Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.519 prodotti)
- Apoptosi(5.787 prodotti)
- Ciclo cellulare/Checkpoint(4.446 prodotti)
- Cromatina/Epigenetica(2.235 prodotti)
- Segnalazione citoscheletrica(1.381 prodotti)
- Danno al DNA/Riparazione del DNA(2.824 prodotti)
- Endocrinologia/Ormoni(3.500 prodotti)
- Enzima(3.639 prodotti)
- Proteina G/GPCR(8.317 prodotti)
- Immunologia e infiammazione(3.516 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.200 prodotti)
- Trasportatore di membrana/canale ionico(2.787 prodotti)
- Metabolismo(9.416 prodotti)
- Microbiologia/Virologia(6.968 prodotti)
- Neuroscienza(9.919 prodotti)
- Altri inibitori(37.928 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.596 prodotti)
- Cellule staminali e Derivati(831 prodotti)
- Adattatori Tirosin-chinasi(2.015 prodotti)
- Ubiquitinazione(1.649 prodotti)
Mostrare 16 più sottocategorie
Trovati 66626 prodotti di "Inibitori"
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ATP synthase inhibitor 2
CAS:<p>ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.</p>Formula:C21H22N2O3SColore e forma:SolidPeso molecolare:382.48CH5447240
CAS:<p>CH5447240: potent hPTHR1 agonist, treats Hypoparathyroidism, EC50 12 nM, 55% oral bioavailability, raises rat serum calcium.</p>Formula:C26H39N5O4SPurezza:98%Colore e forma:SolidPeso molecolare:517.68Anti-inflammatory agent 23
<p>Anti-inflammatory agent 23 blocks LPS-induced NO (IC50: 0.449 μM) and binds p65 well.</p>Formula:C34H49NO6Colore e forma:SolidPeso molecolare:567.76HIF-2α-IN-7
CAS:<p>HIF-2α-IN-7 is a hypoxia inducible factor 2α (HIF-2α) inhibitor.</p>Formula:C18H9F6NO2Colore e forma:SolidPeso molecolare:385.26Intoplicine
CAS:<p>Intoplicine is an inhibitor of DNA topoisomerase I and II.</p>Formula:C21H24N4OPurezza:98%Colore e forma:SolidPeso molecolare:348.44AFP-07 free acid
CAS:<p>AFP 07 free acid is a 7,7-difluoroprostacyclin derivative. It also acts as a selective and highly potent agonist for the IP receptor.</p>Formula:C22H30F2O5Purezza:98%Colore e forma:SolidPeso molecolare:412.47Metocurine chloride
CAS:<p>Metocurine: a muscle relaxant, not for kidney failure patients as it's kidney-excreted.</p>Formula:C40H48Cl2N2O6Colore e forma:SolidPeso molecolare:723.72Motuporin
CAS:<p>Motuporin is an inhibitor of type-1 and type-2A protein phosphatase catalytic subunits (PP-1c and PP-2Ac).</p>Formula:C40H57N5O10Colore e forma:SolidPeso molecolare:767.91(2R,3S)-Azelaprag
CAS:<p>(2R,3S)-N-(4-(2,6-dimethoxyphenyl)-5-(5-methylpyridin-3-yl)-4H-1,2,4-triazol-3-yl)-3-(5-methylpyrimidin-2-yl)butane-2-sulfonamide is an Apelin receptor agonist</p>Formula:C25H29N7O4SPurezza:97.47% - >99.99%Colore e forma:SoildPeso molecolare:523.61Antitumor agent-58
<p>Antitumor agent-58 suppresses tumor growth, colony formation, cell migration, and induces mitochondrial dysfunction in MGC-803 cells.</p>Formula:C27H28F3N9SColore e forma:SolidPeso molecolare:567.63NBD-10007
CAS:NBD-10007 is an inhibitor of HIV-1 entry.Formula:C20H25ClN4O3SPurezza:98%Colore e forma:SolidPeso molecolare:436.96MI-1851
CAS:<p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>Formula:C34H53N15O6Colore e forma:SolidPeso molecolare:767.88Equisetin
CAS:<p>Equisetin: a QSI from Fusarium equiseti, curbs P. aeruginosa virulence, fights Gram-positive bacteria & HIV-1 integrase; not antibacterial to Gram-negative.</p>Formula:C22H31NO4Purezza:98%Colore e forma:SolidPeso molecolare:373.49CXCR2 antagonist 5
<p>CXCR2 antagonist 5 (compound 25) binds strongly (IC50=0.013μM) and mobilizes calcium (IC50=0.1μM).</p>Formula:C15H14F2N4O2SColore e forma:SolidPeso molecolare:352.36DS88790512
CAS:<p>DS88790512, IC50 at 11 nM, is an effective, selective, oral bioeffective TRPC6 inhibitor.</p>Formula:C22H29N3O2Purezza:98%Colore e forma:SolidPeso molecolare:367.48DYRKs-IN-1
CAS:<p>DYRKs-IN-1 has antitumor activity.</p>Formula:C30H30ClN7O4Purezza:98%Colore e forma:SolidPeso molecolare:588.06Dinalbuphine sebacate
CAS:<p>Dinalbuphine sebacate: long-acting nalbuphine prodrug, μ-opioid partial agonist/antagonist, κ-opioid high-efficacy agonist.</p>Formula:C52H68N2O10Colore e forma:SolidPeso molecolare:881.1Onfasprodil
CAS:<p>Onfasprodil, NR2B inhibitor & GABA regulator, potential for Alzheimer's research. (Patent CN111481543A)</p>Formula:C20H23FN2O3Colore e forma:SolidPeso molecolare:358.41G12Si-1
<p>G12Si-1 selectively binds and inhibits K-Ras(G12S) to block oncogenic signaling and nucleotide exchange.</p>Formula:C29H32ClN5O3Colore e forma:SolidPeso molecolare:534.05Steroid sulfatase/17β-HSD1-IN-4
<p>Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ).</p>Formula:C18H17N3O4S2Colore e forma:SolidPeso molecolare:403.48G247
<p>G247 inhibits MsbA by keeping NBDs apart, blocking ATPase activity.</p>Formula:C24H19Cl2FO3Colore e forma:SolidPeso molecolare:445.31Aspochalasin M
