Receptor CGRP
Os receptores de CGRP estão envolvidos na transmissão da dor e na regulação do fluxo sanguíneo. O CGRP é um neuropeptídeo que desempenha um papel crítico na fisiopatologia da enxaqueca, dilatando os vasos sanguíneos e modulando as vias de sinalização da dor. Alvejar os receptores de CGRP tornou-se uma abordagem promissora no desenvolvimento de terapias para enxaqueca. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de CGRP para apoiar sua pesquisa em manejo da dor, neurobiologia e saúde vascular.
Foram encontrados 55 produtos para "Receptor CGRP".
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Adrenomedullin (AM) (22-52), human TFA
Adrenomedullin (AM) human (22-52) is a truncated NH2 TFA-modified adrenal medullary receptor antagonist.Fórmula:C161H253N46F3O50Pureza:98%Cor e Forma:SolidPeso molecular:3690.06Calcitonin (human) acetate
CAS:Calcitonin (human) acetate (21215-62-3, free base) is a synthetic polypeptide hormone composed of 32 amino acids.Fórmula:C153H230N40O47S3Pureza:99.46%Cor e Forma:White SolidPeso molecular:3477.91MK-8825
CAS:MK-8825 is a CGRP receptor antagonist.Fórmula:C31H30F2N6O3Cor e Forma:SolidPeso molecular:572.61Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.Fórmula:C163H267N51O50S2Pureza:98%Cor e Forma:SolidPeso molecular:3805.31Adrenomedullin (11-50), rat
CAS:Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.Fórmula:C194H304N58O59S4Pureza:98%Cor e Forma:SolidPeso molecular:4521.17Ubrogepant-D5
Ubrogepant-D5 is the deuterium-labeled version of Ubrogepant. It is an orally active and selective antagonist of the calcitonin gene-related peptide receptor (CGRP). Ubrogepant (T17194) exhibits high affinity for CGRP receptors in humans and rhesus monkeys, effectively blocking the cAMP response induced by α-CGRP stimulation. This compound is utilized in studies focused on acute migraine.Cor e Forma:Odour Solidα-CGRP(human)
CAS:Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.Fórmula:C163H267N51O49S2Pureza:98%Cor e Forma:SolidPeso molecular:3789.33Adrenomedullin (16-31), human
CAS:Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).Fórmula:C82H129N25O21S2Pureza:98%Cor e Forma:SolidPeso molecular:1865.19Galcanezumab
CAS:Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.Pureza:> 95%Cor e Forma:Transparent LiquidPeso molecular:144.08 kDaα-CGRP(human) TFA
α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as aFórmula:C165H268F3N51O51S2Cor e Forma:SolidPeso molecular:3903.33Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Fórmula:C84H130F3N25O23S2Cor e Forma:SolidPeso molecular:1979.21Adrenotensin (human)
CAS:Adrenotensin: human 153-185 fragment of Adrenomedullin precursor, a 52-amino acid peptide in CGRP hormone family.Fórmula:C143H224N42O43Cor e Forma:SolidPeso molecular:3219.56Calcitonin Gene Related Peptide (CGRP) II, rat TFA
Rat CGRP II TFA: potent vasodilator and CGRP receptor activator for cardiovascular research.Fórmula:C165H268F3N51O52S2Cor e Forma:SolidPeso molecular:3919.33Telcagepant
CAS:Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.Fórmula:C26H27F5N6O3Pureza:98.98% - 98.98%Cor e Forma:SolidPeso molecular:566.52Calcitonin (salmon)
CAS:Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.Fórmula:C145H240N44O48S2Pureza:99.41% - 99.80%Cor e Forma:SolidPeso molecular:3431.85SUN B8155
CAS:SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.Fórmula:C14H15N3O3Pureza:99.38% - 99.99%Cor e Forma:Yellow SolidPeso molecular:273.29Rimegepant
CAS:View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.Fórmula:C28H28F2N6O3Pureza:99.1% - 99.99%Cor e Forma:White SolidPeso molecular:534.56Ref: TM-T4610
10mgA consultar25mgA consultar50mgA consultar100mgA consultar200mgA consultar1mg52,00€5mg92,00€1mL*10mM (DMSO)105,00€β-CGRP, human acetate
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptorFórmula:C164H271N51O50S3Pureza:99.35%Cor e Forma:SolidPeso molecular:3853.46Olcegepant
CAS:Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Fórmula:C38H47Br2N9O5Pureza:96.08% - 97.24%Cor e Forma:SolidPeso molecular:869.65BCTC
CAS:BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)Fórmula:C20H25ClN4OPureza:99.21% - 99.74%Cor e Forma:White SolidPeso molecular:372.89
