Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.523 prodotti)
- Apoptosi(5.792 prodotti)
- Ciclo cellulare/Checkpoint(4.449 prodotti)
- Cromatina/Epigenetica(2.238 prodotti)
- Segnalazione citoscheletrica(1.383 prodotti)
- Danno al DNA/Riparazione del DNA(2.825 prodotti)
- Endocrinologia/Ormoni(3.507 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.333 prodotti)
- Immunologia e infiammazione(3.526 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.202 prodotti)
- Trasportatore di membrana/canale ionico(2.790 prodotti)
- Metabolismo(9.448 prodotti)
- Microbiologia/Virologia(6.981 prodotti)
- Neuroscienza(9.926 prodotti)
- Altri inibitori(37.926 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.597 prodotti)
- Cellule staminali e Derivati(831 prodotti)
- Adattatori Tirosin-chinasi(2.016 prodotti)
- Ubiquitinazione(1.650 prodotti)
Mostrare 16 più sottocategorie
Trovati 66641 prodotti di "Inibitori"
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(Rac)-BI 703704
CAS:<p>(Rac)-BI 703704 is a potent activator of soluble guanylyl cyclase (sGC).</p>Formula:C32H37N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:559.72JAK-2/3-IN-3
<p>JAK-2-/3-IN-3 (ST4j) is a potent JAK2/3 inhibitor for leukemia research, with IC50s: JAK2, 13 nM; JAK3, 14.86 nM; induces apoptosis.</p>Formula:C13H10Cl2N4O2Colore e forma:SolidPeso molecolare:325.15PTP1B-IN-16
<p>PTP1B-IN-16: selective benzimidazole inhibitor of PTP1B, Ki: 12.6 μM, potential for type 2 diabetes research.</p>Formula:C26H18ClN3O4SColore e forma:SolidPeso molecolare:503.96GSK699
CAS:<p>GSK699 is a potent, cell penetrant PCAF/GCN5 PROTAC.</p>Formula:C45H51BrN8O7Colore e forma:SolidPeso molecolare:895.84GNE-203
CAS:<p>GNE-203 is a Met inhibitor.</p>Formula:C30H29Cl2F3N8O3Colore e forma:SolidPeso molecolare:677.50AKT-IN-3
CAS:<p>AKT-IN-3: potent oral Akt inhibitor with low hERG blockage. IC50: 1.4-1.7 nM for Akt1-3. Inhibits AGC kinases like PKA, PKC.</p>Formula:C23H23Cl2F2N5O3Purezza:98%Colore e forma:SolidPeso molecolare:526.36STAT3-IN-9
<p>STAT3-IN-9 hinders STAT3 at Tyr705, doesn't affect STAT1 Tyr701, induces apoptosis, and arrests cells in G2/M phase.</p>Formula:C22H21N3O4Colore e forma:SolidPeso molecolare:391.42Revamilast
CAS:<p>Revamilast, also known as GRC4039, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritis</p>Formula:C18H9Cl2F2N3O4Colore e forma:SolidPeso molecolare:440.18Glucosylceramide synthase-IN-3
<p>Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.</p>Formula:C21H20FN3O3Colore e forma:SolidPeso molecolare:381.4Bizelesin
CAS:<p>Bizelesin, a synthetic antineoplastic agent, binds DNA, disrupts replication, triggers cell-cycle arrest, and induces senescence.</p>Formula:C43H36Cl2N8O5Colore e forma:SolidPeso molecolare:815.7NVP-CGM097 sulfate
CAS:<p>NVP-CGM097 sulfate is a potent and selective inhibitor of MDM2 (hMDM2, IC50 of 1.7±0.1 nM).</p>Formula:C38H49ClN4O8SPurezza:98%Colore e forma:SolidPeso molecolare:757.34MB725
CAS:<p>MB725 is a strong and selective inducer of viability reduction in several cancer cell lines containing the oncogenic p53-Y220C mutation.</p>Formula:C18H21IN4O2SColore e forma:SolidPeso molecolare:484.35Cathepsin C-IN-4
<p>Cathepsin C-IN-4 is a potent inhibitor (IC50: 65.6 nM) of histone C. Cathepsin C-IN-4 inhibits THP-1 cells (IC50: 203.4 nM) and U937 cells (IC50: 177.6 nM).</p>Formula:C21H14ClF3N4SColore e forma:SolidPeso molecolare:446.88DENV-IN-6
CAS:<p>DENV-IN-6, a potent anti-DENV (I-IV) and HIV-1 IIIB inhibitor with EC50 ranging 6.8-17.5 μM for DENV and EC50 0.0181 μM for HIV-1.</p>Formula:C23H26ClFN4OSColore e forma:SolidPeso molecolare:461LSD1/2-IN-3
<p>LSD1/2-IN-3 selectively inhibits LSD1 (Ki 11 nM) over LSD2 (Ki 7 μM), and hinders tumor stem cell proliferation.</p>Formula:C9H8BrF2NColore e forma:SolidPeso molecolare:248.07Symplostatin 1
CAS:<p>Symplostatin 1 is a dolastatin 10 analog from the marine cyanobacterium Symploca hydnoides.</p>Formula:C43H70N6O6SColore e forma:SolidPeso molecolare:799.12Antiangiogenic agent 3
<p>Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.</p>Formula:C19H20O7Colore e forma:SolidPeso molecolare:360.36IRAK4-IN-14
CAS:<p>IRAK4-IN-14 is a selective, potent, orally active IRAK4 inhibitor (IC50: 0.003 μM) with favorable PK parameters in rats and mice. effect.</p>Formula:C25H28FN9OColore e forma:SolidPeso molecolare:489.55Glutaminyl Cyclase Inhibitor 3
CAS:<p>Designed anti-Alzheimer’s compound; potent Glutaminyl Cyclase inhibitor; IC50 at 4.5 nM; reduces brain Aβ; improves cognition.</p>Formula:C24H32N6O2SPurezza:98%Colore e forma:SolidPeso molecolare:468.61Ganoderic acid R
CAS:<p>Ganoderic acid R: potent anticancer, induces apoptosis, cytotoxic to MDR and sensitive tumor cells.</p>Formula:C34H50O6Colore e forma:SolidPeso molecolare:554.76Aplaviroc
