Fosfolipase
As fosfolipases são um grupo de enzimas que hidrolisam fosfolipídios em ácidos graxos e outras substâncias lipofílicas, desempenhando um papel crítico na biologia das membranas e na geração de moléculas sinalizadoras. Inibidores de fosfolipases são usados para estudar seu papel em doenças inflamatórias, distúrbios cardiovasculares e neurodegeneração. Esses inibidores também são valiosos na exploração de vias de sinalização lipídica e suas implicações nos mecanismos de doenças. Na CymitQuimica, oferecemos uma variedade de inibidores de fosfolipases para apoiar sua pesquisa em inflamação, metabolismo lipídico e sinalização celular.
Foram encontrados 84 produtos de "Fosfolipase"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Lansoprazole
CAS:Lansoprazole (A-65006) is a 2, 2, 2-trifluoroethoxypyridyl derivative of timoprazole that is used in the therapy of STOMACH ULCERS and ZOLLINGER-ELLISONFórmula:C16H14F3N3O2SPureza:99.18% - 99.84%Cor e Forma:White Crystalline PowderPeso molecular:369.36ML349
CAS:ML349 is an inhibitor of LYPLA2 (IC50: 144 nM). ML349 is an effective and specific acyl protein thioesterase 2 (APT-2) inhibitor (Ki: 120 nM).Fórmula:C23H22N2O4S2Pureza:99.59% - 99.88%Cor e Forma:SolidPeso molecular:454.56Lp-PLA2-IN-1
CAS:Lp-PLA2-IN-1 suppresses Lp-PLA2, aiding in treating atherosclerosis and Alzheimer's.
Fórmula:C21H17F5N4O3Pureza:99.60%Cor e Forma:SolidPeso molecular:468.38Omeprazole
CAS:Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor.Fórmula:C17H19N3O3SPureza:98.43% - 98.48%Cor e Forma:White SolidPeso molecular:345.42Tris(2,4-di-tert-butylphenyl)phosphate
CAS:Tris(2,4-di-tert-butylphenyl)phosphate (TDTBPP) inhibits secretory phospholipase A2 (sPLA2) with anti-inflammatory effect. Cost-effective and quality-assured.Fórmula:C42H63O4PPureza:99.73%Cor e Forma:SolidPeso molecular:662.92A3373
CAS:A3373 is a novel inhibitor targeting both Phospholipase D1 (PLD1) and Phospholipase D2 (PLD2), demonstrating half maximal inhibitory concentrations (IC50) ofFórmula:C17H9F7N2OPureza:98%Cor e Forma:SoildPeso molecular:390.26Compound 48/80 trihydrochloride
CAS:Compound 48/80 trihydrochloride (C48/80 trihydrochloride) 是 N-甲基对甲氧基苯乙胺和甲醛发生缩合反应后的混合物。Compound 48/80 trihydrochloride 是一种肥大细胞 (mast cell) 脱颗粒剂和组胺 (histamine) 释放剂。Compound 48/80 trihydrochloride 对人血小板磷脂酰肌醇特异性磷脂酶 C (phosphatidylinositol-specific phospholipase C) 活性有抑制作用。
Fórmula:C32H48Cl3N3O3Pureza:98%Cor e Forma:SolidPeso molecular:629.1SB-435495
CAS:SB-435495 is a compound characterized by its potent, selective, reversible, and non-covalent inhibition of Lp-PLA2, demonstrating an IC50 value of 0.06 nM.Fórmula:C38H40F4N6O2SPureza:99.07%Cor e Forma:SolidPeso molecular:720.82nSMase2-IN-1
nSMase2-IN-1 is an orally active inhibitor of Neutral sphingomyelinase 2 (nSMase2) with a potent IC50 value of 0.13 ± 0.06 μM.Fórmula:C12H17N5OPureza:98%Cor e Forma:SolidPeso molecular:247.3LEI110
CAS:LEI110 inhibits PLA2G16 and HRASLS enzymes, Ki 20 nM, selectively targets related thiol hydrolases.Fórmula:C25H23F3N2O3Pureza:98.66% - 98.8%Cor e Forma:SolidPeso molecular:456.46sPLA2 inhibitor 2
sPLA2 inhibitor 2 (compound 6a) is an sPLA2 inhibitor with an IC50 value of 0.0475 μM, making it valuable for diabetes research.Fórmula:C20H18N6O4S2Cor e Forma:SolidPeso molecular:470.52Melittin Acetate
Melittin Acetate, a PLA2 activator, enhances low-weight PLA2 activity but not high-weight PLA2.Fórmula:C133H233N39O33Pureza:99.78%Cor e Forma:SoildPeso molecular:2906.51A4333
A4333, a biotinylated derivative of A3373, selectively inhibits Phospholipase D1 (PLD1) while sparing PLD2.Pureza:98%Cor e Forma:Odour SolidDPTIP
CAS:DPTIP is an effective inhibitor of neutral sphingomyelinase 2 with an IC50 value of 30 nM.Fórmula:C21H18N2O3SPureza:99.88%Cor e Forma:SolidPeso molecular:378.44Ref: TM-T60043
1mg48,00€2mg63,00€5mg96,00€1mL*10mM (DMSO)96,00€10mg153,00€25mg298,00€50mg487,00€100mg710,00€ASM-IN-3
CAS:ASM-IN-3 (Compound 21b) is a selective acid sphingomyelinase (ASM) inhibitor that can penetrate the blood-brain barrier, with an IC50 of 3.37 μM against purified human ASM. By inhibiting ASM activity in the hippocampus and promoting neurogenesis, ASM-IN-3 alleviates depressive-like behavior in reserpine-induced depressive rats.Fórmula:C17H13ClN2O4Cor e Forma:SolidPeso molecular:344.75BIRM 271
CAS:BIRM 271 is a novel arachidonic acid release inhibitor that blocks leukotriene B4 and platelet-activating factor biosynthesis in human neutrophils.
