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DPM-1001 trihydrochloride
DPM-1001 trihydrochloride: Potent PTP1B inhibitor, IC50 100 nM, oral, non-competitive, anti-diabetic.Formula:C35H60Cl3N3O3Colore e forma:SolidPeso molecolare:677.23Altretamine hydrochloride
CAS:Altretamine hydrochloride is an alkylating antineoplastic agent.Formula:C9H19ClN6Colore e forma:SolidPeso molecolare:246.74ATM-3507 trihydrochloride
CAS:ATM-3507 trihydrochloride, a potent inhibitor of tropomyosin, demonstrates inhibition concentration (IC50) values ranging from 3.83 to 6.84 μM across variousFormula:C37H49Cl3FN5O2Colore e forma:SolidPeso molecolare:721.17GS-441524
CAS:GS-441524 treatment of cats with naturally occurring feline infectious peritonitis.Formula:C12H13N5O4Purezza:98.78% - 99.75%Colore e forma:SolidPeso molecolare:291.26DSP-1053 benzenesulfonate
CAS:DSP-1053: Benzylpiperidine-based, potent SERT inhibitor (Ki=1.02nM), partial 5-HT1A receptor agonist (Ki=5.05nM), antidepressant.Formula:C32H38BrNO7SColore e forma:SolidPeso molecolare:660.62PF-06815345 hydrochloride
CAS:PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.Formula:C27H30Cl2FN9O4Colore e forma:SolidPeso molecolare:634.49Anti-inflammatory agent 7
<p>Anti-inflammatory Agent 7 suppresses proinflammatory cytokines by hindering the NF-κB/MAPK signaling pathway in both LPS-treated RAW 264.7 cells and mice.</p>Formula:C36H40N4O9Colore e forma:SolidPeso molecolare:672.72NK1 receptor antagonist 2
CAS:NK1 Receptor Antagonist 2, a compound targeting the NK1 receptor, holds potential for tinnitus and hearing loss research.Formula:C31H35F7N4O2Colore e forma:SolidPeso molecolare:628.62β2AR/M-receptor agonist-2
CAS:<p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>Formula:C36H49ClN4O7SColore e forma:SolidPeso molecolare:717.31PF-4348235 HCl
<p>PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).</p>Formula:C36H50Cl2N4O7SPurezza:98.81%Colore e forma:SolidPeso molecolare:753.78PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Formula:C36H51Cl3N4O7SPurezza:99.85%Colore e forma:SolidPeso molecolare:790.24PI3K/Akt/CREB activator 1
CAS:<p>PI3K/Akt/CREB activator 1 (AE-18) is an iNOS inhibitor that can be used to study vascular dementia and Parkinson's.</p>Formula:C19H15F4NO3Colore e forma:SolidPeso molecolare:381.32Antitrypanosomal agent 10
Antitrypanosomal agent 10, an antitrypanosomal compound, effectively inhibits Trypanosoma cruzi with an IC50 of 0.28 μM.Formula:C17H9F6N5OColore e forma:SolidPeso molecolare:413.28Antitrypanosomal agent 11
<p>Antitrypanosomal Agent 11 is a chemical compound effective against Trypanosoma cruzi, exhibiting an inhibition concentration (IC 50) of 0.23 μM.</p>Formula:C16H10F6N6OColore e forma:SolidPeso molecolare:416.28Gestrinone
CAS:Gestrinone (R 2323) 是一种合成类固醇激素,能够抑制平滑肌瘤(IC50:43.67 μM),有用于子宫内膜异位症的研究潜力。Formula:C21H24O2Purezza:99.21%Colore e forma:Light Yellow SolidPeso molecolare:308.41SARS-CoV-2/MERS Mpro-IN-1