CAS:<p>Aspochalasin M shows moderate activity on HL-60 cells (IC50=20.0 μ M). Aspochalasin M has research potential in leukemia diseases.</p>Formula:C24H35NO4Colore e forma:SolidPeso molecolare:401.54G-9791
CAS:<p>G-9791 is an effective and selective inhibitor of group-I PAK.</p>Formula:C26H26ClFN6O2Purezza:98%Colore e forma:SolidPeso molecolare:508.98IRAK4-IN-12
<p>IRAK4-IN-12 (compound 37) is a potent inhibitor of IRAK4 (IC50: 0.015 μM) with cellular pIRAK4 potency (IC50: 0.5 μM).</p>Formula:C24H31FN8OColore e forma:SolidPeso molecolare:466.55AChE/BChE-IN-1
<p>AChE/BChE-IN-1: dual AChE/BChE inhibitor, IC50 of 1.06 nM/7.3 nM, crosses blood-brain barrier, with antioxidant properties for Alzheimer's research.</p>Formula:C32H35ClN6O3Colore e forma:SolidPeso molecolare:587.11FTI-2148
CAS:<p>FTI-2148 blocks RAS-related FT-1 & GGT-1; IC50: 1.4 nM & 1.7 μM.</p>Formula:C24H28N4O3SPurezza:98%Colore e forma:SolidPeso molecolare:452.57Anti-inflammatory agent 16
<p>Compound 14 is a peptidomimetic that significantly lowers TNFα, NO, CD40, and CD86, showcasing strong anti-inflammatory effects.</p>Formula:C21H23N5O3Colore e forma:SolidPeso molecolare:393.44Purine phosphoribosyltransferase-IN-2
<p>Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.</p>Formula:C11H15N5Na4O10P2Colore e forma:SolidPeso molecolare:531.17C-di-IMP
CAS:<p>Cyclic-di-IMP (C-di-IMP), a STING agonist, serves as a research tool in tumor studies.</p>Formula:C20H22N8O14P2Colore e forma:SolidPeso molecolare:660.38XIAP/cIAP1 antagonist-1
<p>Potent oral XIAP/cIAP1 inhibitor with EC50s: XIAP 5.1 nM, cIAP1 0.32 nM; curbs tumor growth in vivo.</p>Colore e forma:SolidCDK2-IN-8
<p>CDK2-IN-8 is a potent CDK2 inhibitor (IC50= 1.74 μM). CDK2-IN-8 exhibits antiproliferative activity. CDK2-IN-8 can be used for the research of melanoma.</p>Formula:C22H25N5O3Colore e forma:SolidPeso molecolare:407.47CEase-IN-1
<p>CEase-IN-1 (A1H3), potent CEase inhibitor, IC50 0.36μM, for hypercholesterolemia study.</p>Formula:C13H15F3N2O2Colore e forma:SolidPeso molecolare:288.27MI-1481
CAS:<p>MI-1481: potent MML1 inhibitor, IC50 3.6 nM; disrupts menin-MLL1, active in MLL leukemia.</p>Formula:C29H30F3N7O2SPurezza:98%Colore e forma:SolidPeso molecolare:597.65HIV-1 inhibitor-17
<p>HIV-1 inhibitor-18 blocks HIV-1 capsid, acts on NL4-3 strain (EC50: 2.57 μM), has low cytotoxicity (MT-4 CC50: >8.55).</p>Formula:C32H32N4O5SColore e forma:SolidPeso molecolare:584.69Arterolane maleate
CAS:<p>Arterolane, an adenosine triphosphatase inhibitor, is used potentially for the treatment of malaria.</p>Formula:C26H40N2O8Purezza:98%Colore e forma:SolidPeso molecolare:508.612EGFR-IN-34
<p>EGFR-IN-34 is a low-toxicity, acrylamide derivative antitumor agent that is a potent inhibitor of EGFR.</p>Formula:C26H27ClN6O2Colore e forma:SolidPeso molecolare:490.98PKG1α activator 3
<p>PKG1α activator 3 is a PKG1α activator (EC50basal/partial=13/0.52 μM).</p>Formula:C27H26Cl2N2O6Colore e forma:SolidPeso molecolare:545.41LSD1-IN-16
<p>LSD1-IN-16 (4b) inhibits LSD1, MAO-A/B; IC50: 0.015-0.366 μM. Halts prostate cancer cell growth; IC50: 15.2 μM.</p>Formula:C20H18N2OSColore e forma:SolidPeso molecolare:334.43Dot1L-IN-1
CAS:<p>The Ki value of DOT1L-in-1 is 2pm.It is a highly effective, selective and novel Dot1L inhibitor.</p>Formula:C32H36ClN9O2SPurezza:98%Colore e forma:SolidPeso molecolare:646.21SM-433 hydrochloride
<p>SM-433 hydrochloride, a Smac mimetic & IAP inhibitor, binds XIAP BIR3; potent IC50 <1 μM. (Patent WO2008128171A2)</p>Formula:C32H44ClN5O4Colore e forma:SolidPeso molecolare:598.18GNE-886
CAS:<p>GNE-886 has a wide range of applications in life science related research.</p>Formula:C28H30N6O3Purezza:98%Colore e forma:SolidPeso molecolare:498.59CDK4/6-IN-13
CAS:<p>Compounds 10B and 10C: potent cdk4/6 inhibitors with low nM activity, great antiproliferative effects, excellent metabolism, and good pharmacokinetics.</p>Formula:C25H29N7OColore e forma:SolidPeso molecolare:443.54RDN2150
CAS:<p>RDN2150 (Compound 25), a ZAP-70 inhibitor with an IC50 of 14.6 nM, covalently binds to the C346 residue of ZAP-70, suppressing the expression of CD25 and CD69</p>Formula:C28H29ClN8O4Colore e forma:SolidPeso molecolare:577.03Inupadenant HCl
CAS:<p>Inupadenant (EOS-850) is a selective A2a receptor antagonist, targeting immunosuppression in tumors.</p>Formula:C25H27ClF2N8O4S2Colore e forma:SolidPeso molecolare:641.11ZIKV-IN-4
<p>ZIKV-IN-4 is a low cytotoxic, acid-stable anti-ZIKV agent with an EC50 value of 3.49 μM. ZIKV-IN-4 exhibited potent inhibition of ZIKV NS5 MTase.</p>Formula:C33H37NO4Colore e forma:SolidPeso molecolare:511.65AKN-028 acetate
<p>AKN-028 acetate: an oral TK inhibitor for AML research, targets FLT3 with IC50 of 6 nM, inhibits autophosphorylation, and induces apoptosis.</p>Formula:C19H18N6O2Colore e forma:SolidPeso molecolare:362.39Neuraminidase-IN-11