CAS:<p>Aplaviroc (AK 602), a SDP derivative, is a CCR5 antagonist. With IC50s of 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL and HIV-1MOKW.</p>Formula:C33H43N3O6Purezza:97.98% - 98.26%Colore e forma:SolidPeso molecolare:577.71HDAC2-IN-1
<p>HDAC2-IN-1 is an oral HDAC2 inhibitor (IC50: 0.5 μM), crosses the blood-brain barrier, and inhibits HDAC1 and HDAC8.</p>Formula:C22H23ClN4OSColore e forma:SolidPeso molecolare:426.96Vps34-IN-3
<p>Vps34-IN-3 is a potent, selective, and orally bioavailable inhibitor of VPS34 kinase .</p>Formula:C14H20N4O2Colore e forma:SolidPeso molecolare:276.33G-744
CAS:<p>G-744 is a selective and orally active inhibitor of Btk (IC50: 2 nM).</p>Formula:C29H29N5O3SPurezza:98%Colore e forma:SolidPeso molecolare:527.64trans-Doxercalciferol
CAS:<p>trans-Doxercalciferol is an isomer of Doxercalciferol. Doxercalciferol is an activator of the Vitamin D receptor and prevents renal disease.</p>Formula:C28H44O2Purezza:98%Colore e forma:SolidPeso molecolare:412.65LY-2979165
CAS:<p>LY-2979165 is a metabotropic glutamate receptor agonist prodrug.</p>Formula:C13H17N5O5SColore e forma:SolidPeso molecolare:355.37Azonafide-PEABA
CAS:<p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>Formula:C32H33N5O4Purezza:98%Colore e forma:SolidPeso molecolare:551.64Ici D1542
CAS:<p>Ici D1542: potent TXS inhibitor & TXA2 receptor antagonist, effective thromboxane blocker in vitro.</p>Formula:C25H30N2O7Purezza:98%Colore e forma:SolidPeso molecolare:470.51CDK4/6-IN-13
CAS:<p>Compounds 10B and 10C: potent cdk4/6 inhibitors with low nM activity, great antiproliferative effects, excellent metabolism, and good pharmacokinetics.</p>Formula:C25H29N7OColore e forma:SolidPeso molecolare:443.54TTA-P1
CAS:<p>TTA-P1: potent T-type calcium channel inhibitor; impacts neuron firing, hormone secretion, cell growth; potential in absence epilepsy research.</p>Formula:C19H27Cl2FN2OColore e forma:SolidPeso molecolare:389.33FGFR4-IN-9
<p>FGFR4-IN-9 is a selective inhibitor of FGFR4 (IC50: 75.3 nM) that effectively inhibits the growth and angiogenesis of hepatocellular carcinoma cells.</p>Formula:C24H22ClF3N4O4Colore e forma:SolidPeso molecolare:522.9FAAH/MAGL-IN-1
<p>FAAH/MAGL-IN-1 (SIH 3) inhibits FAAH & MAGL with IC50 of 31 & 29 nM, useful in neuropathic pain research.</p>Formula:C15H9Cl2N3O3Colore e forma:SolidPeso molecolare:350.16(-)-Cevimeline hydrochloride hemihydrate
<p>(-)-Cevimeline HCl hemihydrate, a muscarinic agonist, treats Sjogren's xerostomia. Quick absorption, species-dependent metabolism.</p>Formula:C10H19ClNO1·5SPurezza:98%Colore e forma:SolidPeso molecolare:244.78RX 809055AX
CAS:<p>RX 809055AX is a long lasting opioid antagonist at mu and delta receptors.</p>Formula:C29H29ClN2O4Colore e forma:SolidPeso molecolare:505ATM Inhibitor-3
<p>ATM Inhibitor-3 selectively inhibits ATM (IC50: 0.71 nM), targets PI3K kinase family, and is metabolically stable.</p>Formula:C25H29FN6O3Colore e forma:SolidPeso molecolare:480.53Pyripyropene A
CAS:<p>Pyripyropene A is a potent and selective inhibitor of sterol O-acyltransferase 2 (SOAT2)/acyl-coenzyme A:cholesterol acyltransferase 2 (ACAT2)(IC50 of 0.07 μM).</p>Formula:C31H37NO10Purezza:98%Colore e forma:SolidPeso molecolare:583.63MSX-3
CAS:<p>MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2.</p>Formula:C21H23N4Na2O7PPurezza:98%Colore e forma:SolidPeso molecolare:520.389EGFR-IN-62
<p>EGFR-IN-62: IC50 of 10-242 nM for various EGFR mutations, blocks A549/H1975 cell cycle, induces apoptosis, and inhibits cell motility and proliferation.</p>Formula:C30H33N9O2Colore e forma:SolidPeso molecolare:551.64SSR 146977
CAS:<p>NK3 receptor antagonist</p>Formula:C35H42Cl2N4O2Purezza:98%Colore e forma:SolidPeso molecolare:621.64Antitumor agent-54
<p>Compound C11 inhibits 14-3-3η protein (KD: 35 μM), targets liver cancer cells, blocks G1-S phase, and induces apoptosis.</p>Formula:C29H32N2O3Colore e forma:SolidPeso molecolare:456.58(±)-ANAP hydrochloride
CAS:<p>'(±)-ANAP hydrochloride, an unnatural amino acid analog of prodan, serves as a fluorescent probe with enhanced environmental sensitivity.'</p>Formula:C15H17ClN2O3Colore e forma:SolidPeso molecolare:308.76L 767679
CAS:<p>L 767679 is an antagonist of the fibrinogen receptors.</p>Formula:C20H24N4O4Purezza:98%Colore e forma:SolidPeso molecolare:384.43rel-MDM2/4-p53-IN-3
<p>rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.</p>Formula:C25H24Cl2FN3O3Colore e forma:SolidPeso molecolare:504.38HDAC6-IN-3
<p>HDAC6-IN-3 (Compound 14) is an oral anti-prostate cancer agent, inhibiting HDACs and MAO-A, with IC50 of 0.02-1.54 μM.</p>Formula:C19H27N3O3Colore e forma:SolidPeso molecolare:345.44Protopine hydrochloride
