Receptor de Vasopressina
Os receptores de vasopressina são uma família de receptores acoplados à proteína G que mediam os efeitos da vasopressina, um hormônio envolvido na regulação do equilíbrio hídrico, pressão arterial e função renal. Agonistas e antagonistas dos receptores de vasopressina são estudados por seus papéis no tratamento de condições como diabetes insipidus, hiponatremia e insuficiência cardíaca. Esses receptores também são alvos importantes na pesquisa sobre equilíbrio de fluidos e saúde cardiovascular. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de vasopressina de alta qualidade para apoiar sua pesquisa em endocrinologia, nefrologia e biologia cardiovascular.
Foram encontrados 48 produtos de "Receptor de Vasopressina"
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[8-L-arginine] deaminovasopressin
CAS:[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] .Fórmula:C46H64N14O13S2Cor e Forma:SolidPeso molecular:1085.22(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.Fórmula:C52H74N14O12S2Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:1151.38Endolide F
Endolide F (Compound 2) is a proline-containing lactone that serves as a moderate antagonist of the arginine vasopressin V1A receptor.Fórmula:C25H32N4O6Peso molecular:484.23218Velmupressin acetate
CAS:Potent, selective, short-acting peptidic V2R agonist; EC50: 0.07 nM (hV2R), 0.02 nM (rV2R).Fórmula:C44H64ClN11O10S2Pureza:98%Cor e Forma:SolidPeso molecular:1006.63Ornipressin
CAS:Ornipressin is a vasoconstrictor, haemostatic and renal agent.Fórmula:C45H63N13O12S2Pureza:98%Cor e Forma:White PowderPeso molecular:1042.19c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
CAS:c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm: potent, selective V2R agonist; EC50: 0.25 nM (hV2R), 0.05 nM (rV2R).Fórmula:C47H69ClN12O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1045.71V1a/V2 antagonist 1
V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.Fórmula:C25H26ClN5O3Cor e Forma:SolidPeso molecular:479.96Velmupressin
CAS:Peptidic V2R agonist, c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2, with EC50: 0.07 nM (hV2R), 0.02 nM (rV2R); selective, short-acting.Fórmula:C42H60ClN11O8S2Pureza:98%Cor e Forma:SolidPeso molecular:946.58[Lys8] Vasopressin Desglycinamide
CAS:[Lys8] Vasopressin Desglycinamide, a vasopressin analog, supports the maintenance of active and passive avoidance behavior and aids in the facilitation ofFórmula:C44H63N11O12S2Cor e Forma:SolidPeso molecular:1002.17Atosiban
CAS:Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.Fórmula:C43H67N11O12S2Pureza:98%Cor e Forma:SolidPeso molecular:994.19Argipressin
CAS:Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.Fórmula:C46H65N15O12S2Pureza:98%Cor e Forma:White PowderPeso molecular:1084.23Fedovapagon
CAS:Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.Fórmula:C27H34N4O3Pureza:99.46%Cor e Forma:SolidPeso molecular:462.58Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Fórmula:C26H31N3O4Pureza:98.13% - 99.66%Cor e Forma:SolidPeso molecular:449.54Atosiban acetate
CAS:Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.Fórmula:C45H71N11O14S2Pureza:99.84% - 99.92%Cor e Forma:SolidPeso molecular:1054.24Ref: TM-T5148
5mg70,00€10mg109,00€1mL*10mM (DMSO)127,00€25mg166,00€50mg195,00€100mg254,00€500mg625,00€Tolvaptan
CAS:Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
Fórmula:C26H25ClN2O3Pureza:99.78% - >99.99%Cor e Forma:SolidPeso molecular:448.94Felypressin
CAS:Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Fórmula:C46H65N13O11S2Pureza:99.65%Cor e Forma:SolidPeso molecular:1040.22LIXIVAPTAN
CAS:Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Fórmula:C27H21ClFN3O2Pureza:98.36%Cor e Forma:SolidPeso molecular:473.93Ref: TM-T7303
2mg34,00€5mg66,00€1mL*10mM (DMSO)70,00€10mg99,00€25mg205,00€50mg334,00€100mg522,00€200mg743,00€Conivaptan hydrochloride
CAS:Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia andFórmula:C32H26N4O2·HClPureza:98.33% - 99.86%Cor e Forma:SolidPeso molecular:535.04Mozavaptan
CAS:Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.Fórmula:C27H29N3O2Pureza:98.98% - 99.12%Cor e Forma:SolidPeso molecular:427.54Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1bFórmula:C43H77N17O12S2Pureza:99.79%Cor e Forma:SolidPeso molecular:1088.32
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