
Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.524 prodotti)
- Apoptosi(5.793 prodotti)
- Ciclo cellulare/Checkpoint(4.452 prodotti)
- Cromatina/Epigenetica(2.242 prodotti)
- Segnalazione citoscheletrica(1.382 prodotti)
- Danno al DNA/Riparazione del DNA(2.826 prodotti)
- Endocrinologia/Ormoni(3.507 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.333 prodotti)
- Immunologia e infiammazione(3.527 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.203 prodotti)
- Trasportatore di membrana/canale ionico(2.792 prodotti)
- Metabolismo(9.449 prodotti)
- Microbiologia/Virologia(6.981 prodotti)
- Neuroscienza(9.926 prodotti)
- Altri inibitori(37.921 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.597 prodotti)
- Cellule staminali e Derivati(830 prodotti)
- Adattatori Tirosin-chinasi(2.015 prodotti)
- Ubiquitinazione(1.650 prodotti)
Mostrare 16 più sottocategorie
Trovati 66639 prodotti di "Inibitori"
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Sunitinib-d10
CAS:<p>Sunitinib D10, a deuterium-enriched version, inhibits VEGFR2 and PDGFRβ tyrosine kinases (IC50: 80 nM/2 nM).</p>Formula:C22H27FN4O2Purezza:98%Colore e forma:SolidPeso molecolare:408.54Bixin
CAS:<p>Bixin, from Bixa orellana seeds, has anti-tumor, anti-inflammatory effects and boosts heart health by reducing fibrosis and ROS.</p>Formula:C25H30O4Colore e forma:SolidPeso molecolare:394.52'-Fluoro-2'-deoxy-ara-U-3'-phosphoramidite
CAS:<p>2'-Fluoro-2'-deoxy-ara-U-3'-phosphoramidite is a Nucleoside Phosphoramidite; Nucleoside Derivative - Fluoro-modified nucleoside.</p>Formula:C39H46FN4O8PColore e forma:SolidPeso molecolare:748.78Aminooxy-PEG3-C2-NH-Boc
CAS:<p>Aminooxy-PEG3-C2-NH-Boc is a PEG linker for making PROTACs for protein degradation.</p>Formula:C13H28N2O6Colore e forma:SolidPeso molecolare:308.37N4-Benzoyl-3'-O-methylcytidine
CAS:<p>N4-Benzoyl-3'-O-methylcytidine is a Nucleoside Derivative - 3'-Modified nucleoside.</p>Formula:C17H19N3O6Colore e forma:SolidPeso molecolare:361.35(1S)-1,4-Anhydro-1-C-(2,4-difluorophenyl)-D-ribitol
CAS:<p>(1S)-1,4-Anhydro-1-C-(2,4-difluorophenyl)-D-ribitol is a Nucleoside Derivative - C-nucleoside; Fluoro-modified nucleoside.</p>Formula:C11H12F2O4Colore e forma:SolidPeso molecolare:246.21Super Fluor 488
<p>Super Fluor 488: bright green dye, excels with 488 nm laser, pH-stable, high yield & photostable for sensitive bio-imaging.</p>Purezza:98%Colore e forma:SolidPeso molecolare:N/ALoganic acid 6′-O-β-D-glucoside
CAS:<p>Loganic acid 6′-O-β-D-glucoside (8-Epi-Loganic acid-6'-O-β-D-glucoside) is a natural product from Cistanche deserticola and inhibts the production of LPS-</p>Formula:C22H34O15Purezza:98%Colore e forma:SolidPeso molecolare:538.5Cyclopyrimorate
CAS:<p>Cyclopyrimorate is a highly effective bleaching herbicide for weed control in rice fields.</p>Formula:C19H20ClN3O4Colore e forma:SolidPeso molecolare:389.8335-Azidomethyl-2'-β-methyl-2',3',5'-tri-O-benzoyluridine
