Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.524 prodotti)
- Apoptosi(5.793 prodotti)
- Ciclo cellulare/Checkpoint(4.452 prodotti)
- Cromatina/Epigenetica(2.242 prodotti)
- Segnalazione citoscheletrica(1.382 prodotti)
- Danno al DNA/Riparazione del DNA(2.826 prodotti)
- Endocrinologia/Ormoni(3.507 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.333 prodotti)
- Immunologia e infiammazione(3.527 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.203 prodotti)
- Trasportatore di membrana/canale ionico(2.792 prodotti)
- Metabolismo(9.449 prodotti)
- Microbiologia/Virologia(6.981 prodotti)
- Neuroscienza(9.926 prodotti)
- Altri inibitori(37.921 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.597 prodotti)
- Cellule staminali e Derivati(830 prodotti)
- Adattatori Tirosin-chinasi(2.015 prodotti)
- Ubiquitinazione(1.650 prodotti)
Mostrare 16 più sottocategorie
Trovati 66639 prodotti di "Inibitori"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Abarelix acetate
CAS:<p>Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.</p>Formula:C72H95ClN14O14·xC2H4O2Colore e forma:SolidPeso molecolare:1476.14Meclocycline
CAS:<p>Meclocycline: a tetracycline antibiotic, inhibits LDH, reduces cell toxicity from mutant huntingtin, doesn't change protein levels in PC12 cells.</p>Formula:C22H21ClN2O8Colore e forma:SolidPeso molecolare:476.86HIV-1 inhibitor-18
<p>HIV-1 inhibitor-18 blocks HIV-1 capsid, effective on NL4-3 strain (EC50: 5.14 μM), slightly toxic (MT-4CC50>9.51).</p>Formula:C27H31N3O6SColore e forma:SolidPeso molecolare:525.62IL-17 modulator 1 disodium
CAS:<p>Potent, orally active IL-17 Modulator 1 (disodium) from patent WO 2020127685, used in psoriasis and arthritis research.</p>Formula:C28H37N6NaO6PColore e forma:SolidPeso molecolare:607.604Steroid sulfatase/17β-HSD1-IN-3
<p>Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1).</p>Formula:C19H17ClN2O5SColore e forma:SolidPeso molecolare:420.87IRE1α kinase-IN-5
<p>IRE1α kinase-IN-5 (compound 7) is a potent inhibitor of IRE1α (Ki: 98 nM) and is an ATP-competitive ligand for IRE1α.</p>Formula:C28H30N6O3SColore e forma:SolidPeso molecolare:530.64Chitin synthase inhibitor 7
<p>Compound 9c, a chitin synthase inhibitor, has an IC50 of 0.37 nM and is useful for studying fungal infections.</p>Formula:C24H25N3O5Colore e forma:SolidPeso molecolare:435.47Cilazaprilat
CAS:<p>Cilazaprilat is the active metabolite of cilazapril, a pyridazine angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.</p>Formula:C20H27N3O5Colore e forma:SolidPeso molecolare:389.45ZK-Thiazolidinone
CAS:<p>ZK-Thiazolidinone (TAL), ATP-competitive PLK1 inhibitor, disrupts cell division processes in vitro and in vivo, targeting human/mouse tumors.</p>Formula:C23H26F3N5O2SColore e forma:SolidPeso molecolare:493.55sEH inhibitor-1
<p>TCPU (sEH inhibitor-1) is a potent oral human sEH blocker with IC50s of 0.4 nM (human) and 5.3 nM (mouse).</p>Colore e forma:SolidCD73-IN-2
<p>CD73-IN-2 is a potent inhibitor of CD73 (IC50: 0.09 nM).</p>Formula:C17H25ClN5O7PColore e forma:SolidPeso molecolare:477.84CYP11B1-IN-2
<p>CYP11B1-IN-2 selectively inhibits human and rat CYP11B1 (IC50: 9/25 nM) orally to research cortisol-related diseases.</p>Colore e forma:SolidAntifungal agent 28
<p>Antifungal 28 disrupts Candida, hits fluconazole-resistant strains, and inhibits biofilms.</p>Formula:C22H29N5OSColore e forma:SolidPeso molecolare:411.56(±)-HIP-B
CAS:<p>(±)-HIP-B is an excitatory amino acid transporter blocker.</p>Formula:C6H8N2O4Purezza:98%Colore e forma:SolidPeso molecolare:172.14LAF-153
CAS:<p>LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.</p>Formula:C18H32N2O7Colore e forma:SolidPeso molecolare:388.46SAR-114137
CAS:<p>SAR-114137 is a histone sphingomyelin kinase inhibitor used in the study of molluscum arteriosum and peripheral neuropathic pain.</p>Formula:C25H34N4O7SPurezza:99.09% - 99.91%Colore e forma:SolidPeso molecolare:534.63M3258
CAS:<p>LMP7-IN-1 may used in the research of inflammatory and autoimmune diseases, neurodegenerative diseases, proliferative diseases and cancer, is an inhibitor of</p>Formula:C17H20BNO5Purezza:98%Colore e forma:SolidPeso molecolare:329.16Tacrolimus anhydrous 8-epimer
CAS:<p>Tacrolimus anhydrous 8-epimer, an immunosuppressive l-pipecolic acid macrolide, blocks T cell growth by hindering IL-2.</p>Formula:C44H69NO12Colore e forma:SolidPeso molecolare:804.02STAT3-IN-9
<p>STAT3-IN-9 hinders STAT3 at Tyr705, doesn't affect STAT1 Tyr701, induces apoptosis, and arrests cells in G2/M phase.</p>Formula:C22H21N3O4Colore e forma:SolidPeso molecolare:391.42Topoisomerase I inhibitor 8
CAS:<p>Topoisomerase I inhibitor 8, a hexacyclic analogue of camptothecin, is also a potent inhibitor of topoisomerase I and is toxic to tumour cells.</p>Formula:C24H21FN2O4Colore e forma:SolidPeso molecolare:420.43GSK8814