<p>SARS-CoV-2/MERS Mpro-IN-1 is a potent inhibitor of the main proteases in SARS-CoV-2 and MERS, exhibiting IC50 values of 0.10 and 0.06 µM, respectively.</p>Formula:C30H36N4O7Colore e forma:SolidPeso molecolare:564.63SARS-CoV-2/MERS Mpro-IN-2
<p>SARS-CoV-2/MERS Mpro-IN-2 is a potent inhibitor of the main proteases of SARS-CoV-2 and MERS, demonstrating IC50 values of 0.21 and 0.07 µM, respectively.</p>Formula:C28H30Cl2N4O6Colore e forma:SolidPeso molecolare:589.473β-Hydroxy-hop-22(29)-ene
CAS:3β-Hydroxy-hop-22(29)-ene is a potent antiparasitic compound demonstrating moderate efficacy against Trypanosoma cruzi and Leishmania mexicana.Formula:C30H50OColore e forma:SolidPeso molecolare:426.72Antibacterial synergist 2
CAS:"Antibacterial Synergist 2 inhibits biofilms of S. enterica, S. aureus, P. aeruginosa, and C. albicans."Formula:C6H3Br3O2Colore e forma:SolidPeso molecolare:346.8erythro-Austrobailignan-6
CAS:Erythro-Austrobailignan-6: orally active, anti-cancer, inhibits DNA topoisomerases, induces apoptosis, boosts p38/JNK phosphorylation.Formula:C20H24O4Colore e forma:SolidPeso molecolare:328.4JBJ-09-063 hydrochloride
JBJ-09-063 hydrochloride: targeted EGFR inhibitor, effective for various mutations and TKI-resistant lung cancer models.Formula:C31H30ClFN4O3SColore e forma:SolidPeso molecolare:593.11DDO-2093 dihydrochloride
DDO-2093 dihydrochloride: potent MLL1-WDR5 inhibitor, IC50=8.6 nM, Kd=11.6 nM, antitumor.Formula:C29H39Cl3FN9O3Colore e forma:SolidPeso molecolare:687.04Anabasine
CAS:Anabasine ((S)-Anabasine) is from tobacco. Anabasine is a full agonist of nicotinic acetylcholine receptors (nAChRs) with insecticidal activity.Formula:C10H14N2Purezza:99.27%Colore e forma:Colorless Liquid Darkens On Exposure To Air White Fine Crystalline PowderPeso molecolare:162.23Romifidine hydrochloride
CAS:Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.Formula:C9H10BrClFN3Colore e forma:SolidPeso molecolare:294.55Teslexivir hydrochloride
CAS:Teslexivir (BTA074) HCl inhibits HPV 6/11 by blocking E1-E2 protein interaction, vital for DNA replication. Used in condyloma research.Formula:C35H37BrClN3O4Colore e forma:SolidPeso molecolare:679.04DYRKs-IN-1 hydrochloride
CAS:DYRKs-IN-1 HCl inhibits DYRK1A (5 nM IC50) & DYRK1B (8 nM IC50) with antitumor properties.Formula:C30H31Cl2N7O4Colore e forma:SolidPeso molecolare:624.52Cyclic-di-GMP diammonium
CAS:C-di-GMP diammonium activates STING, regulates biofilms, motility, and virulence in bacteria.Formula:C20H30N12O14P2Colore e forma:SolidPeso molecolare:724.47CBB1007 trihydrochloride
CBB1007 trihydrochloride inhibits hLSD1 selectively (IC50=5.27μM), blocks demethylation of H3K4Me2/Me, and activates certain genes.Formula:C27H37Cl3N8O4Colore e forma:SolidPeso molecolare:643.99Fomepizole hydrochloride
CAS:Fomepizole hydrochloride inhibits CYP2E1 and alcohol dehydrogenase, blocking toxic metabolites, and treats methanol/ethylene glycol poisoning.Formula:C4H7ClN2Colore e forma:SolidPeso molecolare:118.56Bicuculline methobromide
