
Canais de Cálcio
Os canais de cálcio são proteínas de membrana que regulam o fluxo de íons de cálcio para dentro e fora das células, o que é essencial para várias funções celulares, incluindo a contração muscular, a liberação de neurotransmissores e a expressão gênica. A desregulação da atividade dos canais de cálcio está associada a condições como hipertensão, arritmias cardíacas e distúrbios neurológicos. Na CymitQuimica, oferecemos uma ampla seleção de moduladores de canais de cálcio para apoiar sua pesquisa em saúde cardiovascular, neurobiologia e transdução de sinais.
Foram encontrados 541 produtos de "Canais de Cálcio"
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(±)-Praeruptorin A
CAS:(±)-Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation.Fórmula:C21H22O7Pureza:98.9% - 99.73%Cor e Forma:SolidPeso molecular:386.40NFAT Inhibitor-2
CAS:NFAT Inhibitor-2 is a compound used as a molecular building block.Fórmula:C22H20F2N2O4SPureza:97.37%Cor e Forma:SolidPeso molecular:446.47Praeruptorin C
CAS:<p>Praeruptorin C: an antioxidant, calcium antagonist, protects neurons, reduces vascular hypertrophy, affects cellular signals.</p>Fórmula:C24H28O7Pureza:99.6% - 99.92%Cor e Forma:SolidPeso molecular:428.47Azumolene sodium anhydrous
CAS:Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.Fórmula:C13H8BrN4NaO3Cor e Forma:SolidPeso molecular:371.13CDN1163
CAS:CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).Fórmula:C20H20N2O2Pureza:99.83% - ≥95%Cor e Forma:SolidPeso molecular:320.39Pinaverium bromide
CAS:Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.Fórmula:C26H41Br2NO4Pureza:99.52%Cor e Forma:White Crystalline PowderPeso molecular:591.42Taurolithocholic acid sodium salt
CAS:Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, butFórmula:C26H44NNaO5SPureza:99.79% - 99.93%Cor e Forma:SolidPeso molecular:505.69FPL64176
CAS:FPL64176 is a L-type calcium channels activator.Fórmula:C22H21NO3Pureza:98.68%Cor e Forma:SolidPeso molecular:347.41Thapsigargin
CAS:Thapsigargin is a natural product, an inhibitor of sarcoplasmic/endoplasmic reticulum Ca2+ ATPase (SERCA) and an endoplasmic reticulum stress inducer.Fórmula:C34H50O12Pureza:99.07% - 99.3%Cor e Forma:Colourless FilmPeso molecular:650.75DHBP dibromide
CAS:DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.Fórmula:C24H38Br2N2Pureza:99.73%Cor e Forma:Yellow To Yellow-Green Powder Or FlakesPeso molecular:514.38Yangambin
CAS:Yangambin: selective PAF antagonist, hypotensive, inhibits Ca2+ influx, induces peripheral vasodilation, affects CNS.Fórmula:C24H30O8Pureza:98.02%Cor e Forma:SolidPeso molecular:446.49SR33805
CAS:<p>SR33805 is a potent antagonist of Ca2+ channel(EC50s of 4.1 nM and 33 nM in depolarized and polarized conditions, respectively)</p>Fórmula:C32H40N2O5SPureza:99.15%Cor e Forma:SolidPeso molecular:564.74OPHIOPOGONIN D
CAS:Ophiopogonin D is a natural product,and is a CYP2J3 inducer that significantly inhibits Ang II induced NF-κB nuclear translocation.Fórmula:C44H70O16Pureza:99.46% - ≥95%Cor e Forma:SolidPeso molecular:855.021-Octanol
CAS:1-Octanol is a saturated fatty alcohol, inhibits T-type Ca²⁺ channels with a 4 μM IC50, and is a potential diesel-like biofuel.Fórmula:C8H18OPureza:99.94%Cor e Forma:Colourless LiquidPeso molecular:130.23Amlodipine mesylate
CAS:Amlodipine mesylate, an oral dihydropyridine Ca2+ blocker, treats angina, hypertension, and may be used in cancer research.Fórmula:C21H29ClN2O8SCor e Forma:SolidPeso molecular:504.98L-Phenylalanine-15N
CAS:L-Phenylalanine-15N, essential amino acid, Ca+ channel and NMDARs antagonist, used in food flavors and pharmaceuticals.Fórmula:C9H11NO2Pureza:98.98%Cor e Forma:SolidPeso molecular:166.18ABT-639 hydrochloride
CAS:ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.Fórmula:C20H21Cl2F2N3O3SCor e Forma:SolidPeso molecular:492.36Bepridil free base
CAS:Bepridil: Class IV anti-arrhythmic, calcium blocker, dilates coronary arteries.Fórmula:C24H34N2OCor e Forma:SolidPeso molecular:366.54Fantofarone
CAS:Fantofarone (SR 33557) is a highly potent antagonist of Calcium Channel.Fórmula:C31H38N2O5SPureza:96.13% - 99.19%Cor e Forma:SolidPeso molecular:550.71Praeruptorin E
CAS:Praeruptorin C/E relaxes arteries, reduces heart contractility, acting like calcium blockers. D/E protect mice from acid lung injury by halting PMNs and IL-6.Fórmula:C24H28O7Pureza:98.04% - 99.95%Cor e Forma:SolidPeso molecular:428.47
