Receptor de estrogénio/progestagénio
Os receptores de estrogênio e progestágeno são receptores hormonais nucleares que mediam os efeitos do estrogênio e da progesterona, respectivamente. Esses receptores regulam vários processos fisiológicos, incluindo função reprodutiva, densidade óssea e saúde cardiovascular. Moduladores dos receptores de estrogênio e progestágeno são amplamente estudados por seus papéis na terapia de reposição hormonal, contracepção e tratamento de cânceres responsivos a hormônios. Na CymitQuimica, oferecemos uma gama abrangente de moduladores de receptores de estrogênio e progestágeno de alta qualidade para apoiar sua pesquisa em endocrinologia, saúde reprodutiva e biologia do câncer.
Foram encontrados 55 produtos de "Receptor de estrogénio/progestagénio"
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(R)-Equol
CAS:(R)-Equol ((+)-Equol) is an ERα and ERβ agonist with Kis of 27.4 and 15.4 nM, respectively.Fórmula:C15H14O3Pureza:99.59%Cor e Forma:SolidPeso molecular:242.27Altrenogest
CAS:<p>Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone.</p>Fórmula:C21H26O2Pureza:98.98% - 99.66%Cor e Forma:Slightly Yellow PowderPeso molecular:310.434,4'-Iminodiphenol
CAS:4,4'-Iminodiphenol (Leucoindophenol) is an inactive estrogen receptor ligand with a diphenylamine backbone.Fórmula:C12H11NO2Pureza:98.68%Cor e Forma:SolidPeso molecular:201.22Promestriene
CAS:Promestriene (3-propyl ethyl) (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation.Fórmula:C22H32O2Pureza:99.35%Cor e Forma:White SolidPeso molecular:328.49Ethynodiol diacetate
CAS:<p>Ethynodiol diacetate (Ethynodiol acetate) is a synthetic progestational hormone used alone or in combination with estrogens as an oral contraceptive.</p>Fórmula:C24H32O4Pureza:99.48% - 99.54%Cor e Forma:SolidPeso molecular:384.51Toremifene
CAS:Toremifene (GTx 006) is a selective estrogen-receptor modulator (SERM).Fórmula:C26H28ClNOPureza:99.77% - >99.99%Cor e Forma:White-To-Off-White SolidPeso molecular:405.96Gestrinone
CAS:Gestrinone (R 2323) 是一种合成类固醇激素，能够抑制平滑肌瘤(IC50:43.67 μM)，有用于子宫内膜异位症的研究潜力。Fórmula:C21H24O2Pureza:99.21%Cor e Forma:Light Yellow SolidPeso molecular:308.41SLU-PP-332
CAS:<p>SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM,</p>Fórmula:C18H14N2O2Pureza:98.3% - 98.60%Cor e Forma:SoildPeso molecular:290.32Clomiphene citrate
CAS:Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.Fórmula:C32H36ClNO8Pureza:98.67% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:598.1Dienestrol
CAS:Dienestrol (Restrol) is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist.Fórmula:C18H18O2Pureza:96.73% - 98%Cor e Forma:Minute Needles From Dilute Alc SolidPeso molecular:266.33Giredestrant
CAS:Giredestrant (GDC-9545) is a potent oral anti-tumor ER antagonist competing with estradiol.Fórmula:C27H31F5N4OPureza:98.96% - 99.56%Cor e Forma:SolidPeso molecular:522.55Mestranol
CAS:Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.Fórmula:C21H26O2Pureza:99.16%Cor e Forma:Crystals From Methanol Or Acetone SolidPeso molecular:310.43Gestodene
CAS:<p>Gestodene (WL 70) is a progestogen hormonal contraceptive.</p>Fórmula:C21H26O2Pureza:98% - 99.68%Cor e Forma:White Crystalline SolidPeso molecular:310.43Ethisterone
CAS:<p>Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.</p>Fórmula:C21H28O2Pureza:97.96% - 99.50%Cor e Forma:Off-White PowderPeso molecular:312.45Quinestrol
CAS:Quinestrol (Ethinylestradiol 3-cyclopentyl ether) is a synthetic estrogen, applied in hormone replacement therapy, and occasionally to use in cancer andFórmula:C25H32O2Pureza:99.36% - 99.72%Cor e Forma:SolidPeso molecular:364.52Panomifene TFA
Panomifene TFA（GYKl13504 TFA） is a antagonist of ERs with anticancer activity that can be used to study breast cancer and musculoskeletal diseases.Fórmula:C27H25F6NO4Pureza:99.74%Cor e Forma:SoildPeso molecular:541.48Methylpiperidino pyrazole