CAS:Bicuculline methobromide: GABAA antagonist, IC50=3μM, induces convulsions, used in epilepsy research.Formula:C21H20BrNO6Colore e forma:SolidPeso molecolare:462.29Ladostigil hydrochloride
CAS:Ladostigil hydrochloride: oral dual cholinesterase and MAO-B/AChE inhibitor; IC50s: 37.1 & 31.8 μM; potential for depression and Alzheimer's research.Formula:C16H21ClN2O2Colore e forma:SolidPeso molecolare:308.8MRS2768 tetrasodium salt
CAS:MRS2768 tetrasodium: a P2Y2 agonist; offers cardioprotection against ischemia.Formula:C15H16N2Na4O18P4Colore e forma:SolidPeso molecolare:728.14BMS-823778 hydrochloride
CAS:<p>BMS-823778 hydrochloride is a potent, selective, and orally active inhibitor of 11β-HSD1 (11β-Hydroxysteroid Dehydrogenase Type 1), demonstrating an IC50 (half</p>Formula:C18H19Cl2N3OColore e forma:SolidPeso molecolare:364.27AnaMorelin hydrochloride
CAS:AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).Formula:C31H43ClN6O3Purezza:99.18% - ≥98%Colore e forma:SolidPeso molecolare:583.164aα,7α,7aα-Nepetalactone
CAS:4aα,7α,7aα-Nepetalactone is a natural terpenoid lactone exhibiting antibacterial activity against E. coli, P. aeruginosa, S. aureus, and others.Formula:C10H14O2Purezza:99.94%Colore e forma:SolidPeso molecolare:166.22RORγt inverse agonist 14
CAS:RORγt inverse agonist 14 (8e) is a potent, selective, and orally active compound with an EC50 of 2.5 nM, exhibiting anti-inflammatory activity.Formula:C26H26F8N2O6S2Purezza:98%Colore e forma:SolidPeso molecolare:678.61AXC-715 trihydrochloride
CAS:AXC-715 trihydrochloride is a TLR7/8 agonist used to make PD-L1 adjuvanted antibody immunocouplings.Formula:C18H28Cl3N5Purezza:99.87%Colore e forma:SolidPeso molecolare:420.81RORγt inverse agonist 26
CAS:RORγt inverse agonist 26, a potent reverse agonist of RORγt, effectively modulates Th17 cell differentiation and suppresses IL-17 production.Formula:C27H21F7N2O5SColore e forma:SolidPeso molecolare:618.52BRM/BRG1 ATP Inhibitor-3
CAS:<p>BRM/BRG1 ATP Inhibitor-3 targets BRM/BRG1 (IC50: 10.4/19.3 nM) for cancer/BAF disorder research.</p>Formula:C26H25N5O2S2Colore e forma:SolidPeso molecolare:503.64BRM/BRG1 ATP Inhibitor-4
CAS:<p>BRM/BRG1 ATP Inhibitor-4, a potent inhibitor of BRG1/BRM, is utilized in the research of cancers and BAF complex-related disorders.</p>Formula:C25H32N6O3SColore e forma:SolidPeso molecolare:496.623-Chlorogentisyl alcohol
CAS:3-Chlorogentisyl alcohol: E. coli β-glucuronidase inhibitor (IC50=0.74µM, Ki=0.58µM), antiproliferative, for anti-cancer/inflammatory research.Formula:C7H7ClO3Colore e forma:SolidPeso molecolare:174.58Antileishmanial agent-13
CAS:Antileishmanial agent-13, a quinoline-isatin hybrid, targets L. Major with IC50s of 0.604 μM (promastigote) and 0.508 μM (amastigote).Formula:C17H10BrClN4OColore e forma:SolidPeso molecolare:401.64Metallo-β-lactamase-IN-9
