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Desidrogenase

Desidrogenase

As desidrogenases são enzimas envolvidas nas reações de oxidação-redução das vias metabólicas, desempenhando um papel central na produção de energia e na respiração celular. Estas enzimas são cruciais para processos como o ciclo do ácido cítrico, a glicólise e a oxidação dos ácidos graxos. Os inibidores de desidrogenases são ferramentas importantes no estudo de doenças metabólicas, câncer e estresse oxidativo. Na CymitQuimica, oferecemos uma seleção abrangente de inibidores de desidrogenases para apoiar sua pesquisa em metabolismo, biologia do câncer e bioquímica.

Foram encontrados 267 produtos de "Desidrogenase"

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  • ML-148

    CAS:
    <p>ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).</p>
    Fórmula:C20H21N3O
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:319.4
  • DS18561882

    CAS:
    <p>DS18561882: Potent MTHFD2 inhibitor (IC50=0.0063), inhibits MTHFD1 (IC50=0.57), good oral kinetics.</p>
    Fórmula:C28H31F3N4O6S
    Pureza:98.19% - >99.99%
    Cor e Forma:Solid
    Peso molecular:608.63
  • Olorofim

    CAS:
    <p>Olorofim(F-901318)is a new selective antifungal compound that inhibits Aspergillus fumigatus DHODH (IC50: 44 nM). Cost-effective and quality-assured.</p>
    Fórmula:C28H27FN6O2
    Pureza:99.28%
    Cor e Forma:Solid
    Peso molecular:498.55
  • Qc1

    CAS:
    <p>Qc1 is an inhibitor of threonine dehydrogenase (TDH) inhibitor and can be used in studies about metabolic diseases.</p>
    Fórmula:C23H16F3N3O2S
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:455.45
  • CPS-11

    CAS:
    <p>CPS-11, a Thalidomide analogue, shows potent, broad antitumor activity, especially in multiple myeloma cells.</p>
    Fórmula:C14H12N2O5
    Pureza:99.8% - 99.98%
    Cor e Forma:Solid
    Peso molecular:288.26
  • ALDH1A3-IN-2

    CAS:
    <p>ALDH1A3-IN-2 is a potent ALDH1A3 inhibitor with an IC50 of 0.30 μM.ALDH1A3-IN-2 has potential for cancer disease research.</p>
    Fórmula:C13H17NO
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:203.28
  • PHGDH-IN-3

    CAS:
    <p>PHGDH-IN-3, an oral PHGDH blocker with 2.8 μM IC50, may help in cancer research.</p>
    Fórmula:C24H18FN3O4S2
    Pureza:97.24% - 98.55%
    Cor e Forma:Solid
    Peso molecular:495.55
  • HSD-016

    CAS:
    <p>HSD-016: Oral 11β-HSD1 inhibitor, active in humans, mice, rats (IC50: 11, 1, 8 nM), potential for type 2 diabetes research.</p>
    Fórmula:C21H21F7N2O3S
    Pureza:99.40% - >99.99%
    Cor e Forma:Solid
    Peso molecular:514.46
  • CM037

    CAS:
    <p>CM037 (A-37) is a selective ALDH1A1 (acetaldehyde dehydrogenase 1A1) inhibitor (IC50; 4.6 µM) with antitumor activity and may be used in studies to eliminate</p>
    Fórmula:C21H25N3O3S2
    Pureza:99.34%
    Cor e Forma:Solid
    Peso molecular:431.57
  • IDH2R140Q-IN-2

    CAS:
    <p>IDH2R140Q-IN-2 is an IDH2R140Q inhibitor indicated for the study of acute myeloid leukaemia (AML).</p>
    Fórmula:C21H18F6N6O
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:484.4
  • IGP-1

    CAS:
    <p>iGP-1 is a cell-permeable mitochondrial sn-Glycerol 3-phosphate dehydrogenase (mGPDH) inhibitor.</p>
    Fórmula:C17H15N3O3
    Pureza:99.12% - 99.15%
    Cor e Forma:Solid
    Peso molecular:309.32
  • PKUMDL-WQ-2101

    CAS:
    <p>PKUMDL-WQ-2101 is a selective allosteric inhibitor of phosphoglycerate dehydrogenase with anti-tumor activity.</p>
    Fórmula:C14H11N3O6
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:317.25
  • hDHODH-IN-7

    CAS:
    <p>hDHODH-IN-7 (DHODH-IN-9) is a nitrogen-containing analog and is a human dihydrorotatory dehydrogenase inhibitor.</p>
    Fórmula:C21H23FN4O
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:366.43
  • BMS-823778

    CAS:
    <p>BMS-823778 is a potent inhibitor of 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1) for the study of type 2 diabetes.</p>
    Fórmula:C18H18ClN3O
    Pureza:99.39% - 99.75%
    Cor e Forma:Solid
    Peso molecular:327.81
  • IMPDH2-IN-2

    CAS:
    <p>IMPDH2-IN-2 is an IMPDH inhibitor with antimicrobial activity and potential anti-tuberculosis activity for the study of inflammation and immune dysfunction.</p>
    Fórmula:C21H15Cl2N3O3
    Pureza:99.02%
    Cor e Forma:Solid
    Peso molecular:428.27
  • G6PD activator AG1

    CAS:
    <p>G6PD activator AG1 is a G6PD agonist that promotes G6PD oligomerization to a catalytically competent form.</p>
    Fórmula:C24H30N4S2
    Pureza:98.38% - 99.51%
    Cor e Forma:Solid
    Peso molecular:438.65
  • DSM421

    CAS:
    <p>DSM421 (DSM-421) is a dihydrodehydrogenase inhibitor (DHODH) that is in preclinical development as a potential treatment option for malaria and has shown</p>
    Fórmula:C14H11F5N6
    Pureza:98.23% - 99.82%
    Cor e Forma:Solid
    Peso molecular:358.27
  • HSD17B13-IN-2

    CAS:
    <p>HSD17B13-IN-2 (compound 1) serves as a potent inhibitor of hydroxysteroid 17ß-dehydrogenase 13 (HSD17B13) with demonstrable activity in cellular experiments [1</p>
    Fórmula:C21H23F2NO4
    Cor e Forma:Solid
    Peso molecular:391.41
  • α-Pyridoin

    CAS:
    <p>α-Pyridoin (α-pyridoin) is an enediol (enediol) compound that acts as a unique antioxidant.</p>
    Fórmula:C12H12N2O2
    Cor e Forma:Solid
    Peso molecular:216.24
  • IDH1 Inhibitor 2

    CAS:
    <p>IDH1 Inhibitor 2 (compound 13) is a potent IDH1 inhibitor via direct covalent modification of His315 (IC50: 110 nM).</p>
    Fórmula:C26H22N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:406.48