CAS:Methylpiperidino pyrazole is an ERα inhibitor and can prevent the BPS-induced Rb phosphorylation and cell cycle progression.Fórmula:C29H31N3O3Pureza:98.84%Cor e Forma:SolidPeso molecular:469.57Bazedoxifene
CAS:Bazedoxifene is an orally active SERM against ERα and ERβ and inhibits IL-6/GP130, applied in postmenopausal osteoporosis and pancreatic cancer research.Fórmula:C30H34N2O3Pureza:98.79%Cor e Forma:SolidPeso molecular:470.61AC-186
CAS:<p>AC-186 is an ERβ agonist with neuroprotective activity for the study of Parkinson's disease.</p>Fórmula:C18H17F3OPureza:99.53%Cor e Forma:SolidPeso molecular:306.32Endoxifen Z-isomer hydrochloride
CAS:Endoxifen Z-isomer hydrochloride (Endoxifen HCl) is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.Fórmula:C25H28ClNO2Cor e Forma:SolidPeso molecular:409.95WAY-200070
CAS:WAY-200070 is a specific agonist of estrogen receptor β (ERRβ, IC50: 2.3 nM).Fórmula:C13H8BrNO3Pureza:99.45% - 99.75%Cor e Forma:SolidPeso molecular:306.11Ulipristal
CAS:Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.Fórmula:C28H35NO3Pureza:99.82%Cor e Forma:SolidPeso molecular:433.584-Hydroxytamoxifen
CAS:<p>4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency.</p>Fórmula:C26H29NO2Pureza:99.37% - 99.93%Cor e Forma:SolidPeso molecular:387.51Elacestrant dihydrochloride
CAS:<p>Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM for</p>Fórmula:C30H40Cl2N2O2Pureza:99.59% - >99.99%Cor e Forma:SolidPeso molecular:531.56Medroxyprogesterone
CAS:Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone used in veterinary practice as an estrus regulator.Fórmula:C22H32O3Pureza:99.18% - 99.51%Cor e Forma:Crystals From Chloroform SolidPeso molecular:344.49Desogestrel
CAS:<p>Desogestrel (Cerazette) is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.</p>Fórmula:C22H30OPureza:99.8%Cor e Forma:Crystals SolidPeso molecular:310.47Ferrous Bisglycinate
CAS:Ferrous Bisglycinate (Bisglycine iron(II) salt) is used in the fortification of infant formulations and foods.Fórmula:C4H8FeN2O4Pureza:≥95%Cor e Forma:SolidPeso molecular:203.96Norgestrel
CAS:<p>Norgestrel (WY-3707), a synthetic progestin, is used for contraception and hinders LH/FSH, thickens mucus, and slows ova transit.</p>Fórmula:C21H28O2Pureza:99.71% - 99.72%Cor e Forma:Crystals From Methanol White Crystalline PowderPeso molecular:312.45GSK5182
CAS:GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)Fórmula:C27H31NO3Pureza:97.63% - 99.42%Cor e Forma:SolidPeso molecular:417.54SNG-1153
CAS:SNG-1153 is a estrogen receptor ER-alpha36 modulator.Fórmula:C21H17F3O5Pureza:99.74%Cor e Forma:SolidPeso molecular:406.35Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-
CAS:<p>Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.</p>Fórmula:C18H18O3Pureza:99.85% - 99.96%Cor e Forma:SolidPeso molecular:282.33Estradiol dipropionate
CAS:Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.Fórmula:C24H32O4Pureza:99.68%Cor e Forma:SolidPeso molecular:384.51Nestoron
CAS:Nestoron (Segesterone Acetate), a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM).Fórmula:C23H30O4Pureza:99.83% - 99.92%Cor e Forma:SolidPeso molecular:370.48PROTAC ERRα ligand 2
CAS:PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)Fórmula:C20H13F6NO4Pureza:≥95%Cor e Forma:SolidPeso molecular:445.31STF-62247
CAS:<p>STF-62247 is TGN inhibitor with IC50 of 0.625 μM and 16 μM in RCC4 and RCC4/VHL cells, respectively.</p>Fórmula:C15H13N3SPureza:99.6% - 99.67%Cor e Forma:SolidPeso molecular:267.35SR 19881
CAS:<p>SR 19881 is a full agonist of ERRγ(EC50 value of 0.39 μM in a binding assay and an EC50 value of 4.7 μM in a cell-based assay).</p>Fórmula:C19H24N2O2Pureza:98.54%Cor e Forma:SolidPeso molecular:312.41Serba-2