CAS:<p>5-Azidomethyl-2'-beta-methyl-2',3',5'-tri-O-benzoyluridine is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside; Azido nucleoside; 2'-Modified</p>Formula:C32H27N5O9Colore e forma:SolidPeso molecolare:625.59MDH1-IN-1
CAS:<p>MDH1-IN-1 is a potent MDH1 inhibitor with potential anticancer activity for the study of diseases related to the immune system.</p>Formula:C21H25NO4Purezza:99.36%Colore e forma:SolidPeso molecolare:355.43Substance P TFA
CAS:<p>Substance P TFA is a CNS neuropeptide, serving as a neurotransmitter and modulator, targeting NK1R.</p>Formula:C65H99F3N18O15SPurezza:98%Colore e forma:SolidPeso molecolare:1461.67AAPH
CAS:<p>AAPH: water-soluble azo, generates free radicals, used in lipid peroxidation studies, and antioxidation tests. Half-life ~175h at 37°C, pH neutral.</p>Formula:C8H20Cl2N6Colore e forma:SolidPeso molecolare:271.192'-Deoxy-2'-fluoro-N6-methyladensoine
CAS:<p>Nucleoside Derivatives - 2’-Modified nucleosides, Fluoro-modified nucleosides, 6-Modified purine nucleosides</p>Formula:C11H14FN5O3Colore e forma:SolidPeso molecolare:283.26m-PEG10-alcohol
CAS:<p>m-PEG10-alcohol, a 10-unit PEG ADC/PROTAC linker, is used in ADC and PROTAC synthesis.</p>Formula:C21H44O11Purezza:98%Colore e forma:SolidPeso molecolare:472.57Propanil
CAS:Propanil is a widely used contact herbicide. It is mainly used in rice production.Formula:C9H9Cl2NOPurezza:98%Colore e forma:Propanil Is A Colorless To Brown Crystals Non Corrosive Used As An HerbicidePeso molecolare:218.08ARD-1676
CAS:<p>ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand with a cereblon ligand.</p>Formula:C44H46ClN7O5Purezza:98%Colore e forma:SolidPeso molecolare:788.332',3',5'-Tri-O-benzoyl-5-iodouridine
CAS:<p>Nucleoside Derivatives - Halo-Nucleosides, 5-Modified pyrimidine nucleosides</p>Formula:C30H23IN2O9Colore e forma:SolidPeso molecolare:682.42OR-1855
CAS:<p>OR-1855 is an active Levosimendan metabolite, has effect on human myometrial contractility.</p>Formula:C11H13N3OPurezza:98%Colore e forma:Pale Yellow SolidPeso molecolare:203.24Sappanchalcone
CAS:<p>Sappanchalcone shows xanthine oxidase inhibitory activity, is a xanthine oxidase inhibitor.</p>Formula:C16H14O5Purezza:97.00% - 98.35%Colore e forma:SolidPeso molecolare:286.28Mozavaptan hydrochloride
CAS:<p>Mozavaptan is a vasopressin receptor antagonist.</p>Formula:C27H30ClN3O2Colore e forma:SolidPeso molecolare:464Propargyl-PEG2-CH2COOH
CAS:<p>Propargyl-PEG2-CH2COOH is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Formula:C9H14O5Colore e forma:SolidPeso molecolare:202.2LIN28 inhibitor LI71 enantiomer
CAS:<p>LIN28 inhibitor LI71 enantiomer, less active than the original, is a cell-permeable LIN28 blocker with a 7 uM IC50.</p>Formula:C21H21NO3Colore e forma:SolidPeso molecolare:335.4032',3',5'-Tri-O-benzoyl-5-difluoromethyluridine