CAS:<p>Protopine inhibits thromboxane, lowers intracellular calcium, and reduces cell adhesion by altering adhesive factors.</p>Formula:C20H20ClNO5Purezza:98%Colore e forma:Prisms From Alc SolidPeso molecolare:389.83Lafadofensine (D-(-)-Mandelic acid)
<p>Lafadofensine D-(-)-Mandelic acid is a monoamines reuptake inhibitor with adequate effects when administered short-term.</p>Formula:C32H32F2N2O6Colore e forma:SolidPeso molecolare:578.6PfPKG-IN-1
<p>PfPKG-IN-1, an imidazole-based inhibitor, targets the Plasmodium falciparum cyclic guanosine monophosphate-dependent protein kinase (PfPKG).</p>Formula:C24H22ClN7OSColore e forma:SolidPeso molecolare:492YCW-E11
CAS:<p>YCW-E11 is an antiapoptotic Bcl-2 family proteins inhibitor.</p>Formula:C25H21Cl2N3O6S2Purezza:98%Colore e forma:SolidPeso molecolare:594.49J-113397
CAS:<p>J-113397 is a potent and selective NOP receptor antagonist (IC50 = 2.3 nM).</p>Formula:C24H37N3O2Purezza:98%Colore e forma:SolidPeso molecolare:399.57GSK3527497
CAS:<p>GSK3527497 is a novel potent and selective inhibitor of transient receptor potential vanilloid-4 (TRPV4).</p>Formula:C17H16ClFN4O4SColore e forma:SolidPeso molecolare:426.85EGFR-IN-48
<p>EGFR-IN-48: potent EGFR inhibitor, oral, IC50: 0.193-66.7 nM, blocks EGFR mutants & BaF3/PC-9 cell proliferation.</p>Colore e forma:SolidMRGPRX1 agonist 3
<p>Compound 1f, a potent MRGPRX1 agonist, has an EC50 of 0.22 μM, useful for neuropathic pain studies.</p>Formula:C14H11FN2OSColore e forma:SolidPeso molecolare:274.31SSM3 TFA
CAS:<p>SSM3 TFA is a potent furin inhibitor, blocking furin-dependent cell surface processing of anthrax protective antigen-83 in vitro..</p>Formula:C22H32N12O2Colore e forma:SolidPeso molecolare:496.57MCTR3
CAS:<p>MCTR3, derived from DHA via maresin 1 in macrophages, hastens tissue healing and reduces inflammation and eicosanoids post-E. coli infection in mice.</p>Formula:C25H37NO5SColore e forma:SolidPeso molecolare:463.63Gougerotin
CAS:<p>Gougerotin is an inhibitor of protein synthesis.</p>Formula:C16H25N7O8Colore e forma:SolidPeso molecolare:443.41EGFR-IN-38
CAS:<p>EGFR-IN-38: low-toxic acrylamide-derived EGFR inhibitor, targets NSCLC, patented for research on EGFR mutation-related diseases.</p>Formula:C25H24ClN7O2Colore e forma:SolidPeso molecolare:489.96Kinamycin B
CAS:<p>Kinamycin B is an antibacterial agent with anticancer activity.</p>Formula:C20H16N2O8Purezza:98%Colore e forma:SolidPeso molecolare:412.35NK-1 Antagonist 1
CAS:<p>NK-1 Antagonist 1 is a NK-1 receptor antagonist.</p>Formula:C25H23F6N5O2Purezza:98%Colore e forma:SolidPeso molecolare:539.47EGFR-IN-23
CAS:<p>EGFR-IN-23, identified as compound 8 in WO2021244502A1, is a potent EGFR tyrosine kinase inhibitor (TKI) demonstrating an inhibitory concentration (IC50) of 8.</p>Formula:C36H44BrN10O3PColore e forma:SolidPeso molecolare:775.68Demethoxyviridin
CAS:<p>Demethoxyviridin inhibits mammalian Ptdlns 3-kinase (p110) and is antifungal.</p>Formula:C19H14O5Purezza:98%Colore e forma:SolidPeso molecolare:322.31Colistin adjuvant-2
<p>Colistin adjuvant-2 is a compound that acts as a potentiation agent for colistin, effectively enhancing its activity against Gram-negative bacteria [1].</p>Formula:C14H7Cl2F3N2OColore e forma:SolidPeso molecolare:347.12GGTI-2154 hydrochloride
CAS:<p>GGTI-2154 hydrochloride: selective GGTase I inhibitor, IC50 21 nM, used in cancer research.</p>Formula:C24H29ClN4O3Colore e forma:SolidPeso molecolare:456.97FR 900452
CAS:<p>FR 900452 is a platelet activating factor antagonist from fermentatiion products of Streptomyces phaeofaciens.</p>Formula:C22H25N3O3SColore e forma:SolidPeso molecolare:411.52SJG-136
CAS:<p>SJG-136 is a DNA cross-linking agent (XL50: 45 nM for pBR322 DNA).</p>Formula:C31H32N4O6Purezza:98%Colore e forma:SolidPeso molecolare:556.61Estrogen receptor antagonist 6
CAS:<p>Estrogen receptor antagonist 6 is a potent blocker of estrogen signaling, regulating various biological effects. (Compound 166)</p>Formula:C25H31F3N2O3Colore e forma:SolidPeso molecolare:464.52HDAC-IN-9
<p>HDAC-IN-9, a dual tubulin/HDAC inhibitor, impedes A549 cell invasion/migration and shows strong anti-tumor/angiogenic effects.</p>Formula:C33H38N2O4Colore e forma:SolidPeso molecolare:526.67Py-MPB-amino-C3-PBD
CAS:<p>Py-MPB-amino-C3-PBD is a cytotoxic agent comprised non-alkylating group,with antimicrobial activity.</p>Formula:C41H44N8O6Purezza:98%Colore e forma:SolidPeso molecolare:744.84α-Amylase-IN-1
CAS:<p>α-Amylase-IN-1 is an α-Amylase inhibitor (IC50: 0.5509 μM).</p>Formula:C18H18N2O3Purezza:99.92%Colore e forma:SoildPeso molecolare:310.35Bafilomycin C1
CAS:<p>vacuolar H+-ATPases (V-ATPases) inhibitor</p>Formula:C39H60O12Purezza:98%Colore e forma:Light Tan SolidPeso molecolare:720.89Topoisomerase II inhibitor 5
