
Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.805 prodotti)
- Apoptosi(6.288 prodotti)
- Ciclo cellulare/Checkpoint(4.815 prodotti)
- Cromatina/Epigenetica(2.486 prodotti)
- Segnalazione citoscheletrica(1.542 prodotti)
- Danno al DNA/Riparazione del DNA(2.945 prodotti)
- Endocrinologia/Ormoni(3.706 prodotti)
- Enzima(3.670 prodotti)
- Proteina G/GPCR(9.023 prodotti)
- Immunologia e infiammazione(3.898 prodotti)
- Virus dell'influenza(302 prodotti)
- Segnalazione JAK/STAT(415 prodotti)
- Segnalazione MAPK(1.248 prodotti)
- Trasportatore di membrana/canale ionico(3.071 prodotti)
- Metabolismo(10.180 prodotti)
- Microbiologia/Virologia(7.620 prodotti)
- Neuroscienza(10.369 prodotti)
- Altri inibitori(35.955 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.442 prodotti)
- Proteasi/Proteasoma(1.719 prodotti)
- Cellule staminali e Derivati(806 prodotti)
- Adattatori Tirosin-chinasi(2.033 prodotti)
- Ubiquitinazione(1.719 prodotti)
Mostrare 16 più sottocategorie
Trovati 66631 prodotti di "Inibitori"
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Sudan Orange G
CAS:SUDAN ORANGE G is a natural product.Formula:C12H10N2O2Purezza:98%Colore e forma:SolidPeso molecolare:214.22PUMA BH3
PUMA BH3 activates Bak, binds Bcl-2; triggers apoptosis via cytochrome C release; Kd 26 nM.Formula:C128H202N42O43SPurezza:98%Colore e forma:SolidPeso molecolare:3049.35-(and-6)-Carboxy SNARF-1, Acetoxymethyl Ester, Acetate
CAS:Carboxy SNARF-1 AM acetate (CAS #126208-13-7), with a pKa ~7.5, shifts from yellow-orange to red fluorescence for pH 7-8 measurement.Formula:C32H25NO9Purezza:98%Colore e forma:SolidPeso molecolare:567.55Laudexium methylsulfate
CAS:Laudexium methylsulfate: neuromuscular blocker for surgery; aids intubation and muscle relaxation.Formula:C53H77N2O12SPurezza:98%Colore e forma:SolidPeso molecolare:966.26Bromo-PEG3-azide
CAS:Bromo-PEG3-azide is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.Formula:C8H16BrN3O3Purezza:98%Colore e forma:SolidPeso molecolare:282.135ONO-8430506
CAS:ONO-8430506 is an orally available, potent autotaxin (ATX)/ENPP2 inhibitor (IC90: 100 nM) that inhibits ATX activity in mouse plasma.Formula:C27H28FN3O3Purezza:98.34%Colore e forma:SolidPeso molecolare:461.53Ref: TM-T38759
1mg103,00€5mg244,00€10mg338,00€25mg510,00€50mg687,00€100mg919,00€1mL*10mM (DMSO)271,00€GADGVGKSA
CAS:GADGVGKSA, a mutant KRAS G12D 9mer peptide, serves as an immunogenic neoantigen for cancer immunotherapy research [1].Formula:C30H52N10O13Colore e forma:SolidPeso molecolare:760.79Bivalirudin TFA
CAS:Bivalirudin TFA, a 20-residue synthetic peptide, reversibly inhibits thrombin, affecting platelet aggregation and thrombin generation.Formula:C98H138N24O33·C2HF3O2Colore e forma:SolidPeso molecolare:2294.34Ascr#8
CAS:Ascr#8 is a dauer-inducing ascaroside isolated from Caenorhabditis elegans. It synergizes with ascr#2 and ascr#3, and strongly enhances male attraction.Formula:C20H27NO7Purezza:98%Colore e forma:SolidPeso molecolare:393.43Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Formula:C84H130F3N25O23S2Colore e forma:SolidPeso molecolare:1979.21pyCTZ hydrochloride
PyCTZ (Pyridyl CTZ) hydrochloride, a pyridyl Coelenterazine (CTZ) analog, serves as an ATP-independent substrate for LumiLuc luciferase, producing intense blueColore e forma:Odour SolidAngiopeptin TFA
CAS:Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.Formula:C58H73F6N11O14S2Colore e forma:SolidPeso molecolare:1326.39Mcl-1 antagonist 1
CAS:Mcl-1 antagonist 1 is a Mcl-1 protein antagonist.Formula:C41H54ClF2N5O8SPurezza:98%Colore e forma:SolidPeso molecolare:850.42m-Acetanisidide, 2-(diethylamino)-4'-(octyloxy)-
