1-[4-[4-Morpholin-4-yl-6-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-1,3,5-triazin-2-yl]phenyl]-3-pyridin-4-ylurea, hydrochloride
CAS: 1463510-35-1
Ref. 3D-NIC51035
1mg | Discontinued | ||
5mg | Discontinued | ||
10mg | Discontinued | ||
25mg | Discontinued | ||
50mg | Discontinued |
Product Information
1-[4-[4-Morpholin-4-yl-6-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-1,3,5-triazin-2-yl]phenyl]-3-pyridin-4-ylurea is a peptide inhibitor that binds to the ATP binding site of protein kinase C (PKC) and blocks its catalytic activity. 1-[4-[4-Morpholin-4-yl-6-(3 -oxa -8 -azabicyclo[3.2.1]octan -8 -yl)-1,3,5 -triazin -2 -yl]phenyl]-3 -pyridin -4 -ylurea has been shown to be an activator of PKCδ with IC50 of 0.5 μM and inhibits PKC γ with IC