Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.687 prodotti)
- Apoptosi(6.097 prodotti)
- Ciclo cellulare/Checkpoint(4.691 prodotti)
- Cromatina/Epigenetica(2.376 prodotti)
- Segnalazione citoscheletrica(1.472 prodotti)
- Danno al DNA/Riparazione del DNA(2.921 prodotti)
- Endocrinologia/Ormoni(3.611 prodotti)
- Enzima(3.655 prodotti)
- Proteina G/GPCR(8.755 prodotti)
- Immunologia e infiammazione(3.765 prodotti)
- Virus dell'influenza(298 prodotti)
- Segnalazione JAK/STAT(407 prodotti)
- Segnalazione MAPK(1.230 prodotti)
- Trasportatore di membrana/canale ionico(2.947 prodotti)
- Metabolismo(9.940 prodotti)
- Microbiologia/Virologia(7.347 prodotti)
- Neuroscienza(10.240 prodotti)
- Altri inibitori(36.533 prodotti)
- Ossidazione-riduzione(43 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.437 prodotti)
- Proteasi/Proteasoma(1.675 prodotti)
- Cellule staminali e Derivati(830 prodotti)
- Adattatori Tirosin-chinasi(2.028 prodotti)
- Ubiquitinazione(1.682 prodotti)
Mostrare 16 più sottocategorie
Trovati 66582 prodotti di "Inibitori"
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Elamipretide Triacetate
CAS:<p>Elamipretide TriTFA, a tetrapeptide, targets mitochondria, associates with cardiolipin, studied for treating Leber's Optic Neuropathy.</p>Formula:C38H61N9O11Purezza:>99.99%Colore e forma:SolidPeso molecolare:819.94Oxindole
CAS:<p>Oxindole (Indolin-2-one) is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic target for anti-cancer drug development.</p>Formula:C8H7NOPurezza:99.34%Colore e forma:Off-White Crystalline PowderPeso molecolare:133.15CTB
CAS:<p>CTB (Cholera Toxin B subunit) is an activator of p300 histone acetyltransferase and induces apoptosis in MCF-7 cells.</p>Formula:C16H13ClF3NO2Purezza:99.82%Colore e forma:SolidPeso molecolare:343.73p-Toluic Acid
CAS:<p>p-Toluic Acid (4-Methylbenzoic acid) belongs to the class of organic compounds known as benzoic acids. 4-Methylbenzoic acid has been primarily detected in saliva. Within the cell, 4-methylbenzoic acid is primarily located in the cytoplasm.</p>Formula:C8H8O2Purezza:99.44%Colore e forma:Physical Description White Powder Sublimes (Ntp 1992)Peso molecolare:136.15Ref: TM-FR14438
Prodotto fuori produzioneSculponeatin O
CAS:<p>Sculponeatin O may have protective effects on the lipid peroxidation-damaged live cells.</p>Formula:C28H40O4Purezza:95.00%Colore e forma:SolidPeso molecolare:440.61Isonicotinic acid
CAS:<p>Isonicotinic acid is a metabolite of Isoniazid.Isonicotinic acid is a useful isomer of nicotinic acid. Isoniazid is converted to Isonicotinic acid by hydrazinolysis, with the biotransformation also to be catalyzed by cytochrome P450 enzymes, such as CYP2C.</p>Formula:C6H5NO2Purezza:99.68%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:123.11Lupinine
CAS:<p>Lupinine is an alkaloid capable of counteracting ethanol anesthesia. Lupinine is an AChE and BChE inhibitor and potential CD69 activator found in species of Loranthus, Calia, and Lupinus. It may also inhibit heparin.</p>Formula:C10H19NOPurezza:99.95%Colore e forma:SolidPeso molecolare:169.26Ammonium Glycyrrhizinate
CAS:<p>Ammonium Glycyrrhizinate (Glycyram) inhibits the cytopathology and growth of several unrelated DNA/RNA viruses.</p>Formula:C42H62O16·NH3Purezza:98.41%Colore e forma:SolidPeso molecolare:839.96Ref: TM-T6384
Prodotto fuori produzioneCompound T69202(SC)
CAS:<p>NBQX (FG9202), an AMPA/kainate receptor blocker, counters glutamate toxicity; water-soluble as disodium salt, has anticonvulsant properties.</p>Formula:C12H6N4Na2O6SColore e forma:SolidPeso molecolare:380.2415Ref: TM-T69202
Prodotto fuori produzioneVonoprazan fumarate
CAS:<p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>Formula:C17H16FN3O2S·C4H4O4Purezza:99.16% - 99.98%Colore e forma:SolidPeso molecolare:461.46Desidustat
CAS:<p>Desidustat is an inhibitor of HIF hydroxylase.</p>Formula:C16H16N2O6Purezza:98%Colore e forma:SolidPeso molecolare:332.31α-Lipoic Acid
CAS:<p>α-Lipoic Acid (Alphalipoic acid) inhibits NF-κB-dependent HIV-1 LTR activation.</p>Formula:C8H14O2S2Purezza:99.83%Colore e forma:Forms Yellowish Flakes SolidPeso molecolare:206.32Elamipretide 2TFA
CAS:<p>Elamipretide 2TFA (RX-31 2TFA) is a novel mitochondrion-targeted antioxidant.</p>Formula:C36H51F6N9O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:867.84Ref: TM-T8831
Prodotto fuori produzioneCoumaran
CAS:<p>Coumaran (2,3-Dihydrobenzofuran) is an acetylcholinesterase (AChE) inhibitor isolated from leaves of L. camara. Coumaran(2,3-Dihydrobenzofuran) can be used as a biopesticide. 2,3-dihydrobenzofuran is a member of the class of 1-benzofurans that is the 2,3-dihydroderivative of benzofuran. It has a role as a metabolite.</p>Formula:C8H8OPurezza:99.61%Colore e forma:LiquidPeso molecolare:120.15Cebranopadol
CAS:<p>Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)</p>Formula:C24H27FN2OPurezza:98.32% - 99.78%Colore e forma:SolidPeso molecolare:378.487-Methoxy-1-tetralone
CAS:<p>7-Methoxy-1-tetralone may have insecticidal activity.</p>Formula:C11H12O2Purezza:99.93%Colore e forma:White CrystalPeso molecolare:176.21Olmutinib
CAS:Olmutinib (BI1482694) is a Novel Epidermal Growth Factor Receptor Tyrosine Kinase InhibitorFormula:C26H26N6O2SPurezza:99.14%Colore e forma:SolidPeso molecolare:486.59Praeruptorin B
