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Sitaxsentan
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Sitaxsentan

CAS: 184036-34-8

Ref. 3D-JHA03634

1mg
148.00 €
10mg
558.00 €
Estimated delivery in United States, on Wednesday 8 Jan 2025

Product Information

Name:
Sitaxsentan
Synonyms:
  • 3-Thiophenesulfonamide, N-(4-chloro-3-methyl-5-isoxazolyl)-2-((6-methyl-1,3-benzodioxol-5-yl)acetyl)-
  • 3-Thiophenesulfonamide, N-(4-chloro-3-methyl-5-isoxazolyl)-2-[2-(6-methyl-1,3-benzodioxol-5-yl)acetyl]-
  • Ipi 1040
  • N-(4-Chloro-3-methyl-1,2-oxazol-5-yl)-2-[2-(6-methyl-2H-1,3-benzodioxol-5-yl)acetyl]thiophene-3-sulfonamide
  • N-(4-Chloro-3-methyl-5-isoxazolyl)-2-((2-methyl-4,5-methylenedioxyphenyl)acetyl)thiophene-3-sulfonamide
  • N-(4-Chloro-3-methyl-5-isoxazolyl)-2-((3,4-(methylenedioxy)-6-methylphenyl)acetyl)-3-thiophenesulfonamide
  • N-(4-Chloro-3-methyl-5-isoxazolyl)-2-[2-(6-methyl-1,3-benzodioxol-5-yl)acetyl]-3-thiophenesulfonamide
  • N-(4-chloro-3-methyl-2H-oxazol-5-yl)-2-[2-(6-methyl-1,3-benzodioxol-5-yl)acetyl]thiophene-3-sulfonamide
  • Sitax
  • Sitaxentan
  • See more synonyms
  • Tbc 11251
Description:

Sitaxsentan is a natriuretic peptide receptor antagonist that blocks the binding of endothelin-1 to its receptors. It has been shown to have efficacy in animal models of pulmonary hypertension, and clinical trials have also been conducted in humans. In vitro assays have shown that sitaxsentan inhibits the production of endothelin, which may be due to its ability to inhibit toll-like receptor 4 signaling. Sitaxsentan has drug interactions with other drugs that are substrates for the P-glycoprotein transporter, such as verapamil, diltiazem, and chloramphenicol. The drug is not metabolized by cytochrome P450 enzymes and does not interact with the renal organic anion transporter (OAT).

Notice:
Our products are intended for lab use only. For any other use, please contact us.
Brand:
Biosynth
Long term storage:
Notes:

Chemical properties

Molecular weight:
454.9 g/mol
Formula:
C18H15ClN2O6S2
Purity:
Min. 95%
Color/Form:
Powder
MDL:
Melting point:
Boiling point:
Flash point:
Density:
Concentration:
EINECS:
Merck:
HS code:

Hazard Info

UN Number:
EQ:
Class:
H Statements:
P Statements:
Forbidden to fly:
Hazard Info:
Packing Group:
LQ:

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