CAS:Metallo-β-lactamase-IN-9 (Compound 23) serves as a broad-spectrum inhibitor of metallo-beta-lactamases (MBL), exhibiting inhibition constants (IC50) of 35 nMFormula:C13H12N6O3SColore e forma:SolidPeso molecolare:332.34Antituberculosis agent-6
CAS:<p>Antituberculosis agent-6: potent against M. tuberculosis (MIC 3.49 μM), antifungal (MIC 62.5 μM), high GI absorption.</p>Formula:C27H20F2N2O3Colore e forma:SolidPeso molecolare:458.46Antituberculosis agent-8
CAS:Antituberculosis agent-8: MIC 3.53 μM vs M. tuberculosis, antifungal MIC 62.50 μM vs A. niger.Formula:C25H19F3N2O3Colore e forma:SolidPeso molecolare:452.43Eltrombopag methyl ester
CAS:Eltrombopag methyl ester, a Tpo receptor agonist derivative, boosts platelet production for thrombocytopenia research.Formula:C26H24N4O4Colore e forma:SolidPeso molecolare:456.49Antitrypanosomal agent 9
CAS:Agent 9 inhibits T. b. brucei (IC50: 1.15 μM), used in HAT research.Formula:C22H27NO3Colore e forma:SolidPeso molecolare:353.45TAK-960 dihydrochloride
<p>TAK-960 dihydrochloride: oral PLK1 inhibitor, IC50 0.8 nM; also Hinders PLK2 and PLK3 (IC50s 16.9/50.2 nM); curbs cancer cell growth.</p>Formula:C27H36Cl2F3N7O3Colore e forma:SolidPeso molecolare:634.52WYE-687 dihydrochloride
CAS:WYE-687 dihydrochloride is an mTOR inhibitor with IC50 of 7 nM, also targeting PI3Kα (81 nM) and PI3Kγ (3.11 μM).Formula:C28H34Cl2N8O3Colore e forma:SolidPeso molecolare:601.53Glibenclamide potassium
CAS:<p>Glibenclamide potassium, a more soluble form of Glibenclamide, exists as anhydrous and hydrate salts.</p>Formula:C23H27ClKN3O5SColore e forma:SolidPeso molecolare:532.09IACS-9571 hydrochloride
CAS:IACS-9571 hydrochloride: potent TRIM24/BRPF1 inhibitor; IC50 = 8 nM (TRIM24); Kd = 31 nM (TRIM24), 14 nM (BRPF1).Formula:C32H43ClN4O8SColore e forma:SolidPeso molecolare:679.22EG01377 dihydrochloride
<p>EG01377 dihydrochloride inhibits NRP1 selectively with Kd 1.32 μM, IC50 609 nM, and has antiangiogenic and antitumor properties.</p>Formula:C26H32Cl2N6O6S2Colore e forma:SolidPeso molecolare:659.6CM-579 trihydrochloride
CM-579 trihydrochloride: reversible G9a/DNMT inhibitor with IC50s 16 nM (G9a) & 32 nM (DNMT); potent against various cancer cells.Formula:C29H43Cl3N4O3Colore e forma:SolidPeso molecolare:602.04Flurandrenolone Acetate
CAS:Flurandrenolone Acetate, a synthetic glucocorticoid derived from Flurandrenolide, is used to study skin issues like eczema and psoriasis.Formula:C26H35FO7Colore e forma:SolidPeso molecolare:478.55PBT434 methanesulfonate
CAS:<p>PBT434 methanesulfonate is an oral α-synuclein aggregation inhibitor, crosses the blood-brain barrier, and may help treat Parkinson's.</p>Formula:C13H17Cl2N3O5SColore e forma:SolidPeso molecolare:398.26Caspase-9 Inhibitor III
CAS:Caspase-9 Inhibitor III (Ac-LEHD-cmk) blocks caspase-9, protects against ischemic heart damage.Formula:C24H35ClN6O9Colore e forma:SolidPeso molecolare:587.02Ebaresdax hydrochloride