CAS:<p>1. Praeruptorin B can inhibit tumor promoter induced phemonenon in vitro.</p>Formula:C24H26O7Purezza:99.96%Colore e forma:SolidPeso molecolare:426.46IGFBP-1 Protein, Rat, Recombinant
<p>IGF-binding proteins prolong the half-life of the IGFs and have been shown to either inhibit or stimulate the growth promoting effects of the IGFs on cell culture. They alter the interaction of IGFs with their cell surface receptors. Promotes cell migration. IGFBP-1 Protein, Rat, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26.9 kDa and the accession number is P21743.</p>Peso molecolare:26.9 kDa (predicted)COR-001
CAS:<p>Ziltivekimab (COR-001) is a human IL-6 antibody, lowers CRP, and may treat inflammation and heart issues in CKD.</p>Purezza:95%Colore e forma:Odour LiquidARGX-112
CAS:<p>Temtokibart is a humanized IgG1 λ2 antibody that specifically targets IL22RA1, and is expressed by cells that are deficient in the glutamine synthetase gene.</p>Colore e forma:Odour LiquidOkadaic acid
CAS:<p>Okadaic acid, a polyether marine toxin, is a highly potent and selective protein phosphatase (PP) inhibitor.</p>Formula:C44H68O13Purezza:98%Colore e forma:White Crystals Or PowderPeso molecolare:805Pazinaclone
CAS:<p>Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.</p>Formula:C25H23ClN4O4Purezza:97.79% - 99.07%Colore e forma:SolidPeso molecolare:478.93CXCR4-IN-1
CAS:<p>CXCR4-IN-1 (Example C5), with an IC50 of 20 nM, is a potent inhibitor of CXCR4, applicable for the research of various conditions such as cancer, HIV, diabetic</p>Formula:C23H32N6Purezza:98%Colore e forma:SolidPeso molecolare:392.54Ref: TM-T79059
Prodotto fuori produzioneFotemustine
CAS:<p>Fotemustine: antineoplastic, chloroethylates DNA, blocks synthesis, causes cell arrest/apoptosis, lipophilic, crosses blood-brain barrier.</p>Formula:C9H19ClN3O5PColore e forma:SolidPeso molecolare:315.69Ref: TM-T21305
Prodotto fuori produzioneHBV-IN-34
CAS:<p>HBV-IN-34 (compound 17i) is a potent inhibitor of HBsAg production, demonstrating remarkable in vitro anti-HBV efficacy with EC50 values of 0.018 μM for HBV DNA</p>Formula:C21H19F2N7Purezza:98%Colore e forma:SolidPeso molecolare:407.42Ref: TM-T79469
Prodotto fuori produzioneFosfonet sodium
CAS:Fosfonet sodium is a sodium salt of phosphonoacetic acid, effective against herpesviruses by inhibiting viral DNA polymerase.Formula:C2H4NaO5PColore e forma:SolidPeso molecolare:162.01Ref: TM-T69345
Prodotto fuori produzionePKUMDL-LTQ-301
CAS:PKUMDL-LTQ-301 is a potent inhibitor of HipA toxin. PKUMDL-LTQ-301 also inhibits E. coli persistence.Formula:C30H28N2O4Purezza:98%Colore e forma:SolidPeso molecolare:480.55Ref: TM-T28423
Prodotto fuori produzioneGlutaminyl Cyclase Inhibitor 4
CAS:Glutaminyl Cyclase Inhibitor 4 is a potent, selective glutaminyl cyclase (QC) inhibitor (IC50: 6.1 nM). It is a potent anti-Alzheimer’s agent.Formula:C22H33N5O3Purezza:98%Colore e forma:SolidPeso molecolare:415.53Ref: TM-T11423
Prodotto fuori produzioneAnti-NASH agent 1
CAS:<p>Anti-NASH Agent 1 (Compound 3d), derived from Elafibranor, serves as a strong PPAR-α/δ agonist aimed at treating nonalcoholic steatohepatitis (NASH).</p>Formula:C26H33NO4Purezza:98%Colore e forma:SolidPeso molecolare:423.54Ref: TM-T79454
Prodotto fuori produzioneLp-PLA2-IN-15
CAS:<p>Lp-PLA2-IN-15 (example 2) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential application in Alzheimer's disease research [1].</p>Formula:C22H17F5N4O3Purezza:98%Colore e forma:SolidPeso molecolare:480.39Ref: TM-T79075
Prodotto fuori produzioneDprE1-IN-8
CAS:<p>DprE1-IN-8 is a potent inhibitor of DprE1, exhibiting an IC50 of less than 0.75 μM.</p>Formula:C19H12F3N5O4SPurezza:98%Colore e forma:SolidPeso molecolare:463.39Ref: TM-T79628
Prodotto fuori produzioneEGFR-IN-82
CAS:<p>EGFR-IN-82 (Compound 8a) is a potent, orally active inhibitor of EGFR, exhibiting IC50 values of 0.09 nM for EGFR L858R/T790M/C797S and 0.06 nM for EGFR Del19/</p>Formula:C32H41BrN9O2PPurezza:98%Colore e forma:SolidPeso molecolare:694.6Ref: TM-T78788
Prodotto fuori produzioneGR 218,231
CAS:GR 218,231 is a selective antagonist of D3 dopamine receptor.Formula:C24H33NO3SPurezza:98%Colore e forma:SolidPeso molecolare:415.59Ref: TM-T27431
Prodotto fuori produzioneCulmerciclib
CAS:<p>Culmerciclib is a cell cycle protein-dependent kinase (CDK) inhibitor that exhibits antitumour effects.</p>Formula:C24H27FN8Colore e forma:SolidPeso molecolare:446.52Ref: TM-T62650
Prodotto fuori produzioneDioxifedrine
CAS:Dioxifedrine is a beta-2 -adrenergic agonist with bronchodilator activity.Formula:C10H15NO3Colore e forma:SolidPeso molecolare:197.23Ref: TM-T71575
Prodotto fuori produzioneAminobutane bisphosphonate
CAS:Aminobutane bisphosphonate curbs bone loss; may manage hypercalcemia in cancer.Formula:C4H13NO6P2Colore e forma:SolidPeso molecolare:233.1Ref: TM-T69443
Prodotto fuori produzioneBenzovindiflupyr
CAS:<p>Benzovindiflupyr: a fungicide that inhibits SDH (IC50=5.2nM), halts S. sclerotiorum growth (EC50=0.011μg/ml), and protects crops like eggplants.</p>Formula:C18H15Cl2F2N3OColore e forma:SolidPeso molecolare:398.23Ceronapril
CAS:Ceronapril (SQ 29852) is an orally active and potent angiotensin-converting enzyme (ACE) inhibitor (IC50 : 36 nM) for the study of dementia and hypertension.Formula:C21H33N2O6PPurezza:97.94%Colore e forma:SolidPeso molecolare:440.47Questiomycin A derivatives 18 TFA
<p>Questiomycin A derivative 18 TFA exhibits antibacterial, anticancer properties and inhibits GRP78.</p>Formula:C16H12F3N3O5Purezza:98.45%Colore e forma:SoildPeso molecolare:383.07Ref: TM-T67717L