CAS:GSK8814 is a selective and ATAD2/2B bromodomain chemical probe and inhibitor (binding constant pKd=8.1 and a pKi=8.9 in BROMOscan).Formula:C28H35F2N5O3Purezza:98%Colore e forma:SolidPeso molecolare:527.61BMS 310705
CAS:<p>BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.</p>Formula:C27H42N2O6SColore e forma:SolidPeso molecolare:522.70EGFR/HER2/DHFR-IN-1
<p>Potent EGFR/HER2/DHFR inhibitor for MCF-7 breast cancer; IC50: 0.153/0.108/0.291 μM; arrests G1/S phase, triggers apoptosis.</p>Formula:C14H11BrN4O2SColore e forma:SolidPeso molecolare:379.23α-Glucosidase-IN-17
CAS:<p>α-Glucosidase-IN-17 (Compound 12B) is a potent and orally active inhibitor of α-glucosidase, demonstrating antidiabetic activity with an inhibitory</p>Formula:C30H27NO2SColore e forma:SolidPeso molecolare:465.61IRAK4-IN-11
<p>IRAK4-IN-11 (compound 6) is a potent inhibitor of IRAK4 with an IC 50 of 0.008 μM. IRAK4-IN-11 exhibits cell pIRAK4 potencies with an IC 50 of 0.19 μM [1].</p>Formula:C16H19N7OColore e forma:SolidPeso molecolare:325.37Pociredir
CAS:<p>Pociredir (FTX-6058), a potent EED inhibitor (KD=0.163 nM), may help in SCD research.</p>Formula:C22H18FN5O2Colore e forma:SolidPeso molecolare:403.41SGLT inhibitor-1
CAS:<p>SGLT inhibitor-1 is a potentsodium glucose co-transporter proteins (SGLTs) dual inhibitor(hSGLT1 and hSGLT2 with IC50s of 43 nM and 9 nM, respectively).</p>Formula:C24H27FO8Purezza:98%Colore e forma:SolidPeso molecolare:462.46Elocalcitol
CAS:<p>Elocalcitol is a calcitriol analog for inhibition of prostate cell growth.</p>Formula:C29H43FO2Colore e forma:SolidPeso molecolare:442.65MEIS-IN-3
<p>MEIS-IN-3 is a potent inhibitor of MEIS.</p>Formula:C25H26N2O4Colore e forma:SolidPeso molecolare:418.48Saphenamycin
CAS:<p>Saphenamycin is an antibiotic from a strain of Streptomyces.</p>Formula:C23H18N2O5Purezza:98%Colore e forma:SolidPeso molecolare:402.40Sinulatumolin E
CAS:<p>Sinulatumolin E, a terpenoid, inhibits TNF-α (IC 50: 3.6 μM); has anti-inflammatory properties.</p>Formula:C15H22O2Colore e forma:SolidPeso molecolare:234.33Topo I-IN-1
<p>Topo I-IN-1 (14d) is a powerful Topo I inhibitor with antitumor effects and DNA intercalation, inducing apoptosis.</p>Formula:C20H14BrN3O2Colore e forma:SolidPeso molecolare:408.25Gabaculine HCl
CAS:<p>Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.</p>Formula:C7H10ClNO2Colore e forma:SolidPeso molecolare:175.61Y1 receptor antagonist 1
CAS:<p>Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.</p>Formula:C28H33N5O3Purezza:98.17%Colore e forma:SolidPeso molecolare:487.59Elacestrant S enantiomer dihydrochloride
<p>Elacestrant (RAD1901) dihydrochloride, an oral ERR degrader, has IC50 of 48 nM (ERα) and 870 nM (ERβ). Its S enantiomer has low activity.</p>Formula:C30H40Cl2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:531.56Ribocil-C R enantiomer
<p>Ribocil-C R enantiomer is the R enantiomer of Ribocil-C. Ribocil-C is a highly selective bacterial riboflavin riboswitches inhibitor.</p>Formula:C21H21N7OSPurezza:98%Colore e forma:SolidPeso molecolare:419.5PIM1-IN-3
<p>PIM1-IN-3 (HL8) selectively blocks PIM1, induces Colo320 cell apoptosis, and may be researched for cancer.</p>Formula:C27H25BrN6OColore e forma:SolidPeso molecolare:529.43DH376
CAS:<p>DH376 inhibits DAGLα in a time and dose dependent manner in mouse brain. DH376 shows picomolar activity.</p>Formula:C31H28F2N4O3Colore e forma:SolidPeso molecolare:542.58GNE-203
CAS:<p>GNE-203 is a Met inhibitor.</p>Formula:C30H29Cl2F3N8O3Colore e forma:SolidPeso molecolare:677.50L-365260 hemihydrate
<p>L-365260 hemihydrate: selective oral CCK-B/gastrin blocker, Ki=1.9/2.0 nM, competes with guinea pig receptors.</p>Formula:C24H24N4O3Colore e forma:SolidPeso molecolare:407.47rel-MDM2/4-p53-IN-3
<p>rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.</p>Formula:C25H24Cl2FN3O3Colore e forma:SolidPeso molecolare:504.38Seco-Duocarmycin SA
CAS:<p>Seco-Duocarmycin SA is a highly potent DNA alkylator used as an ADC cytotoxin.</p>Formula:C25H24ClN3O7Purezza:98%Colore e forma:SolidPeso molecolare:513.93H 218-54
CAS:<p>H 218-54 is a renin inhibitor.</p>Formula:C37H56N2O5SColore e forma:SolidPeso molecolare:640.92AZ-PFKFB3-67 quarterhydrate
<p>AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).</p>Formula:C26H27N5O4Colore e forma:SolidPeso molecolare:460.01TH-6
<p>TH-6, a potent HDAC inhibitor (IC50: HDAC1-0.115, 2-0.135, 3-0.242, 6-0.138, 8-2.120 μM), blocks cell migration, invasion, and has anti-tumor properties.</p>Formula:C22H24FN3O5Colore e forma:SolidPeso molecolare:429.44Saprisartan potassium
CAS:<p>Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.</p>Formula:C25H21BrF3KN4O4SColore e forma:SolidPeso molecolare:649.52HBV-IN-11