<p>Neuraminidase-IN-11 (15e) inhibits H1N1 (IC50: 4.7nM), H5N1 (8.46nM), H5N8 viruses (1.5nM) selectively & potently.</p>Colore e forma:SolidPM-060184
CAS:<p>PM-060184, a tubulin polymerisation inhibitor, is used potentially for the treatment of solid tumours and breast cancer.</p>Formula:C31H45N3O7Purezza:98%Colore e forma:SolidPeso molecolare:571.7Mifepristone methochloride
CAS:<p>Mifepristone methochloride is a glucocorticoid antagonist. This product will be sold for research use only.</p>Formula:C30H38ClNO2Colore e forma:SolidPeso molecolare:480.08LTD4 antagonist 1
CAS:<p>LTD4 antagonist 1 is a potent and orally active antagonist of leukotriene D4 (LTD4; Ki: 0.57 nM).</p>Formula:C31H32F3N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:615.66PF-06263276
CAS:<p>PF-06263276 selectively inhibits pan-JAK with IC50: JAK1 (2.2 nM), JAK2 (23.1 nM), JAK3 (59.9 nM), TYK2 (29.7 nM).</p>Formula:C31H31FN8O2Purezza:98%Colore e forma:SolidPeso molecolare:566.63CYP1B1-IN-2
<p>CYP1B1-IN-2 (compound 9j) is a highly potent and selective inhibitor of CYP1B1, a cytochrome P450 enzyme. It exhibits an IC50 value of 0.52 nM [1].</p>Formula:C20H11F3O2Colore e forma:SolidPeso molecolare:340.3PfPKG-IN-1
<p>PfPKG-IN-1, an imidazole-based inhibitor, targets the Plasmodium falciparum cyclic guanosine monophosphate-dependent protein kinase (PfPKG).</p>Formula:C24H22ClN7OSColore e forma:SolidPeso molecolare:492DC-U4106
CAS:<p>DC-U4106: USP8 inhibitor, Kd 4.7μM, IC50 1.2μM, degrades Erα, low-toxicity tumor suppressor for breast cancer research.</p>Formula:C29H27N5O5Colore e forma:SolidPeso molecolare:525.56Cortistatin A
CAS:<p>Cortistatin A is a potent and selective mediator-associated kinase CDK8 and its paralogue CDK19 inhibitor.</p>Formula:C30H36N2O3Purezza:98%Colore e forma:SolidPeso molecolare:472.62PptT-IN-1
<p>PptT-IN-1, a potent PptT inhibitor (IC50: 2.8 μM), shows promise for tuberculosis research.</p>Formula:C18H29N5O2Colore e forma:SolidPeso molecolare:347.46Tubulin inhibitor 13
CAS:<p>Tubulin inhibitor 13 (E27), IC50 16.1 μM, blocks tubulin polymerization, cancer cell migration, and invasion, induces apoptosis.</p>Formula:C25H21N3O4Colore e forma:SolidPeso molecolare:427.45MY-875
<p>MY-875 inhibits microtubule formation, binds like colchicine (IC50: 0.92 μM), activates Hippo pathway, and induces apoptosis with anticancer properties.</p>Formula:C21H25NO6Colore e forma:SolidPeso molecolare:387.43DNA-PK-IN-2
CAS:<p>DNA-PK-IN-2 is an inhibitor of the DNA-PK enzyme complex, useful in cancer research.</p>Formula:C20H23N5O3Colore e forma:SolidPeso molecolare:381.43EGFR-IN-17
<p>EGFR-IN-17: potent, selective EGFR inhibitor, IC50 of 0.2 nM, overcomes C797S drug resistance.</p>Formula:C27H31ClN7O3PColore e forma:SolidPeso molecolare:568.01AXKO-0046
<p>AXKO-0046 is an indole derivative and small-molecule LDHB selective inhibitor.</p>Formula:C25H33N3Colore e forma:SolidPeso molecolare:375.55Arverapamil
CAS:<p>Arverapamil is a chiral metabolite of Verapamil.</p>Formula:C26H36N2O4Colore e forma:SolidPeso molecolare:440.58Plumbemycin A
CAS:<p>Plumbemycin A is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Formula:C12H20N3O9PColore e forma:SolidPeso molecolare:381.28(S)-Butaprost free acid
CAS:<p>(S)-Butaprost (free acid) is a potent and highly selective EP2 receptor agonist[1].</p>Formula:C23H38O5Colore e forma:SolidPeso molecolare:394.54SARS-CoV-2-IN-24
<p>SARS-CoV-2-IN-24 blocks PLpro, altering its shape and stopping virus replication—useful for SARS-CoV-2 research.</p>Formula:C27H30N4O5Colore e forma:SolidPeso molecolare:490.55GGTI298
CAS:<p>GGTI298 is a potent GGTase I inhibitor; IC50 3μM for Rap1A, >20μM for Ha-Ras.</p>Formula:C27H33N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:479.63BM635 mesylate (1493762-74-5 free base)
<p>BM635 mesylate is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).</p>Formula:C26H33FN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:488.61TTK inhibitor 3
CAS:<p>TTK inhibitor 3 is a potent and selective TTK (an essential spindle assembly checkpoint enzyme) inhibitor with an IC 50 value of 3.0 nM.</p>Formula:C42H49N9O3Colore e forma:SolidPeso molecolare:727.9TGFβ1-IN-1
CAS:<p>TGFβ1-IN-1 is a TGF-β1 inhibitor that inhibits the production of TGF-β1-induced fibrosis markers (α-SMA and fibronectin) and can be used in cancer research.</p>Formula:C22H24N2O3Purezza:99.89% - 99.89%Colore e forma:SolidPeso molecolare:364.438TNP-470
CAS:<p>TNP-470 is a methionine aminopeptidase-2 inhibitor. TNP-470 is also an angiogenesis inhibitor.</p>Formula:C19H28ClNO6Purezza:98%Colore e forma:SolidPeso molecolare:401.88MALT1-IN-5
CAS:<p>MALT1-IN-5 is a potent inhibitor of the MALT1 protease and can be used in cancer research.</p>Formula:C17H17ClF2N6O3Colore e forma:SolidPeso molecolare:426.80GRPR antagonist-2