Prodotto fuori produzioneRadafaxine hydrochloride
CAS:<p>Radafaxine hydrochloride is an inhibitor of DAT and NET transporters, and nAChR family modulator.</p>Formula:C13H19Cl2NO2Purezza:98%Peso molecolare:292.2Mavodelpar free base
CAS:<p>Mavodelpar free acid (REN001 free acid) is an selective agonist of PPARδ.</p>Formula:C31H30FNO5Purezza:98%Colore e forma:SolidPeso molecolare:515.57MitoE10
CAS:MitoE10 is an effective mitochondrial targeting antioxidant.Formula:C42H55O5PSColore e forma:SolidPeso molecolare:702.92Ref: TM-T33406
Prodotto fuori produzioneKBP-7018
CAS:<p>KBP-7018: potent tyrosine kinase inhibitor targeting c-KIT, RET, PDGFR with IC50s of 10, 7.6, 25nM.</p>Formula:C31H30N4O5Colore e forma:SolidPeso molecolare:538.59Ref: TM-T27715
Prodotto fuori produzioneIDX-375
CAS:IDX-375, a HCV NS5B polymerase inhibitor, is used potentially for the treatment of HCV infection.Formula:C29H50N5O7PSPurezza:98%Colore e forma:SolidPeso molecolare:643.78PPARγ-IN-2
CAS:<p>"PPARγ-IN-2 (Compound 5a), a PPARγ inhibitor, exhibits an EC50 of 0.106 μM in inhibiting TG accumulation in 3T3-L1 preadipocytes.</p>Formula:C19H21N5OPurezza:98%Colore e forma:SolidPeso molecolare:335.4Ref: TM-T79678
Prodotto fuori produzione(E)-Crotylbarbital
CAS:<p>(E)-Crotylbarbital, a Crotylbarbital isomer, is a sedative with hypnotic, anticonvulsant properties, aiding sleep and mental stability.</p>Formula:C10H14N2O3Purezza:99.94%Colore e forma:SolidPeso molecolare:210.23BChE-IN-17
CAS:<p>BChE-IN-17 (compound 6n) is a potent, selective inhibitor of butyrylcholinesterase (BChE), demonstrating inhibitory half-maximal inhibitory concentrations (</p>Formula:C23H23BrN2O4S2Colore e forma:SolidPeso molecolare:535.47Ref: TM-T79342
Prodotto fuori produzioneAKOS-22
CAS:<p>AKOS-22: potent VDAC1 inhibitor, Kd=15.4 μM; prevents mitochondrial dysfunction and apoptosis.</p>Formula:C22H21ClF3N3O3Purezza:98%Colore e forma:SolidPeso molecolare:467.87DPX-3778
CAS:DPX-3778, a triethanolamine salt, boosts tobacco callus growth 4-5x at 0.124-2.48 μM and slows aging with IAA and kinetin.Formula:C16H23ClN4O6Colore e forma:SolidPeso molecolare:402.83Ref: TM-T31573
Prodotto fuori produzioneALPK1-IN-2
CAS:<p>ALPK1-IN-2 is a potent inhibitor of ALPK1 (α-kinase 1) (IC50: 95 nM). ALPK1-IN-2 inhibits NF-κB (IC50: 1.31 μM).</p>Formula:C20H18F2N4O2SColore e forma:SolidPeso molecolare:416.44Ref: TM-T62162
Prodotto fuori produzioneBromadoline maleate
CAS:<p>Bromadoline is an opioid analgesic selective for the μ-opioid receptor.</p>Formula:C19H25BrN2O5Purezza:98%Colore e forma:SolidPeso molecolare:441.322Ref: TM-T26908
Prodotto fuori produzioneJAK2-IN-9
CAS:<p>Compound A8, known as JAK2-IN-9, is a selective JAK2 inhibitor with an IC50 of 5 nM.</p>Formula:C20H24N6O2SPurezza:98%Colore e forma:SolidPeso molecolare:412.51Ref: TM-T79581
Prodotto fuori produzioneSR14150
CAS:<p>SR14150 is a partial agonist of high-affinity NOP receptor.</p>Formula:C21H30N2OPurezza:98%Colore e forma:SolidPeso molecolare:326.48Ref: TM-T24828
Prodotto fuori produzionePhenazolam
CAS:<p>Phenazolam is an analytical reference standard categorized as a benzodiazepine. [1] This product is intended for research and forensic applications.</p>Formula:C17H12BrClN4Colore e forma:SolidPeso molecolare:387.66Neurokinin antagonist 1
CAS:<p>Neurokinin antagonist 1 is a potent is a neuropeptide antagonist that can be used to study neurological disorders.</p>Formula:C38H40N4O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:600.75BET-IN-15
CAS:<p>BET-IN-15 (compound 1) is a potent, orally active inhibitor of BET, demonstrating inhibitory IC50 values of 0.64 nM for BRD4-BD1 and 0.25 nM for BRD4-BD2.</p>Formula:C21H18F2N4O3SPurezza:98%Colore e forma:SolidPeso molecolare:444.45Ref: TM-T79167
Prodotto fuori produzioneTrimetoquinol HCl hydrate
CAS:Trimetoquinol hydrochloride possesses differential and selective beta-adrenergic properties.Formula:C19H26ClNO6Colore e forma:SolidPeso molecolare:399.87Ref: TM-T34950
Prodotto fuori produzioneSaxitoxinol
CAS:<p>Saxitoxinol is an analog of saxitoxin, a known voltage-gated sodium channel blocker.</p>Formula:C10H17N7O3Purezza:98%Colore e forma:SolidPeso molecolare:283.29Ref: TM-T68748
Prodotto fuori produzioneMEN11467
CAS:MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist for the study of acute colon cancer.Formula:C38H40N4O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:600.75SB251023
CAS:SB251023 is an agonist of β3-adrenoceptor.Formula:C28H34NO6PColore e forma:SolidPeso molecolare:511.55Cebranopadol ((1α,4α)stereoisomer)
CAS:<p>Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist.</p>Formula:C24H27FN2OPurezza:98%Colore e forma:SolidPeso molecolare:378.48Ref: TM-T10749
Prodotto fuori produzioneLp-PLA2-IN-12
CAS:<p>Lp-PLA2-IN-12 (compound 19), an Lp-PLA2 inhibitor, is utilized in researching neurodegenerative diseases including Alzheimer's disease (AD), glaucoma, age-</p>Formula:C24H23F2N5O3Purezza:98%Colore e forma:SolidPeso molecolare:467.47Ref: TM-T79010
Prodotto fuori produzioneOxitropium Bromide
CAS:Oxitropium bromide, a mAChR blocker, treats asthma and COPD as an anticholinergic bronchodilator.Formula:C19H26BrNO4Purezza:98%Colore e forma:SolidPeso molecolare:412.32Ref: TM-T16417
Prodotto fuori produzioneLp-PLA2-IN-16