CAS:Ebaresdax hydrochloride has analgesic activity and is used in the study of painful diabetic neuropathy caused by type I or type II diabetes.Formula:C12H15ClN2O3SPurezza:99.11% - 99.77%Colore e forma:SolidPeso molecolare:302.78(+)-Dihydrocalanolide A
CAS:DHCal A (NSC 678323) is an oral nonnucleoside Reverse Transcriptase inhibitor for HIV research.Formula:C22H28O5Colore e forma:SolidPeso molecolare:372.45Glucokinase activator 3
CAS:Glucokinase activator 3: potent GK activator, AC50=38 nM, potential for type 2 diabetes research.Formula:C26H33N2O9PS2Colore e forma:SolidPeso molecolare:612.65LC kinetic stabilizer-1
CAS:LC kinetic stabilizer-1: potent, selective for amyloid light chains, EC50: 140 nM (WIL-FL*), 74.1 nM (WIL-FL*T46L/F49Y).Formula:C27H31N5O3Colore e forma:SolidPeso molecolare:473.57LC kinetic stabilizer-2
CAS:LC Kinetic Stabilizer-2 is a powerful stabilizer for amyloidogenic immunoglobulin light chains (LC), demonstrating significant efficacy with an EC50 of 24 nM.Formula:C28H31N3O3Colore e forma:SolidPeso molecolare:457.56Type II TRK inhibitor 1
CAS:Type II TRK Inhibitor 1 is a potent inhibitor targeting multiple tropomyosin receptor kinase (TRK) fusion protein variants as well as the wild type.Formula:C35H33F3N8O3Purezza:98%Colore e forma:SolidPeso molecolare:670.68Mitochondria degrader-1
CAS:Mitochondria degrader-1, a potent autophagy inducer, aids in neurodegenerative, cancer, and aging disease research.Formula:C33H49ClFN7O8SColore e forma:SolidPeso molecolare:758.3Tilpisertib fosmecarbil
CAS:Tilpisertib fosmecarbil is a potent inhibitor of serine/threonine kinases with anti-inflammatory properties.Formula:C35H36ClN8O7PColore e forma:SolidPeso molecolare:747.14S1P5 receptor agonist-1
CAS:S1P5 Receptor Agonist-1 (example 6) is a highly potent and selective agonist for the S1P5 receptor, exhibiting an EC50 value of 20 nM.Formula:C20H24F3NO3Colore e forma:SolidPeso molecolare:383.4VU6036720 hydrochloride
VU6036720 hydrochloride inhibits Kir4.1/5.1. channels with 0.24 μM IC50; used in brain and kidney research.Formula:C20H23Cl2FN4O2SColore e forma:SolidPeso molecolare:473.39Cathepsin K inhibitor 3
CAS:Cathepsin K inhibitor 3: Selective, IC50 of 0.5 nM, good pharmacokinetics, potential for OA research.Formula:C30H31FN4O4SColore e forma:SolidPeso molecolare:562.65Mtb-cyt-bd oxidase-IN-1
<p>Mtb-cyt-bd oxidase-IN-1, a Mycobacterium tuberculosis inhibitor, IC50: 0.13 μM, useful for TB research.</p>Formula:C26H35NO2Colore e forma:SolidPeso molecolare:393.56Mtb-cyt-bd oxidase-IN-3
Mtb-cyt-bd oxidase-IN-3 inhibits M. tuberculosis growth, IC50 0.36 μM, MIC 32 μM, for TB research.Formula:C26H35NO2Colore e forma:SolidPeso molecolare:393.56Mtb-cyt-bd oxidase-IN-4
<p>Mtb-cyt-bd oxidase inhibitor; IC50=0.25μM; MIC=8μM against Mycobacterium tuberculosis; for TB research.</p>Formula:C25H32FNOColore e forma:SolidPeso molecolare:381.53Mtb-cyt-bd oxidase-IN-6