<p>Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.</p>Formula:C26H27N5O4Colore e forma:SolidPeso molecolare:473.52Anti-Influenza agent 3
<p>Compound 11h: Potent, low-toxicity anti-influenza, inhibits M2 ion channels. EC50: 3.29μM (H3N2), 2.45μM (H1N1).</p>Formula:C16H22ClNOSColore e forma:SolidPeso molecolare:311.87(Rac)-Plevitrexed
CAS:<p>(Rac)-Plevitrexed is a racemate of Plevitrexed. Plevitrexed is an orally active and potent inhibitor of thymidylate synthase (TS).</p>Formula:C26H25FN8O4Purezza:98%Colore e forma:SolidPeso molecolare:532.53YKL-04-085
CAS:<p>YKL-04-085 inhibits viral translation effectively, with strong antiviral action at much lower doses than those affecting host-cell growth.</p>Formula:C30H29N5O2Colore e forma:SolidPeso molecolare:491.6ML-SI1
CAS:<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Formula:C23H26Cl2N2O3Colore e forma:SolidPeso molecolare:449.37Daeatal
CAS:<p>Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.</p>Formula:C56H93N19O10Purezza:98%Colore e forma:SolidPeso molecolare:1192.46AMD-7049
CAS:<p>AMD-7049 is a biochemical.</p>Formula:C25H39N5Colore e forma:SolidPeso molecolare:409.61Antibiotic LL Z1640-2
CAS:<p>Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.</p>Formula:C19H22O7Colore e forma:SolidPeso molecolare:362.38MA242 free base
CAS:<p>MA242 free base is a dual MDM2/NFAT1 inhibitor that triggers apoptosis in pancreatic cancer cells.</p>Formula:C24H20ClN3O3SColore e forma:SolidPeso molecolare:465.95Sucistil
<p>Sucistil is an active biochemical. hemoglobin sucistil (bovine) is an oxygen carrier [1].</p>Formula:C9H15NO4SColore e forma:SolidPeso molecolare:233.28MK-7445
CAS:<p>MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.</p>Formula:C21H13Cl2N7OColore e forma:SolidPeso molecolare:450.28(2S,4S)-Sacubitril
CAS:<p>(2S,4S)-Sacubitril (Sacubitril Impurity C) is a stereoisomer derived from Sacubitril which is a potent NEP inhibitor.</p>Formula:C24H29NO5Purezza:98%Colore e forma:SolidPeso molecolare:411.49Lentiginosine
CAS:<p>Lentiginosine is a selective amyloglucosidase inhibitor.</p>Formula:C8H15NO2Colore e forma:SolidPeso molecolare:157.214α-PDD
CAS:<p>4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.</p>Formula:C40H64O8Colore e forma:SolidPeso molecolare:672.93MEK1/2-IN-2
<p>MEK1/2-IN-2 is a potent, ATP-competitive MEK1/2 inhibitor that exhibits equal inhibitory effects on wild-type MEK1/2 and a group of MEK1/2 mutant cells.</p>Formula:C28H22ClFN6OColore e forma:SolidPeso molecolare:512.97LSD1-IN-17
<p>LSD1-IN-17, a potent LSD1/CoREST/MAO inhibitor, IC50: 0.005/0.028/0.820 μM; hinders LNCaP prostate cancer cell growth, IC50: 17.2 μM.</p>Formula:C20H18N2OSColore e forma:SolidPeso molecolare:334.43SZ1676
CAS:<p>SZ1676 is a derivative of SZ1677, which is an agent of neuromuscular blocking.</p>Formula:C37H59BrN2O6Purezza:98%Colore e forma:SolidPeso molecolare:707.78TAK-915
CAS:<p>TAK-915: potent, brain-ready PDE2A inhibitor, 0.61 nM IC50, 4100x selectivity over PDE1A.</p>Formula:C19H18F4N4O5Purezza:98%Colore e forma:SolidPeso molecolare:458.36CYP2C1/CYP2C19-IN-2
<p>CYP2C1/CYP2C19-IN-2 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>Formula:C27H28N2O6SColore e forma:SolidPeso molecolare:508.59PF-4693627
CAS:<p>PF-4693627 is an effective and selective microsomal prostaglandin E synthase-1 inhibitor (IC50=3 nM).</p>Formula:C26H29Cl2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:502.43Aristoforin
CAS:<p>Aristoforin is a SIRT1 and SIRT2 inhibitor that induces cell cycle arrest, shows potent antitumor effects, and inhibits lymphangiogenesis in vivo.</p>Formula:C37H54O6Colore e forma:SolidPeso molecolare:594.82SSTR5 antagonist 2 hydrochloride
<p>SSTR5 antagonist 2 hydrochloride: potent, oral SSTR5 blocker with potential in type 2 diabetes research.</p>Formula:C32H36ClFN2O5Colore e forma:SolidPeso molecolare:583.09Mal-PEG4-VA-PBD
CAS:<p>Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connected</p>Formula:C68H79N9O17Purezza:98%Colore e forma:SolidPeso molecolare:1294.41TRβ agonist 1
CAS:<p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>Formula:C29H25FN2O8Colore e forma:SolidPeso molecolare:548.52NBD-14189
CAS:<p>NBD-14189: Potent HIV-1 entry blocker, binds gp120, IC50: 89 nM, strong antiviral (EC50 <200 nM).</p>Formula:C18H16F4N4O2SColore e forma:SolidPeso molecolare:428.40TAK-637
CAS:<p>TAK-637 is a tachykinin 1 (NK1) receptor antagonist.</p>Formula:C30H25F6N3O2Purezza:98%Colore e forma:SolidPeso molecolare:573.53LH secretion antagonist 1
CAS:<p>LH secretion antagonist 1 is an antagonist of luteinizing hormone secretion with analgesic activity.</p>Formula:C18H24ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:321.84LP 12 hydrochloride hydrate
