Product Information
Name:
ERK5-IN-1
Synonyms:
- 11-Cyclopentyl-2-[[2-ethoxy-4-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one
Description:
Applications ERK5-IN-1 is a potent selective ERK5 inhibitor, inhibiting EGFR-induced ERK5 autophosphorylation and ERK5 enzymatic activity. Orally bioavailable.
References Deng, X. et al. Eur. J. med. Chem., 70, 758 (2013); Elkins, J. et al.: J. Med. Chem., 56, 4413 (2013);
Notice:
Our products are intended for lab use only. For any other use, please contact us.
Brand:
TRC
Long term storage:
Notes:
Chemical properties
Molecular weight:
638.8
Formula:
C38H46N8O3
Color/Form:
Yellow to Dark Yellow Solid
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