<p>GRPR antagonist-2 blocks GRPR, kills some cancer cells, effective on HGC-27 (IC50: 0.77 μM) & Pan02 (IC50: 2.5 μM).</p>Formula:C28H32F3N5O4Colore e forma:SolidPeso molecolare:559.58Scytonemin
CAS:<p>Scytonemin, a cyanobacterial pigment, inhibits cancer cell growth by decreasing Plk1 activity, especially effective on U266 myeloma cells.</p>Formula:C36H20N2O4Colore e forma:SolidPeso molecolare:544.55L-threo-Sphingosine C-18
CAS:<p>L-threo-Sphingosine C-18 is a protein kinase C inhibitor.</p>Formula:C18H37NO2Purezza:98%Colore e forma:SolidPeso molecolare:299.49MC4355
<p>MC4355 is a dual inhibitor of EZH2 and histone deacetylase (HDAC).</p>Formula:C30H36N4O5Colore e forma:SolidPeso molecolare:532.63VU6005806
CAS:<p>VU6005806 is a potent M4 PAM with EC50s: 94 nM (human), 28 nM (rat), 87 nM (dog), 68 nM (cyno); studied for neuropsychiatric disorders.</p>Formula:C17H16F3N7O2SPurezza:98%Colore e forma:SolidPeso molecolare:439.41P300 bromodomain-IN-1
<p>P300 bromodomain-IN-1 blocks c-Myc, induces G1/G0 arrest, apoptosis. Potent EP300 inhibitor (IC50: 49 nM).</p>Formula:C29H31ClN4O4Colore e forma:SolidPeso molecolare:535.03BMS 310705
CAS:<p>BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.</p>Formula:C27H42N2O6SColore e forma:SolidPeso molecolare:522.70LY 292728
CAS:<p>LY 292728 is a highly potent antagonist of leukotriene B4 receptor.</p>Formula:C34H29FO9Purezza:98%Colore e forma:SolidPeso molecolare:600.59Bomedemstat hydrochloride
<p>Bomedemstat (IMG-7289) hydrochloride, an oral LSD1 inhibitor, has anticancer properties, blocking cell growth and triggering apoptosis.</p>Formula:C28H35ClFN7O2Colore e forma:SolidPeso molecolare:556.08STING agonist-20
CAS:<p>STING agonist-20: potent, aids in XMT-2056 synthesis, used as a cancer vaccine adjuvant.</p>Formula:C36H39N11O8Colore e forma:SolidPeso molecolare:753.76T-3861174
CAS:<p>T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.</p>Formula:C26H25FN6O2Colore e forma:SolidPeso molecolare:472.51AChE-IN-8
<p>AChE-IN-8 (Compound 19), potent acetylcholinesterase blocker; IC50 = 1.95 μM; potential Alzheimer's treatment.</p>Formula:C20H22N4O2SColore e forma:SolidPeso molecolare:382.48NPR-C activator 1
CAS:<p>NPR-C activator 1 is an activator of the natriuretic peptide receptor C (NPR-C), which can be used to study cardiovascular diseases.</p>Formula:C18H24N6O3Purezza:98.74%Colore e forma:SolidPeso molecolare:372.42PIM1-IN-3
<p>PIM1-IN-3 (HL8) selectively blocks PIM1, induces Colo320 cell apoptosis, and may be researched for cancer.</p>Formula:C27H25BrN6OColore e forma:SolidPeso molecolare:529.43Ledene
CAS:<p>Ledene (Viridiflorene) is an essential oil produced by viridiflorene synthase.</p>Formula:C15H24Purezza:98%Colore e forma:SolidPeso molecolare:204.35JAK1-IN-9
CAS:<p>JAK1-IN-9 (compound 23a) is a potent, selective inhibitor of JAK1, demonstrating an IC50 of 72 nM.</p>Formula:C16H13IN6Colore e forma:SolidPeso molecolare:416.22Lp-PLA2-IN-10
<p>Lp-PLA2-IN-10, a potent Lp-PLA2 inhibitor, may research neurodegenerative and cardiovascular diseases.</p>Formula:C21H15F5N4O4Colore e forma:SolidPeso molecolare:482.36ZK159222
CAS:<p>ZK159222 is an effective 1α,25-(OH)2D3 receptor (VDR) agonist. ZK159222 has a partial agonistic character.</p>Formula:C32H48O5Purezza:98%Colore e forma:SolidPeso molecolare:512.72CXCR2 antagonist 4
<p>CXCR2 antagonist 4 inhibits CXCR2 (IC50: 0.13 μM) and CXCL8-induced calcium rise (IC50: 27 μM), promising for cancer research.</p>Formula:C15H14F2N4OS2Colore e forma:SolidPeso molecolare:368.42Axl-IN-3
<p>Axl-IN-3 is a selective, potent and orally active inhibitor of AXL kinase (IC50: 41.5 nM) and has a low inhibitory effect on other kinases.</p>Formula:C24H25ClN6O2Colore e forma:SolidPeso molecolare:464.9513(R)-HODE
CAS:<p>13(R)-HODE, produced from linoleic acid, inhibits platelet aggregation (IC50=2.7μM) and is found in bovine endothelial cells.</p>Formula:C18H32O3Colore e forma:SolidPeso molecolare:296.44Antifungal agent 12
<p>Antifungal agent 12 is a new fluconazole-like compound that exhibits good antifungal effects.</p>Formula:C20H16F3N7O2S2Colore e forma:SolidPeso molecolare:507.51CaMKIIα-IN-1
<p>CaMKIIα-IN-1 (Compound 4d) is an orally active inhibitor of Ca 2+ /calmodulin-dependent protein kinase II α (CaMKIIα) with a Kd of 219 nM for CaMKIIα WT hub.</p>Formula:C14H11ClO4Colore e forma:SolidPeso molecolare:278.69PAIR2
CAS:<p>PAIR2 is a selective IRE1α RNase partial antagonist, blocking its ATP site and preventing KIRA from hindering XBP1 splicing.</p>Formula:C27H26F4N6O3SColore e forma:SolidPeso molecolare:590.59ALK-IN-23
<p>ALK-IN-23 inhibits ALK (IC50: 1.6-0.71 nM), hinders cancer cell spread, forms colonies in vitro, and reduces tumors in mice with low toxicity.</p>Formula:C26H29ClN8O3SColore e forma:SolidPeso molecolare:569.08CAII-IN-1
<p>CAII-IN-1 (3n) is a selective bovine CA-II inhibitor with 10.3 μM IC50, used in carbonic anhydrase disorder studies.</p>Formula:C19H21FN4SColore e forma:SolidPeso molecolare:356.46Anti-inflammatory agent 19
