Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.519 prodotti)
- Apoptosi(5.787 prodotti)
- Ciclo cellulare/Checkpoint(4.446 prodotti)
- Cromatina/Epigenetica(2.235 prodotti)
- Segnalazione citoscheletrica(1.381 prodotti)
- Danno al DNA/Riparazione del DNA(2.824 prodotti)
- Endocrinologia/Ormoni(3.500 prodotti)
- Enzima(3.639 prodotti)
- Proteina G/GPCR(8.318 prodotti)
- Immunologia e infiammazione(3.516 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.200 prodotti)
- Trasportatore di membrana/canale ionico(2.787 prodotti)
- Metabolismo(9.416 prodotti)
- Microbiologia/Virologia(6.968 prodotti)
- Neuroscienza(9.920 prodotti)
- Altri inibitori(37.928 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.596 prodotti)
- Cellule staminali e Derivati(831 prodotti)
- Adattatori Tirosin-chinasi(2.015 prodotti)
- Ubiquitinazione(1.649 prodotti)
Mostrare 16 più sottocategorie
Trovati 66627 prodotti di "Inibitori"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
CLR01 sodium
CAS:<p>CLR01 is a tweezer reducing α-synuclein in MSA, inhibits SOD1 in ALS, blocks Ebola/Zika, stabilizes proteins, and lessens mutant p53 toxicity.</p>Formula:C42H30Na2O8P2Colore e forma:SolidPeso molecolare:770.6211AS2575959
CAS:<p>AS2575959 is a novel GPR40 agonist, exhibiting glucose metabolism improvement and synergistic effect with sitagliptin on insulin and incretin secretion.</p>Formula:C32H35NaO7Colore e forma:SolidPeso molecolare:554.6148Teoprolol
CAS:<p>Teoprolol is a blocker of β-adrenergic receptor.</p>Formula:C23H30N6O4Purezza:98%Colore e forma:SolidPeso molecolare:454.52Myxothiazol
CAS:<p>Myxothiazol blocks mitochondrial complex III and triggers SESN2, a gene important for stress response.</p>Formula:C25H33N3O3S2Colore e forma:SolidPeso molecolare:487.68Thielavin B
CAS:<p>Thielavin B, from Thielavia terricola, inhibits prostaglandin E2 synthesis and reduces rat oedema.</p>Formula:C31H34O10Colore e forma:SolidPeso molecolare:566.6Antimalarial agent 9
<p>Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.</p>Formula:C28H32BrN3O2Colore e forma:SolidPeso molecolare:522.48MAO-B-IN-10
<p>MAO-B-IN-10: Potent, selective MAO-B inhibitor; crosses blood-brain barrier; IC50 5.3 μM; reduces Aβ aggregation 58.2%, disaggregates 43.3%.</p>Formula:C23H26N2O4Colore e forma:SolidPeso molecolare:394.46ent-8-iso-15(S)-Prostaglandin F2α
CAS:<p>Isoprostanes are produced by the non-enzymatic, free radical peroxidation of phospholipid-esterified arachidonic acid.</p>Formula:C20H34O5Colore e forma:SolidPeso molecolare:354.48TP-030-1
CAS:<p>TP-030-1, RIPK1 inhibitor: K(i) hRIPK1 at 3.9nM, IC50 mRIPK1 at 4.2μM; targets inflammation, neurodegeneration research.</p>Formula:C23H22N4O3Colore e forma:SolidPeso molecolare:402.45Cathepsin C-IN-3
<p>Cathepsin C-IN-3 is a potent inhibitor of histone C (IC50: 61.79 nM) and also inhibits THP-1 cells (IC50: 101.5 nM) and U937 cells (IC50: 86.5 nM).</p>Formula:C28H21F3N6OSColore e forma:SolidPeso molecolare:546.57Enpp-1-IN-11
<p>Enpp-1-IN-11 inhibits ENPP1 with a 45 nM Ki, is plasma stable, and has low clearance in human/mouse livers, potentially aiding cancer research.</p>Formula:C15H15N5O3SColore e forma:SolidPeso molecolare:345.38MA242
CAS:<p>MA242 is a nuclear factor of activated T cells 1 (NFAT1) for Pancreatic Cancer Therapy and dual inhibitor of murine double minute 2 (MDM2).</p>Formula:C26H21ClF3N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:579.98NS2B/NS3-IN-5
<p>Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.</p>Formula:C14H9IN2O3SColore e forma:SolidPeso molecolare:412.2Osanetant HCl
CAS:<p>Osanetant HCl is the (R)-enantiomer; neurokinin-3 receptor antagonist</p>Formula:C35H42Cl3N3O2Colore e forma:SolidPeso molecolare:643.09AL-6556
CAS:<p>AL-6556 is a prostaglandin DP receptor agonist.</p>Formula:C20H33ClO5Colore e forma:SolidPeso molecolare:388.93Z-FY-CHO
CAS:<p>Pyridoxal (Pyridoxaldehyde), a component of vitamin B6, is an aldehyde obtained by oxidizing pyridoxine and is widely found in plants and animals.</p>Formula:C26H26N2O5Purezza:95.88%Colore e forma:SolidPeso molecolare:446.5FT3967385
<p>FT3967385: New USP30 inhibitor boosts mitochondrial ubiquitylation via PINK1-PARKIN.</p>Formula:C21H19N5O2Colore e forma:SolidPeso molecolare:373.41Nenocorilant
CAS:<p>Nenocorilant (Relacorilant) is an orally active glucocorticoid receptor (GR) antagonist (Ki: 0.15 nM). Nenocorilant can be used to study tumours.</p>Formula:C26H21F4N7O3SColore e forma:SolidPeso molecolare:587.55hCA IX-IN-1
<p>hCA IX-IN-1 inhibits human carbonic anhydrases I, II, IX, and XII with Ki values of 331.4, 28.4, 9.4, 17.8 nM and exhibits anticancer properties.</p>Formula:C19H18N2O3SColore e forma:SolidPeso molecolare:354.42Bafilomycin C1
CAS:<p>vacuolar H+-ATPases (V-ATPases) inhibitor</p>Formula:C39H60O12Purezza:98%Colore e forma:Light Tan SolidPeso molecolare:720.89L-Afegostat
CAS:<p>L-Afegostat (5-epi-Isofagomine), an iminosugar, inhibits glycosidase and β-Glucosidase (K i 30 μM), aids in carbohydrate synthesis.</p>Formula:C6H13NO3Colore e forma:SolidPeso molecolare:147.17S-1033
CAS:<p>S-1033 is an FP receptor agonist.</p>Formula:C20H33NaO4Colore e forma:SolidPeso molecolare:360.4698ABL-001-Amide-PEG3-acid
ABL-001-Amide-PEG3-acid, an analogue to ABL-001, primarily serves as a labeled chemical or fluorescent probe.Formula:C29H33ClF2N6O9Purezza:98%Colore e forma:SolidPeso molecolare:683.06CRM1 degrader 1