CAS:<p>Nucleoside Derivatives - Fluoro-modified nucleosides; 5-Modified pyrimidine nucleosides</p>Formula:C31H24F2N2O9Colore e forma:SolidPeso molecolare:606.535-Cyanouridine
CAS:<p>5-Cyanouridine is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside.</p>Formula:C10H11N3O6Colore e forma:SolidPeso molecolare:269.21Propargyl-PEG5-NHS ester
CAS:<p>Propargyl-PEG5-NHS ester is a cleavable ADC linker used in the synthesis of antibody-drug conjugates (ADCs)[1].</p>Formula:C18H27NO9Purezza:98%Colore e forma:SolidPeso molecolare:401.41Thalidomide-O-C6-NH2 TFA
CAS:<p>Thalidomide-O-C6-NH2 TFA is a synthesized E3 ligase ligand-linker conjugate used in the PROTAC dTAG-13, a degrader of FKBP12F36V and BET[1].</p>Formula:C21H24F3N3O7Purezza:98%Colore e forma:SolidPeso molecolare:487.43Desoxycorticosterone pivalate
CAS:<p>DOCP, a mineralocorticoid, treats dogs with adrenal insufficiency.</p>Formula:C26H38O4Colore e forma:SolidPeso molecolare:414.58Biotin-PEG3-NHS ester
CAS:<p>Biotin-PEG3-NHS ester is a PROTAC linker based on the PEG structure and can be used to prepare PROTAC.</p>Formula:C23H36N4O9SPurezza:97.12% - 98.27%Colore e forma:SolidPeso molecolare:544.62HDAC-IN-4
CAS:<p>HDAC-IN-4 is a selective HDAC6 and HDAC10 inhibitor (pIC50s: 7.2 and 6.8 in BRET assay) with antitumoral activity.</p>Formula:C20H21N3O2Colore e forma:SolidPeso molecolare:335.43'-β-Azido-2',3'-dideoxy-5'-O-(4-methoxytrityl)uridine
CAS:<p>3'-beta-Azido-2',3'-dideoxy-5'-O-(4-methoxytrityl)uridine is a Nucleoside Derivative - 2',3'-Dideoxy nucleoside, 3'-Modified nucleoside, Azido-nucleoside, Xylo-</p>Formula:C29H27N5O5Colore e forma:SolidPeso molecolare:525.56Niazirin
CAS:<p>Moringa oleifera extract with niaziridin and Niazirin may reduce pulmonary hypertension by vasodilation and boosting antioxidants.</p>Formula:C14H17NO5Purezza:98%Colore e forma:SolidPeso molecolare:279.295'-O-DMT-N6-Me-2'-dA
CAS:<p>5'-O-DMT-N6-Me-2'-dA is a nucleoside with protective and modification effects.</p>Formula:C32H33N5O5Colore e forma:SolidPeso molecolare:567.63Mito-apocynin (C11)
CAS:<p>Mito-apocynin (C11)是一种线粒体靶向抗氧化剂,通过靶向和中和细胞呼吸过程中产生的活性氧(ROS)发挥作用。三苯基溴化鏻已被发现能有效预防线粒体功能障碍,线粒体功能障碍是衰老过程和各种疾病的主要原因。它具有抗炎、抗凋亡和抗氧化活性。</p>Formula:C37H44BrO4PPurezza:98%Colore e forma:SolidPeso molecolare:663.62Osimertinib dimesylate
CAS:<p>Osimertinib dimesylate is an irreversible and mutant selective EGFR inhibitor (IC50s: 12 and 1 nM against EGFR L858R and EGFR L858R/T790M).</p>Formula:C30H41N7O8S2Purezza:98%Colore e forma:SolidPeso molecolare:691.82NS 383
CAS:<p>ASIC blocker with varying IC50: 0.12 μM in hASIC1a, and ineffective on hASIC2a/3; <5 μM on rASIC1a/2a/3; alleviates pain in inflamed/CCI rats.</p>Formula:C19H19N3O2Colore e forma:SolidPeso molecolare:321.37Enrofloxacin monohydrochloride
CAS:<p>Enrofloxacin monohydrochloride, an antibiotic, has MIC 90 of 0.312 μg/mL for M. bovis and inhibits vaccinia virus.</p>Formula:C19H23ClFN3O3Colore e forma:SolidPeso molecolare:395.86Drimenol
