Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.523 prodotti)
- Apoptosi(5.792 prodotti)
- Ciclo cellulare/Checkpoint(4.449 prodotti)
- Cromatina/Epigenetica(2.238 prodotti)
- Segnalazione citoscheletrica(1.383 prodotti)
- Danno al DNA/Riparazione del DNA(2.825 prodotti)
- Endocrinologia/Ormoni(3.507 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.333 prodotti)
- Immunologia e infiammazione(3.526 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.202 prodotti)
- Trasportatore di membrana/canale ionico(2.790 prodotti)
- Metabolismo(9.448 prodotti)
- Microbiologia/Virologia(6.981 prodotti)
- Neuroscienza(9.926 prodotti)
- Altri inibitori(37.926 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.597 prodotti)
- Cellule staminali e Derivati(831 prodotti)
- Adattatori Tirosin-chinasi(2.016 prodotti)
- Ubiquitinazione(1.650 prodotti)
Mostrare 16 più sottocategorie
Trovati 66641 prodotti di "Inibitori"
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Physion 8-O-β-D-glucoside
CAS:<p>Physion 8-O-β-D-glucoside is a tumor cell growth inhibitor.</p>Formula:C22H22O10Purezza:95.17% - 99.66%Colore e forma:SolidPeso molecolare:446.4Autocamtide-2-related inhibitory peptide, myristoylated acetate(201422-04-0 free base)
<p>Myristoylated autocamtide-2-related inhibitory peptide acetate is a cell-permeable CaM kinase II inhibitor.</p>Formula:C80H146N22O22Purezza:97.03%Colore e forma:SolidPeso molecolare:1768.15Taurolithocholic acid sodium salt
CAS:<p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>Formula:C26H44NNaO5SPurezza:99.79% - 99.93%Colore e forma:SolidPeso molecolare:505.695-Methylcytidine
CAS:<p>5-Methylcytidine is a modified nucleoside derived from 5-methylcytosine and is a minor constituent of RNA as well as DNA for certain organisms.</p>Formula:C10H15N3O5Purezza:99.02% - 99.88%Colore e forma:SolidPeso molecolare:257.24FRAX486 HCL(1232030-35-1 free base)
<p>FRAX486 HCL is a potent p21-activated kinase (PAK) inhibitor with IC50 values of 14, 33, 39 and 575 nM for PAK1, PAK2, PAK3 and PAK4 respectively.</p>Formula:C25H24Cl3FN6OPurezza:98.85% - 99.82%Colore e forma:SolidPeso molecolare:549.86TW-37
CAS:<p>TW-37 is an nonpeptide inhibitor to recombinant Bcl-2, Bcl-xL and Mcl-1 (Ki: 0.29/1.11/0.26 μM).</p>Formula:C33H35NO6SPurezza:97.06% - ≥95%Colore e forma:SolidPeso molecolare:573.7Atopaxar hydrochloride
CAS:<p>Atopaxar hydrochloride is used in the Treatment of Cardiovascular Disorders.</p>Formula:C29H39ClFN3O5Colore e forma:SolidPeso molecolare:564.1Galanin Receptor Ligand M35 TFA
<p>Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).</p>Formula:C109H154N27F3O28Purezza:99.45%Colore e forma:SolidPeso molecolare:2347.62SR 57227 hydrochloride
CAS:<p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>Formula:C10H14ClN3·HClPurezza:99.89%Colore e forma:SolidPeso molecolare:248.15Cevidoplenib dimesylate hydrochloride
CAS:<p>Cevidoplenib dimesylate hydrochloride is a spleen tyrosine kinase (Syk) inhibitor showing potential immunomodulating and anti-inflammatory properties.</p>Formula:C90H132Cl5N27O12Purezza:97.52%Colore e forma:SolidPeso molecolare:1957.9HNHA
CAS:<p>HNHA is an inhibitor of HDAC.</p>Formula:C17H21NO2SPurezza:98.04%Colore e forma:SolidPeso molecolare:303.42SRT3109
CAS:<p>SRT3109 is a CXCR2 ligand used in the treatment of chemokine mediated diseases and conditions.</p>Formula:C18H23F2N5O4S2Purezza:99.65% - 99.92%Colore e forma:SolidPeso molecolare:475.53FB23
CAS:<p>FB23 binds and inhibits FTO, an enzyme that demethylates m6A in mRNA and aids leukemia development.</p>Formula:C18H14Cl2N2O3Purezza:98.22% - 99.19%Colore e forma:SolidPeso molecolare:377.22Tedizolid Phosphate
CAS:<p>Tedizolid Phosphate (TR-701FA) is an oxazolidinone-class antibiotic. Tedizolid phosphate is a phosphate ester prodrug of the active compound tedizolid.</p>Formula:C17H16FN6O6PPurezza:97.96%Colore e forma:SolidPeso molecolare:450.32AMG 925