<p>CRM1 degrader 1 (1l) is a low-toxic CRM1 degrader that induces apoptosis in gastric carcinoma and selectively inhibits the proliferation of gastric cancer[1].</p>Formula:C16H20O3Colore e forma:SolidPeso molecolare:260.33MSX-3 free acid
CAS:<p>MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.</p>Formula:C21H23N4O7PColore e forma:SolidPeso molecolare:474.40Thioquinapiperifil dihydrochloride
CAS:<p>Thioquinapiperifil dihydrochloride is a potent, selective PDE-5 inhibitor (IC50: 0.074 nM) for research.</p>Formula:C24H29ClN6OSPurezza:98.73%Colore e forma:SolidPeso molecolare:485.05CaMKIIα-IN-1
<p>CaMKIIα-IN-1 (Compound 4d) is an orally active inhibitor of Ca 2+ /calmodulin-dependent protein kinase II α (CaMKIIα) with a Kd of 219 nM for CaMKIIα WT hub.</p>Formula:C14H11ClO4Colore e forma:SolidPeso molecolare:278.69MMSET-IN-1
CAS:<p>MMSET-IN-1 is an inhibitor of multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) .</p>Formula:C18H29N7O5Purezza:98%Colore e forma:SolidPeso molecolare:423.47TAK-637
CAS:<p>TAK-637 is a tachykinin 1 (NK1) receptor antagonist.</p>Formula:C30H25F6N3O2Purezza:98%Colore e forma:SolidPeso molecolare:573.53Milademetan
CAS:<p>Milademetan (DS-3032), an MDM2 inhibitor, exhibits antitumor activity, induces G1 cell cycle arrest and apoptosis, and can be used to study solid tumors.</p>Formula:C30H34Cl2FN5O4Purezza:>99.99%Colore e forma:SolidPeso molecolare:618.53Enbezotinib
CAS:<p>Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.</p>Formula:C21H21FN6O3Purezza:99.84%Colore e forma:SolidPeso molecolare:424.43BMS-986141
CAS:<p>BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614</p>Formula:C27H23N5O5S2Purezza:98.43% - 99.26%Colore e forma:SolidPeso molecolare:561.63AChE-IN-26
CAS:<p>AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).</p>Formula:C21H21BrN2O3Purezza:99.24% - 99.85%Colore e forma:SoildPeso molecolare:429.31Zelasudil
CAS:<p>Zelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.</p>Formula:C22H21F2N7OPurezza:99.15%Colore e forma:SolidPeso molecolare:437.445SB-423562
CAS:<p>SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.</p>Formula:C26H32N2O4Purezza:99.22%Colore e forma:SolidPeso molecolare:436.54Etamicastat hydrochloride
CAS:<p>Etamicastat hydrochloride (BIA 5-453 hydrochloride) is a peripherally selective dopamine beta-hydroxylase inhibitor that reduces hypertension.</p>Formula:C14H16ClF2N3OSPurezza:98.54%Colore e forma:SolidPeso molecolare:347.81AZD 3147
CAS:<p>AZD 3147 inhibits mTORC1 (40.7 nM), mTORC2 (5.75 nM), and PI3Kα/β/δ/γ (912/5495/9333/6310 nM IC50s).</p>Formula:C24H31N5O4S2Purezza:99.99%Colore e forma:SolidPeso molecolare:517.66Aleglitazar
CAS:<p>Aleglitazar (R1439) (R1439) is a potent dual PPARα/γ agonist, with IC50s of 38 nM and 19 nM for human PPARa and PPARγ, respectively.</p>Formula:C24H23NO5SPurezza:99.03%Colore e forma:SolidPeso molecolare:437.51Tuvusertib
CAS:<p>Tuvusertib (M1774), an oral ATR inhibitor (Ki<1µM), selectively blocks CHK1 phosphorylation, disrupts DNA repair, and induces tumor cell apoptosis.</p>Formula:C16H12F2N8OPurezza:98.44% - 99.66%Colore e forma:SolidPeso molecolare:370.32JNJ-6204
CAS:<p>JNJ-6204 is a deuterated compound that efficiently inhibits CSNK1D and CSNK1E.</p>Formula:C19H11D6FN6OPurezza:97.42% - 99.87%Colore e forma:SolidPeso molecolare:370.41CCF0058981
CAS:<p>CCF0058981: noncovalent inhibitor for SARS-CoV-2 & -1 proteases; IC50s: 68 nM (SC2) & 19 nM (SC1). Potential COVID-19 research use.</p>Formula:C24H19ClN6OPurezza:98.94%Colore e forma:SoildPeso molecolare:442.9FABPs ligand 6
CAS:<p>FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.</p>Formula:C28H27FN2O3Purezza:97.45%Colore e forma:SolidPeso molecolare:458.52NRX-103095
CAS:<p>NRX-103095 increases β-catenin binding to SCFβ-TrCP E3 ligase; EC50 is 163 nM for pSer33/Ser37 affinity boost.</p>Formula:C22H16Cl2F3N3O3SPurezza:99.58% - 99.95%Colore e forma:SolidPeso molecolare:530.35IDX184
CAS:<p>IDX184 is a potent, orally active, targeted HCV polymerase inhibitor and nucleoside polymerase.IDX184 effectively inhibits HCV polymerase (IC50=0.31 μM, Ki=52.3</p>Formula:C25H35N6O9PSPurezza:97.15%Colore e forma:SolidPeso molecolare:626.62Cbl-b-IN-3
CAS:<p>Cbl-b-IN-3 is a potent inhibitor of casitas b lineage lymphoma proto-oncogene-b (Cbl-b) (ic50 < 1 nM).Cost-effective and quality-assured.</p>Formula:C30H34F3N5OPurezza:99%Colore e forma:SolidPeso molecolare:537.62USP5-IN-1
<p>USP5-IN-1, a powerful USP5 deubiquitinase inhibitor, selectively binds with 2.8 μM affinity, blocking USP5's di-ubiquitin cleavage.</p>Formula:C19H20ClN3O5SPurezza:99.76%Colore e forma:SoildPeso molecolare:437.9SJ6986
CAS:<p>SJ6986 is a potent, selective and orally active GSPT1/2 degrader. SJ6986 degrades GSPT1 with a DC 50 of 2.1 nM (D max 99%) [1].</p>Formula:C20H14F3N3O7SPurezza:99.73%Colore e forma:SolidPeso molecolare:497.4MAO-B-IN-17
CAS:<p>MAO-B-IN-17 is a selective and potent monoamine oxidase B (MAO-B) inhibitor (IC50: 5.08 μM) for the study of central nervous system disorders like Parkinson's.</p>Formula:C17H17F2NO2Purezza:99.41%Colore e forma:SoildPeso molecolare:305.32USP15-IN-1
CAS:<p>USP15-IN-1 is a potent USP15 inhibitor (IC50 is 3.76 μM).</p>Formula:C22H23N3O3Purezza:99.509% - 99.81%Colore e forma:SolidPeso molecolare:377.44NRX-1532