CAS:m-Acetanisidide, 2-(diethylamino)-4'-(octyloxy)- is a bioactive chemical.Formula:C21H36N2O3Colore e forma:SolidPeso molecolare:364.52Glycosmisic acid
CAS:Glycosmisic acid is a natural product from Nauclea officinalis.Formula:C20H20O7Purezza:98%Colore e forma:SolidPeso molecolare:372.373Amylin (8-37), human
CAS:Human-derived Amylin (8-37) is a vasodilator in rat arteries and forms aggregates linked to type II diabetes.Formula:C138H216N42O45Colore e forma:SolidPeso molecolare:3183.4953-O-Coumaroylasiatic acid
CAS:3-O-Coumaroylasiatic acid is a natural product for research related to life sciences. The catalog number is TN2971 and the CAS number is 143773-52-8.Formula:C39H54O7Purezza:98%Colore e forma:SolidPeso molecolare:634.854(d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin
CAS:'(d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin blocks oxytocin receptors, stopping oxytocin effects on CA1 neuron currents.'Formula:C45H69N9O12S2Colore e forma:SolidPeso molecolare:992.21Anhydro Dihydro Artemisinin
CAS:Anhydro Dihydro Artemisinin is a natural product from Artemisia carvifolia Buch.-Ham. ex Roxb.Formula:C15H22O4Purezza:98%Colore e forma:SolidPeso molecolare:266.337β-Hydroxyrutaecarpine
CAS:7beta-Hydroxyrutaecarpine is a natural product from Euodia ruticarpa.Formula:C18H13N3O2Purezza:98%Colore e forma:SolidPeso molecolare:303.31Thanatin
CAS:Thanatin is an antimicrobial peptide with antifungal properties effective against certain Gram-positive bacteria [1].Formula:C103H177N35O27S3Colore e forma:SolidPeso molecolare:2433.92Taxin B
CAS:Taxin B has toxic effects.Formula:C28H38O10Purezza:98%Colore e forma:SolidPeso molecolare:534.6Ivermectin B1a-d2
Deuterated ivermectin B1aFormula:C48H72D2O14Purezza:98%Colore e forma:SolidPeso molecolare:877.1Apoptosis inducer 12
CAS:Apoptosis Inducer 12 (Compound 3z) is a compound that promotes cell death via the mitochondrial pathway and is utilized in cancer research [1].Formula:C26H27N3O5Colore e forma:SolidPeso molecolare:461.51(Gln22)-Amyloid β-Protein (1-42)
CAS:(Gln22)-Amyloid β-Protein (1-42), a Dutch mutation (E22Q) variant of β-Amyloid (1-42), demonstrates increased fibrillogenic and pathogenic characteristics [1].Formula:C203H312N56O59SColore e forma:SolidPeso molecolare:4513.05Sanfetrinem
CAS:Sanfetrinem (GV104326) sodium is a β-lactamase antibiotic with antimicrobial activity for the study of bacterial infections.Formula:C14H19NO5Purezza:>99.99%Colore e forma:SolidPeso molecolare:281.3NF864
CAS:NF864, a suramin analog, is a P2X1 receptor inhibitor.Formula:C57H28N6Na12O41S12Purezza:98%Colore e forma:SolidPeso molecolare:2113.5Panaxydiol
CAS:<p>Panaxydiol is a natural product for research related to life sciences. The catalog number is TN5804 and the CAS number is 63910-76-9.</p>Formula:C17H24O2Purezza:98%Colore e forma:SolidPeso molecolare:260.37Fluo-3
CAS:Fluo-3 and its derivative, Fluo3/AM, serve as fluorescent indicators for intracellular calcium (Ca2+), facilitating detection through flow cytometry andFormula:C36H30Cl2N2O13Colore e forma:SolidPeso molecolare:769.54Mca-(endo-1a-Dap(Dnp))-TNF-α (-5 to +6) amide (human) TFA
Mca-(endo-1α-Dap(Dnp))-TNF-α(-5 to +6) amide (human) TFA is a peptide that functions as a fluorescence resonance energy transfer (FRET)-based substrate, withFormula:C69H103N23O24·C2HF3O2Colore e forma:SolidGarcinoic acid
CAS:Garcinoic acid is a useful organic compound for research related to life sciences. The catalog number is T123933 and the CAS number is 91893-83-3.Formula:C27H38O4Colore e forma:SolidPeso molecolare:426.597FHD-286
