
Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.524 prodotti)
- Apoptosi(5.793 prodotti)
- Ciclo cellulare/Checkpoint(4.452 prodotti)
- Cromatina/Epigenetica(2.242 prodotti)
- Segnalazione citoscheletrica(1.382 prodotti)
- Danno al DNA/Riparazione del DNA(2.826 prodotti)
- Endocrinologia/Ormoni(3.507 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.333 prodotti)
- Immunologia e infiammazione(3.527 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.203 prodotti)
- Trasportatore di membrana/canale ionico(2.792 prodotti)
- Metabolismo(9.449 prodotti)
- Microbiologia/Virologia(6.981 prodotti)
- Neuroscienza(9.926 prodotti)
- Altri inibitori(37.921 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.597 prodotti)
- Cellule staminali e Derivati(830 prodotti)
- Adattatori Tirosin-chinasi(2.015 prodotti)
- Ubiquitinazione(1.650 prodotti)
Mostrare 16 più sottocategorie
Trovati 66639 prodotti di "Inibitori"
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CAY10735
CAS:<p>CAY10735: Anticancer agent; inhibits growth/migration in various cancer cells; reduces tumor in mouse models. IC50=0.674-11.56μM.</p>Formula:C44H60FN3O4Colore e forma:SolidPeso molecolare:713.979NE97220
CAS:<p>NE97220 is a bioactive chemical.</p>Formula:C7H12N2O6P2Colore e forma:SolidPeso molecolare:282.13VPC44116
CAS:<p>VPC44116 is a bioactive chemical.</p>Formula:C18H31N2O4PColore e forma:SolidPeso molecolare:370.43AI3-10714
CAS:<p>AI3-10714 is a biochemical.</p>Formula:C14H6F17NO2SColore e forma:SolidPeso molecolare:575.24Carbostyril 124
CAS:<p>Carbostyril 124 is a useful organic compound for research related to life sciences. The catalog number is T65062 and the CAS number is 19840-99-4.</p>Formula:C10H10N2OColore e forma:SolidPeso molecolare:174.203HX103
CAS:<p>HX103: Fluorogenic EGFR-TKI probe; inhibits various EGFR mutations; predicts NSCLC treatment response. IC50: 1.3-977 nM.</p>Formula:C26H25ClFN7O5SColore e forma:SolidPeso molecolare:602.04Ref: TM-T75015
Prodotto fuori produzioneMitoquinone
CAS:<p>Mitoquinone is a TPP-based, mitochondrially targeted antioxidant .</p>Formula:C37H44O4PPurezza:98%Colore e forma:SolidPeso molecolare:583.72Chol-N3
CAS:<p>Chol-N3 is a bioorthogonal chol probe capable of integrating with super-resolution fluorescence microscopy (SRM) to enable direct nanoscale imaging of lipid</p>Formula:C24H39N3OColore e forma:SolidPeso molecolare:385.592-Cyclohexen-1-one, 5-(1,5-dimethyl-4-hexen-1-yl)-4-hydroxy-2-methyl-
CAS:<p>1-Hydroxybisabola-2,10-dien-4-one is a natural product for research related to life sciences. The catalog number is TN5398 and the CAS number is 124898-71-1.</p>Formula:C15H24O2Purezza:98%Colore e forma:SolidPeso molecolare:236.35Dabigatran Acyl-β-D-Glucuronide
CAS:<p>Dabigatran acyl-β-D-glucuronide is a major active metabolite of the thrombin inhibitor dabigatran .</p>Formula:C31H33N7O9Colore e forma:SolidPeso molecolare:647.645LY 280748
CAS:<p>LY 280748 is a bio-active chemical.</p>Formula:C23H29N4NaO2Colore e forma:SolidPeso molecolare:416.49Zanamivir-Cholesterol Conjugate
CAS:<p>Zanamivir-cholesterol conjugate is an extended-duration neuraminidase inhibitor highly effective against drug-resistant influenza strains.</p>Formula:C61H104N8O15Colore e forma:SolidPeso molecolare:1189.544PROTAC VEGFR-2 degrader-2
CAS:<p>PROTAC VEGFR-2 degrader-2 has minimal VEGFR-2 inhibition (IC50 > 1μM) and low anti-proliferative effect on EA.hy926 cells (IC50 > 100μM).</p>Formula:C50H56FN9O6SColore e forma:SolidPeso molecolare:930.1STING agonist-9
CAS:<p>STING agonist-9 (Compound 45): potent, EC50 1.2 nM h-STING, 32.82 μM m-STING; antitumor [1].</p>Formula:C39H47N13O6SColore e forma:SolidPeso molecolare:825.94Z-(L-Arg)-AMC (hydrochloride)