<p>NRX-1532 is a small molecule β-catenin:β-TrCP interaction enhancer.</p>Formula:C16H11F3N4O2Purezza:98.95% - 99.68%Colore e forma:SolidPeso molecolare:348.28L-371,257
CAS:<p>L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.</p>Formula:C28H33N3O6Purezza:99.79%Colore e forma:SolidPeso molecolare:507.58NRX-103094
CAS:<p>NRX-103094 boosts β-catenin binding to SCFβ-TrCP ligase with EC50 62 nM and Kd 0.6 nM.</p>Formula:C20H11Cl2F3N2O4SPurezza:99.13%Colore e forma:SolidPeso molecolare:503.28HRO761
CAS:<p>HRO761 is a potent Werne r syndrome RecQ DNA deconjugase (WRN) inhibitor that can be used to study cancers such as colon and stomach cancer.</p>Formula:C31H31ClF3N9O5Purezza:98.74% - 99.62%Colore e forma:SolidPeso molecolare:702.08SY-5609
CAS:<p>SY-5609 (CDK7-IN-3) is a selective non-covalent CDK7 inhibitor, with weak inhibitory activity against CDK2, CDK9 and CDK12.Cost-effective and quality-assured.</p>Formula:C23H26F3N6OPPurezza:99.34% - >99.99%Colore e forma:SolidPeso molecolare:490.46AZD5462
CAS:<p>AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.</p>Formula:C30H41FN2O6Purezza:98.32% - 99.63%Colore e forma:SolidPeso molecolare:544.65DN02
<p>DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).</p>Formula:C22H24FN3O3Purezza:98.22% - 99.74%Colore e forma:SolidPeso molecolare:397.44PF-07258669
CAS:<p>PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.</p>Formula:C25H27FN6O2Purezza:99.9%Colore e forma:SolidPeso molecolare:462.52AZ12601011
CAS:<p>AZ12601011 is a TGFBR1 kinase inhibitor that inhibits the growth of breast tumors.</p>Formula:C19H15N5Purezza:98.81%Colore e forma:SolidPeso molecolare:313.36WAY-213613 hydrochloride
CAS:<p>WAY-213613 hydrochloride: potent, selective GLT-1/EAAT2 inhibitor (IC50 85 nM); weaker for EAAT1/3; inactive at glutamate receptors; research tool for CNS.</p>Formula:C16H13BrF2N2O4Purezza:99.14% - 99.37%Colore e forma:SoildPeso molecolare:415.19Odevixibat
CAS:<p>Odevixibat (A4250) is a selective oral inhibitor for ileal bile acid transport, potentially treating primary biliary cirrhosis.</p>Formula:C37H48N4O8S2Purezza:99.53% - 99.83%Colore e forma:SolidPeso molecolare:740.93LSN3318839
CAS:<p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>Formula:C26H23Cl2N3O2Purezza:99.21%Colore e forma:SolidPeso molecolare:480.39Lometrexol
CAS:<p>Lometrexol (LY 264618) is an antifolate that inhibits GARFT, blocks purine synthesis, induces apoptosis, and has anticancer properties.</p>Formula:C21H25N5O6Purezza:97.76% - 99.56%Colore e forma:SolidPeso molecolare:443.45Elacytarabine
CAS:<p>Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.</p>Formula:C27H45N3O6Purezza:97.69%Colore e forma:SolidPeso molecolare:507.66Suzetrigine
CAS:<p>Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.</p>Formula:C21H20F5N3O4Purezza:98.08% - 99.27%Colore e forma:SolidPeso molecolare:473.39VX-984
CAS:<p>VX-984 (M9831) is an oral DNA-PK inhibitor, crossing the blood-brain barrier, targeting GBM and NSC-LC.</p>Formula:C23H21D2N7OPurezza:97.65% - 99.98%Colore e forma:SolidPeso molecolare:415.49DRF-1042
CAS:<p>DRF-1042 is a camptothecin analog with anticancer and insecticidal activity and is used to study solid tumors such as prostate and colon cancer.</p>Formula:C22H20N2O6Purezza:98.34%Colore e forma:SolidPeso molecolare:408.4Gepotidacin mesylate dihydrate
CAS:<p>Gepotidacin mesylate dihydrate (GSK2140944 mesylate dihydrate) is an antibiotic and an inhibitor of bacterial type II topoisomerase.</p>Formula:C25H36N6O8SPurezza:99.85%Colore e forma:SolidPeso molecolare:580.65KU-60019
CAS:<p>KU-60019 is a specific inhibitor of ATM kinase (IC50: 6.3 nM).</p>Formula:C30H33N3O5SPurezza:98.05% - 98.50%Colore e forma:SolidPeso molecolare:547.67BMS453
CAS:<p>BMS453 (BMS-189453), a synthetic retinoid, is a potent and selective agonist of RARβ and a potent testicular toxin.</p>Formula:C27H24O2Purezza:99.93%Colore e forma:SolidPeso molecolare:380.48Obicetrapib
CAS:<p>Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein.</p>Formula:C32H31F9N4O5Purezza:99.26% - >99.99%Colore e forma:SolidPeso molecolare:722.6Rupintrivir
CAS:<p>Rupintrivirvr (AG7088) is a mimetic peptide inhibitor of rhinovirus (HRV) 3C cysteine protease with antiviral activity for the study of viral infections.</p>Formula:C31H39FN4O7Purezza:97.72% - 99.35%Colore e forma:SolidPeso molecolare:598.66ZD 7155 hydrochloride
CAS:<p>ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.</p>Formula:C26H27ClN6OPurezza:99.8%Colore e forma:SolidPeso molecolare:474.98CP-642931
CAS:<p>CP-642931 (Sorbitol dehydrogenase-IN-1) is a sorbitol dehydrogenase inhibitor used in the study of diabetes mellitus and cardiovascular disease.</p>Formula:C17H25N7OPurezza:99.67% - >99.99%Colore e forma:SolidPeso molecolare:343.43D75-4590
CAS:<p>D75-4590, a β-1,6-Glucan synthetase inhibitor, combats fungal infections by targeting cell walls.</p>Formula:C21H27N5Purezza:98.56% - 98.85%Colore e forma:SolidPeso molecolare:349.47Dual FAAH/sEH-IN-1
CAS:<p>Dual FAAH/sEH-IN-1 inhibits both sEH (IC50: 9.6 nM) and FAAH (IC50: 7 nM), offering potent anti-inflammatory effects.</p>Formula:C25H22ClN3O3S2Purezza:99.89%Colore e forma:SolidPeso molecolare:512.04AKT Kinase Inhibitor
CAS:<p>AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.Cost-effective and quality-assured.</p>Formula:C16H19N7O3Purezza:97.83% - 99.13%Colore e forma:SolidPeso molecolare:357.37NB-360