<p>Anti-inflammatory agent 19: NO inhibitor (IC50: 36μM), blocks HMGB1, for late-stage inflammation, relevant for COVID-19, sepsis.</p>Formula:C30H50O7Colore e forma:SolidPeso molecolare:522.71Mal-PEG4-VA-PBD
CAS:<p>Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connected</p>Formula:C68H79N9O17Purezza:98%Colore e forma:SolidPeso molecolare:1294.41AD012
<p>AD012, a dual cACE/NEP inhibitor, leverages lenopril-tryptophan for potential anti-hypertensive and cardioprotective benefits.</p>Formula:C25H32N2O6Colore e forma:SolidPeso molecolare:456.53MK-7445
CAS:<p>MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.</p>Formula:C21H13Cl2N7OColore e forma:SolidPeso molecolare:450.28Plasma kallikrein-IN-2
<p>Plasma kallikrein-IN-2: PKal inhibitor, IC50=0.1 nM. Used in angioedema, diabetic eye disease research.</p>Formula:C28H24ClF3N8O3Colore e forma:SolidPeso molecolare:612.99HIF-1/2α-IN-1
<p>HIF-1/2α-IN-1, an orally active compound, functions as an inhibitor of HIF-2α.</p>Formula:C17H16N6O4Colore e forma:SolidPeso molecolare:368.35SB 204070 hydrochloride
CAS:<p>SB 204070 hydrochloride is an inhibitor of beta-lactamase, it is isolated from Spondias mombin.</p>Formula:C19H27ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:382.88Carbonic anhydrase inhibitor 9
<p>Carbonic anhydrase inhibitor 9 targets hCA II and IX with Ki of 56.4 and 56.9 nM respectively; shows antiproliferative activity.</p>Formula:C22H20BrN5O4SColore e forma:SolidPeso molecolare:530.39Lobaric acid
CAS:<p>Lobaric acid, from Stereocaulon lichen, has antioxidant and anticancer properties, inhibits PTP1B and 12(S)-LOX, and reduces TMV lesions in plants.</p>Formula:C25H28O8Colore e forma:SolidPeso molecolare:456.48NNTA
CAS:<p>NNTA is a highly selective and potent activator of μ/κ-opioid heteromers.</p>Formula:C31H32N2O4Colore e forma:SolidPeso molecolare:496.60Antileishmanial agent-4
<p>Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].</p>Formula:C17H18N4O4Colore e forma:SolidPeso molecolare:342.35CS-003 HCl
CAS:<p>CS-003 HCl is a TNRA - triple neurokinin receptor antagonist.</p>Formula:C34H39Cl3N2O6SColore e forma:SolidPeso molecolare:710.1Ribocil-C R enantiomer
<p>Ribocil-C R enantiomer is the R enantiomer of Ribocil-C. Ribocil-C is a highly selective bacterial riboflavin riboswitches inhibitor.</p>Formula:C21H21N7OSPurezza:98%Colore e forma:SolidPeso molecolare:419.5α-Glucosidase-IN-14
<p>α-Glucosidase-IN-14 is a potent inhibitor of α-glucosidase (IC50: 5.22 μM).</p>Formula:C24H27N5O4S2Colore e forma:SolidPeso molecolare:513.63Salvinorin A Propionate
CAS:<p>Salvinorin A propionate: partial KOR agonist, Ki=32.6 nM, EC50=4.7 nM; ignores μ/δ/ORL-1, non-opioid receptors; less potent analgesic vs. salvinorin A.</p>Formula:C24H30O8Colore e forma:SolidPeso molecolare:446.49KMN-80
CAS:<p>KMN-80 is a potent, selective EP4 agonist with IC50 3 nM, spurring osteoblast differentiation, and showing in vivo bone repair efficacy.</p>Formula:C21H33NO4Colore e forma:SolidPeso molecolare:363.49PI3K-IN-37
CAS:<p>PI3K-IN-37 inhibits PI3K α/β/δ (IC50: 6/8/4 nM) and mTOR (IC50: 4 nM).</p>Formula:C25H26N6O2Colore e forma:SolidPeso molecolare:442.51Antiproliferative agent-4
<p>Antiproliferative agent-4 suppresses cancer cell growth with low toxicity, inhibits tumors in mice, and induces apoptosis in EC109 cells.</p>Formula:C29H35ClO8Colore e forma:SolidPeso molecolare:547.04IRAK4-IN-14
CAS:<p>IRAK4-IN-14 is a selective, potent, orally active IRAK4 inhibitor (IC50: 0.003 μM) with favorable PK parameters in rats and mice. effect.</p>Formula:C25H28FN9OColore e forma:SolidPeso molecolare:489.55COTC
CAS:<p>COTC is an anticancer bacterial metabolite; inhibits glyoxalase with GSH, halts HeLa cell growth, and fights tumor in Ehrlich murine model.</p>Formula:C11H14O6Colore e forma:SolidPeso molecolare:242.23DC41SMe
CAS:<p>DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.</p>Formula:C38H36ClN5O4S2Purezza:98%Colore e forma:SolidPeso molecolare:726.31CJ-887
CAS:<p>CJ-887 is a STAT3 inhibitor.</p>Formula:C34H45N6O10PColore e forma:SolidPeso molecolare:728.73Ep vinyl quinidine
CAS:<p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>Formula:C20H24N2O2Colore e forma:SolidPeso molecolare:324.42KRAS G12D inhibitor 16
CAS:<p>KRAS G12D inhibitor 16 targets KRAS G12D with IC50 of 0.7 nM and mutant form at 0.35 μM, useful in various cancer studies.</p>Formula:C32H39IN6O3Colore e forma:SolidPeso molecolare:682.59NOS-IN-2
<p>NOS-IN-2: potent, selective imidamide NOS inhibitor, IC50=20μM for iNOS, spares eNOS, low toxicity, useful in inflammation research.</p>Formula:C18H20F3N3O2Colore e forma:SolidPeso molecolare:367.3715(R)-Lipoxin A4
