p>Formula:C14H21NO3Purezza:98%Colore e forma:SolidPeso molecolare:251.32Zorubicin
CAS:<p>Zorubicin, a Daunorubicin derivative, targets topoisomerase II, inhibits DNA polymerase, and researches acute leukemia, sarcomas.</p>Formula:C34H35N3O10Colore e forma:SolidPeso molecolare:645.66Plumbemycin B
CAS:<p>Plumbemycin B is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Formula:C12H21N4O8PColore e forma:SolidPeso molecolare:380.29Bizelesin
CAS:<p>Bizelesin, a synthetic antineoplastic agent, binds DNA, disrupts replication, triggers cell-cycle arrest, and induces senescence.</p>Formula:C43H36Cl2N8O5Colore e forma:SolidPeso molecolare:815.7p38-α MAPK-IN-5
CAS:<p>p38-α MAPK-IN-5: potent p38α inhibitor, IC50s: 0.1 nM (α), 0.2 nM (β), 944 nM (γ), 4100 nM (δ); anti-inflammatory, promising for asthma/COPD research.</p>Formula:C37H49N11O2Colore e forma:SolidPeso molecolare:679.86Rpi 856 C
CAS:<p>Rpi 856 C is a retrovirus protease inhibitor from Streptomyces that is effective against HIV-1 and HTLV-1 proteases.</p>Formula:C39H56N6O10Purezza:98%Colore e forma:SolidPeso molecolare:768.90Saprisartan potassium
CAS:<p>Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.</p>Formula:C25H21BrF3KN4O4SColore e forma:SolidPeso molecolare:649.52O-Propargyl-Puromycin
CAS:<p>O-Propargyl-Puromycin (OP-puro) is a potent protein synthesis inhibitor, a puromycin acetylene analog.</p>Formula:C24H29N7O5Purezza:97.83% - 99.70%Colore e forma:SolidPeso molecolare:495.53BLU2864
CAS:<p>BLU2864: oral PRKACA inhibitor, IC50=0.3 nM, potential in cancer/poly. kidney disease research.</p>Formula:C24H19F3N4O2Purezza:97.58% - 99.92%Colore e forma:SoildPeso molecolare:452.43MAO-B-IN-17
CAS:<p>MAO-B-IN-17 is a selective and potent monoamine oxidase B (MAO-B) inhibitor (IC50: 5.08 μM) for the study of central nervous system disorders like Parkinson's.</p>Formula:C17H17F2NO2Purezza:99.41%Colore e forma:SoildPeso molecolare:305.32BMS453
CAS:<p>BMS453 (BMS-189453), a synthetic retinoid, is a potent and selective agonist of RARβ and a potent testicular toxin.</p>Formula:C27H24O2Purezza:99.93%Colore e forma:SolidPeso molecolare:380.48Glycosyltransferase-IN-1
<p>Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.</p>Formula:C19H21N5OPurezza:99.76%Colore e forma:SolidPeso molecolare:335.4Rupintrivir
CAS:<p>Rupintrivirvr (AG7088) is a mimetic peptide inhibitor of rhinovirus (HRV) 3C cysteine protease with antiviral activity for the study of viral infections.</p>Formula:C31H39FN4O7Purezza:97.72% - 99.35%Colore e forma:SolidPeso molecolare:598.66Iclepertin
CAS:<p>Iclepertin (BI-425809) is a GlyT1 inhibitor.Iclepertin is used for the treatment of Alzheimer;s disease and other CNS disorders.</p>Formula:C20H18F6N2O5SPurezza:98.89% - 98.93%Colore e forma:SolidPeso molecolare:512.42WAY-213613 hydrochloride
CAS:<p>WAY-213613 hydrochloride: potent, selective GLT-1/EAAT2 inhibitor (IC50 85 nM); weaker for EAAT1/3; inactive at glutamate receptors; research tool for CNS.</p>Formula:C16H13BrF2N2O4Purezza:99.14% - 99.37%Colore e forma:SoildPeso molecolare:415.19STK-15
CAS:<p>STK-15 is a candidate for use as a fatty acid binding protein 5 (FABP5) inhibitor.</p>Formula:C34H29NO5Purezza:98.05%Colore e forma:SolidPeso molecolare:531.6Simmitecan hydrochloride
CAS:<p>Simmitecan hydrochloride is a camptothecin derivative, a topoisomerase I inhibitor with anticancer activity, which can be used to study is solid tumors.</p>Formula:C34H39ClN4O6Purezza:98.20% - 98.93%Colore e forma:SolidPeso molecolare:635.15NRX-1532