CAS:<p>Lp-PLA2-IN-16 (Example 1) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential applications in Alzheimer's disease research [1].</p>Formula:C22H17F5N4O3Purezza:98%Colore e forma:SolidPeso molecolare:480.39Ref: TM-T79076
Prodotto fuori produzioneALPK1-IN-1
CAS:<p>ALPK1-IN-1 (A001) strongly inhibits ALPK1, key for innate immunity & NF-κB signaling via TIFA/TRAF.</p>Formula:C25H32N6O2SColore e forma:SolidPeso molecolare:480.63Ref: TM-T63176
Prodotto fuori produzioneanti-TNBC agent-2
CAS:<p>Anti-TNBC agent-2 (3j), a purine derivative, acts as an anti-triple negative breast cancer (TNBC) therapeutic.</p>Formula:C28H37ClFN7OPurezza:98%Colore e forma:SolidPeso molecolare:542.09Ref: TM-T79699
Prodotto fuori produzioneanti-TNBC agent-3
CAS:<p>Anti-TNBC agent-3 (compound 3g) is a compound that induces apoptosis and possesses anti-cancer cell proliferation properties.</p>Formula:C29H39F2N7OColore e forma:SolidPeso molecolare:539.66Ref: TM-T79410
Prodotto fuori produzioneYM 298198 Hydrochloride
CAS:YM 298198 HCl: non-competitive mGlu1 antagonist, Ki=19 nM. Inactive on mGlu2-7, stronger than CPCCOEt.Formula:C18H22N4OSColore e forma:SolidPeso molecolare:342.46Ref: TM-T71764
Prodotto fuori produzioneCK176
CAS:CK176 is an HIV-1 inhibitor, 11x more effective than I-XW-053 in human PBMCs.Formula:C21H12IN3O2Purezza:98%Colore e forma:SolidPeso molecolare:465.24Ref: TM-T27030
Prodotto fuori produzioneCH-100
CAS:CH-100 is a Chinese herbal medicine previously used in the treatment of human hepatitis C.Formula:C14H22ClNO3Colore e forma:SolidPeso molecolare:287.78Ref: TM-T30866
Prodotto fuori produzionePL265
CAS:<p>PL265 is a long-acting dual ENKephalinase inhibitor (DENKi) with analgesic potential.</p>Formula:C27H35N2O9PPurezza:98%Colore e forma:SolidPeso molecolare:562.55D(-)-Octopamine CSA salt
CAS:D(-)-Octopamine CSA salt is an agonist of octopamine receptors.Formula:C18H27NO6SPurezza:98%Colore e forma:SolidPeso molecolare:385.48Ref: TM-T27116
Prodotto fuori produzionePSB-6426
CAS:PSB-6426 is the first potent and selective human nucleoside triphosphate diphosphohydrolase-2 inhibitor.Formula:C22H29N4O10PPurezza:98%Colore e forma:SolidPeso molecolare:540.46Ref: TM-T24681
Prodotto fuori produzioneHPK1-IN-18
CAS:<p>HPK1-IN-18: Potent, specific inhibitor of HPK1, a MAP4K enzyme, for cancer research and treatment.</p>Formula:C24H24N4Colore e forma:LiquidPeso molecolare:368.47Ref: TM-T61449
Prodotto fuori produzionePS372424 HCl
CAS:<p>PS372424 activates CXCR3, triggers ERK phosphorylation, and inhibits CXCL11's effect on CD45+ cell migration in humanized mice.</p>Formula:C33H45ClN6O4Colore e forma:SolidPeso molecolare:625.21Ref: TM-T70411
Prodotto fuori produzionePAD4-IN-2
CAS:<p>PAD4-IN-2 (compound 5i) is a PAD4 inhibitor with an IC50 value of 1.94 μM, shown to suppress tumor growth in mice through specific inhibition of the PAD4-H3cit-</p>Formula:C20H23BClN7O6Colore e forma:SolidPeso molecolare:503.7Ref: TM-T79276
Prodotto fuori produzioneKP372-1
CAS:<p>KP372-1, an Akt inhibitor, blocks PI3K signaling, arrests cell growth, and triggers apoptosis in head/neck squamous cell carcinoma.</p>Formula:C20H8N12O2Colore e forma:SolidPeso molecolare:448.36Erythrityl Tetranitrate
CAS:<p>Erythrityl Tetranitrate, a vasodilator similar to nitroglycerin, was first in "sustained release" tablets; may cause "nitro headache."</p>Formula:C4H6N4O12Colore e forma:SolidPeso molecolare:302.11Ref: TM-T31671
Prodotto fuori produzioneCGP 44532
CAS:CGP 44532 a GABAB receptor agonist.Formula:C4H12NO3PPurezza:98%Colore e forma:SolidPeso molecolare:153.12Ref: TM-T26991
Prodotto fuori produzioneGacyclidine
CAS:Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.Formula:C16H25NSPurezza:99.85% - 99.92%Colore e forma:SolidPeso molecolare:263.44FGFR1 inhibitor-10
CAS:<p>FGFR1 inhibitor-10 (Compound 4i), with an IC50 of 28 nM, effectively inhibits FGFR1 phosphorylation.</p>Formula:C26H30F3N7O2SPurezza:98%Colore e forma:SolidPeso molecolare:561.62Ref: TM-T79686
Prodotto fuori produzioneH 35-25
CAS:H 35-25 is a beta 2-antagonist.Formula:C13H21NOColore e forma:SolidPeso molecolare:207.31Ref: TM-T70895
Prodotto fuori produzioneFostedil
CAS:Fostedil enhances heart function, maintains blood flow during partial/total coronary occlusions, and lowers aortic pressure.Formula:C18H20NO3PSPurezza:98%Colore e forma:SolidPeso molecolare:361.4Ref: TM-T27351
Prodotto fuori produzioneAMPK activator C2
CAS:AMPK activator C2 is an AMPK allosteric activator.Formula:C7H6NO6PPurezza:98%Colore e forma:SolidPeso molecolare:231.1Ref: TM-T23734
Prodotto fuori produzioneAlbuterol stearate
CAS:<p>Albuterol stearate, a salt form of Albuterol, is a selective beta2 agonist for treating asthma and COPD, with 29x preference for beta2 over beta1.</p>Formula:C31H57NO5Purezza:98%Colore e forma:SolidPeso molecolare:523.799Ref: TM-T25030
Prodotto fuori produzioneUBP1112
CAS:group III mGlu receptor antagonistFormula:C10H14NO5PPurezza:98%Colore e forma:SolidPeso molecolare:259.2Ref: TM-T23491
Prodotto fuori produzioneFM-24 HCl
CAS:FM-24 HCl is a long acting beta-adrenergic receptor antagonist.Formula:C19H30ClNO2Colore e forma:SolidPeso molecolare:339.9Ref: TM-T68856
Prodotto fuori produzioneAzilsartan mepixetil potassium
CAS:<p>Azilsartan medoxomil potassium (QR-01019K), an angiotensin II receptor antagonist, exhibits a potent and sustained antihypertensive effect, along with a more</p>Formula:C36H33KN6O8Colore e forma:SolidPeso molecolare:716.78BTK-IN-25
