Naloxone Benzoylhydrazone

CAS: 119630-94-3

Ref. 3D-UEA63094

Product Information

• Name: Naloxone Benzoylhydrazone
• Synonyms: Benzoic acid, 2-[(5α)-4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]hydrazide, Benzoic acid, [(5α)-4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]hydrazide, N'-[(5β,6E)-3,14-dihydroxy-17-(prop-2-en-1-yl)-4,5-epoxymorphinan-6-ylidene]benzohydrazide, Naloxone Benzolyhydrazone K3 Opioid Rece Ptor Ag, [(5alpha)-4,5-Epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-yliden]benzoic acid hydrazide, [(5Α)-4,5-Epoxy-3,14-Dihydroxy-17-(2-Propenyl)Morphinan-6-Ylidene]Hydrazide Benzoic Acid
• CAS: 119630-94-3

Description

Naloxone benzoylhydrazone is a potent opioid antagonist that is used to reverse respiratory depression caused by opioid overdose. It is a benzoylhydrazone derivative of naloxone and has been shown to be highly potent, with an affinity for the kappa-opioid receptor that is 10x greater than its affinity for the mu-opioid receptor. Naloxone benzoylhydrazone also antagonizes δ-opioid receptors and dopamine receptors, which may contribute to its analgesic effects. This drug has been studied in biological studies and has shown efficacy in animal models of chronic pain relief.

• Brand: Biosynth

Chemical properties

• Molecular weight: 445.51 g/mol
• Formula: C₂₆H₂₇N₃O₄
• Purity: Min. 95%