CAS:<p>HBV-IN-11 is a potent inhibitor of HBsAg secretion (EC50: 0.46 μM).</p>Formula:C21H24ClNO6Colore e forma:SolidPeso molecolare:421.87EGFR/BRAF-IN-1
<p>EGFR/BRAF-IN-1 inhibits EGFR/BRAF (BRAFV600E IC50: 45 nM, GI50: 35 nM) and has antioxidant properties.</p>Formula:C26H28ClN3O4Colore e forma:SolidPeso molecolare:481.97MtTMPK-IN-2
CAS:<p>MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).</p>Formula:C23H24ClN3O3Colore e forma:SolidPeso molecolare:425.91NK-1 Antagonist 1
CAS:<p>NK-1 Antagonist 1 is a NK-1 receptor antagonist.</p>Formula:C25H23F6N5O2Purezza:98%Colore e forma:SolidPeso molecolare:539.47Vindeburnol
CAS:<p>Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.</p>Formula:C17H20N2OColore e forma:SolidPeso molecolare:268.35(2R,3S)-Azelaprag
CAS:<p>(2R,3S)-N-(4-(2,6-dimethoxyphenyl)-5-(5-methylpyridin-3-yl)-4H-1,2,4-triazol-3-yl)-3-(5-methylpyrimidin-2-yl)butane-2-sulfonamide is an Apelin receptor agonist</p>Formula:C25H29N7O4SPurezza:97.47% - >99.99%Colore e forma:SoildPeso molecolare:523.61MAFP
CAS:<p>MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase.</p>Formula:C21H36FO2PColore e forma:SolidPeso molecolare:370.48CHF-6366
CAS:<p>CHF-6366: M3 antagonist & β2 agonist (pKi 10.4/11.4), mild Ca channel blocker, used in COPD study.</p>Formula:C42H48N6O8Colore e forma:SolidPeso molecolare:764.87LSD1-IN-18
<p>LSD1-IN-18 inhibits LSD1 (Ki: 0.156 μM, KD: 0.075 μM), blocking THP-1 and MDA-MB-231 cell growth (IC50: 0.16, 0.21 μM).</p>Formula:C31H40N6O2Colore e forma:SolidPeso molecolare:528.69PRMT5-IN-21
<p>PRMT5-IN-21 (compound 1) is a potent inhibitor of cyclonucleoside PRMT5.</p>Formula:C18H18F2N6O3Colore e forma:SolidPeso molecolare:404.37XP5
<p>XP5 is an oral HDAC6 inhibitor, potent against cancer cells, including YCC3/7 (IC50=31 nM to 2.31 μM).</p>Formula:C19H25N3O5SColore e forma:SolidPeso molecolare:407.48KRAS G12C inhibitor 15
CAS:<p>KRAS G12C inhibitor 15 is a potent KRAS G12C inhibitor .</p>Formula:C25H21ClF2N4O3Purezza:98%Colore e forma:SolidPeso molecolare:498.91P053
CAS:<p>P053: potent, selective CerS1 inhibitor, IC50 = 0.5µM, curbs muscle fat oxidation, affects body fat.</p>Formula:C18H21Cl2NO2Purezza:98%Colore e forma:SolidPeso molecolare:354.27Elongation factor P-IN-1
<p>EFP-IN-1: potent β-lysine derivative, inhibits EFP, slows E. coli growth.</p>Formula:C14H31N3O2Colore e forma:SolidPeso molecolare:273.41OMDM169
CAS:<p>OMDM169: potent/selective MAGL inhibitor, raises 2-AG, analgesic via cannabinoid receptors, IC50: 0.13-0.41μM in rat/COS-7, inactive at CB1/CB2.</p>Formula:C25H45NO5Purezza:98%Colore e forma:SolidPeso molecolare:439.63FTO-IN-6
CAS:<p>FTO-IN-6 is a selective inhibitor of fat mass and obesity associated protein (FTO).</p>Formula:C14H12N4O6Colore e forma:SolidPeso molecolare:332.27Antifungal agent 19
<p>Antifungal agent 19 shows the potent antifungal activity ( EC 50 = 0.72 μM).</p>Formula:C19H18F4O2Colore e forma:SolidPeso molecolare:354.34AD5075
CAS:<p>AD5075 is a bioactive chemical.</p>Formula:C22H20N2O5SColore e forma:SolidPeso molecolare:424.47Plumbemycin B
CAS:<p>Plumbemycin B is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Formula:C12H21N4O8PColore e forma:SolidPeso molecolare:380.29Asimicin
CAS:<p>Asimicin is a effective complex I inhibitor.</p>Formula:C37H66O7Purezza:98%Colore e forma:SolidPeso molecolare:622.922-Methylsorbinol
CAS:<p>2-Methylsorbinol is a bioactive chemical.</p>Formula:C12H11FN2O3Colore e forma:SolidPeso molecolare:250.23MsbA-IN-5
<p>MsbA-IN-5 (compound 40) is a potent and highly selective inhibitor of MsbA (IC50: 2 nM). MsbA-IN-5 can be used in Gram-negative studies.</p>Formula:C23H19Cl2N5OColore e forma:SolidPeso molecolare:452.34PKCiota-IN-1
CAS:<p>PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).</p>Formula:C25H22FN5OColore e forma:SolidPeso molecolare:427.47ChE/Aβ1-42-IN-1
<p>ChE/Aβ1-42-IN-1 (compound 28) is a potent aggregation inhibitor of ChE and Aβ 1-42 with excellent BBB permeability.</p>Formula:C19H24N2O3Colore e forma:SolidPeso molecolare:328.41Cacospongionolide B
CAS:<p>Cacospongionolide B from Fasciospongia cavernosa inhibits secretory phospholipase A2, curbing inflammation.</p>Formula:C25H36O4Colore e forma:SolidPeso molecolare:400.55HIV-1 inhibitor-44
<p>HIV-1 inhibitor-44 (compound 11l) is an HIV-1 reverse transcriptase inhibitor that exhibits activity against wild-type HIV-1 strains (EC50: 0.209 μM).</p>Formula:C23H26N2O4SColore e forma:SolidPeso molecolare:426.5314α-Demethylase/DNA Gyrase-IN-1
<p>14α-Demethylase/DNA Gyrase-IN-1 (Compound 7c) is a potent inhibitor of 14α-Demethylase/DNA Gyrase with antibacterial activity.</p>Formula:C26H22N4O4Colore e forma:SolidPeso molecolare:454.48VU6005806
CAS:<p>VU6005806 is a potent M4 PAM with EC50s: 94 nM (human), 28 nM (rat), 87 nM (dog), 68 nM (cyno); studied for neuropsychiatric disorders.</p>Formula:C17H16F3N7O2SPurezza:98%Colore e forma:SolidPeso molecolare:439.41BMS-986034