CAS:Mtb-cyt-bd oxidase-IN-6, a potent inhibitor of Mycobacterium tuberculosis (Mtb) cytochrome bd (cyt-bd) oxidase (MtbCyt-bd Oxidase), exhibits an inhibitoryFormula:C20H27NOColore e forma:SolidPeso molecolare:297.43Antibacterial agent 124
CAS:Antibacterial agent 124 inhibits Sa ProRS with an IC50 of 0.18 μM.Formula:C16H17ClFN3O2Colore e forma:SolidPeso molecolare:337.78Antibacterial agent 126
Antibacterial agent 126 combats biofilm, disrupts membranes, and boosts ROS/RNS to prevent drug resistance.Formula:C21H24NO6PColore e forma:SolidPeso molecolare:417.39Mtb-cyt-bd oxidase-IN-7
Mtb-cyt-bd oxidase-IN-7 inhibits Cyt-bd with 4.17 μM affinity and has anti-tuberculosis properties.Formula:C18H14F3NO2Colore e forma:SolidPeso molecolare:333.3Mycobacterial Zmp1-IN-1
Zmp1-IN-1: An inhibitor of mycobacterial Zmp1 with dose-dependent anti-tuberculosis effects.Formula:C26H27N3O7SColore e forma:SolidPeso molecolare:525.57Antibacterial agent 131
Antibacterial agent 131 is a compound with antibacterial properties.Formula:C24H17ClN4OSPurezza:99.63%Colore e forma:SolidPeso molecolare:444.94Antibacterial agent 132
CAS:<p>Antibacterial agent 132 showed antimicrobial activity against C.</p>Formula:C24H17ClN4OSPurezza:98%Colore e forma:SolidPeso molecolare:444.94SARS-CoV-2 3CLpro-IN-10
SARS-CoV-2 3CLpro-IN-10(5d) inhibits 3CL protease: 190 nM (SARS-CoV-2), 790 nM (SARS-CoV-1), 70 nM (MERS-CoV), and has broad-spectrum antiviral effects.Formula:C24H33FN3NaO8SColore e forma:SolidPeso molecolare:565.59SARS-CoV-2 3CLpro-IN-11
SARS-CoV-2 3CLpro-IN-11, potent inhibitor: IC50 of 140nM for 3CLpro; 240nM for SARS-CoV-1; 70nM for MERS-CoV; broad-spectrum antiviral.Formula:C25H36N3NaO9SColore e forma:SolidPeso molecolare:577.62α-Synuclein inhibitor 8
CAS:α-Synuclein inhibitor 8 effectively impedes α-Synuclein aggregation and disaggregation with an IC50 of 2.5 µM, demonstrating substantial reduction in neuronalFormula:C24H20N2O6Colore e forma:SolidPeso molecolare:432.43Caspase-3/7 activator 2
Caspase-3/7 activator 2 triggers apoptosis with tumor selectivity and anti-proliferative properties.Formula:C32H34N2O7Colore e forma:SolidPeso molecolare:558.62Caspase-3/7 activator 3
Caspase-3/7 activator 3 triggers apoptosis with tumor selectivity and anti-proliferative effects.Formula:C24H27NO5Colore e forma:SolidPeso molecolare:409.47CEP-28122 mesylate salt
<p>CEP-28122 mesylate, a diaminopyrimidine, selectively inhibits ALK with IC50 of 1.9 nM and exhibits antitumor effects.</p>Formula:C29H39ClN6O6SColore e forma:SolidPeso molecolare:635.17Trandolaprilate hydrate
CAS:Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.Formula:C22H32N2O6Colore e forma:SolidPeso molecolare:420.5Lewis y tetrasaccharide
CAS:<p>Lewis Y tetrasaccharide, a derivative of Lewis X, is an antigen linked to ovarian cancer metastasis and bad prognosis.</p>Formula:C26H45NO19Colore e forma:SolidPeso molecolare:675.63AZ13705339 hemihydrate