CAS:<p>AMG 925 is a potent and orally bioavailable dual FLT3/CDK4 inhibitor with IC50 of 1 nM and 3 nM, respectively.</p>Formula:C26H29N7O2Purezza:99.75%Colore e forma:SolidPeso molecolare:471.55[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS:<p>Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).</p>Formula:C39H65N9O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:803.99DUPA
CAS:<p>DUPA (N,N''-Carbonylbis[L-glutamic acid]) is used as the targeting moiety to actively deliver DTX for treatment of Prostate-Specific Membrane Antigen (PSMA)</p>Formula:C11H16N2O9Purezza:99.56%Colore e forma:SolidPeso molecolare:320.25MLS000532223
CAS:<p>MLS000532223 is a selectiveRho family GTPases inhibitor(EC50 : 16 μM to 120 μM).</p>Formula:C15H9NO3Purezza:98.6%Colore e forma:SolidPeso molecolare:251.2420(R)-Ginsenoside Rg2
CAS:<p>20(R)-Ginsenoside Rg2 (20R-Ginsenoside Rg2) is a compound with anti-oxidant and anti-apoptosis.</p>Formula:C42H72O13Purezza:99.7% - 99.86%Colore e forma:SolidPeso molecolare:785.01Ki16425
CAS:<p>Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.</p>Formula:C23H23ClN2O5SPurezza:97.6% - 97.78%Colore e forma:SolidPeso molecolare:474.96EST64454 free base
CAS:<p>EST64454: σ1R antagonist for pain, high solubility, permeable, BCS class I, metabolically stable.</p>Formula:C18H22F2N4O2Colore e forma:SolidPeso molecolare:364.39Lodoxamide
CAS:<p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>Formula:C11H6ClN3O6Purezza:99.13% - 99.81%Colore e forma:SolidPeso molecolare:311.632-Acetylthiazole
CAS:<p>2-Acetylthiazole (2-Acetylthiazole;2 Acetylthiazole) is used in the preparation of chiral alcohols, triazolothiazoles, it is also used in aldol condensation</p>Formula:C5H5NOSPurezza:98.32%Colore e forma:Clear ColorlessPeso molecolare:127.16CX-5461 dihydrochloride
<p>CX-5461 dihydrochloride: Oral Pol I inhibitor, HCT-116 (IC50: 142 nM), A375 (IC50: 113 nM), MIA PaCa-2 (IC50: 54 nM), weak on Pol II (IC50 ≥ 25 μM).</p>Formula:C27H29Cl2N7O2SColore e forma:SolidPeso molecolare:586.54Br-Mmc
CAS:<p>Br-Mmc (4-Bromomethyl-7-methoxycoumarin) is used as a new fluorescence label for fatty acids. It is used for the determination of fatty acids by HPLC or TLC.</p>Formula:C11H9BrO3Purezza:98.15%Colore e forma:Light Green-Yellow CrystalsPeso molecolare:269.09SPOP-IN-6b hydrochloride
CAS:<p>SPOP-IN-6b hydrochloride is a highly effective inhibitor of speckle-type POZ protein (SPOP), exhibiting an IC50 value of 3.58 μM.</p>Formula:C28H33ClN6O3Colore e forma:SolidPeso molecolare:537.06Raffinose
CAS:<p>Raffinose, an indigestible trisaccharide of galactose, glucose, and fructose, is found in plants and hydrolyzed by α-GAL.</p>Formula:C18H32O16Purezza:99.9%Colore e forma:WetsolidPeso molecolare:504.44Drofenine
CAS:<p>Drofenin: anticonvulsant, anticholinergic, neurotropic, musculotropic, FIASMA.</p>Formula:C20H31NO2Colore e forma:SolidPeso molecolare:317.47Phanquinone
CAS:<p>Phanquinone is active against a wide range of Gram-positive and Gram-negative organisms.</p>Formula:C12H6N2O2Purezza:97.79%Colore e forma:SolidPeso molecolare:210.19Paroxetine maleate
CAS:<p>Paroxetine maleate is a selective inhibitor of serotonin reuptake and an antidepressant.</p>Formula:C23H24FNO7Colore e forma:SolidPeso molecolare:445.443LED209
CAS:<p>LED209, a specific inhibitor of quorum sensor QseC of GNB, can generate a multifunctional agent PAMAM-LED209.</p>Formula:C19H17N3O2S2Purezza:97.35%Colore e forma:SolidPeso molecolare:383.492-hydroxymethyl benzoic acid
CAS:<p>2-hydroxymethyl benzoic acid is a principal metabolite of the phthalidyl moiety in man.</p>Formula:C8H8O3Purezza:98.36%Colore e forma:SolidPeso molecolare:152.15Larotrectinib sulfate
CAS:<p>Larotrectinib sulfate (LOXO-101 sulfate) is an oral active and specific ATP-competitive inhibitor of tropomyosin receptor kinases (TRK).</p>Formula:C21H22F2N6O2·H2O4SPurezza:98.62% - 99.76%Colore e forma:SolidPeso molecolare:526.51Aplidine
