Oclacitinib Maleate
CAS: 1640292-55-2
Ref. 3D-QQC29255
5mg | Discontinued | ||
10mg | Discontinued | ||
25mg | Discontinued | ||
50mg | Discontinued | ||
100mg | Discontinued |
Product Information
Oclacitinib Maleate is an orally-bioavailable small molecule drug candidate that inhibits the activity of the protein tyrosine kinase, which is a key signaling molecule in many cancers. Studies have shown that oclacitinib binds to the phosphate group on the ATP-binding site of the enzyme, preventing it from binding to its receptor. Oclacitinib has been shown to be safe and well tolerated for long-term use in diabetic patients. This drug has also been shown to inhibit PDL1 expression and inhibit insulin-like growth factor 1 (IGF1).