CAS:<p>BMS-986034 is a GPR119 agonist.</p>Formula:C24H24Cl2N6O4Colore e forma:SolidPeso molecolare:531.39MraY-IN-1
<p>MraY-IN-1 inhibits MraY (IC50: 140μM), fights E. coli K12, B. subtilis W23, P. fluorescens (MIC50: 7-46μg/ml), for antimicrobial research.</p>Formula:C35H46N3O5Colore e forma:SolidPeso molecolare:588.76LP-284
CAS:<p>LP-284 is a DNA alkylating agent effective against solid tumors and hematologic cancers like MCL.</p>Formula:C16H20N2O4Colore e forma:SolidPeso molecolare:304.34Resolvin D1 methyl ester
CAS:<p>Resolvin D1, from docosahexaenoic acid via 15-/5-lipoxygenase, curbs acute inflammation; EC50 ~30 nM. Its methyl ester may enhance bioavailability.</p>Formula:C23H34O5Colore e forma:SolidPeso molecolare:390.51DL-Buthionine-(S,R)-sulfoximine hydrochloride
<p>DL-Buthionine-(S,R)-sulfoximine hydrochloride (Buthionine sulfoximine hydrochloride) is a potent and specific glutamylcysteine synthetase biosynthesis inhibitor</p>Formula:C8H19ClN2O3SColore e forma:SolidPeso molecolare:258.77Sacibertinib
CAS:<p>Sacibertinib inhibits Trk, targeting EGFR-TK (EC50 110 nM) & HER2 (EC50 244 nM), with anticancer properties.</p>Formula:C32H31ClN6O4Colore e forma:SolidPeso molecolare:599.08AKR1C3-IN-5
<p>AKR1C3-IN-5 inhibits AKR1C3, key in prostate/breast cancers, with MCF-7 cell IC50 of 9.6 μM.</p>Formula:C34H44N2O7Colore e forma:SolidPeso molecolare:592.72MDL-27210
CAS:<p>MDL-27210 is the ethyl ester prodrug of a potent angiotensin-converting enzyme inhibitor, MDL-27088.</p>Formula:C27H32N2O5Colore e forma:SolidPeso molecolare:464.55Orvepitant
CAS:<p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>Formula:C31H35F7N4O2Colore e forma:SolidPeso molecolare:628.62Unoprostone isopropyl
CAS:<p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>Formula:C25H44O5Purezza:98%Colore e forma:SolidPeso molecolare:424.61Bleomycin Free Base
CAS:<p>Bleomycin Free Base, a glycopeptide antibiotic, halts DNA function and treats solid tumors.</p>Formula:C55H84N17O21S3Colore e forma:SolidPeso molecolare:1415.55STA 2
CAS:<p>STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.</p>Formula:C21H34O3SColore e forma:SolidPeso molecolare:366.56KT2-962
CAS:<p>KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.</p>Formula:C23H27ClNNaO5S2Colore e forma:SolidPeso molecolare:520.04TRPC5-IN-4
CAS:<p>TRPC5-IN-4: Potent, safe inhibitor; IC50 14.07 nM (TRPC5), 65 nM (TRPC4); non-toxic to liver/kidney cells; for CKD research.</p>Formula:C18H11ClF4N4O3Colore e forma:SolidPeso molecolare:442.75LIT-001 free base
CAS:<p>LIT-001, a nonpeptide OT-R agonist, enhances mouse autism-like behavior, with EC50=55 nM and Ki=226 nM.</p>Formula:C28H33N7O2SPurezza:98%Colore e forma:SolidPeso molecolare:531.676-trans-12-epi-Leukotriene B4
CAS:<p>6-trans-12-epi-Leukotriene B4, a metabolite of arachidonic acid, serves as a potent anti-inflammatory agent.</p>Formula:C20H32O4Colore e forma:SolidPeso molecolare:336.47Antitumor agent-76
CAS:<p>Antitumor agent-76 is a water-soluble, orally active, rapid-release prodrug of Triptolide that exhibits anticancer effects.</p>Formula:C28H36ClNO10Colore e forma:SolidPeso molecolare:582.04TRPA1 Antagonist 1
CAS:<p>TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate prodrug which converts to its active parent drug.</p>Formula:C24H20F6N5Na2O7PSPurezza:98%Colore e forma:SolidPeso molecolare:713.45AChE/GSK-3β-IN-1
CAS:<p>AChE/GSK-3β-IN-1 is a potent dual AChE/GSK-3β inhibitor that crosses the blood-brain barrier and acts on hAChE (IC50: 1.2 nM), hBChE (IC50: 149.8 nM) and hGSK-</p>Formula:C31H35N7O3SColore e forma:SolidPeso molecolare:585.72TRPC4/5-IN-1
<p>TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.</p>Formula:C21H21N3OColore e forma:SolidPeso molecolare:331.41Avibactam sodium dihydrate
<p>Avibactam sodium dihydrate (NXL-104) is a reversible covalent inhibitor for CTX-M-15 and TEM-1 β-lactamases with IC50s of 5 nM and 8 nM.</p>Formula:C7H14N3NaO8SColore e forma:SolidPeso molecolare:323.26PXS-5153A monohydrochloride
CAS:<p>PXS-5153A is an oral, fast-acting LOXL2/3 inhibitor with IC50 <40 nM for LOXL2 and 63 nM for LOXL3, potentially treating fibrosis.</p>Formula:C20H25Cl2FN4O2SPurezza:98%Colore e forma:Odour SolidPeso molecolare:475.41PLP_Snyder530
<p>PLP_Snyder530, a potent PL pro inhibitor, halts SARS-CoV-2 by triggering protease conformation changes.</p>Formula:C24H24N2O2Colore e forma:SolidPeso molecolare:372.46KNI 10033
CAS:<p>KNI 10033 is a potent inhibitor of HIV protease</p>Formula:C40H45N5O7S2Colore e forma:SolidPeso molecolare:771.95Quinagolide Free Base
CAS:<p>Quinagolide Free Base is a non-ergot dopamine D(2)-agonist.</p>Formula:C20H33N3O3SColore e forma:SolidPeso molecolare:395.565α-reductase-IN-1