CAS:<p>Lipid-derived lipoxins are produced at the site of vascular and mucosal inflammation where they down-regulate polymorphonuclear leukocyte recruitment and</p>Formula:C20H32O5Colore e forma:SolidPeso molecolare:352.47PI3K-IN-26
CAS:<p>PI3K-IN-26 is an effective PI3K inhibitor. PI3K-IN-26 inhibits the proliferation of SU-DHL-6 cells, IC50= 36 nM.</p>Formula:C21H18N6OSColore e forma:SolidPeso molecolare:402.47BRD-7880
CAS:<p>BRD-7880 is a potent and highly specific inhibitor of aurora kinases B and C.</p>Formula:C32H38N4O7Colore e forma:SolidPeso molecolare:590.67Cenicriviroc Sulfone
CAS:<p>Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.</p>Formula:C41H52N4O5SColore e forma:SolidPeso molecolare:712.9414α-Demethylase/DNA Gyrase-IN-1
<p>14α-Demethylase/DNA Gyrase-IN-1 (Compound 7c) is a potent inhibitor of 14α-Demethylase/DNA Gyrase with antibacterial activity.</p>Formula:C26H22N4O4Colore e forma:SolidPeso molecolare:454.48LP-284
CAS:<p>LP-284 is a DNA alkylating agent effective against solid tumors and hematologic cancers like MCL.</p>Formula:C16H20N2O4Colore e forma:SolidPeso molecolare:304.34GR-112000
CAS:<p>GR-112000 is a peptide-based tachykinin NK2 receptor antagonist.</p>Formula:C30H36N6O3Colore e forma:SolidPeso molecolare:528.65Epiderstatin
CAS:<p>Epiderstatin is isolated from Streptomyces pulveraceus subsp. epiderstagenes; inhibits mitogenic activity of epidermal growth factor.</p>Formula:C15H20N2O4Colore e forma:SolidPeso molecolare:292.33Fumarranol
CAS:<p>Fumarranol inhibits angiogenesis and malaria growth by targeting PfMAP2.</p>Formula:C16H24O4Colore e forma:SolidPeso molecolare:280.36URAT1 inhibitor 2
<p>URAT1 inhibitor 2: oral URAT1/CYP blocker, IC50 of 1.36μM (URAT1), 16.97μM (CYP1A2), 5.22μM (CYP2C9); potential gout treatment.</p>Formula:C21H18BrN3O2SColore e forma:SolidPeso molecolare:456.36VEGFR-2-IN-10
<p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>Formula:C20H21N3O2Colore e forma:SolidPeso molecolare:335.4Anticancer agent 29
<p>Compound E/Z-6f, anticancer, IC50: CDK2 (0.054 μM), CDK1 (0.127 μM), CDK4 (0.129 μM), CDK6 (0.396 μM).</p>Formula:C22H15ClFNOColore e forma:SolidPeso molecolare:363.81HPK1-IN-31
<p>HPK1-IN-31 inhibitor with an IC 50 value of 0.8 nM. HPK1-IN-31 has anti-tumour activity and has great potential for immunotherapy .</p>Formula:C30H33N7O3Colore e forma:SolidPeso molecolare:539.63Antitubercular agent-15
<p>Antitubercular agent-15 (5n): low toxicity, fights M. tuberculosis strains; MIC90 values range 0.73-18.8 μg/mL.</p>Formula:C21H29FN2Colore e forma:SolidPeso molecolare:328.47LXR agonist 2
<p>LXR agonist 2 is a potent agonist of the LXR (liver X receptor). LXR agonist 2 stabilises NCOA1 (coactivator), which in turn agonises the LXR.</p>Formula:C35H40ClN3O3Colore e forma:SolidPeso molecolare:586.16HPK1-IN-21
<p>HPK1-IN-21 is a potent, orally active HPK1 kinase inhibitor with a Ki value of 0.8 nM.</p>Formula:C22H25ClFN5O2Colore e forma:SolidPeso molecolare:445.92HBV-IN-31
CAS:<p>HBV-IN-31: strong cccDNA inhibitor, anti-HBV, IC50=0.13 µM HBsAg, hampers cell growth.</p>Formula:C23H18ClNO6Colore e forma:SolidPeso molecolare:439.85HPK1-IN-14
CAS:<p>HPK1-IN-14 is a potent inhibitor of HPK1. HPK1-IN-14 has potential for the study of HPK1-related diseases.</p>Formula:C24H23FN6O2Colore e forma:SolidPeso molecolare:446.48Pamiparib maleate
CAS:<p>Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.</p>Formula:C44H42F2N8O14Purezza:98%Colore e forma:SolidPeso molecolare:944.859BILA 1906 BS
CAS:<p>BILA 1906 BS is an inhibitor of substrate analog protease.</p>Formula:C41H52N6O4SPurezza:98%Colore e forma:SolidPeso molecolare:724.95FAK-IN-3
<p>FAK-IN-3 inhibits FAK, reduces PA-1 cell migration/invasion, and tumor growth, with no major side effects.</p>Formula:C28H28N6O4Colore e forma:SolidPeso molecolare:512.56NB-533
CAS:<p>NB-533 is a macrocyclic peptidic BACE-1 inhibitor.</p>Formula:C33H55N3O4Colore e forma:SolidPeso molecolare:557.819(S),10(S),13(S)-TriHOME
CAS:<p>9(S),10(S),13(S)-TriHOME is an oxylipin derived from linoleic acid. It has been detected in beer and in bronchoalveolar lavage fluid (BALF) from female smokers.</p>Formula:C18H34O5Colore e forma:SolidPeso molecolare:330.46L-697639
CAS:<p>L-697639 inhibits of HIV-1 reverse transcriptase and HIV-1 replication.</p>Formula:C18H21N3O2Colore e forma:SolidPeso molecolare:311.38LasR-IN-1
<p>LasR-IN-1 (9g) strongly inhibits LasR, potent vs E. coli, with a 28.13 μM MIC against P. aeruginosa.</p>Formula:C23H21N3O2Colore e forma:SolidPeso molecolare:371.43PD-L1-IN-1
<p>PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.</p>Formula:C21H23N5O2Colore e forma:SolidPeso molecolare:377.44L 734217
CAS:<p>L 734217 is an antagonist of the fibrinogen receptor.</p>Formula:C18H31N3O4Purezza:98%Colore e forma:SolidPeso molecolare:353.46Tubulin polymerization-IN-32
<p>Tubulin polymerization-IN-32: a cancer cell growth inhibitor used for research in cancers like lymphoma.</p>Formula:C29H30N2O7Colore e forma:SolidPeso molecolare:518.56NLRP3-IN-7