CAS:<p>NB-360: potent, brain-penetrant BACE1/2 inhibitor; IC50s: 5-6 nM; high selectivity vs pepsin, cathepsin E/D.</p>Formula:C21H19F4N5O2Purezza:99.72%Colore e forma:SolidPeso molecolare:449.4Cort108297
CAS:<p>Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.</p>Formula:C26H25F4N3O3SPurezza:98.36% - 99.94%Colore e forma:SolidPeso molecolare:535.55AChE/BChE-IN-10
CAS:<p>AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.</p>Formula:C26H30N2O2Purezza:99.55% - 99.88%Colore e forma:SoildPeso molecolare:402.53Aldometanib
CAS:<p>Aldometanib (LXY-05-029) is an oral aldolase inhibitor that maintains metabolic balance by blocking FBP and activating lysosomal AMPK.</p>Formula:C27H43Cl2IN2Purezza:99.32% - 99.55%Colore e forma:SolidPeso molecolare:593.46Umibecestat
CAS:<p>Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM & 10 nM), potentially for Alzheimer's research.</p>Formula:C19H15ClF7N5O2Purezza:99.88%Colore e forma:SolidPeso molecolare:513.8LLY-283
CAS:<p>LLY-283, PRMT5 inhibitor, IC50 22 nM, Kd 6 nM, oral, selective, with antitumor effects.</p>Formula:C17H18N4O4Purezza:99.49%Colore e forma:SolidPeso molecolare:342.35Simmitecan hydrochloride
CAS:<p>Simmitecan hydrochloride is a camptothecin derivative, a topoisomerase I inhibitor with anticancer activity, which can be used to study is solid tumors.</p>Formula:C34H39ClN4O6Purezza:98.20% - 98.93%Colore e forma:SolidPeso molecolare:635.15ALOX15-IN-2
CAS:<p>ALOX15-IN-2: Potent ALOX15 inhibitor. IC50: 1.55 μM for LA; 2.79 μM for AA. Stops linoleic/arachidonic acid oxidation.</p>Formula:C23H29N3O4SPurezza:98.10%Colore e forma:SolidPeso molecolare:443.56SYM2206
CAS:<p>SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated</p>Formula:C20H22N4O3Purezza:99.88%Colore e forma:SolidPeso molecolare:366.41BDZ-g
CAS:<p>BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.</p>Formula:C21H21N5O2SPurezza:99.97%Colore e forma:SolidPeso molecolare:407.49Vofopitant dihydrochloride
CAS:<p>Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.</p>Formula:C21H25Cl2F3N6OPurezza:98.99%Colore e forma:SolidPeso molecolare:505.36Treprostinil diethanolamine
CAS:<p>Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,</p>Formula:C27H45NO7Purezza:99.86%Colore e forma:SolidPeso molecolare:495.65Vecabrutinib
CAS:<p>Vecabrutinib (SNS-062) is a potent and noncovalent BTK and ITK inhibitor (Kd: 0.3 nM and 2.2 nM, respectively). Vecabrutinib displays an IC50 of 24 nM for ITK.</p>Formula:C22H24ClF4N7O2Purezza:99.74%Colore e forma:SolidPeso molecolare:529.92O-Propargyl-Puromycin
CAS:<p>O-Propargyl-Puromycin (OP-puro) is a potent protein synthesis inhibitor, a puromycin acetylene analog.</p>Formula:C24H29N7O5Purezza:97.83% - 99.70%Colore e forma:SolidPeso molecolare:495.53NDI-034858
CAS:<p>NDI-034858 (TAK-279) is a tyrosine kinase 2 (TYK2) inhibitor (Kd<200 pM) that targets the JH2 structural domain of Tyk2 for the treatment of autoimmune diseases</p>Formula:C23H24N8O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:460.49Evixapodlin
CAS:<p>Evixapodlin (PD-1/PD-L1-IN 7) is a human PD-1/PD-L1 protein/protein interaction inhibitor (IC50: 0.213).Evixapodlin has anticancer and antiviral activities.</p>Formula:C34H36Cl2N8O4Purezza:99.07%Colore e forma:SolidPeso molecolare:691.61BMS 299897
CAS:<p>BMS 299897, a sulfonamide γ-secretase inhibitor, inhibits Aβ production with an IC50 of 7 nM in HEK293 cells overexpressing APP.</p>Formula:C24H21ClF3NO4SPurezza:99.82%Colore e forma:SolidPeso molecolare:511.94AZD-5672
CAS:<p>AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.</p>Formula:C32H38F2N2O5S2Purezza:98.1%Colore e forma:SolidPeso molecolare:632.78BQ-788
CAS:<p>BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.</p>Formula:C34H51N5O7Purezza:98.81%Colore e forma:SolidPeso molecolare:641.8BODIPY FL prazosin
CAS:<p>BODIPY FL prazosin is an α1-adrenergic antagonist that inhibits α1a-AR and α1b-AR.</p>Formula:C28H32BF2N7O3Purezza:97.27%Colore e forma:SolidPeso molecolare:563.41Glycosyltransferase-IN-1
<p>Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.</p>Formula:C19H21N5OPurezza:99.76%Colore e forma:SolidPeso molecolare:335.4Dazostinag disodium
CAS:<p>Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.</p>Formula:C21H20F2N8Na2O10P2S2Purezza:98.84% - 99.96%Colore e forma:SolidPeso molecolare:754.48STK-15
CAS:<p>STK-15 is a candidate for use as a fatty acid binding protein 5 (FABP5) inhibitor.</p>Formula:C34H29NO5Purezza:98.05%Colore e forma:SolidPeso molecolare:531.6Eravacycline dihydrochloride
CAS:<p>Eravacycline dihydrochloride (TP-434-046) is a potent and broad-spectrum antibacterial agent against six E. coli (MICs: 0.125-0.25 mg/L).</p>Formula:C27H33Cl2FN4O8Purezza:94.59% - 95%Colore e forma:SolidPeso molecolare:631.48KI696
CAS:<p>KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.</p>Formula:C28H30N4O6SPurezza:99.74%Colore e forma:SolidPeso molecolare:550.63Tigemonam
CAS:<p>Tigemonam is a monobactam, a novel orally administered monobactam that protects against gram-negative aerobic bacterial pathogens. Cost-effective and quality-assured.</p>Formula:C12H15N5O9S2Purezza:99.03% - >99.99%Colore e forma:SolidPeso molecolare:437.41Cap-dependent endonuclease-IN-1