CAS:<p>BTK-IN-25 (compound 71) is a potent BTK inhibitor, demonstrating an IC50 of 0.77 nM against BTK(C481S) and achieving an IC50 of 1 nM in DOHH2 cells [1].</p>Formula:C28H27F2N3O5Purezza:98%Colore e forma:SolidPeso molecolare:523.53BTK-IN-27
CAS:<p>BTK-IN-27 (example 8), a potent BTK inhibitor with an IC50 of 0.2 nM, demonstrates anti-proliferative effects in TMD8 cells with an IC50 of less than 5 nM.</p>Formula:C31H35N7O2Purezza:98%Colore e forma:SolidPeso molecolare:537.66AEF0117
CAS:<p>AEF0117 is a signaling inhibitor of CB1-SSi that inhibits cannabinoid self-administration and can be used to study cannabis withdrawal.</p>Formula:C29H40O3Purezza:99.58%Colore e forma:SolidPeso molecolare:436.63RIOK2-IN-2
CAS:<p>RIOK2-IN-2 (8) functions as an inhibitor of RIOK2, exhibiting IC50 values of 3.02 μM in MKN-1 cells and 5.34 μM in MOLT4 cells [1].</p>Formula:C27H23F3N6O2Colore e forma:SolidPeso molecolare:520.51APG-2449
CAS:<p>APG-2449 is an orally active inhibitor targeting ALK, ROS1, and FAK, demonstrating antitumor efficacy in mouse models of non-small cell lung cancer (NSCLC) [1].</p>Formula:C33H42ClN5O4SPurezza:98%Colore e forma:SolidPeso molecolare:640.24Ref: TM-T79363
Prodotto fuori produzioneAntitumor photosensitizer-1
CAS:<p>Antitumor Photosensitizer-1 (Compound 8) is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-toxicity,</p>Formula:C42H51N5O6Colore e forma:SolidPeso molecolare:721.88Mal-VC-PAB-PNP-CDN-A
CAS:<p>Mal-VC-PAB-PNP-CDN-A is a conjugate comprised of an agent and a linker, utilized in antibody-drug conjugates (ADC) [1] [2].</p>Formula:C51H67N17O20P2Colore e forma:SolidPeso molecolare:1300.13I5B2
CAS:<p>I5B2 is a novel phosphorus-containing angiotensin I converting enzyme inhibitor. Angiotensin I converting enzyme is produced by Actinomadura sp.</p>Formula:C23H32N3O7PPurezza:98%Colore e forma:SolidPeso molecolare:493.49Ref: TM-T25515
Prodotto fuori produzioneLerzeparib
CAS:<p>Lerzeparib is a PARP (ADP-ribose polymerase) inhibitor that exhibits antineoplastic activity [1].</p>Formula:C21H20FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:365.4JAK-IN-34
CAS:<p>JAK-IN-34 (compound 11n) is a potent inhibitor of Janus kinases (JAKs), demonstrating IC50 values of 0.40 nM for JAK1, 0.83 nM for JAK2, 2.10 nM for JAK3,</p>Formula:C27H26N6OPurezza:98%Colore e forma:SolidPeso molecolare:450.53BCR-ABL-IN-8
CAS:<p>BCR-ABL-IN-8 (compound 26f) is a BCR-ABL inhibitor featuring a trimethoxy group [1].</p>Formula:C30H33N7O5Purezza:98%Colore e forma:SolidPeso molecolare:571.63Bumetanide sodium
CAS:Bumetanide sodium, a potent diuretic, blocks NKCC1 (IC50: 0.68 μM) and NKCC2 (IC50: 4.0 μM).Formula:C17H19N2NaO5SColore e forma:SolidPeso molecolare:386.4Ref: TM-T61713
Prodotto fuori produzioneL 689037
CAS:L 689037 is an inhibitor of leukotriene biosynthesis.Formula:C36H37ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:597.14Ref: TM-T24337
Prodotto fuori produzioneImmune cell migration-IN-1
CAS:<p>Immune cell migration-IN-1 (compound 2) serves as a potent inhibitor of immune cell migration, with potential research applications for mitigating conditions</p>Formula:C30H25ClN4O6SColore e forma:SolidPeso molecolare:605.06YK-029A
CAS:<p>YK-029A, an orally active EGFR mutant inhibitor, targets both EGFR T790M and EGFRex20ins mutations.</p>Formula:C27H32N8O2Purezza:98%Colore e forma:SolidPeso molecolare:500.6Ref: TM-T79461
Prodotto fuori produzionediMal-O-CH2COOH
CAS:<p>DiMal-O-CH2COOH is a cleavable linker utilized in antibody-drug conjugates (ADCs).</p>Formula:C13H12N2O7Colore e forma:SolidPeso molecolare:308.24Py-MAA-Val-Cit-PAB-MMAE
CAS:<p>Py-MAA-Val-Cit-PAB-MMAE (AAJ8D6-PY-Val-Cit-MMAE) serves as an ADC linker for Zapadcine-3a, a broad-spectrum anti-TRAILR2 ADC with antineoplastic properties.</p>Formula:C72H111N13O16SColore e forma:SolidPeso molecolare:1446.79IDO1-IN-22
CAS:<p>IDO1-IN-22 (Compound 3) is an inhibitor of IDO1, demonstrating potent activity with biochemical hIDO1 IC50 of 67.4 nM and HeLa hIDO1 IC50 of 17.6 nM.</p>Formula:C12H12BrFN6O3Purezza:98%Colore e forma:SolidPeso molecolare:387.16LM2I
CAS:<p>LM2I, a derivative of Spinosyn A (SPA), serves both as an argininosuccinate synthase (ASS1) enzyme activator and a tumor inhibitor through direct interaction</p>Formula:C47H77N3O11Colore e forma:SolidPeso molecolare:860.13FAP-IN-2
CAS:<p>FAP-IN-2 is a 99mTc-labeled, isonitrile-containing derivative of a fibroblast activation protein (FAPI) inhibitor suitable for tumor imaging [1].</p>Formula:C24H28F2N6O3Colore e forma:SolidPeso molecolare:486.51Antibacterial agent 157
CAS:<p>Compound B12 (Antibacterial agent 157) is a fungicidal agent that can impact protein synthesis in Botrytis cinerea.</p>Formula:C26H23BrF4N2O3Colore e forma:SolidPeso molecolare:567.37Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE
CAS:<p>Compound S6, Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE, is a potent anticancer agent specifically activated by the tumor microenvironment; it demonstrates efficacy</p>Formula:C67H101N11O16Purezza:98%Colore e forma:SolidPeso molecolare:1316.58STAT3-IN-18
CAS:<p>STAT3-IN-18 (compound SPP), a platinum (IV) complex featuring an axial ligand from sandalwood, suppresses the JAK2-STAT3 pathway in breast cancer (BC) cells and</p>Formula:C18H24Cl2N2O6PtPurezza:98%Colore e forma:SolidPeso molecolare:630.38Insecticidal agent 6