CAS:<p>5α-reductase-IN-1 is a potent inhibitor of the enzyme 5α-reductase.</p>Formula:C31H37NO5Purezza:98%Colore e forma:SolidPeso molecolare:503.63RO5461111
CAS:<p>RO5461111: Oral Cathepsin S inhibitor, IC50 of 0.4 nM (human) & 0.5 nM (mouse), reduces T/B cell activation, treats lung inflammation & lupus nephritis.</p>Formula:C27H24F6N4O4SColore e forma:SolidPeso molecolare:614.56LasR-IN-2
<p>LasR-IN-2 blocks LasR via H-bond with TRY-56, useful in bacterial infection and CF research.</p>Formula:C21H16ClN3O2Colore e forma:SolidPeso molecolare:377.82HDAC6-IN-3
<p>HDAC6-IN-3 (Compound 14) is an oral anti-prostate cancer agent, inhibiting HDACs and MAO-A, with IC50 of 0.02-1.54 μM.</p>Formula:C19H27N3O3Colore e forma:SolidPeso molecolare:345.44SphK2-IN-1
CAS:<p>SphK2-IN-1 is an SphK2 inhibitor with an IC50 value of 0.359 μM. SphK2-IN-1 can be used to study cancer, inflammation, neurological and cardiovascular diseases.</p>Formula:C23H22ClF3N8OColore e forma:SolidPeso molecolare:518.92P-gp modulator 3
<p>P-gp modulator 3 (Compound 37) is a potent, competitive, metabotropic P-glycoprotein (P-gp) modulator.</p>Formula:C31H37N3O5Colore e forma:SolidPeso molecolare:531.64NMDAR/HDAC-IN-1
<p>Compound 9d is a dual NMDAR and HDAC inhibitor with high NMDAR affinity (Ki=0.59 μM) and inhibits HDAC1-3,6,8; crosses the blood-brain barrier.</p>Formula:C22H28N2O3Colore e forma:SolidPeso molecolare:368.47nNOS-IN-25
CAS:<p>nNOS-IN-25 is an effective, selective, and cell-permeable inhibitor of neuronal nitric oxide synthase.</p>Formula:C21H22N4Purezza:98%Colore e forma:SolidPeso molecolare:330.43Aplaviroc hydrochloride
CAS:<p>Aplaviroc, a potent CCR5 inhibitor, binds selectively, blocking HIV entry and specific monoclonal antibody attachment in vitro.</p>Formula:C33H44ClN3O6Colore e forma:SolidPeso molecolare:614.17Anti-inflammatory agent 6
<p>Anti-inflammatory agent 6 blocks IKKα/β, IκBα, and NF-κB p65 phosphorylation, key to controlling inflammation.</p>Formula:C22H20O12Colore e forma:SolidPeso molecolare:476.39PX-316
CAS:<p>PX-316: AKT inhibitor, reduces Akt activity by 78% in HT-29 xenografts, effective against MCF-7 and HT-29 cancers, well-tolerated intravenously.</p>Formula:C28H57O10PColore e forma:SolidPeso molecolare:584.72PF-06648671
CAS:<p>PF-06648671 is a γ-secretase modulator for the treatment of neurodegenerative and/or neurological disorders.</p>Formula:C25H23ClF4N4O3Purezza:98%Colore e forma:SolidPeso molecolare:538.92DNA crosslinker 2 dihydrochloride
CAS:<p>Potent DNA crosslinker 2 binds minor groove, increases Tm by 1.2°C, and inhibits NCI-H460, A2780, MCF-7 cancer cells.</p>Formula:C15H22Cl2N8OColore e forma:SolidPeso molecolare:401.29JAK3-IN-13
<p>JAK3-IN-13: Oral JAK3 inhibitor, selective & potent. Acts on NK1, JNK2, JNK3, Tyk2. Anti-tumor. IC50: JNK3, 8 nM; Tyk2, 365 nM; JNK2, 2039 nM; NK1, 4728 nM.</p>Formula:C25H33ClN6O5Colore e forma:SolidPeso molecolare:533.02GSK2945 hydrochloride
<p>GSK2945 HCl is a specific Rev-erbα antagonist, EC50: 21.5 μM (mouse), 20.8 μM (human), increases cholesterol 7α-hydroxylase.</p>Formula:C20H19Cl3N2O2SColore e forma:SolidPeso molecolare:457.8Trypanothione synthetase-IN-4
<p>Trypanothione synthetase-IN-4, an L. infantum inhibitor, has potent anti-leishmanicidal properties (EC50: 0.6 μM).</p>Formula:C29H52INO2Colore e forma:SolidPeso molecolare:573.63(S)-Purvalanol B
CAS:<p>(S)-Purvalanol B is the S enantiomer of Purvalanol B. Purvalanol B is an inhibitor of cyclin-dependent kinase(CDK) .</p>Formula:C20H25ClN6O3Purezza:98%Colore e forma:SolidPeso molecolare:432.9PF-4693627
CAS:<p>PF-4693627 is an effective and selective microsomal prostaglandin E synthase-1 inhibitor (IC50=3 nM).</p>Formula:C26H29Cl2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:502.43MEK4 inhibitor-2
CAS:<p>MEK4 Inhibitor-2, a novel MEK4 inhibitor, demonstrates efficacy against pancreatic adenocarcinoma, exhibiting an IC50 value of 83 nM.</p>Formula:C20H15FN4O3SColore e forma:SolidPeso molecolare:410.42ATM Inhibitor-2
<p>ATM Inhibitor -2 is a potent and selective inhibitor of ATM (IC50<1 nM).</p>Formula:C26H31N7O3Colore e forma:SolidPeso molecolare:489.57CV 5975
CAS:<p>CV 5975 is a nonsulfhydryl ACE inhibitor that was investigated for use in hypertension and heart failure.</p>Formula:C22H31N3O5SColore e forma:SolidPeso molecolare:449.56Artemisiane E
CAS:<p>Artemisiane E is a potent PI3K/AKT pathway inhibitor with an IC 50 of 8.9 μM .</p>Formula:C20H22O5Colore e forma:SolidPeso molecolare:342.39Terpendole E
CAS:<p>Terpendole E is an atypical L5 site inhibitor.</p>Formula:C28H39NO3Colore e forma:SolidPeso molecolare:437.61SOS1-IN-6
CAS:<p>SOS1-IN-6 (compound 33-P1) is a potent inhibitor of SOS1, acting on SOS1-G12D (IC50: 14.9 nM) and SOS1-G12V (IC50: 73.3 nM).</p>Formula:C26H28F3N3O2Colore e forma:SolidPeso molecolare:471.51LpxA-IN-1
