Receptor GABA
Os receptores de GABA são os principais receptores de neurotransmissores inibitórios no sistema nervoso central, desempenhando um papel crítico na regulação da excitabilidade neuronal e na manutenção do equilíbrio entre excitação e inibição. A disfunção dos receptores de GABA está implicada em vários distúrbios neurológicos e psiquiátricos, incluindo epilepsia, ansiedade e depressão. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de GABA para apoiar sua pesquisa em neurobiologia, saúde mental e desenvolvimento terapêutico.
Foram encontrados 364 produtos de "Receptor GABA"
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(1S,3R)-3-Aminocyclopentane carboxylic acid
CAS:<p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>Fórmula:C6H11NO2Cor e Forma:SolidPeso molecular:129.16Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Fórmula:C19H38ClN5O2SCor e Forma:SolidPeso molecular:436.06Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Cor e Forma:Odour SolidAHN-683
CAS:AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.Fórmula:C42H32FN3O7Pureza:98%Cor e Forma:SolidPeso molecular:709.72GABAA receptor modulator-3
GABAA receptor modulator-3 (compound 3b) is a positive allosteric modulator (PAM). It inhibits the peak current and steady-state current of α1β3γ2 GABAAR with IC50 values of 671 μM and 64 μM, respectively.Fórmula:C18H22O2Cor e Forma:SolidPeso molecular:270.37RuBi-GABA
CAS:Ruthenium-bipyridine-triphenylphosphine caged GABAFórmula:C42H39F6N5O2P2RuPureza:98%Cor e Forma:SolidPeso molecular:922.8Lesogaberan napadisylate
CAS:Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.Fórmula:C13H17FNO5PSCor e Forma:SolidPeso molecular:349.31S-8510 free base
CAS:S-8510 is a GABA-A receptor inverse agonist enhancing memory, LTP, and neurotransmitters in rats.Fórmula:C12H10N4O2Cor e Forma:SolidPeso molecular:242.23MRK-016
CAS:MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.Fórmula:C17H20N8O2Pureza:99.76%Cor e Forma:SolidPeso molecular:368.39Etifoxine
CAS:Etifoxine targets β2/β3 GABAA receptors, is anxiolytic in humans/rodents, boosts GABAA, binds TSPO, aids axon regeneration, no sedative effects.Fórmula:C17H17ClN2OPureza:98%Cor e Forma:SolidPeso molecular:300.78Padsevonil
CAS:Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy.Fórmula:C14H14ClF5N4O2SPureza:99.63%Cor e Forma:SolidPeso molecular:432.80CGP 36742
CAS:CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Fórmula:C7H18NO2PCor e Forma:SolidPeso molecular:179.2Valnoctamide
CAS:Valnoctamide (Valmethamide) has antiepileptic and anticonvulsant activity and may be used in the study of neurological disorders.Fórmula:C8H17NOPureza:98%Cor e Forma:SolidPeso molecular:143.23Vigabatrin Hydrochloride
CAS:Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.Fórmula:C6H11NO2·HClPureza:98%Cor e Forma:SolidPeso molecular:165.62Dipropofol
CAS:<p>Dipropofol (4,4-Bis(2,6-di-isopropylphenol)) is a small molecule GABAA receptor agonist that can be used to study epilepsy.</p>Fórmula:C24H34O2Pureza:99.51%Cor e Forma:SolidPeso molecular:354.53L-655708
CAS:L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.Fórmula:C18H19N3O4Pureza:99.36%Cor e Forma:PowderPeso molecular:341.36(-)-α-Pinene
CAS:(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) enhances the quantity of NREMS without affecting the intensity of NREMS by prolonging GABAergic synaptic transmission,Fórmula:C10H16Pureza:98.02% - 98.60%Cor e Forma:Colourless LiquidPeso molecular:136.23Furosemide-d5
CAS:Furosemide-d5 is a deuterium marker for Furosemide and used in isotope tracer experiments. orally active inhibitor of Na+/K+/2Cl- (NKCC) diuretic reagent.Fórmula:C12H11ClN2O5SCor e Forma:SolidPeso molecular:335.78Primidone (Standard)
CAS:Primidone (Standard) is the standard substance of Primidone, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Primidone (NCI-C56360) is a potent anticonvulsant agent. It is a neuronal voltage-gated sodium channel blocker and has value in the study of epilepsy, essential tremor, and psychiatric disorders.Fórmula:C12H14N2O2Peso molecular:218.25