CAS:<p>Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.</p>Formula:C27H22F2N2O6SPurezza:98.88% - 99.09%Colore e forma:SolidPeso molecolare:540.54Moiramide B
CAS:<p>Moiramide B is an acetyl coenzyme A carboxylase inhibitor with antimicrobial activity, strongly inhibiting Gram-positive bacteria.</p>Formula:C25H31N3O5Purezza:98.53% - 99.90%Colore e forma:SolidPeso molecolare:453.53AM103
CAS:<p>AM103 is an effective and selective inhibitor of FLAP (IC50 = 4.2 nM).</p>Formula:C36H38N3NaO4SPurezza:99.75%Colore e forma:SolidPeso molecolare:631.76Pocenbrodib
CAS:<p>Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP/p300 family with potential antitumour activity and is palatable for cancer research.</p>Formula:C28H32FN3O6Purezza:98.48% - 99.54%Colore e forma:SolidPeso molecolare:525.57SDZ 220-040
CAS:<p>SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂，可诱导根系生长的部分无重力模式 。</p>Formula:C16H16Cl2NO6PPurezza:98.13%Colore e forma:SolidPeso molecolare:420.18Picrotoxinin
CAS:<p>Picrotoxinin blocks chloride channels, antagonizes GABAA noncompetitively (IC50: 1.15 μM, α1β2γ2L), and induces convulsions.</p>Formula:C15H16O6Purezza:98.07%Colore e forma:SolidPeso molecolare:292.28LY2979165
CAS:<p>LY2979165 (mGlu2 agonist) is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.</p>Formula:C13H22N6O6SPurezza:98.41%Colore e forma:SolidPeso molecolare:390.42BLU2864
CAS:<p>BLU2864: oral PRKACA inhibitor, IC50=0.3 nM, potential in cancer/poly. kidney disease research.</p>Formula:C24H19F3N4O2Purezza:97.58% - 99.92%Colore e forma:SoildPeso molecolare:452.43MIV-247
CAS:<p>MIV-247 is a cathepsin S inhibitor that attenuates mechanically abnormal pain in preclinical neuropathic pain models and can be used to study myocardial injury.</p>Formula:C17H24F3N3O4Purezza:99.27%Colore e forma:SolidPeso molecolare:391.39Iclepertin
CAS:<p>Iclepertin (BI-425809) is a GlyT1 inhibitor.Iclepertin is used for the treatment of Alzheimer;s disease and other CNS disorders.</p>Formula:C20H18F6N2O5SPurezza:98.89% - 98.93%Colore e forma:SolidPeso molecolare:512.42EZM0414
CAS:<p>EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM in SETD2 biochemical assay and IC50 of 34 nM in a cellular assay.</p>Formula:C22H29FN4O2Purezza:99.58%Colore e forma:SolidPeso molecolare:400.49Darizmetinib
CAS:<p>Darizmetinib (HRX215) is an MKK4 inhibitor.</p>Formula:C21H17F2N5O3SPurezza:98.03% - 99.57%Colore e forma:SolidPeso molecolare:457.45JTK-109
CAS:<p>JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.</p>Formula:C37H33ClFN3O4Purezza:98.48% - 99.68%Colore e forma:SolidPeso molecolare:638.13Emprumapimod
CAS:<p>Emprumapimod, an oral p38α MAPK inhibitor, targets RPMI-8226 cells, curbs LPS-induced IL-6; IC50: 100 pM; for cardiomyopathy, acute pain.</p>Formula:C24H29F2N5O3Purezza:99.21% - >99.99%Colore e forma:SolidPeso molecolare:473.52BAY-3827
CAS:<p>BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.</p>Formula:C27H25FN6OPurezza:99.90%Colore e forma:SolidPeso molecolare:468.53Dersimelagon
CAS:<p>Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.</p>Formula:C36H45F4N3O5Purezza:97.35% - 98.23%Colore e forma:SolidPeso molecolare:675.75Vofopitant
CAS:<p>Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).</p>Formula:C21H23F3N6OPurezza:97.86%Colore e forma:SolidPeso molecolare:432.44PREP inhibitor-1
CAS:<p>PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.</p>Formula:C22H28N4O2Purezza:98.78%Colore e forma:SoildPeso molecolare:380.48GLPG0974
CAS:<p>GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.</p>Formula:C25H25ClN2O4SPurezza:99.8%Colore e forma:SolidPeso molecolare:484.99GSK3368715 dihydrochloride
CAS:<p>GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study of advanced solid tumors.</p>Formula:C20H40Cl2N4O2Purezza:99.66% - 99.66%Colore e forma:SolidPeso molecolare:439.46ELOVL1-IN-2
CAS:<p>ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).</p>Formula:C18H15FN2OPurezza:99.84%Colore e forma:SolidPeso molecolare:294.32BE1218
CAS:<p>BE1218 is a liver X receptor (LXR) inverse agonist active on LXRα and LXRβ with an IC50 of 9 nM and 7 nM, respectively.</p>Formula:C30H30FNO4S2Purezza:99.7%Colore e forma:SoildPeso molecolare:551.69INCB054329
CAS:<p>INCB054329 is a BET inhibitor targeting BRD2/3/4 and BRDT with IC50s ranging from 1-119 nM.</p>Formula:C19H16N4O3Purezza:99.52%Colore e forma:SolidPeso molecolare:348.36BCL6-IN-3
CAS:<p>BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.</p>Formula:C24H31ClF2N6O2Purezza:98.17%Colore e forma:SolidPeso molecolare:508.99(+)-Tetrabenazine
CAS:<p>(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold</p>Formula:C19H27NO3Purezza:98.31%Colore e forma:SolidPeso molecolare:317.42NRX-252114
CAS:<p>NRX-252114 promotes mutant β-catenin degradation, binding it to E3 ligase SCFβ-TrCP (EC50: 6.5 nM; Kd: 0.4 nM).</p>Formula:C22H12Cl2F3N3O2SPurezza:99.70%Colore e forma:SolidPeso molecolare:510.32Zotizalkib
CAS:<p>TPX-0131: potent, selective, CNS-ready, oral ALK inhibitor (WT IC50: 1.4nM, G1202R/L1196M IC50: 0.3nM) with robust antitumor effects.</p>Formula:C21H20F3N5O3Purezza:98.7%Colore e forma:SolidPeso molecolare:447.41SB-224289 hydrochloride
CAS:<p>SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.</p>Formula:C32H33ClN4O3Purezza:97.82% - 98.99%Colore e forma:SolidPeso molecolare:557.08DRB18
CAS:<p>DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.</p>Formula:C22H23ClN2O2Purezza:99.54%Colore e forma:SolidPeso molecolare:382.88HOIPIN-8 sodium
