Pirenzepine-d10 Dihydrochloride

CAS: 29868-97-1

Ref. TR-P508503

Product Information

• Name: Pirenzepine-d10 Dihydrochloride
• Synonyms: 5,11-Dihydro-11-[2-(4-methyl-1-piperazinyl-d10)acetyl]-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one Dihydrochloride, Duogastral-d10 Dihydrochloride, Durapirenz-d10 Dihydrochloride, Gasteril-d10 Dihydrochloride, Gastrozepin-d10 Dihydrochloride, Leblon-d10 Dihydrochloride, Maghen-d10 Dihydrochloride, Renzepin-d10 Dihydrochloride, Tabe-d10 Dihydrochloride, 11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one dihydrochloride, 11-[2-(4-methylpiperazin-1-yl)acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one hydrate hydrochloride, 5,11-Dihydro-11-((4-methylpiperazin-1-yl)acetyl)-6H-pyrido(2,3-b)-(1,4)benzodiazepin-6-one dihydrochloride, 5,11-Dihydro-11-[(4-methyl-1-piperazinyl)acetyl]-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one dihydrochloride, 6H-Pyrido[2,3-b][1,4]benzodiazepin-6-one, 5,11-dihydro-11-[(4-methyl-1-piperazinyl)acetyl]-, dihydrochloride, 6H-Pyrido[2,3-b][1,4]benzodiazepin-6-one, 5,11-dihydro-11-[2-(4-methyl-1-piperazinyl)acetyl]-, hydrochloride (1:2), Duogastral, Durapirenz, Gasteril, Gastricur, Gastrozepin, L-S 519, LS 519Cl₂, LS 59Cl2, Leblon, Maghen, Pirenzepine HCL, Pirenzepine Hcl Hydrate, Pirenzepine Hydrochloride, Renzepin, Ulcosan, Ulcuforton

Description

Applications Pirenzepine-d10 Dihydrochloride is an analogue of Pirenzepine (P508500), an antiucerative agent that works by inhibiting tricyclic gastric-acid secretion.
References Fliri, A . F., et al.: J. Med. Chem., 52, 8038 (2009); Eberlein, W., et al.: Arzneimittel-Forsch., 27, 356 (1977), Hellerr, G., et al.: Verh. Deut. Ges. Inn. Med., 84, 991 (1978), Carmine, A.A., et al.: Drugs, 30,85 (1985), El-Obeid, H.A., et al.: Anal. Profiles Drug Subs., 16, 445 (1987), Homon, C.A., et al.: Ther. Drug Monit., 9, 236 (1987),

• Brand: TRC

Chemical properties

• Molecular weight: 435.39
• Formula: C₁₉H₁₂D₁₁Cl₂N₅O₂
• Color/Form: Neat
• InChI: InChI=1S/C19H21N5O2.2ClH/c1-22-9-11-23(12-10-22)13-17(25)24-16-7-3-2-5-14(16)19(26)21-15-6-4-8-20-18(15)24;;/h2-8H,9-13H2,1H3,(H,21,26);2*1H/i1D3,9D2,10D2,11D2,12D2