CAS:<p>Drimenol inhibits Botrytis cinerea (EC50: 80 ppm) and quorum sensing.</p>Formula:C15H26OPurezza:98%Colore e forma:SolidPeso molecolare:222.37HTS01037
CAS:<p>HTS01037 is an inhibitor of fatty acid-binding. HTS01037 is a competitive antagonist of protein-protein interactions mediated by AFABP/aP2 (Ki: 0.67 μM).</p>Formula:C14H11NO5S2Colore e forma:SolidPeso molecolare:337.37N-desmethyl Enzalutamide D6
<p>N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.</p>Formula:C20H8D6F4N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:456.456-(β-D-5-O-(4,4'-Dimethoxytrityl)-2-deoxyribofuranosyl)-3,4-dihydro-8H-pyrimido[4,5-c][1,2]oxazin-7-one
CAS:<p>Nucleoside Derivatives - Bi-/Tricyclic nucleosides; Protected nucleosides w/NH2/OH open</p>Formula:C32H33N3O7Colore e forma:SolidPeso molecolare:571.62Methotrexate Diglutamate
CAS:<p>Methotrexate Diglutamate Small molecule compound present in the liver that acts as a partially purified human dihydrofolate reductase inhibitor.</p>Formula:C25H29N9O8Purezza:98.51%Colore e forma:SolidPeso molecolare:583.55Octanoic acid
CAS:<p>Octanoic acid (Caprylic acid) is found naturally in coconuts and breast milk. Caprylic acid is used in the production of esters used in perfumery.</p>Formula:C8H16O2Purezza:97.43% - 99.90%Colore e forma:Colourless Liquid OilyPeso molecolare:144.21Ayanin
CAS:<p>Ayanin: a vasorelaxant with potential in allergic asthma treatment; IL-4 inhibition IC50 of 2.2µM; non-selective PDE1-4 inhibitor for respiratory research.</p>Formula:C18H16O7Purezza:99.65%Colore e forma:SolidPeso molecolare:344.32KY-05009
CAS:<p>KY-05009 blocks TGF-β1 EMT in lung cancer cells, inhibits TNIK, Wnt genes, induces apoptosis, and is an ATP-competitive TNIK inhibitor (Ki = 100 nM).</p>Formula:C18H16N4O2SPurezza:99.89%Colore e forma:SolidPeso molecolare:352.41Glucosamine sulfate
CAS:<p>Glucosamine sulfate (D-Glucosaminesulfate) was extracted from synthetic product;Store the product in sealed, cool and dry condition.</p>Formula:C6H13NO5·H2SO4Purezza:99.64%Colore e forma:White CrystalPeso molecolare:277.25Guanine
CAS:<p>Guanine (2-Aminohypoxanthine) is a purine base that is a constituent of nucleotides occurring in nucleic acids.</p>Formula:C5H5N5OPurezza:99.89%Colore e forma:Several Desmotropic Forms; Usually Amorphous SolidPeso molecolare:151.13Emtricitabine
CAS:<p>Emtricitabine is a nucleoside reverse transcriptase inhibitor with anti-human immunodeficiency virus (HIV) and hepatitis B virus activity.Cost-effective and quality-assured.</p>Formula:C8H10FN3O3SPurezza:99.15% - 99.78%Colore e forma:White PowderPeso molecolare:247.25Angiotensin 1/2 + A (2 - 8) Acetate
<p>Angiotensin 1/2 + A (2 - 8) Acetate is a Vasoconstrictor.</p>Formula:C51H75N13O12Purezza:98.55%Colore e forma:SolidPeso molecolare:1062.22Ac2-26 acetate
<p>Ac2-26 acetate is an active N-terminal peptide of annexin A1(AnxA1).</p>Formula:C141H210N32O44SPurezza:98%Colore e forma:SolidPeso molecolare:3089.43