<p>LP 12 hydrochloride hydrate: potent, selective 5-HT7 agonist (Ki: 0.13 nM); less affinity for D2, 5-HT1A/2A receptors.</p>Formula:C32H39N3O·HCl·xH2OColore e forma:SolidJAK-IN-23
<p>"JAK-IN-23: oral dual JAK/STAT & NF-κB inhibitor; JAK1 (IC50: 8.9 nM), JAK2 (15 nM), JAK3 (46.2 nM); for IBD research."</p>Formula:C23H22Cl2N4OColore e forma:SolidPeso molecolare:441.3511-trans Leukotriene E4
CAS:<p>Slow isomerization of the C-11 double bond of LTE4 leads to the formation of 11-trans LTE4. 11-trans LTE4 is equipotent to LTE4 in contracting guinea pig ileum.</p>Formula:C23H37NO5SColore e forma:SolidPeso molecolare:439.61(S)-JDQ-443
CAS:<p>(S)-JDQ-443, an isomer of JDQ-443, is a selective, potent oral KRAS G12C inhibitor with antitumor properties.</p>Formula:C29H28ClN7OColore e forma:SolidPeso molecolare:526.03BPTF-IN-BZ1
<p>BPTF-IN-BZ1 is a BPTF inhibitor that possesses a high potency with a Kd of 6.3 nM.</p>Formula:C13H15ClN4OColore e forma:SolidPeso molecolare:278.74Esorubicin
CAS:<p>Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.</p>Formula:C27H29NO10Colore e forma:SolidPeso molecolare:527.52Mifepristone methochloride
CAS:<p>Mifepristone methochloride is a glucocorticoid antagonist. This product will be sold for research use only.</p>Formula:C30H38ClNO2Colore e forma:SolidPeso molecolare:480.08U 75875
CAS:<p>U 75875 is a protease inhibitor.</p>Formula:C45H61N7O7Colore e forma:SolidPeso molecolare:812.01PDE4B-IN-3
<p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>Formula:C30H35N3O4S2Colore e forma:SolidPeso molecolare:565.75Neuraminidase-IN-4
<p>Neuraminidase-IN-4 inhibits neuraminidase (EC50: 1.59 μM) and has strong anti-H5N1 activity.</p>Formula:C21H20N2O6SColore e forma:SolidPeso molecolare:428.46Miaosporone A
<p>Miaosporone A: angucyclic quinone, cytotoxic to MCF-7, NCI-H187, Vero cells; anti-TB and anti-malaria with IC50 of 2.4 μM, 2.5 μM.</p>Formula:C19H18O5Colore e forma:SolidPeso molecolare:326.34FWM-1
<p>FWM-1 blocks SARS-CoV-2 NSP13, hinders ATP binding, with -328.6 kcal/mol binding energy.</p>Formula:C15H11ClN4O4S2Colore e forma:SolidPeso molecolare:410.86trans-RdRP-IN-5
<p>Trans-RdRP-IN-5 is a potent inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), with applications in influenza virus research.</p>Formula:C23H21N3O5Colore e forma:SolidPeso molecolare:419.43KRAS G12C inhibitor 46
CAS:<p>KRAS G12C inhibitor 46 is a potent inhibitor of KRAS G12C.</p>Formula:C32H33F2N7O2Colore e forma:SolidPeso molecolare:585.65Gallinamide A
CAS:<p>Gallinamide A is a potent inhibitor of cathepsin L with an IC 50 value of 17.6 pM.</p>Formula:C31H52N4O7Colore e forma:SolidPeso molecolare:592.77Flutimide
CAS:<p>Flutimide: Endonuclease inhibitor, IC50 = 3μM, for research on acute respiratory diseases like influenza.</p>Formula:C12H18N2O3Colore e forma:SolidPeso molecolare:238.28FCE-24379
CAS:<p>FCE-24379 is a selective antagonist of vascular serotonin receptors that has been shown to lowers blood pressure in hypertensive rats.</p>Formula:C20H22N4O2Colore e forma:SolidPeso molecolare:350.41Epolactaene
CAS:<p>Epolactaene: neuritogenic, inhibits mammalian DNA polymerases & human DNA topoisomerase II.</p>Formula:C21H27NO6Colore e forma:SolidPeso molecolare:389.44MtDTBS-IN-1
<p>MtDTBS-IN-1 is a notably potent binder (K_D = 57 nM) and inhibitor (K_i = 5 μM) of MtDTBS.</p>Formula:C16H16N4O5Colore e forma:SolidPeso molecolare:344.32MS8815
CAS:<p>MS8815 is a selective EZH2 PROTAC degrader with IC50 of 8.6 nM, used in triple-negative breast cancer research.</p>Formula:C65H87N9O8SColore e forma:SolidPeso molecolare:1154.51Heme Oxygenase-2-IN-1
<p>Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).</p>Formula:C19H17N3O2Colore e forma:SolidPeso molecolare:319.36Galectin-8-IN-1
<p>Galectin-8-IN-1 selectively binds galectin-8N with 48 μM affinity, 15x more than galectin-3.</p>Formula:C16H18N2O6Colore e forma:SolidPeso molecolare:334.32BRD50837
CAS:<p>BRD50837 is a potent and selective inhibitor of Sonic Hedgehog (Shh).</p>Formula:C26H32ClN3O6SPurezza:98%Colore e forma:SolidPeso molecolare:550.07sEH inhibitor-4
<p>Compound B15: potent sEH inhibitor (0.03 nm), reduces inflammation & pain.</p>Formula:C27H28Cl2N4O3Colore e forma:SolidPeso molecolare:527.44Cleistanthin
CAS:<p>Cleistanthin, a toxic Cleistanthus collinus compound, has antihypertensive, alpha-antagonist, and diuretic properties; a modified naphthofuran-xylose.</p>Formula:C28H28O11Colore e forma:SolidPeso molecolare:540.52IRAK4-IN-18
<p>IRAK4-IN-18: Potent IRAK4 inhibitor (IC50: 15 nM), reduces IL23 in cells, prevents rat arthritis.</p>Formula:C24H25FN6O3Colore e forma:SolidPeso molecolare:464.49HIV-1 inhibitor-44