CAS:<p>Compound Im (Insecticidal agent 6) is a potent inhibitor of insect ryanodine receptors (RyRs), exhibiting an EC50 of 0.6308 µM against S.</p>Formula:C19H14BrCl2N5O4Purezza:98%Colore e forma:SolidPeso molecolare:527.16Canlitinib
CAS:<p>Canlitinib, a tyrosine kinase inhibitor, holds potential for cancer research.</p>Formula:C33H31F2N3O7Purezza:98%Colore e forma:SolidPeso molecolare:619.61JAK1-IN-11
CAS:<p>JAK1-IN-11 (compound 11) serves as a potent inhibitor of Janus kinases, exhibiting nanomolar inhibitory concentrations with IC50 values of 0.02 nM (JAK1) and 0.</p>Formula:C26H36N6O4SPurezza:98%Colore e forma:SolidPeso molecolare:528.67TrkB-IN-1
CAS:<p>TrkB-IN-1 is a potent, orally active agonist of the TrkB receptor, with favorable pharmacokinetic (PK) properties.</p>Formula:C19H16N2O6Purezza:98%Colore e forma:SolidPeso molecolare:368.34SARS-CoV-2-IN-68
CAS:<p>SARS-CoV-2-IN-68 (compound 6C) is a covalent inhibitor of both SARS-CoV-2 PLpro and Mpro, exhibiting potent antiviral properties by targeting the Zn-finger</p>Formula:C14H12N2OSePurezza:98%Colore e forma:SolidPeso molecolare:303.22Mal-cyclohexane-Gly-Gly-Phe-Gly-Exatecan
CAS:<p>Mal-cyclohexane-Gly-Gly-Phe-Gly-Exatecan is a linker molecule employed in the synthesis of antibody-drug conjugates (ADCs), demonstrating potent antitumor</p>Formula:C55H60FN9O13Colore e forma:SolidPeso molecolare:1074.12URAT1&XO inhibitor 1
CAS:<p>URAT1&XO Inhibitor 1 (compound 29) serves as a dual inhibitor with IC50 values of approximately 10 μM for URAT1 and 1.01 μM for Xanthine Oxidase.</p>Formula:C20H13N5O3SPurezza:98%Colore e forma:SolidPeso molecolare:403.41Ref: TM-T79175
Prodotto fuori produzioneDiaFluo
CAS:<p>DiaFluo is a probe for protein S-sulfinylation from cells.</p>Formula:C32H32N4O9SColore e forma:SolidPeso molecolare:648.69CIAC001
CAS:<p>CIAC001, a pyruvate kinase PKM2 inhibitor, exhibits anti-neuroinflammatory properties.</p>Formula:C20H25N3O2Colore e forma:SolidPeso molecolare:339.43Ref: TM-T79637
Prodotto fuori produzioneSHP2-IN-14
CAS:<p>SHP2-IN-14 (compound 27) is a potent, orally active allosteric inhibitor of SHP2, displaying strong anti-tumor activity with an IC50 of 7 nM.</p>Formula:C22H20Cl2N8OColore e forma:SolidPeso molecolare:483.35Ref: TM-T79108
Prodotto fuori produzioneEstrogen receptor modulator 8
CAS:<p>Estrogen Receptor Modulator 8 (compound 4) is an orally active inhibitor targeting Estrogen Receptor/ERR α with potent efficacy (IC50 = 0.437 nM in MCF-7 cells</p>Formula:C25H24F4N2O2Purezza:98%Colore e forma:SolidPeso molecolare:460.46ATR-IN-24
CAS:<p>ATR-IN-24 (Compound 1) is an ATR inhibitor with demonstrated anticancer activity [1].</p>Formula:C23H26N6O2Purezza:98%Colore e forma:SolidPeso molecolare:418.49Ref: TM-T79058
Prodotto fuori produzioneAntitumor agent-104
CAS:<p>Antitumor Agent-104 (Compound 9) serves as an antineoplastic by impeding DNA repair mechanisms in tumor cells, primarily through the inhibition of PARP1 enzyme</p>Formula:C31H33FN6O3Purezza:98%Colore e forma:SolidPeso molecolare:556.63URAT1 inhibitor 5
CAS:<p>URAT1 Inhibitor 5 (compound 16) serves as a powerful inhibitor of URAT1 and is utilized in hyperuricemia research [1].</p>Formula:C18H14BrN3O2SColore e forma:SolidPeso molecolare:416.29Antibacterial agent 160
CAS:<p>Antibacterial Agent 160 is a potent antibacterial agent that rapidly eradicates bacteria and inhibits the formation of bacterial biofilms.</p>Formula:C29H27ClFN3O6Colore e forma:SolidPeso molecolare:567.99BBDDL2059
CAS:<p>BBDDL2059 is a selective covalent inhibitor targeting EZH2, exhibiting an IC50 of 1.5 nM against the EZH2-Y641F mutant.</p>Formula:C27H36N4O4SPurezza:98%Colore e forma:SolidPeso molecolare:512.66Ref: TM-T79200
Prodotto fuori produzioneCap-dependent endonuclease-IN-9
CAS:<p>Cap-dependent endonuclease-IN-9, a strong influenza inhibitor, shows low toxicity, good pharmacokinetics, and dynamic action.</p>Formula:C29H22F2N4O7SPurezza:98%Colore e forma:SolidPeso molecolare:608.57Ref: TM-T72125
Prodotto fuori produzioneSyk-IN-8
CAS:<p>Syk-IN-8 (compound 19q) functions as a Syk inhibitor with demonstrated antiproliferative effects on a variety of hematological tumor cells.</p>Formula:C23H26N10Purezza:98%Colore e forma:SolidPeso molecolare:442.52VISTA-IN-2
CAS:<p>VISTA-IN-2 (Compound 1) is a V-domain Ig suppressor of T-cell activation (VISTA) inhibitor that promotes the degradation of VISTA in cells via autophagy,</p>Formula:C23H23N3OPurezza:98%Colore e forma:SolidPeso molecolare:357.45Ref: TM-T79653
Prodotto fuori produzioneAnti-MI/R injury agent 1
CAS:<p>Anti-MI/R injury agent 1 (compound 18), derived from Panaxatriol, represents an orally administered, potent agent against myocardial ischemia/reperfusion (MI/R</p>Formula:C32H49NO6Colore e forma:SolidPeso molecolare:543.73Omeprazole acid
CAS:Omeprazole treats GERD, ulcers, Zollinger-Ellison syndrome, prevents GI bleeding; it's a proton pump inhibitor.Formula:C34H32N6Na2O10S2Colore e forma:SolidPeso molecolare:794.76Ref: TM-T71980
Prodotto fuori produzioneTauro-Obeticholic Acid sodium
CAS:<p>Tauro-obeticholic acid, a farnesoid X receptor (FXR) agonist and semisynthetic derivative of chenodeoxycholic acid, is an active metabolite of obeticholic acid.</p>Formula:C28H48NO6S·NaColore e forma:SolidPeso molecolare:549.74Igermetostat