<p>NRX-1532 is a small molecule β-catenin:β-TrCP interaction enhancer.</p>Formula:C16H11F3N4O2Purezza:98.95% - 99.68%Colore e forma:SolidPeso molecolare:348.28MIV-247
CAS:<p>MIV-247 is a cathepsin S inhibitor that attenuates mechanically abnormal pain in preclinical neuropathic pain models and can be used to study myocardial injury.</p>Formula:C17H24F3N3O4Purezza:99.27%Colore e forma:SolidPeso molecolare:391.39Evixapodlin
CAS:<p>Evixapodlin (PD-1/PD-L1-IN 7) is a human PD-1/PD-L1 protein/protein interaction inhibitor (IC50: 0.213).Evixapodlin has anticancer and antiviral activities.</p>Formula:C34H36Cl2N8O4Purezza:99.07%Colore e forma:SolidPeso molecolare:691.61L-371,257
CAS:<p>L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.</p>Formula:C28H33N3O6Purezza:99.79%Colore e forma:SolidPeso molecolare:507.58VX-984
CAS:<p>VX-984 (M9831) is an oral DNA-PK inhibitor, crossing the blood-brain barrier, targeting GBM and NSC-LC.</p>Formula:C23H21D2N7OPurezza:97.65% - 99.98%Colore e forma:SolidPeso molecolare:415.49Emprumapimod
CAS:<p>Emprumapimod, an oral p38α MAPK inhibitor, targets RPMI-8226 cells, curbs LPS-induced IL-6; IC50: 100 pM; for cardiomyopathy, acute pain.</p>Formula:C24H29F2N5O3Purezza:99.21% - >99.99%Colore e forma:SolidPeso molecolare:473.52CCF0058981
CAS:<p>CCF0058981: noncovalent inhibitor for SARS-CoV-2 & -1 proteases; IC50s: 68 nM (SC2) & 19 nM (SC1). Potential COVID-19 research use.</p>Formula:C24H19ClN6OPurezza:98.94%Colore e forma:SoildPeso molecolare:442.9Zelasudil
CAS:<p>Zelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.</p>Formula:C22H21F2N7OPurezza:99.15%Colore e forma:SolidPeso molecolare:437.445HRO761
CAS:<p>HRO761 is a potent Werne r syndrome RecQ DNA deconjugase (WRN) inhibitor that can be used to study cancers such as colon and stomach cancer.</p>Formula:C31H31ClF3N9O5Purezza:98.74% - 99.62%Colore e forma:SolidPeso molecolare:702.08USP15-IN-1
CAS:<p>USP15-IN-1 is a potent USP15 inhibitor (IC50 is 3.76 μM).</p>Formula:C22H23N3O3Purezza:99.509% - 99.81%Colore e forma:SolidPeso molecolare:377.44NRX-103094
CAS:<p>NRX-103094 boosts β-catenin binding to SCFβ-TrCP ligase with EC50 62 nM and Kd 0.6 nM.</p>Formula:C20H11Cl2F3N2O4SPurezza:99.13%Colore e forma:SolidPeso molecolare:503.28CP-642931
CAS:<p>CP-642931 (Sorbitol dehydrogenase-IN-1) is a sorbitol dehydrogenase inhibitor used in the study of diabetes mellitus and cardiovascular disease.</p>Formula:C17H25N7OPurezza:99.67% - >99.99%Colore e forma:SolidPeso molecolare:343.43Treprostinil diethanolamine
CAS:<p>Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,</p>Formula:C27H45NO7Purezza:99.86%Colore e forma:SolidPeso molecolare:495.65BAY-3827
CAS:<p>BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.</p>Formula:C27H25FN6OPurezza:99.90%Colore e forma:SolidPeso molecolare:468.53Lometrexol
CAS:<p>Lometrexol (LY 264618) is an antifolate that inhibits GARFT, blocks purine synthesis, induces apoptosis, and has anticancer properties.</p>Formula:C21H25N5O6Purezza:97.76% - 99.56%Colore e forma:SolidPeso molecolare:443.45Vofopitant
CAS:<p>Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).</p>Formula:C21H23F3N6OPurezza:97.86%Colore e forma:SolidPeso molecolare:432.44GLPG0974
CAS:<p>GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.</p>Formula:C25H25ClN2O4SPurezza:99.8%Colore e forma:SolidPeso molecolare:484.99NDI-034858
CAS:<p>NDI-034858 (TAK-279) is a tyrosine kinase 2 (TYK2) inhibitor (Kd<200 pM) that targets the JH2 structural domain of Tyk2 for the treatment of autoimmune diseases</p>Formula:C23H24N8O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:460.49Cbl-b-IN-3