CAS:<p>LpxA-IN-1, a novel UDP-N-acetylglucosamine acyltransferase (LpxA) inhibitor exhibiting potent activity (IC 50 2 nM), effectively targets Pseudomonas aeruginosa</p>Formula:C21H11D7F3N5O3Colore e forma:SolidPeso molecolare:452.44(1R,3S)-THCCA-Asn
<p>(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.</p>Formula:C24H24N4O6Colore e forma:SolidPeso molecolare:464.47PDE4-IN-12
<p>PDE4-IN-12 is a potent and safe PDE4 ubiquitous inhibitor that acts on PDE4 (IC50: 3.5 nM, SI: 2.71) and PDE7 (IC50: 15 nM, SI: 4.27).</p>Formula:C34H35NO6Colore e forma:SolidPeso molecolare:553.64Cap-dependent endonuclease-IN-2
<p>Cap-dependent endonuclease-IN-2 strongly blocks influenza A virus RNA polymerase; it's a CEN inhibitor.</p>Formula:C30H24FN3O7SColore e forma:SolidPeso molecolare:589.59Danshenxinkun D
CAS:<p>Danshenxinkun D has antituberculosis H_(37)Rv activity in vitro.</p>Formula:C21H20O4Purezza:98%Colore e forma:SolidPeso molecolare:336.38Anticancer agent 68
CAS:<p>Compound 12, an anticancer agent, halts G2/M phase, triggers cell death, and activates p53 & PTEN for tumor suppression.</p>Formula:C20H18ClNO5Colore e forma:SolidPeso molecolare:387.81HPK1-IN-30
CAS:<p>HPK1-IN-30 is a potent inhibitor of HPK1. HPK1-IN-30 has potential for cancer disease research.</p>Formula:C25H23FN6Colore e forma:SolidPeso molecolare:426.49Pefcalcitol
CAS:<p>Pefcalcitol is a novel antipsoriatic prodrug candidate containing a 16-en-22-oxa-vitamin D3 structure.</p>Formula:C26H34F5NO4Colore e forma:SolidPeso molecolare:519.54Estrogen receptor antagonist 7
CAS:<p>ER antagonist 7, compound 13, inhibits ERs, halts breast/ovarian cancer cell growth, has anticancer properties.</p>Formula:C23H17N3O4Colore e forma:SolidPeso molecolare:399.4NVP-CFC218
CAS:<p>NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.</p>Formula:C37H45ClN4O4Colore e forma:SolidPeso molecolare:645.23BRD0418
CAS:<p>BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.</p>Formula:C29H32N2O5Purezza:99.57%Colore e forma:SolidPeso molecolare:488.57Tipelukast
CAS:<p>Tipelukast (KCA 757), an oral drug for asthma research, blocks leukotrienes and fights inflammation and fibrosis.</p>Formula:C29H38O7SPurezza:>99.99%Colore e forma:SolidPeso molecolare:530.67VEGFR-IN-3
CAS:<p>VEGFR-IN-3 inhibits cancer cell growth (OVCAR-4, MDA-MB-468) with IC50s: 0.29, 0.35μM. Used in cancer research.</p>Formula:C27H28N2O6Colore e forma:SolidPeso molecolare:476.52(-)-Mesembrine
CAS:<p>Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4).</p>Formula:C17H23NO3Colore e forma:SolidPeso molecolare:289.37STAT3-IN-8
CAS:<p>"STAT3-IN-8 (compound H172) is a potent inhibitor of STAT3 with potential applications in cancer research [1]."</p>Formula:C19H7F7N2O3Purezza:98%Colore e forma:SolidPeso molecolare:444.26Anti-inflammatory agent 10
<p>Tilomisole-derived benzimidazole-thiazole, orally active, favors COX-2 inhibition over COX-1.</p>Formula:C17H13BrN4O3S2Colore e forma:SolidPeso molecolare:465.34CLR01 sodium
CAS:<p>CLR01 is a tweezer reducing α-synuclein in MSA, inhibits SOD1 in ALS, blocks Ebola/Zika, stabilizes proteins, and lessens mutant p53 toxicity.</p>Formula:C42H30Na2O8P2Colore e forma:SolidPeso molecolare:770.6211Mepixetil
<p>Mepixetil is a potent angiotensin II receptor antagonist[1].</p>Formula:C12H18N2O3Colore e forma:SolidPeso molecolare:238.289(R)-HETE
CAS:<p>9(R)-HETE, 50% of racemic mix, activates RXRγ 1.5x at 300 nM; identified by HPLC comparison.</p>Formula:C20H32O3Colore e forma:SolidPeso molecolare:320.47BChE-IN-2
<p>BChE-IN-2, a pyrimidine/pyridine derivative, potently inhibits BChE (Ki 0.099 μM) and shows promise in AD research.</p>Formula:C22H31N5Colore e forma:SolidPeso molecolare:365.52LH secretion antagonist 1
CAS:<p>LH secretion antagonist 1 is an antagonist of luteinizing hormone secretion with analgesic activity.</p>Formula:C18H24ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:321.84CHNQD-01255
CAS:<p>CHNQD-01255 is an orally active inhibitor of Arf-GEFs that is effective against hepatocellular carcinoma (HCC).</p>Formula:C23H29NO6Colore e forma:SolidPeso molecolare:415.48Chitinase-IN-5
<p>Chitinase-IN-5 (8i) blocks OfChi-h (IC50: 0.051 μM), has insecticidal qualities, useful for eco-friendly pest control.</p>Formula:C20H21ClFN7Colore e forma:SolidPeso molecolare:413.88mTOR/HDAC6-IN-1
<p>mTOR/HDAC6-IN-1 inhibits HDAC6 (IC50: 56 nM) & mTOR (IC50: 133.7 nM), may treat TNBC by inducing autophagy and apoptosis.</p>Formula:C20H20ClN5O2Colore e forma:SolidPeso molecolare:397.86IAA65
CAS:<p>IAA65 is a potent inhibitor of T-type calcium channels, exhibiting an IC50 value of 18.9 μM, and holds potential for use in epilepsy research [1].</p>Formula:C16H13F6NO2Colore e forma:SolidPeso molecolare:365.27MLKL-IN-6