CAS:Serba-2 is an agonist of benzopyran selective estrogen receptor beta.Fórmula:C18H18O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:282.33Fulvestrant-d3
<p>Fulvestrant-d3 is a isotope labeled compound of Fulvestrant.an estrogen receptor (ER) antagonist and GPR30 agonist thatinduces apoptosis and autophagy.</p>Fórmula:C32H47F5O3SCor e Forma:SolidPeso molecular:609.79ERRα antagonist-1
CAS:ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα).Fórmula:C21H19N3S2Pureza:99.66%Cor e Forma:SolidPeso molecular:377.53Capesaris
CAS:<p>Capesaris (GTX-758) is an oral estrogen receptor α agonist, used in prostate cancer research.</p>Fórmula:C19H13F2NO3Pureza:99.65%Cor e Forma:SolidPeso molecular:341.31ERRγ Inverse Agonist 1
CAS:ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].Fórmula:C30H38Cl2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:529.54Norethisterone enanthate
CAS:Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.Fórmula:C27H38O3Pureza:99.23%Cor e Forma:SolidPeso molecular:410.59NXT629
CAS:NXT629 is a PPAR-α antagonist with anticancer activity, inhibiting PPARδ, and can be used in ovarian cancer and melanoma research.Fórmula:C35H39N5O3SPureza:99.07% - 99.07%Cor e Forma:SolidPeso molecular:609.78OP-1074
CAS:<p>OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.</p>Fórmula:C29H31NO4Pureza:98%Cor e Forma:SolidPeso molecular:457.56Bisphenol Z
CAS:Bisphenol Z is a bisphenol compound and high-performance monomer used in advanced engineering plastics, having antagonistic activity towards ERα.Fórmula:C18H20O2Pureza:99.88%Cor e Forma:SolidPeso molecular:268.35SIM-688
CAS:SIM-688 is a selective and orally active estrogen receptor inhibitor of NF-κB transcriptional activity (IC50 = 122 nM in HAECT-1 cells).Fórmula:C34H31F3N2O2Pureza:99.56%Cor e Forma:SolidPeso molecular:556.62DS20362725
CAS:DS20362725 is a selective estrogen-related receptor alpha (ERRα) agonist, commonly used in the study of metabolic disorders.Fórmula:C19H22N2O2Pureza:99.34%Cor e Forma:SolidPeso molecular:310.39Estrogen receptor antagonist 8
CAS:Estrogen Receptor Antagonist 8 is an ER antagonist with anti-uterine activity and may be used in the study of ovarian dysfunction.CASNETIN SODIUM (CasN)Fórmula:C25H21N3O4Pureza:98.48%Cor e Forma:SolidPeso molecular:427.45LY88074
CAS:<p>LY88074, a raloxifene analog sans basic side chain, is an ERβ agonist (EC50 = 232 nM) that promotes uterine cell growth.</p>Fórmula:C21H14O4SPureza:98.31%Cor e Forma:SolidPeso molecular:362.4Palazestrant
CAS:Palazestrant, an antiestrogen and antineoplastic agent, effectively targets ER+/HER2+ cancer when used in conjunction with a HER2 inhibitor.Fórmula:C28H36FN3OPureza:97.55%Cor e Forma:SolidPeso molecular:449.6Zindoxifene
CAS:Zindoxifene (D 16726) is an anti-estrogenic compound with antitumor activity that can be used in studies of breast and prostate cancer.Fórmula:C21H21NO4Pureza:98.99%Cor e Forma:SolidPeso molecular:351.4H3B-6545
CAS:H3B-6545 is a selective and oral estrogen receptor covalent antagonist (SERCA) used in the research of metastatic ER-positive, HER2-negative breast cancer.Fórmula:C30H29F4N5O2Cor e Forma:SolidPeso molecular:567.58ERRα antagonist-2
CAS:ERRα antagonist-2 is an estrogen-related receptor α inverse agonist, inhibiting migration and invasion in ER-negative MDA-MB-231,breast cancer.Fórmula:C19H16N2O6SPureza:99.26%Cor e Forma:SolidPeso molecular:400.41(E/Z)-GSK5182
CAS:GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.Fórmula:C27H31NO3Pureza:97.58%Cor e Forma:SolidPeso molecular:417.54ERB-196
CAS:Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.Fórmula:C17H10FNO2Pureza:98%Cor e Forma:SolidPeso molecular:279.27
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