CAS:<p>Cbl-b-IN-3 is a potent inhibitor of casitas b lineage lymphoma proto-oncogene-b (Cbl-b) (ic50 < 1 nM).Cost-effective and quality-assured.</p>Formula:C30H34F3N5OPurezza:99%Colore e forma:SolidPeso molecolare:537.62Picrotoxinin
CAS:<p>Picrotoxinin blocks chloride channels, antagonizes GABAA noncompetitively (IC50: 1.15 μM, α1β2γ2L), and induces convulsions.</p>Formula:C15H16O6Purezza:98.07%Colore e forma:SolidPeso molecolare:292.28Enbezotinib
CAS:<p>Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.</p>Formula:C21H21FN6O3Purezza:99.84%Colore e forma:SolidPeso molecolare:424.43AChE-IN-26
CAS:<p>AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).</p>Formula:C21H21BrN2O3Purezza:99.24% - 99.85%Colore e forma:SoildPeso molecolare:429.31SYM2206
CAS:<p>SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated</p>Formula:C20H22N4O3Purezza:99.88%Colore e forma:SolidPeso molecolare:366.41AKT Kinase Inhibitor
CAS:AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.Cost-effective and quality-assured.Formula:C16H19N7O3Purezza:97.83% - 99.13%Colore e forma:SolidPeso molecolare:357.37FABPs ligand 6
CAS:<p>FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.</p>Formula:C28H27FN2O3Purezza:97.45%Colore e forma:SolidPeso molecolare:458.52Suzetrigine
CAS:Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.Formula:C21H20F5N3O4Purezza:98.08% - 99.27%Colore e forma:SolidPeso molecolare:473.39Etamicastat hydrochloride
CAS:<p>Etamicastat hydrochloride (BIA 5-453 hydrochloride) is a peripherally selective dopamine beta-hydroxylase inhibitor that reduces hypertension.</p>Formula:C14H16ClF2N3OSPurezza:98.54%Colore e forma:SolidPeso molecolare:347.81ELOVL1-IN-2
CAS:<p>ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).</p>Formula:C18H15FN2OPurezza:99.84%Colore e forma:SolidPeso molecolare:294.32SJ6986
CAS:SJ6986 is a potent, selective and orally active GSPT1/2 degrader. SJ6986 degrades GSPT1 with a DC 50 of 2.1 nM (D max 99%) [1].Formula:C20H14F3N3O7SPurezza:99.73%Colore e forma:SolidPeso molecolare:497.4JNJ-6204
CAS:<p>JNJ-6204 is a deuterated compound that efficiently inhibits CSNK1D and CSNK1E.</p>Formula:C19H11D6FN6OPurezza:97.42% - 99.87%Colore e forma:SolidPeso molecolare:370.41Moiramide B
CAS:Moiramide B is an acetyl coenzyme A carboxylase inhibitor with antimicrobial activity, strongly inhibiting Gram-positive bacteria.Formula:C25H31N3O5Purezza:98.53% - 99.90%Colore e forma:SolidPeso molecolare:453.53(+)-Tetrabenazine
CAS:(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-foldFormula:C19H27NO3Purezza:98.69%Colore e forma:SolidPeso molecolare:317.42DRB18
CAS:<p>DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.</p>Formula:C22H23ClN2O2Purezza:99.54%Colore e forma:SolidPeso molecolare:382.88Cort108297
CAS:<p>Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.</p>Formula:C26H25F4N3O3SPurezza:98.36% - 99.94%Colore e forma:SolidPeso molecolare:535.55GSK3368715 dihydrochloride
CAS:<p>GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study of advanced solid tumors.</p>Formula:C20H40Cl2N4O2Purezza:99.66% - 99.66%Colore e forma:SolidPeso molecolare:439.46KU-60019
CAS:<p>KU-60019 is a specific inhibitor of ATM kinase (IC50: 6.3 nM).</p>Formula:C30H33N3O5SPurezza:98.05% - 98.50%Colore e forma:SolidPeso molecolare:547.67SDZ 220-040
CAS:<p>SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂，可诱导根系生长的部分无重力模式 。</p>Formula:C16H16Cl2NO6PPurezza:98.13%Colore e forma:SolidPeso molecolare:420.18Vecabrutinib
CAS:<p>Vecabrutinib (SNS-062) is a potent and noncovalent BTK and ITK inhibitor (Kd: 0.3 nM and 2.2 nM, respectively). Vecabrutinib displays an IC50 of 24 nM for ITK.</p>Formula:C22H24ClF4N7O2Purezza:99.74%Colore e forma:SolidPeso molecolare:529.92Darizmetinib