<p>MLKL-IN-6 (compound P28) is a mixed lineage kinase inhibitor that specifically targets the Mixed Lineage Kinase domain-like (MLKL) protein.</p>Formula:C20H18N4O5Purezza:98%Colore e forma:SolidPeso molecolare:394.38DD04107
CAS:<p>DD04107 inhibits α-CGRP release, targets Synaptotagmin 1 in sensory neurons.</p>Formula:C48H88N14O12SColore e forma:SolidPeso molecolare:1085.36GW311616
CAS:<p>GW-311616 is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).</p>Formula:C19H31N3O4SColore e forma:SolidPeso molecolare:397.53PARP10/15-IN-3
<p>Compound 8a, a dual PARP10 & PARP15 inhibitor, has IC50s: PARP10 at 0.14μM & PARP15 at 0.40μM; it's cell-permeable & anti-apoptotic.</p>Formula:C12H12N2O3Colore e forma:SolidPeso molecolare:232.24Demethoxyviridin
CAS:<p>Demethoxyviridin inhibits mammalian Ptdlns 3-kinase (p110) and is antifungal.</p>Formula:C19H14O5Purezza:98%Colore e forma:SolidPeso molecolare:322.31YEATS4 binder-1
<p>YEATS4 binder-1(4e) is an effective and selective compound that targets the KAc recognition site within the YEATS structural domain, exhibiting a binding</p>Formula:C23H34N4O3Colore e forma:SolidPeso molecolare:414.54Kinamycin B
CAS:<p>Kinamycin B is an antibacterial agent with anticancer activity.</p>Formula:C20H16N2O8Purezza:98%Colore e forma:SolidPeso molecolare:412.35Aniline-MPB-amino-C3-PBD
CAS:<p>Aniline-MPB-amino-C3-PBD is a cytotoxic agent comprised of the non-alkylating group. It is a sequence-selective DNA minor-groove binding agent.</p>Formula:C42H46N8O6Purezza:98%Colore e forma:SolidPeso molecolare:758.86GPR81 agonist 2
CAS:<p>GPR81 agonist 2 is a potent agonist targeting the GPR81 receptor, demonstrating EC50 values of 0.023 µM for hGPR81 and 0.123 µM for hGPR109A, respectively.</p>Formula:C26H27ClN6O5S2Colore e forma:SolidPeso molecolare:603.11Antibacterial agent 75
<p>Antibacterial agent 75 re-sensitizes VRSA to vancomycin.</p>Formula:C22H28N6OColore e forma:SolidPeso molecolare:392.5HIV-1 inhibitor-17
<p>HIV-1 inhibitor-18 blocks HIV-1 capsid, acts on NL4-3 strain (EC50: 2.57 μM), has low cytotoxicity (MT-4 CC50: >8.55).</p>Formula:C32H32N4O5SColore e forma:SolidPeso molecolare:584.69MRGPRX1 agonist 3
<p>Compound 1f, a potent MRGPRX1 agonist, has an EC50 of 0.22 μM, useful for neuropathic pain studies.</p>Formula:C14H11FN2OSColore e forma:SolidPeso molecolare:274.31Leukotriene F-4 sulfone
CAS:<p>Leukotriene F-4 sulfone induces vascular permeability changes.</p>Formula:C28H44N2O10SColore e forma:SolidPeso molecolare:600.72NAZ2329
CAS:<p>NAZ2329: Cell-permeable, targets R5 RPTPs, inhibits hPTPRZ1 (IC50=7.5 μM) & hPTPRG (IC50=4.8 μM), hampers glioblastoma growth, affects stem cell traits.</p>Formula:C21H18F3NO4S3Colore e forma:SoildPeso molecolare:501.56Macbecin I
CAS:<p>Hsp90 inhibitor</p>Formula:C30H42N2O8Purezza:98%Colore e forma:SolidPeso molecolare:558.66EBI-1051
CAS:<p>EBI-1051 is a highly potent and orally efficacious inhibitor of MEK (IC50: 3.9 nM).</p>Formula:C18H15F2IN2O5Purezza:98%Colore e forma:SolidPeso molecolare:504.22Mal-PEG4-VA-PBD
CAS:<p>Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connected</p>Formula:C68H79N9O17Purezza:98%Colore e forma:SolidPeso molecolare:1294.41Rodatristat ethyl
CAS:<p>Rodatristat ethyl is an oral TPH1 inhibitor reducing 5-HT levels & lowering PAH at low doses.</p>Formula:C29H31ClF3N5O3Purezza:98%Colore e forma:SolidPeso molecolare:590.04GSK579289A
CAS:<p>GSK579289A is an inhibitor of benzimidazole thiophene.</p>Formula:C26H27ClN4O3SPurezza:98%Colore e forma:SolidPeso molecolare:511.04PSMA-1007
CAS:<p>PSMA-1007 is a novel Glu-Ureido-type prostate-specific membrane antigen (PSMA) inhibitor.</p>Formula:C49H55FN8O16Colore e forma:SolidPeso molecolare:1030.01Carmegliptin dihydrochloride
CAS:<p>Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.</p>Formula:C20H30Cl2FN3O3Colore e forma:SolidPeso molecolare:450.38ORP-101
CAS:<p>ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.</p>Formula:C60H84N2O8Colore e forma:SolidPeso molecolare:961.32CBP/p300-IN-2
CAS:<p>CBP/EP300-IN-2 is an inhibitor of CBP/EP300 (IC50s: 1.07 nM and 5.96 nM for CBP/HTRF and Myc).</p>Formula:C27H29F2N7O2Purezza:98%Colore e forma:SolidPeso molecolare:521.56GNTI dihydrochloride
CAS:<p>κ opioid receptor antagonist</p>Formula:C27H30ClN5O3Purezza:98%Colore e forma:SolidPeso molecolare:508.01Gallinamide A
CAS:<p>Gallinamide A is a potent inhibitor of cathepsin L with an IC 50 value of 17.6 pM.</p>Formula:C31H52N4O7Colore e forma:SolidPeso molecolare:592.77Topo I/COX-2-IN-1
<p>Topo I/COX-2-IN-1: potent dual inhibitor; IC50 0.24μM (COX-2), 4.42μM (Topo I); anti-cancer; induces apoptosis, halts migration.</p>Formula:C21H18ClFN2O3Colore e forma:SolidPeso molecolare:400.83U 75875