<p>NLRP3-IN-7 (Compound 36) is a selective inhibitor of the NLRP3 inflammasome and is able to assemble the NLRP3 inflammasome.</p>Formula:C18H15ClN2O4S3Colore e forma:SolidPeso molecolare:454.97Ranakinin
CAS:<p>Ranakinin is a novel tachykinin receptor agonist; from the brain of frog, Rana ridibunda.</p>Formula:C62H95N17O15SColore e forma:SolidPeso molecolare:1350.59FAAH/MAGL-IN-3
<p>FAAH/MAGL-IN-3 irreversibly inhibits FAAH (IC50: 179 nM) & MAGL (IC50: 759 nM) with low PAMPA permeability.</p>Formula:C21H25N3O6SColore e forma:SolidPeso molecolare:447.5LXRβ agonist-3
CAS:<p>LXRβ agonist-3 is a potent and selective LXRβ (liver X receptor β) agonist (EC50: 0.095 μM).</p>Formula:C30H33N3O6SColore e forma:SolidPeso molecolare:563.66HPK1-IN-3
<p>HPK1-IN-3: Selective HPK1 inhibitor, ATP-competitive, IC50=0.25nM; boosts IL-2 in PBMCs, EC50=108nM.</p>Formula:C23H22F4N6O2Colore e forma:SolidPeso molecolare:490.45Lumirubin
CAS:<p>Lumirubin is a water-soluble photoproduct of bilirubin formed in vivo during phototherapy.</p>Formula:C33H36N4O6Colore e forma:SolidPeso molecolare:584.66BAY-7598
CAS:<p>BAY-7598 is a potent, selective, and orally bioavailable MMP12 inhibitor (IC50s: 0.085, 0.67, and 1.1 nM for human/murine/rat MMP12).</p>Formula:C28H31N3O6Purezza:98%Colore e forma:SolidPeso molecolare:505.56GNE-616
CAS:<p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>Formula:C24H23F4N5O3SPurezza:98%Colore e forma:SolidPeso molecolare:537.53Fasitibant
CAS:<p>Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.</p>Formula:C36H49Cl2N6O6SColore e forma:SolidPeso molecolare:764.78Antitumor agent-77
<p>Antitumor agent-77 suppresses cancer cell growth, migration, induces apoptosis, and hinders EMT.</p>Formula:C7H11F3N2O5PtColore e forma:SolidPeso molecolare:455.25Dyrk1A/α-synuclein-IN-1
<p>Dyrk1A/α-synuclein-IN-1 (Compound b1) is a dual inhibitor of Dyrk1A (IC50: 177 nM) and α-synuclein aggregation (IC50: 10.5 μM).</p>Formula:C20H21N5O3SColore e forma:SolidPeso molecolare:411.48CD73-IN-7
CAS:<p>CD73-IN-7: potent inhibitor of CD73, blocks adenosine production to treat tumors.</p>Formula:C13H11ClN4O2Colore e forma:SolidPeso molecolare:290.75-cis Carbaprostacyclin
CAS:<p>5-cis Carbaprostacyclin: a PGI2 stable analog; poor human platelet aggregation inhibitor (IC50: 2.8 μM); weakens rabbit artery relaxation (EC50: 104 μM).</p>Formula:C21H34O4Colore e forma:SolidPeso molecolare:350.49Adecypenol
CAS:<p>Adecypenol is a unique adenosine deaminase inhibitor. It shows effective inhibitory activity against calf intestinal adenosine deaminase.</p>Formula:C12H16N4O4Purezza:98%Colore e forma:SolidPeso molecolare:280.28HBV-IN-18
<p>HBV-IN-18 (Compound 3) is an HBV capsid assembly modulator (CpAM) (EC50: 2790 nM).</p>Formula:C17H15F6N5O2Colore e forma:SolidPeso molecolare:435.32PTP1B-IN-17
<p>PTP1B-IN-17, a benzimidazole derivative, inhibits PTP1B (Ki: 30.2 μM) and may help study type 2 diabetes.</p>Formula:C26H19N3O4SColore e forma:SolidPeso molecolare:469.51Antibacterial agent 69
<p>Antibacterial agent 69 is a novel structural antimicrobial modulator that can be used against lethal multidrug-resistant bacterial infections (MIC: 2.978 μM).</p>Formula:C24H19N3O4SColore e forma:SolidPeso molecolare:445.49GDC-6036-NH
CAS:<p>GDC-6036-NH is a precursor of compound 17a /b, which is a RAS inhibitor that can be used in cancer research.</p>Formula:C26H30ClF4N7OPurezza:99.84%Colore e forma:SolidPeso molecolare:568.01HDAC6-IN-9
CAS:<p>HDAC6-IN-9 is a γ-secretase modulator that can significantly reduce the level of Aβ42 in mouse brain and can be used to study neurological diseases.</p>Formula:C19H16N2O3Purezza:98.84%Colore e forma:SolidPeso molecolare:320.34Amdinocillin methylacetate
CAS:<p>Amdinocillin methylacetate is a Synthetic penicillin.</p>Formula:C18H27N3O4SColore e forma:SolidPeso molecolare:381.49Antibacterial agent 80
<p>Antibacterial agent 80 (compound 20) has antibacterial activity [1].</p>Formula:C14H21N3S2Colore e forma:SolidPeso molecolare:295.47MsbA-IN-1
<p>MsbA-IN-1: Potent MsbA inhibitor (IC50: 4 nM), anti-E. coli (MIC: 79 μM), penetrates Gram-negative bacteria.</p>Formula:C23H18Cl2FNO3Colore e forma:SolidPeso molecolare:446.3Antimalarial agent 9
<p>Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.</p>Formula:C28H32BrN3O2Colore e forma:SolidPeso molecolare:522.48DIDS
CAS:<p>DIDS inhibits anion exchangers reversibly then irreversibly and blocks RAD51.</p>Formula:C16H10N2O6S4Purezza:98%Colore e forma:SolidPeso molecolare:454.52AD013
<p>AD013 is a selective ACE inhibitor and NEP inhibitor with potential anti-hypertensive and cardioprotective benefits.</p>Formula:C24H28N2O5Colore e forma:SolidPeso molecolare:424.49CXCR7 antagonist-1 hydrochloride
