
Canais de Cálcio
Os canais de cálcio são proteínas de membrana que regulam o fluxo de íons de cálcio para dentro e fora das células, o que é essencial para várias funções celulares, incluindo a contração muscular, a liberação de neurotransmissores e a expressão gênica. A desregulação da atividade dos canais de cálcio está associada a condições como hipertensão, arritmias cardíacas e distúrbios neurológicos. Na CymitQuimica, oferecemos uma ampla seleção de moduladores de canais de cálcio para apoiar sua pesquisa em saúde cardiovascular, neurobiologia e transdução de sinais.
Foram encontrados 541 produtos de "Canais de Cálcio"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
CGP 28392
CAS:CGP 28392 is used as a partial calcium channel agonist.Fórmula:C18H17F2NO5Pureza:98%Cor e Forma:SolidPeso molecular:365.33Kadethrin
CAS:Kadethrin is a synthetic pyrethroid. It was used as a pesticide.Fórmula:C23H24O4SPureza:98%Cor e Forma:Yellow-Brown Viscous Oil SolidPeso molecular:396.5N-Salicyloyltryptamine
CAS:N-Salicyloyltryptamine (STP): a tryptamine with anticonvulsant, anti-inflammatory, analgesic effects; inhibits Na+, Ca2+, K+ channels (IC50 34.6 μM).Fórmula:C17H16N2O2Cor e Forma:SolidPeso molecular:280.32YS-035 hydrochloride
CAS:inhibitor of outward K+ currentsFórmula:C21H30ClNO4Pureza:98%Cor e Forma:SolidPeso molecular:395.92Norbormide
CAS:Norbormide is a toxic compound used as a rodenticide. It has several mechanisms of action, acting as a vasoconstrictor and calcium channel blocker.Fórmula:C33H25N3O3Pureza:98%Cor e Forma:Crystals From Methylene Chloride + Ether Norbormide Is A Colorless To Off-White Crystalline Powder Used As A Selective Rat Poison (Epa 1998)Peso molecular:511.57Anipamil
CAS:Anipamil is a long-acting blocker of calcium channel,and for the treatment of cardiovascular disease.Fórmula:C34H52N2O2Pureza:98%Cor e Forma:SolidPeso molecular:520.79(S)-Lercanidipine hydrochloride
CAS:(S)-Lercanidipine hydrochloride is the S-enantiomer of Lercanidipine hydrochloride. (S)-lercanidipine hydrochloride is a potent blocker of calcium channel.Fórmula:C36H42ClN3O6Pureza:98%Cor e Forma:SolidPeso molecular:648.19SOCE inhibitor 1
CAS:SOCE inhibitor 1 is a inhibitor of store-operated calcium entry (SOCE)(IC50 of 4.4 μM).Fórmula:C25H22F3N5O4Pureza:98%Cor e Forma:SolidPeso molecular:513.47GSK-5498A
CAS:GSK-5498A: Selective CARC blocker, inhibits release of mediators from mast cells and cytokines from T-cells (IC50, 1 μM).Fórmula:C18H11F6N3OCor e Forma:SolidPeso molecular:399.29Lemildipine
CAS:Lemildipine is a new blocker of dihydropyridine calcium entry.Fórmula:C20H22Cl2N2O6Cor e Forma:SolidPeso molecular:457.3GSK-5503A
CAS:GSK-5503A is a novel channel blocker of CRAC.Fórmula:C23H17F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:405.4ORM-10962
CAS:ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55Fórmula:C27H29N3O4Pureza:98%Cor e Forma:SolidPeso molecular:459.54PD-217014 HCl
CAS:PD-217014, a GABA analog, blocks (3)H-gabapentin on alpha(2)delta calcium channels (K(i) 18 nmol/l), and is a visceral analgesic.Fórmula:C11H19NO2Pureza:98%Cor e Forma:SolidPeso molecular:197.27A 39355
CAS:A 39355 may specifically overcome multidrug resistance without the serious hypotensive effects associated with calcium antagonists.Fórmula:C28H39Cl2N3OPureza:98%Cor e Forma:SolidPeso molecular:504.54NP-252
CAS:NP-252 is a calcium channel antagonist potentially for the treatment of angina pectoris and congestive heart failure.Fórmula:C26H35N3O5Pureza:98%Cor e Forma:SolidPeso molecular:469.57KB-130015
CAS:KB-130015, a activator of hERG1 potassium channels, blocks native and recombinant hERG1 channels at high voltages.Fórmula:C18H14I2O4Pureza:98%Cor e Forma:SolidPeso molecular:548.11Watanidipine dihydrochloride
CAS:Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.Fórmula:C41H44Cl2N4O6Pureza:98%Cor e Forma:SolidPeso molecular:759.73Gallopamil, (-)-
CAS:Gallopamil, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.Fórmula:C28H40N2O5Pureza:98%Cor e Forma:SolidPeso molecular:484.63AK-2-38
CAS:AK-2-38 is a nifedipine analogue with potent smooth muscle calcium antagonist action and partial agonist effects on isolated guinea pig left atrium.Fórmula:C26H30N2O4Pureza:98%Cor e Forma:SolidPeso molecular:434.53Falipamil
CAS:Falipamil, a verapamil derivative, is a calcium channel blocker with antitachycardic and potential antianginal effects.Fórmula:C24H32N2O5Pureza:98%Cor e Forma:SolidPeso molecular:428.52