CAS:<p>Igermetostat, an EZH2 inhibitor, is utilized both in vivo and in vitro for cancer research [1].</p>Formula:C32H46N4O4Purezza:98%Colore e forma:SolidPeso molecolare:550.73CYY292
CAS:<p>CYY292 is a chemical compound acting as an inhibitor of PDGFRα, PDGFRβ, FGFR1, -2, and -3, with respective IC50 values of 5.35, 4.6, 28, 28, and 78 nM.</p>Formula:C24H28N8OColore e forma:SolidPeso molecolare:444.53BET-IN-14
CAS:<p>BET-IN-14 is a pan BET inhibitor with an IC50 of 5.35 nM, demonstrating oral activity and anticancer properties [1].</p>Formula:C30H37N7O2Purezza:98%Colore e forma:SolidPeso molecolare:527.66Yhhu6669
CAS:<p>Yhhu6669 is an anti-HBV agent that suppresses viral DNA and replication by promoting DNA-free capsid assembly, effectively reducing HBV DNA and HBcAg levels in</p>Formula:C29H28ClFN6O3Purezza:98%Colore e forma:SolidPeso molecolare:563.02Ref: TM-T78756
Prodotto fuori produzioneDDO-2213
CAS:<p>DDO-2213 is a potent, orally active inhibitor of the WDR5-MLL1 interaction, demonstrating an IC50 of 29 nM and a Kd of 72.9 nM against WDR5.</p>Formula:C24H27ClFN7OColore e forma:SolidPeso molecolare:483.97And1-IN-1
CAS:<p>And1-IN-1, also known as compound III, is a potent inhibitor of And1 [1].</p>Formula:C15H11BCl2O2Colore e forma:SolidPeso molecolare:304.96MDVN1003
CAS:MDVN1003 inhibits BTK & PI3Kδ in B cells, blocking NHL growth; it kills lymphoma cells, not erythroblasts.Formula:C22H20FN7OPurezza:98%Colore e forma:SolidPeso molecolare:417.44Ref: TM-T28008
Prodotto fuori produzioneEST73502
CAS:<p>EST73502 is a compound that functions as a dual agonist for the μ-opioid receptor (MOR) and an antagonist for the σ1 receptor (σ1R). It is selective, orally active, and possesses the ability to penetrate the blood-brain barrier (BBB). The compound exhibits a Ki value of 64 nM for the MOR and 118 nM for the σ1R. Additionally, EST73502 demonstrates antinociceptive activity [1].</p>Formula:C19H26F2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:352.426(αR)-Cyclopropaneacetamide-Exatecan
CAS:<p>(αR)-Cyclopropaneacetamide-Exatecan (compound 2-A), an Exenotecan derivative, serves as a cytotoxic agent that effectively inhibits the proliferation of U87MG</p>Formula:C29H28FN3O6Colore e forma:SolidPeso molecolare:533.55MOR agonist-1
CAS:<p>MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associated</p>Formula:C22H26ClFN2O2Purezza:98%Colore e forma:SolidPeso molecolare:404.91S-72
CAS:<p>S-72 acts as a microtubule polymerization inhibitor, effective in cell-free assays at concentrations of 1, 3, and 10 µM.</p>Formula:C20H22N4O3SColore e forma:SolidPeso molecolare:398.50Ref: TM-T83874
Prodotto fuori produzioneFLT3-IN-19
CAS:<p>FLT3-IN-19 (Comp 50) is a potent, selective inhibitor of FLT3, demonstrating an IC50 value of 0.213 nM, and is applicable in research pertaining to acute</p>Formula:C22H26N8OColore e forma:SolidPeso molecolare:418.49VMAT2-IN-2 tosylate
CAS:<p>VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].</p>Formula:C27H36F3NO6SPurezza:98%Colore e forma:SolidPeso molecolare:559.64Ref: TM-T79061
Prodotto fuori produzioneXilmenolone
CAS:<p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>Formula:C26H37N3O2Purezza:98%Colore e forma:SolidPeso molecolare:423.59Ref: TM-T78670
Prodotto fuori produzioneLT-540-717
CAS:<p>LT-540-717 (compound 32), a potent FLT3 inhibitor (IC50=0.62 nM), exhibits antiproliferative activity and effectively inhibits various acquired FLT3 mutations,</p>Formula:C24H24N8O2Colore e forma:SolidPeso molecolare:456.5Ref: TM-T79490
Prodotto fuori produzioneBelfosdil
CAS:Belfosdil is a blocker of antihypertensive calcium channel.Formula:C27H50O7P2Purezza:98%Colore e forma:SolidPeso molecolare:548.63Ref: TM-T26764
Prodotto fuori produzioneDPP
CAS:<p>DPP, a Platinum(IV) complex with a pterostilbene-derived axial ligand, inhibits the JAK2-STAT3 pathway in breast cancer (BC) cells, demonstrating</p>Formula:C36H40Cl2N2O10PtPurezza:98%Colore e forma:SolidPeso molecolare:926.7Davelizomib
CAS:<p>Davelizomib is a proteasome inhibitor that exhibits antineoplastic activity [1].</p>Formula:C21H26BF2N3O7Purezza:98%Colore e forma:SolidPeso molecolare:481.25JAK-IN-27
CAS:<p>JAK-IN-27, also known as compound 1, is an orally active, potent inhibitor of the JAKS family kinases, displaying inhibitory concentrations (IC50s) of 3.0 nM</p>Formula:C20H21F2N7OPurezza:98%Colore e forma:SolidPeso molecolare:413.42IDO/Tubulin-IN-2
CAS:<p>IDO/Tubulin-IN-2 inhibits TDO/tubulin, effective on U87, HepG2, A549, HCT-116, LO2 cancer cells; IC50 values 0.036-1.04 μM, boosts antitumor action.</p>Formula:C48H40N6O10Colore e forma:SolidPeso molecolare:860.87Ref: TM-T74536
Prodotto fuori produzioneS1P1 agonist 6
CAS:<p>Compound I (S1P1 agonist 6) is an S1P1 agonist that mitigates autoimmune activity by inhibiting lymphocyte trafficking and has potential as an immunosuppressive</p>Formula:C25H26F3NO3Purezza:98%Colore e forma:SolidPeso molecolare:445.47FOXM1-IN-2
CAS:<p>FOXM1-IN-2, a FOXM1 inhibitor, exhibits antineoplastic activity [1].</p>Formula:C48H47F4N7O12SColore e forma:SolidPeso molecolare:1021.99I-BET282
CAS:<p>BET-IN-1 is a bromodomain inhibitor extracted from patent WO/2013024104A1 (example 2, plC50: 6.0 - 7.0).</p>Formula:C25H30N4O4Purezza:98%Colore e forma:SolidPeso molecolare:450.53Tibremciclib
CAS:<p>Tibremciclib is a cyclin-dependent kinase 4 (CDK4) inhibitor that exhibits antineoplastic properties [1].</p>Formula:C28H32F2N8Purezza:98%Colore e forma:SolidPeso molecolare:518.6ALPK1-IN-3