CAS:<p>Z-(L-Arg)-AMC releases fluorescent AMC upon cleavage by trypsin, cathepsins B & H, used to measure their activity (Ex/Em: 340-360/440-460 nm).</p>Formula:C24H28ClN5O5Colore e forma:SolidPeso molecolare:501.97Thalidomide-C2-amido-C2-COOH
CAS:<p>Thalidomide-C2-amido-C2-COOH is a compound that includes a CRBN ligand for the E3 ubiquitin ligase, as well as a linker.</p>Formula:C19H20N4O7Purezza:98%Colore e forma:SolidPeso molecolare:416.38A031
CAS:<p>A031: PROTAC AR degrader, IC50 < 0.25 μM, inhibits prostate cancer growth in zebrafish.</p>Formula:C50H61ClN10O7SColore e forma:SolidPeso molecolare:981.6OVA Peptide 323-339
<p>OVA Peptide (323-339) is an Ovalbumin epitope crucial for hypersensitivity in BALB/c mice.</p>Formula:C74H120N26O25Purezza:98%Colore e forma:SolidPeso molecolare:1773.91N-Deacetyllapaconitine
<p>N-Deacetyllapaconitine is a useful organic compound for research related to life sciences and the catalog number is T131546.</p>Formula:C30H42N2O7Colore e forma:SolidPeso molecolare:542.673AT-1002 TFA
<p>AT-1002 TFA, a 6-mer synthetic peptide, functions as a tight junction regulator and absorption enhancer.</p>Formula:C34H54F3N9O9SColore e forma:SolidPeso molecolare:821.91HA-CD44 interaction inhibitor 1
<p>Antitumor agent-109 (compound 6) is a dual-function inhibitor that targets hyaluronic acid and CD44, which are involved in tumor progression and invasion.</p>Colore e forma:Odour SolidPROTAC eEF2K degrader-1
CAS:<p>PROTAC eEF2K degrader-1 (11l) targets eEF2K, induces apoptosis in MDA-MB-231 cells, and degrades eEF2K.</p>Formula:C31H33N9O11Colore e forma:SolidPeso molecolare:707.65Nutlin carboxylic acid
CAS:<p>Nutlin carboxylic acid is a Nutlin 3-based MDM2 ligand; used with a linker to create PROTACs.</p>Formula:C32H32Cl2N4O6Purezza:98%Colore e forma:SolidPeso molecolare:639.53Ref: TM-T17874
Prodotto fuori produzioneAzido-PEG12-t-butyl ester
CAS:<p>Azido-PEG12-t-butyl ester, a soluble PEG with azide/reactive t-butyl, forms triazoles via Click Chemistry; deprotectable in acid.</p>Formula:C31H62N3O14Colore e forma:SolidPeso molecolare:700.84Praluzatamab ravtansine
CAS:<p>Sirtratumab vedotin (ASG15-ME) is an antibody-drug conjugate (ADC) that links a SLITRK6-specific human gamma 2 antibody (Igγ2) to the microtubule disruption agent monomethyl auristatin E (MMAE) through a protease-cleavable linker [1].</p>Purezza:99.40%Colore e forma:SoildMicrocystin-LY
CAS:<p>Microcystin-LY, from Microcystis aeruginosa, is a heptapeptide toxin that triggers oxidative stress by activating the Nrf2 pathway, most effective at 3μM.</p>Formula:C52H71N7O13Colore e forma:SolidPeso molecolare:1002.16Oroxin A
CAS:<p>Oroxin A, a partial PPARγ agonist, activates PPARγ, inhibits α-glucosidase, and has antioxidant properties.</p>Formula:C21H20O10Purezza:98%Colore e forma:SolidPeso molecolare:432.38Ref: TM-TWS0787
Prodotto fuori produzionePROTAC BRD4 Degrader-17
CAS:<p>Compound 13i is a potent PROTAC BRD4 degrader with IC50s: 29.54 nM (BD1), 3.82 nM (BD2), impedes G2/M progression, and induces apoptosis in MV-4-11 cells.</p>Formula:C49H47N7O9Colore e forma:SolidPeso molecolare:877.94AS-604850
<p>AS-604850: PI3Kγ inhibitor, ATP-competitive, IC50=2.5μM, 30x> PI3Kδ/β, 18x> PI3Kα.</p>Formula:C11H5F2NO4SPurezza:98%Colore e forma:SolidPeso molecolare:285.22C12 NBD Sphingomyelin
CAS:<p>C12 NBD sphingomyelin, a fluorescent sphingomyelin derivative, serves as a sphingomyelinase substrate (Ex=470 nm, Em=525 nm).</p>Formula:C41H73N6O9PColore e forma:SolidPeso molecolare:825.03Ref: TM-T75371
Prodotto fuori produzioneIDO1-IN-20
CAS:<p>IDO1-IN-20 is an enzyme that catalyzes the oxidative metabolism of tryptophan. It can immunosuppress tumors in the tumor microenvironment.</p>Formula:C15H19BrFN7O4SColore e forma:SolidPeso molecolare:492.32α-Conotoxin GI
