6-Bromoimidazo[1,2-a]pyrazine
CAS: 912773-24-1
Ref. 3D-FB140690
5g | Discontinued | ||
10g | Discontinued | ||
25g | Discontinued | ||
50g | Discontinued | ||
100g | Discontinued |
Product Information
- 6-Bromoimidazo[1,2-A]Pyrazine
6-Bromoimidazo[1,2-a]pyrazine is a potent inhibitor of the enzyme phosphatidylinositol-3 kinase (PI3K). It has been used in drug development and has shown to be a reversible inhibitor of PI3K. 6-Bromoimidazo[1,2-a]pyrazine binds to the ATP site on the enzyme and prevents phosphorylation by blocking access to this site. The binding of 6-bromoimidazo[1,2-a]pyrazine is reversible due to its ability to dissociate when ATP is removed. This drug has been shown to inhibit the growth of cancer cells in vitro.