CAS:<p>HOIPIN-8 sodium is a LUBAC inhibitor for the study of inflammatory and immune diseases.</p>Formula:C23H15F2N4NaO3Purezza:97.34%Colore e forma:SolidPeso molecolare:456.38TGFβRI-IN-3
CAS:<p>TGFβRI-IN-3 inhibits TGFβR1 with an IC 50 of 0.79 nM with 2000-fold selectivity against MAP4K4.</p>Formula:C28H23N3O2SPurezza:99.85%Colore e forma:SoildPeso molecolare:465.57BAY-8400
<p>BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy in</p>Formula:C21H17F2N5OPurezza:99.53%Colore e forma:SolidPeso molecolare:393.39BRD0639
CAS:<p>BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.</p>Formula:C21H22ClN5O4SPurezza:99.85%Colore e forma:SolidPeso molecolare:475.95Rolapitant hydrochloride
CAS:<p>Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.</p>Formula:C25H27ClF6N2O2Purezza:98.35% - 99.79%Colore e forma:SolidPeso molecolare:536.94JAK2-IN-7
CAS:<p>JAK2-IN-7 selectively inhibits JAK2 (IC50: 3 nM), shows 14-fold selectivity over JAK1/3, FLT3, induces G0/G1 arrest, apoptosis, and has antitumor effects.</p>Formula:C26H33N7OPurezza:99.54%Colore e forma:SolidPeso molecolare:459.5910-Methoxycamptothecin
CAS:<p>10-Methoxycamptothecin is a natural bioactive derivative of camptothecin (CPT) isolated from Camptotheca acuminata and possesses high anti-cancer properties.</p>Formula:C21H18N2O5Purezza:98.36%Colore e forma:SolidPeso molecolare:378.38CK2 inhibitor 2
CAS:<p>CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.</p>Formula:C21H17ClN4O2Purezza:99.02%Colore e forma:SolidPeso molecolare:392.84FGI-106 tetrahydrochloride
CAS:<p>FGI-106 tetrahydrochloride demonstrates potent inhibitory activity across a broad spectrum of viruses, including those causing hemorrhagic fevers such as Ebola</p>Formula:C28H42Cl4N6Purezza:99.68%Colore e forma:SolidPeso molecolare:604.48PD 151746
CAS:<p>PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.</p>Formula:C11H8FNO2SPurezza:98.63% - ≥95%Colore e forma:SolidPeso molecolare:237.25SR 11302
CAS:<p>SR 11302 is an inhibitor of activator protein-1 (AP-1).</p>Formula:C26H32O2Purezza:98.65%Colore e forma:SolidPeso molecolare:376.53Durlobactam sodium salt
CAS:<p>Durlobactam sodium salt (ETX2514) have an IC50 values of 4, 14 and 190 nM against class A KPC-2, class C AmpC and class D OXA-24.Cost-effective and quality-assured.</p>Formula:C8H10N3NaO6SPurezza:97.01% - 99.03%Colore e forma:SolidPeso molecolare:299.23(E/Z)-GSK5182
CAS:<p>GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.</p>Formula:C27H31NO3Purezza:97.58%Colore e forma:SolidPeso molecolare:417.54Rineterkib
CAS:<p>Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.</p>Formula:C26H27BrF3N5O2Purezza:99.73%Colore e forma:SolidPeso molecolare:578.42ARN19702
CAS:<p>ARN19702: orally active, brain-penetrant, selective NAAA inhibitor, IC50 230 nM, broad analgesic profile.</p>Formula:C21H22FN3O3S2Purezza:99.86%Colore e forma:SolidPeso molecolare:447.55Sinefungin
CAS:<p>Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viral</p>Formula:C15H23N7O5Purezza:98.12%Colore e forma:SolidPeso molecolare:381.39LY3143921 hydrate
CAS:<p>LY3143921 ((S)-Example 2) hydrate is an orally active CDC7 kinase inhibitor with broad in vitro anticancer activity [1].</p>Formula:C16H14FN5O2Purezza:98.43%Colore e forma:SolidPeso molecolare:327.31Gemcitabine elaidate hydrochloride
CAS:<p>CP-4126, a lipophilic pro-drug of Gemcitabine, converts to active form by esterases, allowing oral administration with dose-dependent effects.</p>Formula:C27H44ClF2N3O5Purezza:98.50% - 99.6%Colore e forma:SolidPeso molecolare:564.11XMD-17-51 Trifluoroacetate
CAS:<p>XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that regulates protein kinases.</p>Formula:C23H25F3N8O3Purezza:99.65%Colore e forma:SolidPeso molecolare:518.49Sebetralstat
CAS:<p>Sebetralstat (KVD900) is an inhibitor of plasma kallikrein and can be used in studies about metabolic diseases.</p>Formula:C26H26FN5O4Purezza:99.85%Colore e forma:SolidPeso molecolare:491.51LSZ-102
CAS:<p>LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.</p>Formula:C25H17F3O4SPurezza:98.56%Colore e forma:SolidPeso molecolare:470.46INCB086550
CAS:<p>INCB086550 (PD-1/PD-L1-IN-8) (example 24) is a PD-1/PD-L1 inhibitor, with an IC50 <= 10 nM.</p>Formula:C41H39N7O4Purezza:98.49%Colore e forma:SolidPeso molecolare:693.79FX-11
CAS:<p>FX-11: potent LDHA inhibitor (Ki 8 μM), activates PKM2, reduces ATP, induces oxidative stress/ROS, cell death, shows antitumor effects.</p>Formula:C22H22O4Purezza:98.95%Colore e forma:SolidPeso molecolare:350.41Clorophene
CAS:<p>Clorophene (Clorofene) is an antimicrobial agent and can be used in personal care products.</p>Formula:C13H11ClOPurezza:99.87%Colore e forma:White To Light Tan Or Pink Flakes Phenolic Odor (Ntp 1992)Peso molecolare:218.68TCblR Protein, Human, Recombinant (His)
<p>TCblR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 32-58 KDa and the accession number is Q9NPF0.</p>Colore e forma:SolidPeso molecolare:32-58 KDa (reducing condition)Ref: TM-TMPJ
Prodotto fuori produzioneGAS6 Protein, Human, Recombinant (His)