CAS:<p>α-conotoxin GI, a conopeptide isolated from the venom of the cone snail Conus geographus, is a competitive antagonist of the muscle-type nicotinic acetylcholine</p>Formula:C55H80N20O18S4Purezza:98%Colore e forma:SolidPeso molecolare:1437.61Questiomycin A derivatives 14
<p>Questiomycin A derivatives 14 is a Questiomycin A derivative.</p>Formula:C18H18N2O3Purezza:99.73%Colore e forma:SoildPeso molecolare:310.35Ajadine
CAS:<p>Ajadine is a Norditerpenoid alkaloid.</p>Formula:C35H48N2O10Colore e forma:SolidPeso molecolare:656.773Phenol, m-(2-(methylamino)ethyl)-, hydrochloride
CAS:<p>Phenol, m-(2-(methylamino)ethyl)-, hydrochloride is a biaoctive chemical.</p>Formula:C9H14ClNOColore e forma:SolidPeso molecolare:187.67MB-07803
CAS:<p>MB07803 is an orally available prodrug of an effective, noncompetitive inhibitor of fructose 1,6-bisphosphatase (FBPase) (EC50: 140 nM and t1/2 of 7.6±2.9 h).</p>Formula:C24H37N4O7PSPurezza:98%Colore e forma:SolidPeso molecolare:556.61Ref: TM-T16017
Prodotto fuori produzioneMCA17-1
CAS:<p>MCA17-1 exhibits superior bioactivity compared to the positive control, obeticholic acid (OCA), in the treatment of liver fibrosis.</p>Formula:C14H15NO5Colore e forma:SolidPeso molecolare:277.276Rhizocticin A
CAS:<p>Rhizocticin A is a potential inhibitor of threonine synthase.</p>Formula:C11H22N5O6PPurezza:98%Colore e forma:SolidPeso molecolare:351.3Decafentin
CAS:<p>Decafentin is a biochemical be used for fungicide, bactericide, wood Preservative and herbicide.</p>Formula:C46H51BrClPSnColore e forma:SolidPeso molecolare:868.95Chloracetophos
CAS:<p>Chloracetophos is a Agricultural Chemical.</p>Formula:C6H10Cl3O5PColore e forma:SolidPeso molecolare:299.47mTORC1-IN-1
<p>mTORC1-IN-1 (T1), a rapamycin homologue (rapalog) and selective inhibitor of mTORC1, controls cell growth and metabolism, with implications in various diseases</p>Purezza:98%Colore e forma:Odour SolidCarbamic acid, N-(O,O-dimethylphosphorothioyl)-N-methyl-, m-isopropylphenyl ester
CAS:<p>Carbamic acid, N-(O,O-dimethylphosphorothioyl)-N-methyl-, m-isopropylphenyl ester is a bioactive chemical.</p>Formula:C13H20NO4PSColore e forma:SolidPeso molecolare:317.34PD-1/PD-L1-IN 5 TFA
CAS:<p>PD-1/PD-L1-IN 5 is an inhibitor of PD-1/PD-L1 protein/protein interaction (IC50 of ≤100 nM).</p>Formula:C22H18N4O3S·xC2HF3O2Purezza:98%Colore e forma:SolidABT-491 free base
CAS:<p>ABT-491 free base is a bio-active chemical. Detailed information has not been published.</p>Formula:C28H22FN5O2Colore e forma:SolidPeso molecolare:479.51(Rac)-IBT6A hydrochloride
CAS:<p>(Rac)-IBT6A HCl: racemic Ibrutinib impurity; for IBT6A dimers/adducts; Ibrutinib is a Btk inhibitor (IC50=0.5nM).</p>Formula:C22H23ClN6OColore e forma:SolidPeso molecolare:422.91Cap-dependent endonuclease-IN-12
CAS:<p>Cap-dependent endonuclease-IN-12 (EXP-35) is a potent inhibitor with low toxicity, active against H1N1.</p>Formula:C55H46F4N6O14S2Colore e forma:SolidPeso molecolare:1155.112-Oleoylglycerol
CAS:<p>2-Oleoylglycerol is a lipid found in palm kernels that acts as a GPR119 agonist with neuroprotective properties and can be used in steatohepatitis modeling.</p>Formula:C21H40O4Purezza:98%Colore e forma:SolidPeso molecolare:356.54Pulcherriminic acid
CAS:<p>Pulcherriminic acid, a cyclic dipeptide, chelates Fe3+, forms pulcherrimin, and has antimicrobial properties used in food, agriculture, and medicine.</p>Formula:C12H20N2O4Colore e forma:SolidPeso molecolare:256.30TPPS
CAS:<p>Tetraphenylporphine sulfonate (TPPS) serves as a non-cytotoxic probe suitable for tumor localization detection [1].</p>Formula:C44H30N4O12S4Purezza:98%Colore e forma:SolidPeso molecolare:934.99