<p>HIV-1 inhibitor-44 (compound 11l) is an HIV-1 reverse transcriptase inhibitor that exhibits activity against wild-type HIV-1 strains (EC50: 0.209 μM).</p>Formula:C23H26N2O4SColore e forma:SolidPeso molecolare:426.53HIF-2α-IN-7
CAS:<p>HIF-2α-IN-7 is a hypoxia inducible factor 2α (HIF-2α) inhibitor.</p>Formula:C18H9F6NO2Colore e forma:SolidPeso molecolare:385.26Asukamycin
CAS:<p>Asukamycin, from S. nodosus asukaensis, is a polyketide antibiotic inhibiting tumor cells by activating caspases 8 and 3.</p>Formula:C31H34N2O7Colore e forma:SolidPeso molecolare:546.61Antimalarial agent 2
<p>Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.</p>Formula:C27H25N3O5Colore e forma:SolidPeso molecolare:471.5ALOX15-IN-1
<p>ALOX15-IN-1 (8b) inhibits rabbit/human ALOX15; IC50: 0.04 μM for LA, 2.06 μM for AA.</p>Formula:C24H31N3O5SColore e forma:SolidPeso molecolare:473.59UB 165
CAS:<p>Subtype-selective nicotinic agonist</p>Formula:C13H15ClN2Purezza:98%Colore e forma:SolidPeso molecolare:234.72PF-06648671
CAS:<p>PF-06648671 is a γ-secretase modulator for the treatment of neurodegenerative and/or neurological disorders.</p>Formula:C25H23ClF4N4O3Purezza:98%Colore e forma:SolidPeso molecolare:538.92TCMDC-125431
<p>TCMDC-125431 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystals.</p>Formula:C25H27N3O2SColore e forma:SolidPeso molecolare:433.57USP7-IN-10
CAS:<p>USP7-IN-10 is a potent inhibitor of ubiquitin-specific protease 7 (USP7), exhibiting an inhibition concentration half-maximal (IC50) value of 13.39 nM.</p>Formula:C26H29ClN4O3SColore e forma:SolidPeso molecolare:513.05SR 33805 oxalate
CAS:<p>Ca2+ channel antagonist</p>Formula:C34H42N2O9SPurezza:98%Colore e forma:SolidPeso molecolare:654.77Lamivudine, (+/-)-trans-
CAS:<p>Lamivudine, a drug for HIV-1 and HBV, inhibits reverse transcriptase and resembles zalcitabine.</p>Formula:C8H11N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:229.26Cortistatin A
CAS:<p>Cortistatin A is a potent and selective mediator-associated kinase CDK8 and its paralogue CDK19 inhibitor.</p>Formula:C30H36N2O3Purezza:98%Colore e forma:SolidPeso molecolare:472.62TY 11345
CAS:<p>TY 11345 is a proton pump inhibitor.</p>Formula:C18H18N3NaO2SColore e forma:SolidPeso molecolare:363.41BTK-IN-15
<p>BTK-IN-15: Oral BTK inhibitor, IC50 0.7 nM, induces cancer cell apoptosis, selective with anti-tumor effects.</p>Formula:C28H24FN5O2Colore e forma:SolidPeso molecolare:481.52Tipelukast
CAS:<p>Tipelukast (KCA 757), an oral drug for asthma research, blocks leukotrienes and fights inflammation and fibrosis.</p>Formula:C29H38O7SPurezza:>99.99%Colore e forma:SolidPeso molecolare:530.67OPC-167832
CAS:<p>OPC-167832: oral dprE1 inhibitor, IC50 0.258 μM, anti-tuberculosis, for Mycobacterium tuberculosis research.</p>Formula:C21H20ClF3N2O4Colore e forma:SolidPeso molecolare:456.845-Iminodaunorubicin hydrochloride
CAS:<p>5-Iminodaunorubicin HCl: quinone-modified anthracycline with antitumor properties, induces DNA breaks in cancer cells.</p>Formula:C27H31ClN2O9Colore e forma:SolidPeso molecolare:563.00Mf 268
CAS:<p>Mf 268 is a pseudo-reversible carbamate-type inhibitor which interacts with the catalytic and regulatory anionic site of the enzyme.</p>Formula:C28H46N4O3Colore e forma:SolidPeso molecolare:486.69HDAC-IN-34
<p>HDAC-IN-34 inhibits HDAC1 (IC50: 0.022 μM) & HDAC6 (IC50: 0.45 μM), binds DNA causing damage, and halts HCT-116 cell growth (IC50: 1.41 μM).</p>Formula:C24H26N6O3Colore e forma:SolidPeso molecolare:446.5FAK-IN-2
<p>FAK-IN-2: potent oral FAK inhibitor, IC50 35 nM, reduces tumor growth, migration, and induces cell death.</p>Formula:C28H31ClN8O3Colore e forma:SolidPeso molecolare:563.059(S)-HEPE
CAS:<p>9(S)-HEPE is a monohydroxy fatty acid derived from EPA. The biological activity of 9(S)-HEPE has not been documented.</p>Formula:C20H30O3Colore e forma:SolidPeso molecolare:318.45CH5447240
CAS:<p>CH5447240: potent hPTHR1 agonist, treats Hypoparathyroidism, EC50 12 nM, 55% oral bioavailability, raises rat serum calcium.</p>Formula:C26H39N5O4SPurezza:98%Colore e forma:SolidPeso molecolare:517.68Purine phosphoribosyltransferase-IN-2
<p>Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.</p>Formula:C11H15N5Na4O10P2Colore e forma:SolidPeso molecolare:531.17Anti-inflammatory agent 10
<p>Tilomisole-derived benzimidazole-thiazole, orally active, favors COX-2 inhibition over COX-1.</p>Formula:C17H13BrN4O3S2Colore e forma:SolidPeso molecolare:465.34Lavendomycin
CAS:<p>Lavendomycin can be extracted from Streptomyces lavendulae and has active against Gram-positive bacteria.</p>Formula:C29H50N10O8Colore e forma:SolidPeso molecolare:666.77MAO-B-IN-10
<p>MAO-B-IN-10: Potent, selective MAO-B inhibitor; crosses blood-brain barrier; IC50 5.3 μM; reduces Aβ aggregation 58.2%, disaggregates 43.3%.</p>Formula:C23H26N2O4Colore e forma:SolidPeso molecolare:394.46Elongation factor P-IN-1
