CAS 143675-79-0

fragmento de (pglu5,D-trp7,9,10)-substância*P

Fórmula: C₅₇H₆₄N₁₂O₉S

InChI: InChI=1S/C57H64N12O9S/c1-79-24-23-42(51(59)72)64-55(76)46(26-33-29-60-39-16-8-5-13-36(33)39)69-57(78)48(28-35-31-62-41-18-10-7-15-38(35)41)68-54(75)45(25-32-11-3-2-4-12-32)66-56(77)47(27-34-30-61-40-17-9-6-14-37(34)40)67-53(74)44(19-21-49(58)70)65-52(73)43-20-22-50(71)63-43/h2-18,29-31,42-48,60-62H,19-28H2,1H3,(H2,58,70)(H2,59,72)(H,63,71)(H,64,76)(H,65,73)(H,66,77)(H,67,74)(H,68,75)(H,69,78)/t42-,43-,44-,45-,46+,47+,48+/m0/s1

Chave InChI: WSYRBHQWMXTCHQ-SFIKJRKMSA-N

SMILES: CSCC[C@@H](C(=O)N)NC(=O)[C@@H](CC1=CNC2=CC=CC=C21)NC(=O)[C@@H](CC3=CNC4=CC=CC=C43)NC(=O)[C@H](CC5=CC=CC=C5)NC(=O)[C@@H](CC6=CNC7=CC=CC=C76)NC(=O)[C@H](CCC(=O)N)NC(=O)[C@@H]8CCC(=O)N8

Sinónimos:

• G Protein Antagonist
• Pyr-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH2

G-Protein antagonist peptide

CAS: 143675-79-0

Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.

Fórmula: C₅₇H₆₄N₁₂O₉S

Pureza: 98%

Cor e Forma: Solid

Peso molecular: 1093.27

Ref: TM-TP1902

Gxa0Protein Antagonist

CAS: 143675-79-0

Fórmula: C₅₇H₆₄N₁₂O₉S

Peso molecular: 1093.26

Ref: 7W-GK3748

G Protein Antagonist Pyr-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH2

CAS: 143675-79-0

G protein antagonist Pyr-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH2 is a synthetic peptide that inhibits the activity of cyclase enzymes. It has been shown to inhibit skin cancer cells and has been shown to bind intracellular targets, such as protein kinase C, with high affinity. G protein antagonist Pyr-Gln-D-Trp-Phe-D-Trp-D-Trp--Met--NH2 has also been shown to inhibit the guanine nucleotide binding proteins (G proteins), which are necessary for cell signaling. G protein antagonist Pyr--Gln--D--Trp--Phe--D--Trp--D---Trp---Met---NH2 may also be used as an inhibitor of neurokinin 1 receptor activation and whole cell recordings have shown this drug to be potent antagonists of α subunit. G protein antagonist Pyr--Gln--D

Fórmula: C₅₇H₆₄N₁₂O₉S

Pureza: Min. 95%

Peso molecular: 1,093.26 g/mol

Ref: 3D-FG110327