<p>GAS6 (Growth arrest-specific protein 6) is also known as AXL receptor tyrosine kinase ligand, AXLLG, is a multimodular protein that is up-regulated by a wide variety of cell types in response to growth arrest. Gas6 binds and induces signaling through the receptor tyrosine kinases Axl, Dtk, and Mer whose signaling is implicated in cell growth and survival, cell adhesion and cell migration. GAS6/AXL signaling plays a role in various processes such as endothelial cell survival during acidification by preventing apoptosis, optimal cytokine signaling during human natural killer cell development, hepatic regeneration, gonadotropin-releasing hormone neuron survival and migration, platelet activation, or regulation of thrombotic responses. GAS6 Protein, Human, Recombinant (His) is expressed in HEK293 cells.</p>Purezza:＞99.90%Colore e forma:SoildPeso molecolare:72.7 KDa (Predicted), 80-90 KDa (Reducing conditions)TEM1/CD248 Protein, Mouse, Recombinant (His)
<p>TEM1/CD248 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 73.6 kDa and the accession number is Q91V98.</p>Colore e forma:SolidPeso molecolare:73.6 kDa (predicted). Due to glycosylation, the protein migrates to 75-140 kDa based on Tris-Bis PAGE result.EGFR-IN-7
CAS:<p>EGFR-IN-7 (TQB3804) is a selective and potent EGFR kinase inhibitor.</p>Formula:C32H41BrN9O2PPurezza:95.32% - 99.64%Colore e forma:SolidPeso molecolare:694.62'-Hydroxy-4'-methylacetophenone
CAS:<p>2'-Hydroxy-4'-methylacetophenone, a phenolic compound isolated from Angelicae koreana roots possesses acaricidal property. 2'-Hydroxy-4'-methylacetophenone has acaricidal activity, it could be used in the preparation of 4'-methyl-2'-[(p-tolylsulfonyl) oxy] acetophenone.</p>Formula:C9H10O2Purezza:99.88%Colore e forma:Black LiquidPeso molecolare:150.17PRGL493
CAS:<p>PRGL493 blocks ACSL4, halts PC3/MDA-MB-231 cancer cell spread, and inhibits MA-10 tumor progesterone. Effective in mouse PC3 tumor model at 0.25 mg/kg.</p>Formula:C25H21N7O2Purezza:98.80% - 99.11%Colore e forma:SolidPeso molecolare:451.48(-)-Isopulegol
CAS:<p>Isopulegol has antioxidant, and neuroactive properties. It also has gastroprotective effects induced by isopulegol appear to be mediated, at least in part, by endogenous prostaglandins, K+ATP channel opening and antioxidant proprieties related to GSH increased.</p>Formula:C10H18OPurezza:99.89%Colore e forma:LiquidPeso molecolare:154.253-Methoxyphenylacetic acid
CAS:<p>3-Methoxyphenylacetic acid belongs to the class of organic compounds known as anisoles. 3-Methoxyphenylacetic acid is slightly soluble (in water) and a weakly acidic compound (based on its pKa).3-Methoxyphenylacetic acid (m-Methoxyphenylacetic acid), a m-hydroxyphenylacetic acid (m-OHPAA) derivative, is a phytotoxin in Rhizoctonia solani. 3-Methoxyphenylacetic acid is used to develop a toxin-mediated bioassay for resistance to rhizoctonia root rot</p>Formula:C9H10O3Purezza:98.61%Colore e forma:White SolidPeso molecolare:166.17α-Terpineol
CAS:<p>Terpineol possesses antifungal activity against Trichophyton mentagrophytes, it also exhibits strong antimicrobial activity against periodontopathic and cariogenic bacteria. α-Terpineol (Terpineol) shows anticonvulsant, and anti-inflammatory activities, it inhibits the gene expression of the IL-6 receptor.</p>Formula:C10H18OPurezza:97.55%Colore e forma:Colorless LiquidPeso molecolare:154.25Ref: TM-FR14115
Prodotto fuori produzioneAnisylacetone
CAS:<p>Anisylacetone (Anisylacetone) is an effective lure for the male melon fly.</p>Formula:C11H14O2Purezza:99.74%Colore e forma:LiquidPeso molecolare:178.23Ref: TM-FR12339
Prodotto fuori produzione4-Ethoxycoumarin
CAS:<p>4-Ethoxycoumarin has antimicrobial activity.</p>Formula:C11H10O3Purezza:99.64%Colore e forma:SolidPeso molecolare:190.2Ref: TM-FR12662
Prodotto fuori produzioneRelacorilant
CAS:<p>Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.</p>Formula:C27H22F4N6O3SPurezza:98.53% - 99%Colore e forma:SolidPeso molecolare:586.563-Acetylcoumarin
CAS:<p>3-Acetylcoumarin as a practical ligand for copper-catalyzed CN coupling reactions at room temperature. It has neuroprotective and acaricidal properties.</p>Formula:C11H8O3Purezza:99.41%Colore e forma:Yellow Crystalline PowderPeso molecolare:188.1820-HETE
CAS:<p>20-HETE is a CYP450 product, vasoconstrictor, modulates K+ channels, affects NADPH, ROS, NF-κB, NO synthase, and cell apoptosis/proliferation.</p>Formula:C20H32O3Purezza:99.79%Colore e forma:SolidPeso molecolare:320.47Stephalonine L
CAS:<p>Stephalonine L is a natural product for research related to life sciences. The catalog number is TN6290 and the CAS number is 2379277-60-6.</p>Formula:C30H35NO10Purezza:98%Colore e forma:SolidPeso molecolare:569.6Ref: TM-TN6290
Prodotto fuori produzionePodoblastin A (D-mannitol)
<p>Podoblastin A (D-mannitol) is a useful organic compound for research related to life sciences and the catalog number is TSP-41077145.</p>Formula:C20H34O4Peso molecolare:338.49Pomalidomide-amido-PEG3-C2-NH2
CAS:<p>Cereblon Ligand-Linker 22: A pomalidomide-based E3 ligase conjugate with a PEG3 linker for PROTACs.</p>Formula:C22H28N4O8Purezza:98%Colore e forma:SolidPeso molecolare:476.48Ref: TM-T18553
Prodotto fuori produzioneL-Histidinyl-D-penicillaminatocobalt(III)
CAS:<p>L-Histidinyl-D-penicillaminatocobalt(III) can provide a model for the binding of D-penicillamine to metal ions.</p>Formula:C11H15CoN4O5SColore e forma:SolidPeso molecolare:374.26m-PEG1-acid