Fórmula:C21H25N3OPureza:99.64%Cor e Forma:SoildPeso molecular:335.44VU533
CAS:VU533 is a NAPE-PLD activator, EC50=0.30 µM, boosts macrophage activity, potential in cardiometabolic diseases.Fórmula:C21H22FN3O3S2Pureza:99.87%Cor e Forma:SolidPeso molecular:447.55DPTIP hydrochloride
CAS:DPTIP hydrochloride is a potent inhibitor of neutral sphingomyelinase (N-SMase 2) that can cross the blood-brain barrier. It acts as an exosome inhibitor with an IC50 value of 30 nM.Fórmula:C21H19ClN2O3SCor e Forma:SolidPeso molecular:414.91PLA2-IN-1
PLA2-IN-1 (Compound 7) is a potent and selective inhibitor of phospholipase A (PLA2) with an IC50 value of 1 nM. It effectively inhibits PLA2-induced coagulation disorders in vitro and shows potential for use as an antidote for snake bites caused by cobra venom.Cor e Forma:Odour Solid1-Myristoyl-2-Linoleoyl-sn-glycero-3-PC
CAS:1-Myristoyl-2-Linoleoyl-sn-glycero-3-PC is a phospholipid identified in human plasma, characterized by the presence of Myristic acid and Linoleic acid at the sn-1 and sn-2 positions, respectively.Fórmula:C40H76NO8PCor e Forma:SolidPeso molecular:730.01AACOCF3
CAS:AACOCF3 (Arachidonyl trifluoromethyl ketone) is a cell-permeable trifluoromethyl ketone analog of arachidonic acid.Fórmula:C21H31F3OPureza:99% - 99%Cor e Forma:Yellow LiquidPeso molecular:356.47MJ33 lithium salt
CAS:MJ33 lithium salt is an inhibitor of NADPH oxidase type 2-mediated ROS generation, inhibits PLA2 activity, and can be used to study acute lung injury.Fórmula:C22H43F3LiO6PPureza:99%Cor e Forma:SolidPeso molecular:498.48BMS493
CAS:BMS493 is an inverse agonist of RAR that inhibits retinoic acid-induced differentiation and inhibits the increase in phospholipase A2 activity.Fórmula:C29H24O2Pureza:99.12% - >99.99%Cor e Forma:SolidPeso molecular:404.5PACOCF3
CAS:PACOCF3, a phospholipase A2 inhibitor, hinders Ca2+ signaling with an IC50 of 3.8 μM in renal cells.Fórmula:C17H31F3OPureza:99.93%Cor e Forma:SolidPeso molecular:308.42Phospholipase A2
CAS:Phospholipase A2 (PLA2) is an enzyme that hydrolyzes fatty acids present in the sn-2 position of phospholipids and is closely related to lipid metabolism.Cor e Forma:SolidLEI-401
CAS:LEI-401 is a NAPE-PLD inhibitor.LEI-401 reduces the level of n-acyl ethanolamines in the brain of free-ranging mice and modulates their emotional behaviour.Fórmula:C24H31N5O2Pureza:99.79% - 99.79%Cor e Forma:SolidPeso molecular:421.54Bromoenol lactone
CAS:NeurokininBromoenol lactone ((6E)-Bromoenol lactone) is an iPLA2β and serine protease inhibitor that attenuates nicotine-induced breast cancer cell proliferation.Fórmula:C16H13BrO2Cor e Forma:SolidPeso molecular:317.18AA26-9
CAS:AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.Fórmula:C7H10N4OPureza:99.88%Cor e Forma:SolidPeso molecular:166.18Ref: TM-T3990
1mg34,00€2mg49,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg113,00€25mg200,00€50mg333,00€100mg495,00€N-(p-amylcinnamoyl) Anthranilic Acid
CAS:N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.Fórmula:C21H23NO3Pureza:99.35% - 99.67%Cor e Forma:SolidPeso molecular:337.41Rhamnetin
CAS:Rhamnetin (beta-Rhamnocitrin), a quercetin derivative found in Coriandrum sativum, has antioxidant and anti-inflammatory activities.Fórmula:C16H12O7Pureza:99.61% - 99.905%Cor e Forma:SolidPeso molecular:316.26Ref: TM-TN1419
1mg60,00€5mg130,00€1mL*10mM (DMSO)137,00€10mg200,00€25mg338,00€50mg497,00€100mg708,00€hnps-PLA Inhibitor
CAS:Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).
