Transferase
As transferases são uma grande classe de enzimas que catalisam a transferência de grupos funcionais, como metil, glicosil e fosfato, de uma molécula para outra. Inibidores de transferases são usados para estudar uma ampla gama de processos biológicos, incluindo transdução de sinal, metabolismo e expressão gênica. Esses inibidores são ferramentas essenciais em áreas de pesquisa como câncer, doenças metabólicas e epigenética, onde a desregulação da atividade das transferases está implicada. Na CymitQuimica, oferecemos uma seleção abrangente de inibidores de transferases para apoiar sua pesquisa em enzimologia, sinalização celular e mecanismos de doenças.
Foram encontrados 42 produtos para "Transferase".
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Opicapone
CAS:Opicapone (BIA 9-1067), a potent COMT inhibitor for Parkinson's studies, lowers cell ATP (IC50: 98 μM).Fórmula:C15H10Cl2N4O6Pureza:98.17% - 99.36%Cor e Forma:SolidPeso molecular:413.169Cycloleucine
CAS:Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.Fórmula:C6H11NO2Pureza:99.90%Cor e Forma:SolidPeso molecular:129.157CAIF
CAIF is an irreversible and selective allosteric covalent inhibitor of fucosyltransferase 8 (FUT8) with an IC50 of 5.7 μM. It hinders core fucosylation modification in cancer cells, thereby inhibiting their invasion and migration. CAIF is applicable in cancer research.β-1,4-GALT1-IN-1
β-1,4-GALT1-IN-1 (Compound 6) is a β-1,4-GALT1 inhibitor with an IC50 value of 6.2 μM. It is applicable in studying various pathological conditions, including cancer, autoimmune diseases, and viral infections.Fórmula:C29H23NO10Cor e Forma:SolidPeso molecular:545.494J6-3
J6-3 is an inhibitor of ICMT with an IC50 of 0.6 μM, exhibiting anticancer properties. The compound inhibits MDA-MB231 cells with an IC50 of 3.4 μM.Fórmula:C28H40N2Cor e Forma:SolidPeso molecular:404.31915L-739750 2HCl
L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.Fórmula:C23H41Cl2N3O6S2Pureza:97.01% - 99.16%Cor e Forma:SolidPeso molecular:590.621,3-β-Oligoglucan phosphorylase
1,3-β-Oligoglucanphosphorylase (EC 2.4.1.30) is a member of the glycosyltransferase family, specifically classified as a hexosyltransferase. This enzyme utilizes two substrates, (1,3-β-D-glucosyl) n and phosphate, to produce (1,3-β-D-glucosyl) n-1 and α-D-glucose-1-phosphate as its two products.Histamine glutarimide
CAS:Histamine glutarimide is a novel QPCT inhibitor that targets inflammatory processes like eosinophil migration, showing anti-asthmatic effects in animal models.Fórmula:C10H13N3O2Pureza:99.79%Cor e Forma:SolidPeso molecular:207.23R1-11
R1-11 is an indole-based ICMT inhibitor with an IC50 of 0.6 μM, exhibiting anticancer properties. It inhibits MDA-MB231 and PC3 cells with IC50 values of 2.2 μM and 2.0 μM, respectively.Fórmula:C25H37N5Cor e Forma:SolidPeso molecular:407.30491,4-α-Glucan 6-α-glucosyltransferase
1,4-α-Glucan 6-α-glucosyltransferase (EC 2.4.1.24) is part of the glycosyltransferase family, specifically classified as a hexosyltransferase.Sinbaglustat
CAS:Sinbaglustat (OGT2378), an oral N-alkyl iminosugar, inhibits GCS/GBA2 and treats lysosomal storage and neurodegenerative disorders.Fórmula:C11H23NO4Pureza:99.97%Cor e Forma:SolidPeso molecular:233.3046Squalene synthase-IN-2
Squalene synthase-IN-2 (compound isomer A-(1S, 3R)-14i) is an orally active inhibitor of squalene synthase, with IC50 values of 3.4 nM for squalene synthase and 99 nM for cholesterol synthesis enzymes. Squalene synthase-IN-2 effectively reduces plasma cholesterol and triglycerides.Fórmula:C31H39ClN2O6Cor e Forma:SolidPeso molecular:570.24966FTI-277
CAS:FTI-277, an FTase inhibitor, blocks H-Ras/K-Ras signaling and HDV infection; mimics Ras CAAX peptide.Fórmula:C22H29N3O3S2Pureza:99.63%Cor e Forma:White SolidPeso molecular:447.61BAY-593
CAS:BAY-593 is an orally active GGTase-I inhibitor capable of blocking YAP1/TAZ signaling in vivo, exhibiting antitumor activity.Fórmula:C26H31F3N2O3Cor e Forma:SolidPeso molecular:476.53PD 128042
CAS:PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.Fórmula:C23H39NO4Pureza:99.79%Cor e Forma:SolidPeso molecular:393.56Tipifarnib (S enantiomer)
CAS:Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).Fórmula:C27H22Cl2N4OPureza:99.2%Cor e Forma:SolidPeso molecular:489.396Nitecapone
CAS:Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)Fórmula:C12H11NO6Pureza:98.39%Cor e Forma:SolidPeso molecular:265.2188Ibiglustat
CAS:Ibiglustat (GZ402671) inhibits Glucosylceramide synthase, may treat Fabry disease by preventing GL-3 synthesis.Fórmula:C20H24FN3O2SPureza:97.97% - 98.81%Cor e Forma:White SolidPeso molecular:389.487Entacapone
CAS:Entacapone (OR-611) is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT).Fórmula:C14H15N3O5Pureza:98.80% - >99.99%Cor e Forma:Yellow Crystalline SolidPeso molecular:305.29CP-609754
CAS:CP-609754 shows selective inhibition of farnesyltransferase.Fórmula:C29H22ClN3O2Pureza:99.86% - 99.87%Cor e Forma:SolidPeso molecular:479.957
