Hydroxy vardenafil

CAS: 224785-98-2

Ref. 3D-FH24158

Product Information

• Name: Hydroxy vardenafil
• Synonyms: 2-[2-Ethoxy-5-[[4-(2-hydroxyethyl)-1-piperazinyl]sulfonyl]phenyl]-5-methyl-7-propylimidazo[5,1-f][1,2,4]triazin-4(1H)-one4-[[3-(1,4 -Dihydro-5-methyl-4-oxo-7-propylimidazo[5,1-f][1,2,4]triazin-2-yl)-4-ethoxyphenyl]sulfonyl]-1-piperazineethanol, Imidazo[5,1-f][1,2,4]triazin-4(1H)-one, 2-[2-ethoxy-5-[[4-(2-hydroxyethyl)-1-piperazinyl]sulfonyl]phenyl]-5-methyl-7-propyl-, Hydroxyvardenafil, 2-[2-Ethoxy-5-[[4-(2-hydroxyethyl)-1-piperazinyl]sulfonyl]phenyl]-5-methyl-7-propylimidazo[5,1-f][1,2,4]triazin-4(1H)-one, 1-Piperazineethanol, 4-[[3-(1,4-dihydro-5-methyl-4-oxo-7-propylimidazo[5,1-f][1,2,4]triazin-2-yl)-4-ethoxyphenyl]sulfonyl]-

Description

Hydroxy vardenafil is a dietary supplement that belongs to the group of sildenafil analogs. It is structurally similar to sildenafil and inhibits phosphodiesterase type-5 (PDE-5) in human liver cells. The hydroxy group at position 3 of vardenafil is responsible for its stability and long half-life, which allows it to be administered as a single dose. Hydroxy vardenafil has been shown to have a matrix effect on the plasma concentration of sildenafil and other PDE-5 inhibitors. Hydroxy vardenafil was found to be more potent than sildenafil in inhibiting PDE-5 activity in human liver cells.

• Brand: Biosynth

Chemical properties

• Molecular weight: 504.6 g/mol
• Formula: C₂₃H₃₂N₆O₅S
• Purity: Min. 95%
• InChI: InChI=1S/C23H32N6O5S/c1-4-6-20-24-16(3)21-23(31)25-22(26-29(20)21)18-15-17(7-8-19(18)34-5-2)35(32,33)28-11-9-27(10-12-28)13-14-30/h7-8,15,30H,4-6,9-14H2,1-3H3,(H,25,26,31)
• InChI key: InChIKey=KZFHUILKKFVOMB-UHFFFAOYSA-N
• SMILES: CCCc1nc(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCN(CCO)CC4)ccc3OCC)nn12