CAS:<p>U 75875 is a protease inhibitor.</p>Formula:C45H61N7O7Colore e forma:SolidPeso molecolare:812.01Aristoforin
CAS:<p>Aristoforin is a SIRT1 and SIRT2 inhibitor that induces cell cycle arrest, shows potent antitumor effects, and inhibits lymphangiogenesis in vivo.</p>Formula:C37H54O6Colore e forma:SolidPeso molecolare:594.82Rodatristat
CAS:<p>Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).</p>Formula:C27H27ClF3N5O3Purezza:98%Colore e forma:SolidPeso molecolare:561.98TLR7/8 antagonist 2
<p>TLR7/8 antagonist 2: potent, orally active, IC50: 4.9 nM (TLR7), 0.6 nM (TLR8); potential for lupus therapy research.</p>Formula:C22H26FN5Colore e forma:SolidPeso molecolare:379.47IRAK4-IN-9
CAS:<p>IRAK4-IN-9 is a potent IRAK4 inhibitor with an IC50 of 1.5 nM, promising for inflammatory, autoimmune diseases, and cancer research.</p>Formula:C22H25N7Colore e forma:SolidPeso molecolare:387.48Tofacitinib Prodrug-1
<p>Tofacitinib Prodrug-1: an oral prodrug reducing Tofacitinib's side effects, treats ulcerative colitis in mice effectively with low toxicity.</p>Formula:C36H39ClN10O7Colore e forma:SolidPeso molecolare:759.21DHU-Se1
<p>DHU-Se1: potent anti-inflammatory, releases reactive selenium from macrophages, inhibits iNOS/TNF-α, blocks M0 to M1 polarization.</p>Formula:C23H23N3OSSeColore e forma:SolidPeso molecolare:468.47CVS-1578
CAS:<p>CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.</p>Formula:C20H30N6O5SColore e forma:SolidPeso molecolare:466.55PF-00489791
CAS:<p>PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy.</p>Formula:C20H28N8O4SPurezza:99.97%Colore e forma:SolidPeso molecolare:476.55MAP3K14-IN-173
CAS:<p>MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.</p>Formula:C29H31N7O2Colore e forma:SolidPeso molecolare:509.60RdRP-IN-4
<p>RdRP-IN-4, an oral arylbenzohydrazide, inhibits influenza A/B by targeting PB1 of RdRP, with EC50s of 53 nM (H1N1) and 20 nM (Flu B), and aids infected mice.</p>Formula:C17H17Br2N3O2Colore e forma:SolidPeso molecolare:455.14Revexepride
CAS:<p>Revexepride, a 5-HT4 agonist, may boost CYP3A4, used for treating GERD.</p>Formula:C21H32ClN3O4Purezza:98%Colore e forma:SolidPeso molecolare:425.95Atorvastatin 3-Deoxyhept-2E-Enoic Acid
CAS:<p>Atorvastatin 3-Deoxyhept-2E-Enoic Acid, an impurity in Atorvastatin, lowers blood lipids as an HMG-CoA reductase inhibitor.</p>Formula:C33H33FN2O4Purezza:98%Colore e forma:SolidPeso molecolare:540.62HBV-IN-24
<p>HBV-IN-24 inhibits HBV DNA, HBsAg, HBeAg (EC50: 0.6, 0.6, 4.6 nM), and has antiviral properties with neurotoxicity mitigation.</p>Formula:C23H27NO6Colore e forma:SolidPeso molecolare:413.46Dehydrocrenatidine
CAS:<p>Dehydrocrenatidine (Kumujian G) is an inhibitor of JAK and induces cell apoptosis.</p>Formula:C15H14N2O2Purezza:98%Colore e forma:SolidPeso molecolare:254.28HPK1-IN-16
CAS:<p>HPK1-IN-16, a potent HPK1 inhibitor, useful for cancer research and treatment.</p>Formula:C28H27FN4OColore e forma:SolidPeso molecolare:454.54OSI-7904L free acid
CAS:<p>OSI-7904L is a folate-based thymidylate synthase inhibitor. It also has antimalarial and antitumor properties.</p>Formula:C27H24N4O6Purezza:98%Colore e forma:SolidPeso molecolare:500.5K027
<p>K027 is a potent organophosphate (OP) inhibitor of acetylcholinesterase (AChE) reactivation. k027 can be used to study Alzheimer's disease.</p>Formula:C15H18Br2N4O2Colore e forma:SolidPeso molecolare:446.1412(S)-HETE
CAS:<p>Enpatoran hydrochloride (M5049 hydrochloride) is a TLR7/8 inhibitor with antiviral activity that is used in the study of autoimmune diseases.</p>Formula:C20H32O3Colore e forma:SolidPeso molecolare:320.47PF1070A
CAS:<p>PF1070A is a natural cyclic tetrapeptide HDAC Inhibitor through the inhibition of PfHDAC1 catalytic activity, potently inducing the synthesis of metallothionein</p>Formula:C31H44N4O6Colore e forma:SolidPeso molecolare:568.7Pparδ agonist 5
<p>Pparδ agonist 5 is a selective, orally active PPARδ agonist with an EC50 of 0.335 μM and better selectivity than GW0742.</p>Formula:C23H21F3N2O2SColore e forma:SolidPeso molecolare:446.49BAA473
<p>BAA473, a bile acid analog, activates the pyrin inflammasome, triggering IL-18 secretion in myeloid and intestinal cells.</p>Formula:C36H62O5Purezza:98%Colore e forma:SolidPeso molecolare:574.87Mt KARI-IN-1
<p>Mt KARI-IN-1 inhibits Mtb KARI with a 3.06 μM Ki, targeting tuberculosis.</p>Formula:C14H11N5O4S2Colore e forma:SolidPeso molecolare:377.4PPARγ phosphorylation inhibitor 1
<p>PPARγ phosphorylation inhibitor 1 (Compound 10) is a potent PPARγ binding agent (IC50: 24 nM) with antidiabetic effects.</p>Formula:C22H14Cl2N2O4Colore e forma:SolidPeso molecolare:441.26EFdA-TP tetrasodium
CAS:<p>EFdA-TP tetrasodium is a potent HIV-1 inhibitor that blocks DNA synthesis as an ICT or DCT.</p>Formula:C12H11FN5Na4O12P3Purezza:98%Colore e forma:SolidPeso molecolare:621.12