CAS:<p>M-PEG1-acid, a soluble PEG derivative, has a terminal carboxylic acid for forming amide bonds with primary amines using activators like EDC, DCC.</p>Formula:C4H8O3Purezza:98%Colore e forma:SolidPeso molecolare:104.10Patecibart
CAS:<p>Patecibart is a humanized immunoglobulin G4-kappa monoclonal antibody that functions as an antagonist to the endothelin receptor A (EDNRA).</p>Purezza:98%Colore e forma:LiquidRef: TM-T81538
Prodotto fuori produzioneFirefly Luciferase circRNA
<p>Firefly Luciferase circRNA, originally isolated from Photinus pyralis (Firefly), expresses a luciferase protein and serves as an optimal marker for monitoring</p>Colore e forma:Odour SolidTripeptide-41
CAS:<p>Tripeptide-41 (CG-Lipoxyn) is a bioactive peptide known for its ability to reduce fat accumulation.</p>Formula:C29H30N4O5Purezza:98%Colore e forma:SolidPeso molecolare:514.57Kbz probe 1
CAS:<p>Kbz probe 1, an adaptable probe utilized for examining histone benzoylation and interactions within living cells, showcases extensive versatility.</p>Formula:C13H17ClF2N2O3Colore e forma:SolidPeso molecolare:322.73FGFR-IN-1
CAS:<p>FGFR-IN-1 targets FGFR1-3 with IC50 <100 nM. (US20130338134A1, ex 219)</p>Formula:C26H24F2N4O6SColore e forma:SolidPeso molecolare:558.55(Rac)-IBT6A hydrochloride
CAS:<p>(Rac)-IBT6A HCl: racemic Ibrutinib impurity; for IBT6A dimers/adducts; Ibrutinib is a Btk inhibitor (IC50=0.5nM).</p>Formula:C22H23ClN6OColore e forma:SolidPeso molecolare:422.91(±)5-HETE
CAS:<p>(±)5-HETE is one of the six monohydroxy fatty acids produced by the non-enzymatic oxidation of arachidonic acid.</p>Formula:C20H32O3Colore e forma:SolidPeso molecolare:320.47Apoptosis inducer 4
CAS:<p>Apoptosis Inducer 4 (Compound 12b) is a compound that induces apoptosis and exhibits anticancer properties [1].</p>Formula:C41H50O11S3Colore e forma:SolidPeso molecolare:815.02Aflatoxin M1
CAS:<p>Aflatoxin M1, a toxic metabolite of Aflatoxin B1, is produced by Aspergillus fungi, with a toxicity order: B1 > M1 > G1 > B2 > M2 > G2.</p>Formula:C17H12O7Colore e forma:SolidPeso molecolare:328.276m-Ciaamp
CAS:<p>3-Carboxyphenyl((N-((4-iodophenyl)acetyl)amino)methyl)phosphonate is a bioactive chemical.</p>Formula:C16H15INO6PColore e forma:SolidPeso molecolare:475.175Cap-dependent endonuclease-IN-15
CAS:<p>Cap-dependent endonuclease-IN-15: potent CEN inhibitor, halts influenza virus replication, aids viral research.</p>Formula:C27H23F2N3O7SeColore e forma:SolidPeso molecolare:618.44Ref: TM-T72117
Prodotto fuori produzioneDeutetrabenazine metabolite M4
CAS:<p>Deutetrabenazine's metabolite M4 depletes monoamines by reversibly inhibiting VMAT2, affecting nerve terminals.</p>Formula:C19H21D6NO4Purezza:98%Colore e forma:SolidPeso molecolare:339.46TLQP-21 TFA
<p>TLQP-21 TFA is a VGF-derived peptide, C3aR1 agonist (mouse EC50: 10.3μM; human EC50: 68.8μM), that raises intracellular Ca2+ for nociception research.</p>Purezza:98%Colore e forma:LiquidSKF 89748
CAS:<p>SKF 89748 is an agonists of alpha 1-adrenoceptor.</p>Formula:C12H17NOSPurezza:98%Colore e forma:SolidPeso molecolare:223.337-(Diethylamino)-4-methyl-2H-chromen-2-one
CAS:<p>7-(Diethylamino)-4-methyl-2H-chromen-2-one is a useful organic compound for research related to life sciences.</p>Formula:C14H17NO2Colore e forma:SolidPeso molecolare:231.30GEM-5
CAS:<p>GEM-5, a gemcitabine conjugate with HIF-1α inhibitor YC-1 (IC50=30 nM), down-regulates HIF-1α, up-regulates p53, and induces A2780 cell apoptosis.</p>Formula:C32H29F2N5O8Colore e forma:SolidPeso molecolare:649.60Endoplasmic reticulum dye 1
CAS:<p>Endoplasmic reticulum dye 1: a live cell imaging agent for exocytosis at the plasma membrane with low cytotoxicity and high photobleaching resistance.</p>Formula:C21H12N7O3ReColore e forma:SolidPeso molecolare:596.58m-PEG11-Tos
<p>m-PEG11-Tos is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs[1].</p>Formula:C28H50O13SPurezza:98%Colore e forma:SolidPeso molecolare:626.75OVA Peptide 323-339
<p>OVA Peptide (323-339) is an Ovalbumin epitope crucial for hypersensitivity in BALB/c mice.</p>Formula:C74H120N26O25Purezza:98%Colore e forma:SolidPeso molecolare:1773.91Yhhu 3792
<p>Activates Notch pathway, boosts NSC self-renewal and neurogenesis, enhances mice memory.</p>Colore e forma:Solid2',3'-cGAMP-C2-SH
CAS:<p>2', 3'-cGAMP-C2-SH is a ADC cytotoxin.</p>Formula:C22H28N10O12P2SColore e forma:SolidPeso molecolare:718.53(D)-PPA 1
CAS:<p>PD-1/PD-L1 binder, Kd 0.51 μM; blocks interaction in flow cytometry at 1 mg/mL; inhibits tumors, extends mouse survival.</p>Formula:C70H98N20O21Purezza:98%Colore e forma:SolidPeso molecolare:1555.67Antitubercular agent-10
CAS:<p>Antitubercular agent-10 shows potent antitubercular activity with a MIC value of 30 nM.</p>Formula:C19H15N5O6S2Colore e forma:SolidPeso molecolare:473.481,6,8-Trihydroxy-2,7-dimethoxy-3-methylanthraquinone
<p>1,6,8-Trihydroxy-2,7-dimethoxy-3-methylanthraquinone is a useful organic compound for research related to life sciences and the catalog number is T125250.</p>Formula:C34H26O14Colore e forma:SolidPeso molecolare:658.5685-hydroxy-Nω-methyl Tryptamine (oxalate)
CAS:<p>5-hydroxy-Nω-methyl Tryptamine is a metabolite of serotonin in humans that has also been found in plants.</p>Formula:C13H16N2O5Colore e forma:SolidPeso molecolare:280.28Ref: TM-T37212
Prodotto fuori produzioneBPH-675
CAS:<p>BPH-675 is a bioactive chemical.</p>Formula:C24H23NO9P2SColore e forma:SolidPeso molecolare:563.45