CAS:Darizmetinib (HRX215) is an MKK4 inhibitor.Formula:C21H17F2N5O3SPurezza:98.03% - 99.57%Colore e forma:SolidPeso molecolare:457.45Cap-dependent endonuclease-IN-1
CAS:<p>Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.</p>Formula:C27H22F2N2O6SPurezza:98.88% - 99.09%Colore e forma:SolidPeso molecolare:540.54Dazostinag disodium
CAS:<p>Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.</p>Formula:C21H20F2N8Na2O10P2S2Purezza:98.84% - 99.96%Colore e forma:SolidPeso molecolare:754.48HOIPIN-8 sodium
CAS:<p>HOIPIN-8 sodium is a LUBAC inhibitor for the study of inflammatory and immune diseases.</p>Formula:C23H15F2N4NaO3Purezza:97.34%Colore e forma:SolidPeso molecolare:456.38SB-423562
CAS:<p>SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.</p>Formula:C26H32N2O4Purezza:99.22%Colore e forma:SolidPeso molecolare:436.54LSN3318839
CAS:<p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>Formula:C26H23Cl2N3O2Purezza:99.21%Colore e forma:SolidPeso molecolare:480.39AM103
CAS:AM103 is an effective and selective inhibitor of FLAP (IC50 = 4.2 nM).Formula:C36H38N3NaO4SPurezza:99.75%Colore e forma:SolidPeso molecolare:631.76Vofopitant dihydrochloride
CAS:Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.Formula:C21H25Cl2F3N6OPurezza:98.99%Colore e forma:SolidPeso molecolare:505.36BCL6-IN-3
CAS:BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.Formula:C24H31ClF2N6O2Purezza:98.17%Colore e forma:SolidPeso molecolare:508.99BE1218
CAS:<p>BE1218 is a liver X receptor (LXR) inverse agonist active on LXRα and LXRβ with an IC50 of 9 nM and 7 nM, respectively.</p>Formula:C30H30FNO4S2Purezza:99.7%Colore e forma:SoildPeso molecolare:551.69NB-360
CAS:<p>NB-360: potent, brain-penetrant BACE1/2 inhibitor; IC50s: 5-6 nM; high selectivity vs pepsin, cathepsin E/D.</p>Formula:C21H19F4N5O2Purezza:99.72%Colore e forma:SolidPeso molecolare:449.4AChE/BChE-IN-10
CAS:<p>AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.</p>Formula:C26H30N2O2Purezza:99.55% - 99.88%Colore e forma:SoildPeso molecolare:402.53AZD5462
CAS:<p>AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.</p>Formula:C30H41FN2O6Purezza:98.32% - 99.63%Colore e forma:SolidPeso molecolare:544.65Elacytarabine
CAS:<p>Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.</p>Formula:C27H45N3O6Purezza:97.69%Colore e forma:SolidPeso molecolare:507.66Dersimelagon
CAS:<p>Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.</p>Formula:C36H45F4N3O5Purezza:97.35% - 98.23%Colore e forma:SolidPeso molecolare:675.75ALOX15-IN-2
CAS:<p>ALOX15-IN-2: Potent ALOX15 inhibitor. IC50: 1.55 μM for LA; 2.79 μM for AA. Stops linoleic/arachidonic acid oxidation.</p>Formula:C23H29N3O4SPurezza:98.10%Colore e forma:SolidPeso molecolare:443.56JTK-109
CAS:<p>JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.</p>Formula:C37H33ClFN3O4Purezza:98.48% - 99.68%Colore e forma:SolidPeso molecolare:638.13AZD 3147
CAS:<p>AZD 3147 inhibits mTORC1 (40.7 nM), mTORC2 (5.75 nM), and PI3Kα/β/δ/γ (912/5495/9333/6310 nM IC50s).</p>Formula:C24H31N5O4S2Purezza:99.99%Colore e forma:SolidPeso molecolare:517.66IDX184
CAS:<p>IDX184 is a potent, orally active, targeted HCV polymerase inhibitor and nucleoside polymerase.IDX184 effectively inhibits HCV polymerase (IC50=0.31 μM, Ki=52.3</p>Formula:C25H35N6O9PSPurezza:97.15%Colore e forma:SolidPeso molecolare:626.62PREP inhibitor-1
CAS:PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.Formula:C22H28N4O2Purezza:98.78%Colore e forma:SoildPeso molecolare:380.48
