
ATPase
As ATPases são enzimas que catalisam a decomposição do ATP em ADP e um íon fosfato livre, uma reação que libera energia usada para impulsionar muitos processos dentro da célula, incluindo o transporte ativo através das membranas. As ATPases desempenham papéis cruciais na manutenção da homeostase celular, equilíbrio de pH e gradientes iônicos. Disfunções na atividade da ATPase estão associadas a doenças como insuficiência cardíaca, hipertensão e neurodegeneração. Na CymitQuimica, fornecemos inibidores e moduladores de ATPase de alta qualidade para apoiar sua pesquisa em energética celular, transporte de membranas e patologia de doenças.
Foram encontrados 100 produtos de "ATPase"
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Transdermal Peptide Disulfide Acetate
<p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>Fórmula:C42H68N14O18S2Pureza:99.97%Cor e Forma:SolidPeso molecular:1121.2Prilocaine
CAS:Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread ofFórmula:C13H20N2OPureza:98.49%Cor e Forma:Needles SolidPeso molecular:220.31(-)-Blebbistatin
CAS:(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.Fórmula:C18H16N2O2Pureza:99.38% - 99.61%Cor e Forma:SolidPeso molecular:292.33CB-5083
CAS:CB-5083 is a potent, selective, and orally bioavailable p97 AAA ATPase inhibitor ( IC50=11 nM).Fórmula:C24H23N5O2Pureza:95.95% - 99.92%Cor e Forma:SolidPeso molecular:413.47Tenatoprazole
CAS:Tenatoprazole (TU-199), a prodrug of the proton pump inhibitor (PPI) class, can inhibit proton transport (IC50: 3.2 μM).Fórmula:C16H18N4O3SPureza:99.57%Cor e Forma:White Crystalline PowderPeso molecular:346.4Rabeprazole sodium
CAS:Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.Fórmula:C18H20N3NaO3SPureza:98% - 99.912%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:381.42Esomeprazole Magnesium
CAS:Esomeprazole Magnesium (NEXIUM) is the S-isomer of omeprazole, can reduce gastric acid secretion with selective and irreversible proton pump inhibitor activity.Fórmula:C34H36MgN6O6S2Pureza:98.76% - 99.73%Cor e Forma:SolidPeso molecular:713.12Revaprazan hydrochloride
CAS:Revaprazan hydrochloride (YH1885) is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity.Fórmula:C22H24ClFN4Pureza:99.62% - 99.91%Cor e Forma:SolidPeso molecular:398.9FCCP
CAS:FCCP (Trifluoromethoxy carbonylcyanide phenylhydrazone) is an oxidative phosphorylation (OXPHOS) inhibitor and mitochondrial proton carrier uncoupler.Fórmula:C10H5F3N4OPureza:98% - 99.65%Cor e Forma:White SolidPeso molecular:254.17Chloroprocaine
CAS:Chloroprocaine: Na,K-ATPase inhibitor, IC50=13 mM, local anesthetic.Fórmula:C13H19ClN2O2Cor e Forma:SolidPeso molecular:270.76KM 91104
CAS:KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.Fórmula:C14H12N2O4Pureza:99.04%Cor e Forma:SolidPeso molecular:272.26PF 03716556
CAS:PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal refluxFórmula:C22H26N4O3Pureza:99.79% - 99.95%Cor e Forma:SolidPeso molecular:394.47Tetradifon
CAS:Tetradifon is a broad-spectrum organochlorine acaricide that inhibits mitochondrial OSCP, blocking energy production (IC50=4.5-27nmoL/mg) with oligomycin-like effects.Fórmula:C12H6Cl4O2SPureza:99.84%Cor e Forma:Yellowish Odorless OilPeso molecular:356.05Istaroxime oxalate
CAS:<p>Istaroxime (PST-2744) is a positive inotrope that inhibits Na+/K+ ATPase, raising intracellular sodium and calcium levels.</p>Fórmula:C23H34N2O7Cor e Forma:SolidPeso molecular:450.53FCPT
CAS:FCPT is an ATP competitive kinesin-5 inhibitor.Fórmula:C17H13FN2SPureza:98%Cor e Forma:SolidPeso molecular:296.36RS 029
CAS:RS 029 is a nitroimidazole that has been exhibited to significantly inhibit (Na+K+) ATP-ase activity.Fórmula:C13H16N6O6Pureza:98%Cor e Forma:SolidPeso molecular:352.3Azeloprazole
CAS:Azeloprazole, a proton pump inhibitor, is used potentially for the treatment of gastroesophageal reflux disease (GERD).Fórmula:C22H27N3O4SPureza:98%Cor e Forma:SolidPeso molecular:429.53Ro18-5362
CAS:Ro18-5362 is the less active prodrug of Ro 18-5364.Fórmula:C22H25N3O2SPureza:98%Cor e Forma:SolidPeso molecular:395.52Laurinterol
CAS:Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.Fórmula:C15H19BrOCor e Forma:SolidPeso molecular:295.21Bifenazate
CAS:<p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>Fórmula:C17H20N2O3Pureza:99.62%Cor e Forma:Solid CrystallinePeso molecular:300.35