CAS:<p>CXCR7 antagonist-1 hydrochloride blocks SDF-1 and I-TAC from CXCR7; may prevent cancer and inflammation.</p>Formula:C21H20ClFN6OColore e forma:SolidPeso molecolare:426.87AL 6598
CAS:<p>AL 6598, a prodrug of PGD2 agonist AL 6556, reduces IOP by 53% at 1μg twice daily in monkeys; binds DP receptors with Ki of 3.2μM.</p>Formula:C23H39ClO5Colore e forma:SolidPeso molecolare:431.01VEGFR-2-IN-15
<p>VEGFR-2-IN-15 (Compound 14b) is a potent inhibitor of VEGFR-2. VEGFR-2-IN-15 inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.</p>Formula:C23H18ClN3O4SColore e forma:SolidPeso molecolare:467.92PDHK-IN-4
<p>PDHK-IN-4 inhibits PDHK2 (IC50: 0.0051 μM) & PDHK4 (IC50: 0.0122 μM), with potential for cancer research.</p>Formula:C24H25N5O3Colore e forma:SolidPeso molecolare:431.49AGN-204396
CAS:<p>AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).</p>Formula:C32H44FN3O4Colore e forma:SolidPeso molecolare:553.71Tubulin inhibitor 19
<p>Tubulin inhibitor 19 (9b), a potent indole chalcone, strongly blocks tubulin, valuable in cancer studies.</p>Formula:C21H23NO5Colore e forma:SolidPeso molecolare:369.41LasR-IN-3
<p>LasR-IN-3 inhibits LasR in Pseudomonas, disrupting its dimer, causing loss of function.</p>Formula:C22H19N3O2Colore e forma:SolidPeso molecolare:357.41Homopteroic Acid
CAS:<p>Homopteroic Acid, a precursor to Homofolic Acid, inhibits L1210 mouse leukemia growth by targeting folate uptake.</p>Formula:C15H14N6O3Colore e forma:SolidPeso molecolare:326.31LRRK2-IN-3
CAS:<p>LRRK2-IN-3: potent, selective oral LRRK2 blocker, BBB-penetrant, IC50 of 0.6 nM in hPBMCs, for Parkinson's research.</p>Formula:C25H29ClF2N6O2Colore e forma:SolidPeso molecolare:518.99PF-9404C
CAS:<p>PF-9404C: S-S diastereoisomer, beta-blocker with vasodilation, boosts cyclic GMP in rat aorta cells from 3 to 53 pmol/mg protein.</p>Formula:C16H25N3O9Purezza:98%Colore e forma:SolidPeso molecolare:403.38Antimalarial agent 7
<p>Antimalarial agent 7 is a potent and effective inhibitor of PfATP4. Antimalarial agent 7 has potential for the study of the human plasmodium falciparum.</p>Formula:C23H22F2N4O3Colore e forma:SolidPeso molecolare:440.44Nikkomycin Z
CAS:<p>Nikkomycin Z (Nikkomycin Z from Streptomyces tendae) is a competitive chitin synthase inhibitor.It inhibitor of the growth of filamentous fungi, insects,</p>Formula:C20H25N5O10Purezza:98%Colore e forma:SolidPeso molecolare:495.44FT3967385
<p>FT3967385: New USP30 inhibitor boosts mitochondrial ubiquitylation via PINK1-PARKIN.</p>Formula:C21H19N5O2Colore e forma:SolidPeso molecolare:373.41KNT-127
CAS:<p>KNT-127 is an agonist of δ-Opioid receptor.</p>Formula:C24H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:372.46CRM1 degrader 1
<p>CRM1 degrader 1 (1l) is a low-toxic CRM1 degrader that induces apoptosis in gastric carcinoma and selectively inhibits the proliferation of gastric cancer[1].</p>Formula:C16H20O3Colore e forma:SolidPeso molecolare:260.33CXCR4 probe 1
CAS:<p>CXCR4 probe 1, a specific PET tracer, targets CXCR4 with antagonist TN14003 (IC50: 6.9 nM), aiding in imaging CXCR4-related diseases and tumors.</p>Formula:C24H30FN5O4SColore e forma:SolidPeso molecolare:502.59CDK7-IN-17
CAS:<p>CDK7-IN-17, a pyrimidine-based CDK7 inhibitor, shows promise for various cancers, especially with abnormal transcription.</p>Formula:C24H26F3N6OPColore e forma:SolidPeso molecolare:502.47AKT-IN-10
CAS:<p>AKT-IN-10, a potent AKT inhibitor, has potential for breast and prostate cancer research, impacting cell growth and survival pathways.</p>Formula:C26H34ClN5O2Colore e forma:SolidPeso molecolare:484.03KUS121
CAS:<p>KUS121: VCP ATPase activity inhibitor (IC50=330 nM), protects cells from ER stress, assists in cerebral ischemia, and preserves vision in retinitis pigmentosa.</p>Formula:C22H17FN4NaO3SColore e forma:SolidPeso molecolare:459.45CDK8-IN-5
CAS:<p>CDK8-IN-5: potent CDK8 inhibitor, IC50=72 nM, boosts IL-10 by 43%, may aid inflammatory bowel disease research.</p>Formula:C26H22N2O4Colore e forma:SolidPeso molecolare:426.46OM-153
CAS:<p>OM-153 blocks tankyrase 1 (IC50: 13 nM) and 2 (IC50: 2 nM), stifling WNT signaling and COLO 320DM cell growth.</p>Formula:C28H24FN7O2Colore e forma:SolidPeso molecolare:509.53Antibiotic LL Z1640-2
CAS:<p>Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.</p>Formula:C19H22O7Colore e forma:SolidPeso molecolare:362.38A 70450
CAS:<p>A 70450, an inhibitor of aspartyl proteinase, can be used as an antifungal agent and may have a role in HIV protease inhibition therapy.</p>Formula:C42H71ClN6O5Purezza:98%Colore e forma:SolidPeso molecolare:775.50L-Afegostat
CAS:<p>L-Afegostat (5-epi-Isofagomine), an iminosugar, inhibits glycosidase and β-Glucosidase (K i 30 μM), aids in carbohydrate synthesis.</p>Formula:C6H13NO3Colore e forma:SolidPeso molecolare:147.17BACE1-IN-2
CAS:<p>BACE1-IN-2 is a BACE1 inhibitor (IC50: 22 nM).</p>Formula:C19H15F4N5O2Purezza:98%Colore e forma:SolidPeso molecolare:421.35