CAS:FHD-286 is an inhibitor of BRM/BRG1 ATPase and can be used for studies on the treatment of BAF-related disorders such as acute myeloid leukemia.Formula:C24H30N6O6S2Purezza:99.73%Colore e forma:SolidPeso molecolare:562.66Ref: TM-T9749
1mg144,00€5mg283,00€10mg454,00€25mg615,00€50mg777,00€100mg1.064,00€1mL*10mM (DMSO)359,00€Thalidomide-O-amido-PEG1-(C1-PEG)2-C2-NH2
CAS:<p>Thalidomide-O-amido-PEG1-(C1-PEG)2-C2-NH2 is a synthetic conjugate compound that combines a Thalidomide-based cereblon ligand and a linker, which is commonly</p>Formula:C25H34N4O9Purezza:98%Colore e forma:SolidPeso molecolare:534.566Lys-Gln-Ala-Gly-Asp-Val
CAS:KQAGDV is a fibrinogen γ-chain cell adhesion peptide, targeting α2bβ3 integrin, and binds SMCs.Formula:C25H44N8O10Colore e forma:SolidPeso molecolare:616.665,5'-Dimethoxysecoisolariciresinol
CAS:5,5'-Dimethoxysecoisolariciresinol is a natural product from Podocarpus spicata.Formula:C22H30O8Purezza:98%Colore e forma:SolidPeso molecolare:422.47IDR-1
CAS:IDR-1: Antimicrobial peptide, combats Gram-positive/negative bacteria, modulates immunity, non-toxic, anti-inflammatory, regulates chemokines/cytokines.Formula:C65H118N18O15Colore e forma:SolidPeso molecolare:1391.77Boc-aminooxy-amide-PEG4-propargyl
CAS:Boc-aminooxy-amide-PEG4-propargyl is a 4-unit PEG linker for ADC synthesis.Formula:C18H32N2O8Purezza:98%Colore e forma:SolidPeso molecolare:404.46β-Lipotropin (60-65)
CAS:<p>β-Lipotropin (60-65) (β-LPH (60-65)), an opioid agonist, is a significant [1] opioid peptide.</p>Formula:C33H47N9O8SColore e forma:SolidPeso molecolare:729.85egg white lysozyme (19-36) [Gallus gallus]
Hen egg-white lysozyme, ~14.6 kDa with 129 amino acids, catalyzes hydrolysis of bacterial cell walls' glycosidic bonds.Formula:C86H144N28O23S2Purezza:98%Colore e forma:SolidPeso molecolare:2002.375-Ethoxy-10-Gingerol
CAS:5-Ethoxy-10-Gingerol is a natural productFormula:C23H38O4Purezza:98%Colore e forma:SolidPeso molecolare:378.55Dactimicin sulfate
CAS:Dactimicin is a new aminoglycoside. It also has in vitro activity, post-antibiotic effect, and interaction with other antibiotics.Formula:C18H40N6O14S2Colore e forma:SolidPeso molecolare:628.67Mitoclomine
CAS:Mitoclomine is a biochemical.Formula:C16H19Cl2NOColore e forma:SolidPeso molecolare:312.23Prafnosbart
CAS:Prafnosbart (DS-6016A) is a humanized IgG1-kappa monoclonal antibody targeting ACVR1 (activin A receptor type 1, ACVRLK2, ALK2, ACVR1A, SKR1), utilized inColore e forma:LiquidEnterocin K1
CAS:Enterocin K1 (EntK1) is a ribosomally synthesized bacteriocin that exerts potent antibacterial activity against Vancomycin-resistant Enterococcus (VRE).Formula:C218H321N53O51S2Colore e forma:SolidPeso molecolare:4564.34Honyucitrin
CAS:Honyucitrin is a natural product of Citrus, Rutaceae.Formula:C25H26O5Purezza:98%Colore e forma:SolidPeso molecolare:406.47Amyloid Precursor C-Terminal Peptide
Amyloid precursor peptide involved in Alzheimer's forms plaques; sequence Gly-Tyr-Glu-Asn-Pro-Thr-Y-Lys-Phe-F-Glu-Gln-M-Gln-Asn. Linked to astrocytosis.Formula:C86H118N20O27S1Purezza:98%Colore e forma:SolidPeso molecolare:1896.04Eicosanyl caffeate
CAS:Eicosanyl caffeate has anti-ulcer and moderate antioxidant properties, it exhibits potent elastase inhibitory activity, with the IC(50) value of 0.99 microg/mL.Formula:C29H48O4Purezza:98%Colore e forma:SolidPeso molecolare:460.69(+)-N-Methylallosedridine
CAS:(+)-N-Methylallosedridine is a natural product for research related to life sciences. The catalog number is TN4612 and the CAS number is 41447-16-9.Formula:C9H19NOPurezza:98%Colore e forma:SolidPeso molecolare:157.25Leprolomin
CAS:Leprolomin is a bioactive chemical.Formula:C20H22O8Colore e forma:SolidPeso molecolare:390.38

