Receptor GABA
Os receptores de GABA são os principais receptores de neurotransmissores inibitórios no sistema nervoso central, desempenhando um papel crítico na regulação da excitabilidade neuronal e na manutenção do equilíbrio entre excitação e inibição. A disfunção dos receptores de GABA está implicada em vários distúrbios neurológicos e psiquiátricos, incluindo epilepsia, ansiedade e depressão. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de GABA para apoiar sua pesquisa em neurobiologia, saúde mental e desenvolvimento terapêutico.
Foram encontrados 337 produtos de "Receptor GABA"
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Aminooxyacetic acid hemihydrochloride
CAS:<p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>Fórmula:C2H5NO3·5HClPureza:98.03%Cor e Forma:Light Beige Crystalline PowderPeso molecular:109.3Amentoflavone
CAS:<p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>Fórmula:C30H18O10Pureza:98.21% - 99.22%Cor e Forma:Odourless Whitish SolidPeso molecular:538.46U93631
CAS:<p>GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.</p>Fórmula:C17H21N3O2Pureza:99.65% - 99.76%Cor e Forma:SolidPeso molecular:299.37α-Thujone
CAS:<p>α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.</p>Fórmula:C10H16OPureza:97.02% - 98.41%Cor e Forma:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Peso molecular:152.23Darigabat
CAS:<p>Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.</p>Fórmula:C22H21FN4O3SPureza:98.42% - 99.29%Cor e Forma:SolidPeso molecular:440.49Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Fórmula:C8H5F3N2OSPureza:99.71% - 99.88%Cor e Forma:PowderPeso molecular:234.2CGP 36216 hydrochloride
CAS:<p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>Fórmula:C5H14NO2PPureza:98%Cor e Forma:SolidPeso molecular:151.14β-CCB
CAS:<p>benzodiazepine receptor ligand</p>Fórmula:C16H16N2O2Pureza:98%Cor e Forma:SolidPeso molecular:268.31NO 711
CAS:<p>NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.</p>Fórmula:C21H22N2O3Pureza:99.70%Cor e Forma:SolidPeso molecular:350.41(±)-Homoproline Hydrochloride
CAS:<p>(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can Trust</p>Fórmula:C6H12ClNO2Pureza:99.69%Cor e Forma:SolidPeso molecular:165.62CP-457920
CAS:<p>CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.</p>Fórmula:C18H17N3O3Pureza:99.06% - 99.74%Cor e Forma:SolidPeso molecular:323.35Ro 41-3290
CAS:Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.Fórmula:C24H21ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:420.89PF-0713
CAS:<p>PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.</p>Fórmula:C14H22OPureza:98%Cor e Forma:SolidPeso molecular:206.32HZ166
CAS:<p>HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.</p>Fórmula:C21H16N4O2Pureza:98%Cor e Forma:SolidPeso molecular:356.38Pregabalin arenacarbil
CAS:<p>Pregabalin arenacarbil is a gabamimetic.</p>Fórmula:C15H27NO6Cor e Forma:SolidPeso molecular:317.38NCS-382
CAS:<p>γ-Hydroxybutyric acid antagonist</p>Fórmula:C13H14O3Pureza:98%Cor e Forma:SolidPeso molecular:218.25Ro 19-4603
CAS:<p>Benzodiazepine inverse agonist</p>Fórmula:C15H17N3O3SPureza:98%Cor e Forma:SolidPeso molecular:319.38GABAA receptor agent 4
CAS:<p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>Fórmula:C17H24N2OCor e Forma:SolidPeso molecular:272.39mGAT3/4-IN-1
CAS:<p>mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.</p>Fórmula:C26H31ClN2O2S2Cor e Forma:SolidPeso molecular:503.12CGP11952
CAS:<p>CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.</p>Fórmula:C21H21Cl2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:446.33