CAS:<p>ALPK1-IN-3,serves as an ALPK1 inhibitor that dampens proinflammatory gene expression in the kidney and enhances survival in animal models of sepsis-induced</p>Formula:C20H16F2N4OSPurezza:98%Colore e forma:SolidPeso molecolare:398.43ROCK2-IN-6
CAS:<p>ROCK2-IN-6 (Comp A) is a selective inhibitor of ROCK2, applicable in the study and treatment of ROCK-mediated, autoimmune, and inflammatory diseases [1].</p>Formula:C26H21F2N7OPurezza:98%Colore e forma:SolidPeso molecolare:485.49CGP 56999A
CAS:CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.Formula:C19H30NO5PPurezza:98%Colore e forma:SolidPeso molecolare:383.42Ref: TM-T26993
Prodotto fuori produzioneHPK1-IN-38
CAS:<p>HPK1-IN-38 (compound 15) is an inhibitor of MAP4K1/HPK1, suitable for research into disorders related to HPK1 [1].</p>Formula:C29H29N5O3Colore e forma:SolidPeso molecolare:495.57PI3Kδ-IN-13
CAS:<p>PI3Kδ-IN-13 (compound 89), with an IC50 value of 2.6 nM, is an inhibitor of PI3Kδ, applicable for researching diseases involving cell proliferation, including</p>Formula:C27H39N7O4S2Colore e forma:SolidPeso molecolare:589.77Antitumor photosensitizer-2
CAS:<p>Compound 11, also known as Antitumor Photosensitizer-2, is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-</p>Formula:C40H47N5O7Colore e forma:SolidPeso molecolare:709.83Civorebrutinib
CAS:<p>Civorebrutinib (WS-413) is an inhibitor of Bruton's tyrosine kinase that exhibits antineoplastic activity [1].</p>Formula:C23H22ClN7O2Colore e forma:SolidPeso molecolare:463.92HBV-IN-38
CAS:<p>HBV-IN-38 (Example 193), an HBV DNA inhibitor with an EC50 value of ≤100 nM, serves as a research tool for investigating viral infections [1].</p>Formula:C18H16F3N5O4S2Purezza:98%Colore e forma:SolidPeso molecolare:487.48JAK1-IN-10
CAS:<p>JAK1-IN-10 (compound 9), a cyano-substituted cyclic hydrazine derivative, functions as a potent and selective inhibitor of JAK1 [1].</p>Formula:C15H17N7Purezza:98%Colore e forma:SolidPeso molecolare:295.34JDB175
CAS:<p>JDB175, a selective BTK inhibitor with oral bioavailability, demonstrates excellent penetration through the blood-brain barrier.</p>Formula:C26H21F3N4O2Purezza:98%Colore e forma:SolidPeso molecolare:478.47MDL-811
CAS:<p>MDL-811, an allosteric activator of SIRT6, markedly enhances the deacetylation of histone H3 at lysine residues 9, 18, and 56 (H3K9Ac, H3K18Ac, and H3K56Ac),</p>Formula:C25H25BrCl2FN3O5S2Purezza:98%Colore e forma:SolidPeso molecolare:681.42LFS-1107
CAS:<p>LFS-1107, a reversible CRM1 inhibitor (Kd: 12.5 pM), selectively targets and eliminates ENKTL cells, offering potential for cancer research applications [1].</p>Formula:C12H11N5OS2Purezza:98%Colore e forma:SolidPeso molecolare:305.38Sakura 6
CAS:<p>Sakura 6, a synthetic serotonin transporter (SERT)-binding peptide, enhances the interaction between SERT and neuronal nitric oxide synthase.</p>Formula:C31H45N5O7Colore e forma:SolidPeso molecolare:599.73Bi-Mc-VC-PAB-MMAE
CAS:<p>Bi-Mc-VC-PAB-MMAE is an agent-linker conjugate for antibody-drug conjugates (ADCs), featuring the linker (Fmoc-Val-Cit-PAB) and the potent tubulin inhibitor (</p>Formula:C71H104N12O18Colore e forma:SolidPeso molecolare:1413.66PHI-101
CAS:<p>PHI-101 is a checkpoint kinase 2 (Chk2) inhibitor that can be used for the study of refractory acute myeloid leukemia (AML) and ovarian cancer.</p>Formula:C19H19FN4O2SPurezza:99.4%Colore e forma:SolidPeso molecolare:386.44ALS-I-41
CAS:ALS-I-41 is a novel, potent and selective antagonist of oxytocin receptor.Formula:C30H38FN3O6SPurezza:98%Colore e forma:SolidPeso molecolare:587.7Ref: TM-T26602
Prodotto fuori produzioneDG026
CAS:DG026 selectively inhibits IRAP, reducing its cross-presentation in dendritic cells without affecting ERAP1.Formula:C35H40N3O4PPurezza:98%Colore e forma:SolidPeso molecolare:597.68Ref: TM-T27160
Prodotto fuori produzioneIfetroban
CAS:<p>Ifetroban is a potent and selective TxA2/PGH2 receptor antagonist.</p>Formula:C25H32N2O5Colore e forma:SolidPeso molecolare:440.53Ref: TM-T27588
Prodotto fuori produzioneROCK-IN-6
CAS:<p>ROCK-IN-6, a selective ROCK2 inhibitor, exhibits potent inhibition with an IC50 of 2.19 nM and holds promise for research into glaucoma and retinal diseases [1</p>Formula:C19H19N5O8SPurezza:98%Colore e forma:SolidPeso molecolare:477.45Ref: TM-T79077
Prodotto fuori produzioneBPH-628
CAS:<p>BPH-628 is a bioactive chemical.</p>Formula:C20H20O7P2Colore e forma:SolidPeso molecolare:434.32Cortivazol
CAS:Cortivazol is an Anti-Inflammatory Drug.Formula:C32H38N2O5Purezza:98%Colore e forma:SolidPeso molecolare:530.65Ref: TM-T25271
Prodotto fuori produzioneIfetroban sodium
CAS:<p>Ifetroban sodium (BMS-180291), oral TXA2/PGH2 antagonist for researching heart, stroke, BP, thrombosis.</p>Formula:C25H31N2NaO5Colore e forma:SolidPeso molecolare:462.522Ref: TM-T62924
Prodotto fuori produzioneDimethandrolone Undecanoate
CAS:Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.Formula:C31H50O3Purezza:99.65% - >99.99%Colore e forma:SolidPeso molecolare:470.73Ref: TM-T27176
Prodotto fuori produzionehDHODH-IN-8
<p>hDHODH-IN-8 is a potent human dihydroorotic dehydrogenase (hDHODH) inhibitor (IC50: 16 nM) that exhibits potent antiproliferative effects and has good water solubility, with potential for oncology studies, especially in lymphoma.</p>Formula:C21H15F6N3O4Purezza:98%Peso molecolare:487.35