CAS:<p>Aplidine possesses antiviral activity against SARS-CoV-2(IC90 = 0.88 nM).</p>Formula:C57H87N7O15Purezza:99.86%Colore e forma:SolidPeso molecolare:1110.34Persicogenin
CAS:<p>Persicogenin has anticancer, antimutagenic, and antileishmanial activities, it can inhibit the proliferation of mouse tsFT210 cancer cells, it mainly inhibits</p>Formula:C17H16O6Purezza:97.8% - 98.47%Colore e forma:SolidPeso molecolare:316.31Isoacteoside
CAS:<p>Isoacteoside has the anti-inflammatory effect, mediated by action on caspase-1, mitogen-activated protein kinases (c-Jun N-terminal kinase, p38, extracellular</p>Formula:C29H36O15Purezza:97.71% - 99.48%Colore e forma:SolidPeso molecolare:624.59Hydroxy-Dynasore
CAS:<p>Hydroxy-Dynasore (Dyngo-4a) , a effective dynamin inhibitor, inhibits withDynI (brain), DynI (rec), and DynII (rec) of IC50 of 0.38 μM, 1.1 μM, and 2.3 μM,</p>Formula:C18H14N2O5Purezza:97.60% - >99.99%Colore e forma:SolidPeso molecolare:338.319-Ethyladenine
CAS:<p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>Formula:C7H9N5Purezza:99.35% - 99.41%Colore e forma:SolidPeso molecolare:163.182-O-α-D-Glucopyranosyl-L-ascorbic Acid
CAS:<p>2-O-α-D-Glucopyranosyl-L-ascorbic Acid (ASCORBYL GLUCOSIDE) is a glucoside derivative of ascorbic acid that can be enzymatically hydrolysed to ascorbic acid.</p>Formula:C12H18O11Purezza:98.56% - 99.73%Colore e forma:SolidPeso molecolare:338.26COG 133 Acetate
<p>COG 133 Acetate, (C97H181N37O19) is a peptide with the sequence Ac-Leu-Arg-Val-Arg-Leu-Ala-Ser-His-Leu-Arg-Lys-Leu-Arg-Lys-Arg-Leu-Leu-amide.</p>Formula:C99H185N37O21Purezza:99.73%Colore e forma:SolidPeso molecolare:2229.76Arabinose
CAS:<p>Arabinose, a pentose sugar, is found in feces, cytoplasm, eukaryotes, sweet basil, and tamarind.</p>Formula:C5H10O5Purezza:98.71% - 99.93%Colore e forma:Monoclinic Needles Or Prisms White Fine Crystalline PowderPeso molecolare:150.13GSK-114
CAS:<p>GSK-114, a TNNI3K inhibitor with a 25 nM IC50, is 40x more selective than B-Raf and good for in vivo studies.</p>Formula:C19H23N5O4SPurezza:99.51%Colore e forma:SolidPeso molecolare:417.483'-Deoxyguanosine
CAS:<p>3'-Deoxyguanosine is a ligand that can be complexed with enzymes, such as purine nucleoside phosphorylase, and receptors.</p>Formula:C10H13N5O4Purezza:98.85% - 98.96%Colore e forma:SolidPeso molecolare:267.24Parishin
CAS:<p>Parishin (Parishin A) A is isolated from the rhizomes of Gastrodia elata. It has good neuroprotective effects against brain disorders.</p>Formula:C45H56O25Purezza:98.56% - 99.58%Colore e forma:SolidPeso molecolare:996.91ZM-447439
CAS:<p>ZM 447439 selectively inhibits Aurora A/B (IC50: 110/130 nM); 8x less effective on MEK1, Src, Lck; minimal impact on CDK1/2/4, Plk1, Chk1.</p>Formula:C29H31N5O4Purezza:99.11% - 99.59%Colore e forma:Pale Yellow SolidPeso molecolare:513.59PRX-07034 hydrochloride
CAS:<p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>Formula:C21H29Cl2N3O4SPurezza:98.5%Colore e forma:SolidPeso molecolare:490.44CPI-444
CAS:<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Formula:C20H21N7O3Purezza:98.78%Colore e forma:SolidPeso molecolare:407.434-Acetamidobenzenesulfonamide
CAS:<p>4-Acetamidobenzenesulfonamide used in proteomics research and is an anti-infective agent</p>Formula:C8H10N2O3SPurezza:99.86%Colore e forma:Solid Solid CrystallinePeso molecolare:214.24Isoxazole
CAS:<p>Isoxazole (1,2-oxazole) is the inhibitor of acetylcholinesterase (AChE). The ligands of Isoxazole bind to and inhibit the Sxc- antiporter.</p>Formula:C3H3NOPurezza:99.34%Colore e forma:Colorless LiquidPeso molecolare:69.06Imepitoin
CAS:<p>Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.</p>Formula:C13H14ClN3O2Purezza:99.82%Colore e forma:SolidPeso molecolare:279.72
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