AZ13705339 hemihydrate: potent PAK1 inhibitor (IC50: 0.33 nM), also binds PAK1/2 (Kd: 0.28/0.32 nM), for cancer research.Formula:C33H36FN7O3SH2OColore e forma:SolidPeso molecolare:638.77R 59-022 hydrochloride
CAS:<p>R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.</p>Formula:C27H27ClFN3OSPurezza:97.7%Colore e forma:SolidPeso molecolare:496.04Antiarrhythmic agent-1
CAS:Antiarrhythmic agent-1 (example I), functioning as an antiarrhythmic agent and an IKr potassium channel blocker (IC 50 <1 μM), effectively inhibits cardiacFormula:C25H27N3O4SColore e forma:SolidPeso molecolare:465.56Lagociclovir valactate
CAS:Lagociclovir valactate is a prodrug of Lagociclovir . Lagociclovir valactate is an orally active anti- HBV agent [1] .Formula:C18H25FN6O6Colore e forma:SolidPeso molecolare:440.43(-)-15-Deoxyspergualin
CAS:(-)-15-Deoxyspergualin is a potent antitumor agent that demonstrates significant inhibition against mouse leukemia L-1210.Formula:C17H37N7O3Colore e forma:SolidPeso molecolare:387.52Cyclopropenone probe 1
<p>Cyclopropenone probe 1 targets and covalently modifies triple-negative breast cancer enzyme GSTP1 at its active site.</p>Formula:C12H8O2Colore e forma:SolidPeso molecolare:184.19Antibacterial agent 19
CAS:Antibacterial agent 19 targets K. pneumoniae and multi-resistant S. aureus with MICs: 0.022 and 0.045 mg/mL.Formula:C16H16F2N2O4Colore e forma:SolidPeso molecolare:338.31Antibacterial agent 64
CAS:Potent antibacterial, YycG inhibitor with 6.1 µM IC50. Synergistic with ampicillin against biofilm bacteria.Formula:C29H20ClN3O6S2Colore e forma:SolidPeso molecolare:606.07KRAS G12C inhibitor 28
CAS:KRAS G12C Inhibitor 28 is a compound that effectively inhibits the KRAS G12C mutation, exhibiting potent antitumor effects with an inhibitory concentration (Formula:C33H36F2N5O4PColore e forma:SolidPeso molecolare:635.64KRAS G12C inhibitor 32
CAS:KRAS G12C Inhibitor 32, an eight-membered heterocyclic compound with nitrogen, acts as a potent inhibitor of KRAS G12C [1].Formula:C29H30Cl3FN6O3Purezza:98%Colore e forma:SolidPeso molecolare:635.94KRAS G12C inhibitor 45
CAS:KRAS G12C inhibitor 45 is a potent KRAS G12C inhibitor .Formula:C32H33F2N5O5SColore e forma:SolidPeso molecolare:637.7Plasma kallikrein-IN-2
Plasma kallikrein-IN-2: PKal inhibitor, IC50=0.1 nM. Used in angioedema, diabetic eye disease research.Formula:C28H24ClF3N8O3Colore e forma:SolidPeso molecolare:612.99KRAS G12C inhibitor 35
CAS:<p>KRAS G12C inhibitor 35 targets KRAS G12C in cancer research (CN112920183A, compound 3).</p>Formula:C31H27ClF2N6O3Colore e forma:SolidPeso molecolare:605.035-Amino-2-chloropyridine
CAS:<p>5-Amino-2-chloropyridine is Pyridine intermediates</p>Formula:C5H5ClN2Purezza:>99.99%Colore e forma:SoildPeso molecolare:128.5600KRAS G12C inhibitor 37
CAS:KRAS G12C inhibitor 37 targets a key signaling protein, showing promise for cancer research involving KRAS G12C.Formula:C35H39F3N8O2Colore e forma:SolidPeso molecolare:660.73

