
Enzima
Os inibidores de enzimas são moléculas que se ligam a enzimas e diminuem sua atividade. Esses inibidores são amplamente utilizados em pesquisas para estudar a cinética enzimática, regulação e o papel de enzimas específicas nas vias metabólicas. Os inibidores de enzimas também são cruciais no desenvolvimento de medicamentos, pois muitos agentes terapêuticos funcionam inibindo enzimas envolvidas em processos patológicos. Ao direcionar enzimas, esses inibidores podem modular vias bioquímicas e oferecer tratamentos potenciais para várias doenças. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de enzimas de alta qualidade para apoiar sua pesquisa em bioquímica, farmacologia e descoberta de medicamentos.
Subcategorias de "Enzima"
- Anidrase carbónica(178 produtos)
- Hidroxilase(30 produtos)
- MPO(2 produtos)
- Redutase(52 produtos)
- Tirosinase(67 produtos)
Foram encontrados 3587 produtos de "Enzima"
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hCAI/II-IN-3
CAS:<p>"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."</p>Fórmula:C16H18N4O4S2Cor e Forma:SolidPeso molecular:394.47WES-1
CAS:<p>WES-1 (Compound 8g), a carbonic anhydrase IX inhibitor (Ki: 55.9 μM), exhibits broad-spectrum antiproliferative activity against various cancer cell lines,</p>Fórmula:C20H20N4O3SPureza:98%Cor e Forma:SolidPeso molecular:396.46L 662583
CAS:<p>L 662583 is a topical inhibitor of carbonic anhydrase.</p>Fórmula:C13H17ClN2O5S3Pureza:98%Cor e Forma:SolidPeso molecular:412.93PGDS Protein, Human, Recombinant
<p>Hematopoietic Prostaglandin D Synthase (HPGDS) belongs to the GST superfamily and Sigma family.</p>Cor e Forma:Lyophilized PowderPeso molecular:26 KDa (reducing condition)hCAI/II-IN-1
CAS:<p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>Fórmula:C18H29N5O3S3Cor e Forma:SolidPeso molecular:459.65L-693612
CAS:<p>L-693612 is an inhibitor of carbonic anhydrase.</p>Fórmula:C14H24N2O5S3Pureza:98%Cor e Forma:SolidPeso molecular:396.55GV2-20
CAS:<p>GV2-20 is an effective carbonic anhydrase 2 inhibitors.</p>Fórmula:C15H13N3O6Pureza:98%Cor e Forma:SolidPeso molecular:331.28hCAIX-IN-6
CAS:<p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>Fórmula:C18H12N2O4SCor e Forma:SolidPeso molecular:352.36hCAIX-IN-11
CAS:<p>hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.</p>Fórmula:C21H15ClN4O3Cor e Forma:SolidPeso molecular:406.82hCAIX/XII-IN-2
CAS:<p>Compound 6a: Selective hCAIX/XII inhibitor; Ki: 30 nM (hCAIX), 3.6 nM (hCAXII); >10,000 nM (hCAI/II).</p>Fórmula:C19H14N2O4Cor e Forma:SolidPeso molecular:334.33hCAII-IN-1
CAS:<p>hCAII-IN-1 (7f) inhibits CA II/IX with Kis 1.2 nM/113.6 nM, potential for cancer treatment.</p>Fórmula:C21H21BrN6O4SCor e Forma:SolidPeso molecular:533.4HCAIX-IN-2
CAS:<p>HCAIX-IN-2 (compound 9d) is a selective inhibitor of carbonic anhydrase and acts on hCA IX (Ki: 24.6 nM) and hCA XII (Ki: 45.3 nM).</p>Fórmula:C19H16N8O4SCor e Forma:SolidPeso molecular:452.45hCAXII-IN-2
CAS:<p>hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.</p>Fórmula:C21H18ClN3O4Cor e Forma:SolidPeso molecular:411.84DTP348
CAS:<p>DTP348: Oral carbonic anhydrase IX inhibitor & hypoxic cell radiosensitizer with sulfamide & 5-nitroimidazole components.</p>Fórmula:C6H11N5O4SCor e Forma:SolidPeso molecular:249.25hCA I-IN-1
CAS:<p>hCA I-IN-1 inhibits hCA I (Ki: 38.3 nM), II (Ki: 716.4 nM), IX (Ki: 940.1 nM), XII (Ki: 192.8 nM).</p>Fórmula:C27H23N5O4SCor e Forma:SolidPeso molecular:513.57hCAXII-IN-4
CAS:<p>hCAXII-IN-4 is a selective and potent CA XII inhibitor with a Ki value of 6.4 nM for human CA XII.</p>Fórmula:C22H27N5O6SCor e Forma:SolidPeso molecular:489.54PPIE Protein, Human, Recombinant (His)
<p>Peptidyl-prolyl cis-trans isomerase E, also known as Cyclophilin E, Cyclophilin-33, Rotamase E, CYP33, PPIE, is an enzyme which belongs to the cyclophilin-type</p>Cor e Forma:Lyophilized PowderPeso molecular:34 KDa (reducing condition)hCAI/II-IN-2
CAS:<p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>Fórmula:C12H12N4O5S2Cor e Forma:SolidPeso molecular:356.38Tyrosinase-IN-7
CAS:<p>Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.</p>Fórmula:C15H10O5Pureza:99%Cor e Forma:SolidPeso molecular:270.24hCA IX-IN-2
<p>hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative</p>Fórmula:C23H24N2O4STeCor e Forma:SolidPeso molecular:552.11