<p>EFP-IN-1: potent β-lysine derivative, inhibits EFP, slows E. coli growth.</p>Formula:C14H31N3O2Colore e forma:SolidPeso molecolare:273.41AHR antagonist 5 hemimaleate
<p>Potent oral AHR antagonist with IC50 < 0.5 μM, hinders tumor growth with anti-PD-1.</p>Formula:C29H28FN7O4Colore e forma:SolidPeso molecolare:499.55Cdc7-IN-8
CAS:<p>Cdc7-IN-8, inhibits Cdc7 kinase, key in DNA replication, and is promising for cancer research. (WO2021032170A1)</p>Formula:C19H21N5O2Colore e forma:SolidPeso molecolare:351.40Anti-Trypanosoma cruzi agent-2
<p>Compd 3b: anti-trypanosomal, IC50 0.51 μM (NINOA), 3.06 μM (INC-5), also combats T. gondii.</p>Formula:C17H10ClNO5Colore e forma:SolidPeso molecolare:343.72BAY-091
CAS:<p>BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.</p>Formula:C26H21FN4O2Purezza:97.66% - 99.23%Colore e forma:SoildPeso molecolare:440.47G-9791
CAS:<p>G-9791 is an effective and selective inhibitor of group-I PAK.</p>Formula:C26H26ClFN6O2Purezza:98%Colore e forma:SolidPeso molecolare:508.98EGFR-IN-45
<p>EGFR-IN-45: Strong EGFR/CDK2 inhibitor (IC50s: 0.4 & 1.6 μM), halts cancer cell cycle pre-G1, prompts apoptosis, also targets Topo I/II.</p>Formula:C28H23N7OColore e forma:SolidPeso molecolare:473.53Antibacterial agent 113
<p>Antibacterial agent 113 targets multiple bacteria including P. aeruginosa and E. coli, showing efficacy at MIC 15625 μM.</p>Formula:C29H18ClN5OColore e forma:SolidPeso molecolare:487.94GW311616 hydrochloride
CAS:<p>GW-311616 hydrochloride is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).</p>Formula:C19H32ClN3O4SPurezza:98%Colore e forma:SolidPeso molecolare:433.99PPARα/γ agonist 1
<p>PPARα/γ agonist 1 is a potent and dual PPARα/γ partial agonist which is a promising prototype for the research of dyslipidemia and diabetes.</p>Formula:C18H19NO2Colore e forma:SolidPeso molecolare:281.35XP5
<p>XP5 is an oral HDAC6 inhibitor, potent against cancer cells, including YCC3/7 (IC50=31 nM to 2.31 μM).</p>Formula:C19H25N3O5SColore e forma:SolidPeso molecolare:407.48Neuraminidase-IN-11
<p>Neuraminidase-IN-11 (15e) inhibits H1N1 (IC50: 4.7nM), H5N1 (8.46nM), H5N8 viruses (1.5nM) selectively & potently.</p>Colore e forma:SolidMV061194
CAS:<p>MV061194 is a potent and selective cathepsin K (Cat K) inhibitor.</p>Formula:C28H37N5O4SColore e forma:SolidPeso molecolare:539.69AZ-PFKFB3-67 quarterhydrate
<p>AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).</p>Formula:C26H27N5O4Colore e forma:SolidPeso molecolare:460.01Anticancer agent 68
CAS:<p>Compound 12, an anticancer agent, halts G2/M phase, triggers cell death, and activates p53 & PTEN for tumor suppression.</p>Formula:C20H18ClNO5Colore e forma:SolidPeso molecolare:387.81Dyrk1A-IN-4
CAS:<p>Dyrk1A-IN-4, compound 48, is an oral DYRK1A/DYRK2 inhibitor with IC50s: 2 nM (DYRK1A), 6 nM (DYRK2), anticancer properties.</p>Formula:C14H13F3N6Colore e forma:SolidPeso molecolare:322.29AKN-028 acetate
<p>AKN-028 acetate: an oral TK inhibitor for AML research, targets FLT3 with IC50 of 6 nM, inhibits autophosphorylation, and induces apoptosis.</p>Formula:C19H18N6O2Colore e forma:SolidPeso molecolare:362.39HCV-IN-7
CAS:<p>HCV-IN-7: potent oral HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.</p>Formula:C40H48N8O6SPurezza:98%Colore e forma:SolidPeso molecolare:768.92VRT-18858
CAS:<p>VRT-18858 is a metabolite of VX-740.</p>Formula:C24H25N5O7Colore e forma:SolidPeso molecolare:495.48MrgprX2 antagonist-7
<p>MrgprX2 antagonist-7 is an anti-allergic agent with significant anti-allergic effects and inhibits mast cell degranulation.</p>Formula:C24H22ClF3N6O3Colore e forma:SolidPeso molecolare:534.92CB 30900
CAS:<p>CB30900 is a novel and effective thymidylate synthase inhibitor.</p>Formula:C31H32FN5O9Colore e forma:SolidPeso molecolare:637.61Antitumor agent-72
CAS:<p>Antitumor agent-72 (compound 6w) is a potent anticancer agent that exhibits its anticancer activity by inducing apoptosis via caspase-3 activation and PARP</p>Formula:C25H20ClNO6Colore e forma:SolidPeso molecolare:465.88Monoamine oxidase/Aromatase-IN-1
<p>Compound 2q: Dual MAO/aromatase inhibitor; IC50: 39 nM (MAO-B), 31 nM (aromatase). Useful in neurological/breast cancer research.</p>Formula:C19H19N3O3SColore e forma:SolidPeso molecolare:369.44CHK-IN-1
CAS:<p>CHK-IN-1 is a dual inhibitor of CHK1 and CHK2 with antiproliferative activity.</p>Formula:C18H19ClFN5OSPurezza:>99.99%Colore e forma:SolidPeso molecolare:407.89BRD4 Inhibitor-17
<p>BRD4 Inhibitor-17: Potent with 0.33 μM IC50; modulates gene expression, may counter arsenic toxicity.</p>Formula:C16H16FN3O3SColore e forma:SolidPeso molecolare:349.38Suloctidil HCl
