
cAMP
cAMP é um segundo mensageiro importante em muitos processos biológicos, incluindo a regulação do metabolismo, expressão gênica e crescimento celular. Na via de sinalização MAPK, o cAMP pode modular a atividade de várias quinases, incluindo a PKA, que por sua vez influencia a cascata MAPK. A desregulação da sinalização de cAMP está implicada em várias doenças, incluindo câncer e distúrbios cardiovasculares. Na CymitQuimica, oferecemos uma variedade de moduladores de cAMP para apoiar sua pesquisa em transdução de sinal, metabolismo e patologia de doenças.
Foram encontrados 47 produtos de "cAMP"
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Bucladesine sodium
CAS:<p>Bucladesine sodium (DC2797) is a cAMP analog with cell-permeable properties.</p>Fórmula:C18H23N5NaO8PPureza:96.56% - 99.76%Cor e Forma:White PowderPeso molecular:491.37HJC0197
CAS:HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.Fórmula:C19H21N3OSPureza:98.05%Cor e Forma:SolidPeso molecular:339.45MR-L2
CAS:MR-L2 is a reversible and noncompetitive allosteric activator of long-isoform phosphodiesterase-4 (PDE4).Fórmula:C19H16Cl3FN4OPureza:98.09% - 98.94%Cor e Forma:SolidPeso molecular:441.71JNJ-39758979
CAS:<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Fórmula:C11H19N5Pureza:98.33% - 99.62%Cor e Forma:SolidPeso molecular:221.3A-3 hydrochloride
CAS:<p>A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.</p>Fórmula:C12H14Cl2N2O2SPureza:99.32%Cor e Forma:SolidPeso molecular:321.22CE3F4
CAS:CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of 10.7 μM and 66 μM for Epac1 and Epac2(B), respectively).Fórmula:C11H10Br2FNOPureza:97.15% - 98.06%Cor e Forma:SolidPeso molecular:351.01ESI-05
CAS:ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.Fórmula:C16H18O2SPureza:97.22%Cor e Forma:SolidPeso molecular:274.38Mirabegron
CAS:<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Fórmula:C21H24N4O2SPureza:99.64%Cor e Forma:Light Yellow To Yellow SolidPeso molecular:396.51Bithionol
CAS:Bithionol (Actamer), formerly marketed as an active ingredient in various topical drug products, was shown to be a potent photosensitizer with the potential toFórmula:C12H6Cl4O2SPureza:99.04%Cor e Forma:White Or Grayish-White Crystalline Powder Phenolic Odor (Ntp 1992)Peso molecular:356.05MRS-1706
CAS:MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.Fórmula:C27H29N5O5Pureza:99.00%Cor e Forma:SolidPeso molecular:503.55OX04528
CAS:OX04528 is an orally active and potent GPR84 biased agonist.OX04528 inhibits cAMP signaling and may be useful in cancer research.Fórmula:C16H13F6NO2Pureza:99.74%Cor e Forma:SoildPeso molecular:365.27BC 11-38
CAS:<p>BC 11-38 is a potent, selective PDE biodepressant which is mainly effective against PDE11 (IC50 : 0.28 μM).</p>Fórmula:C15H16N2OS2Pureza:98.95% - 99.28%Cor e Forma:SolidPeso molecular:304.432-PCCA hydrochloride
CAS:<p>2-PCCA hydrochloride, a racemate, is a potent and selective GPR88 receptor agonist showing inhibition of GPR88-mediated cAMP production in HEK293 cells with an</p>Fórmula:C30H39Cl2N3OPureza:97.54% - 99.36%Cor e Forma:SoildPeso molecular:528.56Adenosine 3'-monophosphate (sodium salt hydrate)
Adenosine 3'-monophosphate (sodium salt hydrate) (3'-AMP) is a nucleotide and cAMP-generating agonist that elevates cAMP levels in NG108-15 cells.Fórmula:C10H15N5NaO8PCor e Forma:SolidPeso molecular:387.22Anti-Cathelicidin/Camp Polyclonal Antibody
Antibody Type: Rabbit Polyclonal<br> Application: ELISA,ICC/IF,IF,IHC-Fr,IHC-P<br> Reactivity: (predicted:Mouse,Rat)Cor e Forma:LiquidPeso molecular:Theoretical: 19 kDa.GLP-1R modulator L7-028
CAS:GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.Fórmula:C24H28N2O3Pureza:98.76% - >99.99%Cor e Forma:SolidPeso molecular:392.49Pinoresinol 4-O-β-D-glucopyranoside
CAS:(+)-Pinoresinol-β-D-glucoside, also known as (+)-pinor, is a major active lignan furanoid found in Forsythia.Fórmula:C26H32O11Pureza:99.32% - >99.99%Cor e Forma:SolidPeso molecular:520.53Ro 20-1724
CAS:Ro 20-1724 (4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone) is a widely used inhibitor of cyclic nucleotide phosphodiesterase with IC50 of 2.0 μM and Ki of 3.1Fórmula:C15H22N2O3Pureza:98.82% - 99.79%Cor e Forma:SolidPeso molecular:278.35SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Fórmula:C15H13ClN4O2S2Pureza:97.82% - 98%Cor e Forma:SolidPeso molecular:380.87RS-25344 hydrochloride
CAS:RS 25344 hydrochloride is a phosphodiesterase (PDE) 4 inhibitorFórmula:C19H14ClN5O4Pureza:99.25%Cor e Forma:SolidPeso molecular:411.8

