Triptorelin Acetate

CAS: 140194-24-7

Ref. TR-T815800

Product Information

• Name: Triptorelin Acetate
• Synonyms: Luteinizing hormone-releasing factor (swine), 6-D-tryptophan-, acetate (1:1), Luteinizing hormone-releasing factor (pig), 6-D-tryptophan-, monoacetate (salt), Luteinizing hormone-releasing factor (swine), 6-D-tryptophan-, monoacetate (salt) (9CI), BIM 21003C, Decapeptyl-Depot, OvuGel, 5-Oxo-L-prolyl-L-histidyl-L-tryptophyl-L-seryl-L-tyrosyl-D-tryptophyl-L-leucyl-L-arginyl-L-prolylglycinamide, Glycinamide, 5-oxo-L-prolyl-L-histidyl-L-tryptophyl-L-seryl-L-tyrosyl-D-tryptophyl-L-leucyl-L-arginyl-L-prolyl-, Triptelin Acetate
• CAS: 140194-24-7

Description

Stability Hygroscopic
Applications Synthetic peptide agonist analog of LH-RH. Triptoreline is a potent agonist of LH-releasing hormone, currently used in the treatment of prostatic cancer where therapy may be required over months or years. Antineoplastic (hormonal). Used in the treatment of endometriosis and infertility.
References Sanders, L., et al.: Eur. J. Drug Metab. Pharmacokinet., 15, 95 (1990), Chiba, M., et al.: Biomaterials, 18, 893 (1997), Blanco, D., et al.: Eur. J. Pharm. Biopharm., 45, 285 (1998), Sinha, V., et al.: J. Control. Rel., 90, 261 (2003),

• Brand: TRC

Chemical properties

• Molecular weight: 1371.50
• Formula: C₆₆H₈₆N₁₈O₁₅
• Color/Form: Neat
• InChI: 1H3,(H,3,4)/t44-,45-,46-,47-,48+,49-,50-,51-,52-, InChI=1S/C64H82N18O13.C2H4O2/c1-34(2)23-46(56(88)75-45(13-7-21-69-64(66)67)63(95)82-22-8-14-52(82)62(94)72-31-53(65)85)76-58(90)48(25-36-28-70-42-11-5-3-9-40(36)42)78-57(89)47(24-35-15-17-39(84)18-16-35)77-61(93)51(32-83)81-59(91)49(26-37-29-71-43-12-6-4-10-41(37)43)79-60(92)50(27-38-30-68-33-73-38)80-55(87)44-19-20-54(86)74-44, /m0./s1, 1-2(3)4/h3-6,9-12,15-18,28-30,33-34,44-52,70-71,83-84H,7-8,13-14,19-27,31-32H2,1-2H3,(H2,65,85)(H,68,73)(H,72,94)(H,74,86)(H,75,88)(H,76,90)(H,77,93)(H,78,89)(H,79,92)(H,80,87)(H,81,91)(H4,66,67,69)
• InChI key: InChIKey=CYNQIKSKCVESCU-FWWMSABFSA-N
• SMILES: Cc1ccc(C(=O)OC2COC3COC(c4ccccc4)O[C@@H]3C2)cc1