CAS:<p>Suloctidil HCl is a peripheral vascular dilator.</p>Formula:C20H36ClNOSColore e forma:SolidPeso molecolare:374.02Factor B-IN-4
CAS:<p>Factor B-IN-4 is a potent inhibitor (IC50: 1 μM) of complement factor B. Factor B-IN-4 can be used to study inflammatory and immune-related diseases.</p>Formula:C27H32N2O4Colore e forma:SolidPeso molecolare:448.55Antibacterial agent 99
CAS:<p>Compound 7b (Antibacterial agent 99) is an effective agent with antibacterial, antifungal properties and no haemolytic activity.</p>Formula:C27H27BrN2Colore e forma:SolidPeso molecolare:459.42MraY-IN-3
<p>MraY-IN-3 (12a) is a potent inhibitor of the bacterial translocase MraY (IC50: 140 μM). 46 μg/ml).</p>Formula:C35H45N3O5Colore e forma:SolidPeso molecolare:587.75U92016A hydrochloride
CAS:<p>U92016A hydrochloride: potent, orally active 5-HT1A agonist, metabolically stable, high intrinsic activity, Ki=0.2 nM.</p>Formula:C19H26ClN3Colore e forma:SolidPeso molecolare:331.89L5-DA
<p>L5-DA, a G-quadruplex ligand, stabilizes G4s in HeLa cells, induces apoptosis, and is cytotoxic with an IC50 of 4.3 μM.</p>Formula:C32H34N6O2Colore e forma:SolidPeso molecolare:534.65COX-2/NO-IN-1
<p>COX-2/NO-IN-1: oral iNOS & NO blocker (IC50=3.52μM), COX-2 supressor, anti-inflammatory, protects kidneys.</p>Formula:C15H15NO3Colore e forma:SolidPeso molecolare:257.28ZLMT-12
<p>ZLMT-12: tacrine derivative, inhibits CDK2/CDK9, weak on AChE/BuChE, anti-proliferative, low toxicity, blocks S/G2/M phase, induces apoptosis.</p>Formula:C26H31ClN6OColore e forma:SolidPeso molecolare:479.02TIM-3-IN-1
<p>TIM-3-IN-1 is a useful tool to enable further studies on the biology of TIM-3 immunoregulation in cancer.</p>Formula:C20H16ClN7O3SColore e forma:SolidPeso molecolare:469.9MDL-43291
CAS:<p>MDL-43291 is a leukotriene receptor antagonist.</p>Formula:C25H42O4SColore e forma:SolidPeso molecolare:438.66ACT-672125
CAS:<p>ACT-672125: Potent CXCR3 blocker, may treat autoimmunity, safe with dose-dependent efficacy in lung inflammation.</p>Formula:C25H25F3N10O2SColore e forma:SolidPeso molecolare:586.59THR-β agonist 4
CAS:<p>THR-β agonist 4 is a potent agonist of THR-β.</p>Formula:C16H11Cl2F2N5O6SColore e forma:SolidPeso molecolare:510.26Antibacterial agent 82
<p>Antibacterial agent 82 (compound 7p) is an antibacterial agent [1].</p>Formula:C22H18N2O2Colore e forma:SolidPeso molecolare:342.39K252d
CAS:<p>K252d: indolocarbazole alkaloid in Nocardiopsis; inhibits PKC in rat brain and bovine heart phosphodiesterase.</p>Formula:C26H23N3O5Colore e forma:SolidPeso molecolare:457.48LY367385 hydrochloride
CAS:<p>LY367385 hydrochloride: selective mGluR1a antagonist, IC50 = 8.8 μM, neuroprotective, anticonvulsant, antiepileptic.</p>Formula:C10H12ClNO4Colore e forma:SolidPeso molecolare:245.66SPR-00305
CAS:<p>SPR-00305 is a novel potent inhibitor of the mvfr pathway</p>Formula:C24H19ClN2O3Colore e forma:SolidPeso molecolare:418.87COX-2-IN-12
<p>COX-2-IN-12: Potent, selective COX-2 inhibitor, IC50=19.98μM, safe anti-inflammatory with low acute toxicity.</p>Formula:C17H19NO3Colore e forma:SolidPeso molecolare:285.34U 80215
CAS:<p>U 80215 is an enzyme-competitive inhibitor.</p>Formula:C42H60N8O6SColore e forma:SolidPeso molecolare:805.04HIV-IN-3
<p>HIV-IN-3 (Compound 22a) is a potent inhibitor of HIV (IC50: 1.5 μM). HIV-IN-3 has potential for the study of HIV-related diseases.</p>Formula:C21H32ClN7O3Colore e forma:SolidPeso molecolare:465.98Quinagolide Free Base
CAS:<p>Quinagolide Free Base is a non-ergot dopamine D(2)-agonist.</p>Formula:C20H33N3O3SColore e forma:SolidPeso molecolare:395.56A1AR antagonist 1
<p>Compound 18g, a potent A1AR blocker with Ki: 2.08 nM (hA1), 6.91 nM (hA2A), 31.2 nM (hA2B).</p>Formula:C18H14N4OColore e forma:SolidPeso molecolare:302.33NLRP3-IN-4
<p>NLRP3-IN-4 is an effective, oral NLRP3 inflammasome inhibitor with potent anti-inflammatory effects on colitis.</p>Formula:C22H22N2O5Colore e forma:SolidPeso molecolare:394.42MK-6913
CAS:<p>MK-6913 is a potent and selective agonist of estrogen receptor β.</p>Formula:C25H27N3O2Purezza:98%Colore e forma:SolidPeso molecolare:401.5Sapintoxin D
CAS:<p>Sapintoxin D is a fluorescent phorbol ester and selective activator of protein kinase C.</p>Formula:C30H37NO8Colore e forma:SolidPeso molecolare:539.62PCSK9-IN-16
CAS:<p>PCSK9-IN-16, holds potential for research into hypercholesterolemia and other cardiovascular diseases [1].</p>Formula:C16H20N6O2S3Colore e forma:SolidPeso molecolare:424.56FCE-27262
CAS:<p>FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist.</p>Formula:C23H31N3O3Colore e forma:SolidPeso molecolare:397.51Encephalitic alphavirus-IN-1
<p>Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) & EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.</p>Formula:C27H25FN6O2Colore e forma:SolidPeso molecolare:484.52
