Receptor GABA
Os receptores de GABA são os principais receptores de neurotransmissores inibitórios no sistema nervoso central, desempenhando um papel crítico na regulação da excitabilidade neuronal e na manutenção do equilíbrio entre excitação e inibição. A disfunção dos receptores de GABA está implicada em vários distúrbios neurológicos e psiquiátricos, incluindo epilepsia, ansiedade e depressão. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de GABA para apoiar sua pesquisa em neurobiologia, saúde mental e desenvolvimento terapêutico.
Foram encontrados 365 produtos de "Receptor GABA"
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6-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFórmula:C11H11N3OPureza:99.03%Cor e Forma:SolidPeso molecular:201.22Fipronil
CAS:Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Fórmula:C12H4Cl2F6N4OSPureza:97.21%Cor e Forma:Solid PowderPeso molecular:437.15Acetoxyvalerensre
CAS:<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Fórmula:C17H24O4Pureza:98.22%Cor e Forma:SolidPeso molecular:292.374-Acetamidobutanoic acid
CAS:4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Fórmula:C6H11NO3Pureza:98.51%Cor e Forma:SolidPeso molecular:145.16α-Asarone
CAS:alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Fórmula:C12H16O3Pureza:99.64% - 99.64%Cor e Forma:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecular:208.25Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Fórmula:C15H18BrN3O3Pureza:98.51% - 99.24%Cor e Forma:SolidPeso molecular:368.23Gaboxadol hydrochloride
CAS:Gaboxadol (hydrochloride) is a GABAA receptor agonist.Fórmula:C6H9ClN2O2Pureza:99.39%Peso molecular:176.601SKF89976A HCl
CAS:SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Fórmula:C22H25NO2Cor e Forma:SolidPeso molecular:335.442'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Fórmula:C16H14O4Pureza:98.75%Cor e Forma:SolidPeso molecular:270.28Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Fórmula:C20H25NO2S2Pureza:99.25% - 99.67%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:375.55AZD-6280
CAS:AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Fórmula:C20H22N4O3Pureza:98.99%Cor e Forma:SolidPeso molecular:366.41CL 218872
CAS:CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Fórmula:C13H9F3N4Pureza:99.92%Cor e Forma:SolidPeso molecular:278.23Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Fórmula:C30H18O10Pureza:98.21% - 99.22%Cor e Forma:Odourless Whitish SolidPeso molecular:538.46Piperazine
CAS:Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Fórmula:C4H10N2Cor e Forma:SolidPeso molecular:86.14AZD7325
CAS:<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Fórmula:C19H19FN4O2Pureza:99.83%Cor e Forma:SolidPeso molecular:354.382'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFórmula:C17H14O3Pureza:99.28% - 99.63%Cor e Forma:SolidPeso molecular:266.29Tiagabine hydrochloride hydrate
CAS:Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Fórmula:C20H28ClNO3S2Cor e Forma:SolidPeso molecular:430.02rac-BHFF
CAS:<p>rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.</p>Fórmula:C17H21F3O3Pureza:99.69% - >99.99%Cor e Forma:SolidPeso molecular:330.34Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Fórmula:C22H31NO3Pureza:98% - 99.92%Cor e Forma:SolidPeso molecular:357.49Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFórmula:C2H5NO3·5HClPureza:98.03%Cor e Forma:Light Beige Crystalline PowderPeso molecular:109.3