Fórmula:C21H21N3O4Pureza:99.68%Cor e Forma:SolidPeso molecular:379.41Varespladib
CAS:Varespladib (LY315920) inhibits hnsPLA2 effectively (IC50=7 nM), studied for sickle cell, VOC, and acute coronary syndrome.Fórmula:C21H20N2O5Pureza:99.97%Cor e Forma:SolidPeso molecular:380.39Ref: TM-T2044
1mg46,00€1mL*10mM (DMSO)81,00€5mg87,00€10mg144,00€25mg227,00€50mg338,00€100mg487,00€200mg705,00€BAPTA
CAS:BAPTA is a neuroprotective agent in cerebral ischemia, acting as an intercellular Ca2+ chelator.Fórmula:C22H24N2O10Pureza:97.21% - ≥95%Cor e Forma:White SolidPeso molecular:476.43Rapanone
CAS:Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) is a natural benzoquinone that is a potent and selective inhibitor of human synovial PLA2.Fórmula:C19H30O4Pureza:99.56%Cor e Forma:SolidPeso molecular:322.44U-73343
CAS:U-73343 is an inactive analog of U-73122 and can be used as a negative control. U-73122 dose-dependently inhibits acid secretion irrespective of the stimulant.Fórmula:C29H42N2O3Pureza:99.06%Cor e Forma:SolidPeso molecular:466.66Tanshinone I
CAS:Tanshinone I (Tanshinone A), an active principle isolated from the herbal medicine Salvia miltiorrhiza, displays cytotoxicity against tumor cells.Fórmula:C18H12O3Pureza:98.31% - 98.70%Cor e Forma:SolidPeso molecular:276.29ML348
CAS:ML348 (GNF-Pf-1127) is a selective and reversible lysophospholipase 1 (LYPLA1) inhibitor (IC50 = 210 nM).Fórmula:C18H17ClF3N3O3Pureza:99% - 99.88%Cor e Forma:SolidPeso molecular:415.79Ref: TM-T3439
2mg44,00€5mg65,00€10mg92,00€25mg215,00€50mg334,00€100mg537,00€200mg750,00€500mg1.134,00€FIPI
CAS:FIPI, a halopemide derivative, strongly blocks PLD1 and PLD2 (IC50s: 25 nM, 20 nM) and hinders PLD-mediated cell activity.Fórmula:C23H24FN5O2Pureza:97.21% - 98.68%Cor e Forma:SolidPeso molecular:421.47ML-298
CAS:ML-298 (CID53393915) is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).Fórmula:C22H23F3N4O2Pureza:99.35%Cor e Forma:SolidPeso molecular:432.441-Naphthaleneacetic acid
CAS:1-Naphthaleneacetic acid, an auxin-like synthetic plant hormone, boosts rooting in horticulture.Fórmula:C12H10O2Pureza:98.67%Cor e Forma:Needles From Water White To Off White CrystalsPeso molecular:186.21ST271
CAS:ST271 is an effective protein tyrosine kinase (PTK) inhibitor.
Fórmula:C16H20N2O2Pureza:98.94%Cor e Forma:SolidPeso molecular:272.34Darapladib
CAS:Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.Fórmula:C36H38F4N4O2SPureza:99.82% - >99.99%Cor e Forma:SolidPeso molecular:666.77Ref: TM-T6109
200mgA consultar1mg42,00€2mg52,00€5mg87,00€1mL*10mM (DMSO)116,00€10mg125,00€25mg180,00€50mg309,00€100mg499,00€RHC 80267
CAS:RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)Fórmula:C20H34N4O4Pureza:99.54%Cor e Forma:White SolidPeso molecular:394.51GW4869
CAS:GW4869 (GW69A) is a selective and non-competitive inhibitor of neutral sphingomyelinase N-SMase (IC50=1 μM).Fórmula:C30H30Cl2N6O2Pureza:98.12% - 98.47%Cor e Forma:SolidPeso molecular:577.5Anti-Inflammatory Peptide 1 Acetate
Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) inhibits PLA2 to reduce inflammation and pain.Fórmula:C47H86N12O16S2Pureza:98.95%Cor e Forma:SolidPeso molecular:1139.391-Linoleoyl Glycerol
CAS:1-Linoleoyl Glycerol (Monolinolein) is fatty acid glycerol that has been isolated from Saururus Chinensis roots.Fórmula:C21H38O4Pureza:98.95% - 99.15%Cor e Forma:Less Oil Colourless OilPeso molecular:354.52ONO-RS-082
CAS:ONO-RS-082 is a Ca2+-independent phospholipase A2 inhibitor.Fórmula:C21H22ClNO3Pureza:99.35%Cor e Forma:SolidPeso molecular:371.86Ref: TM-T21815
2mg39,00€5mg58,00€1mL*10mM (DMSO)64,00€10mg96,00€25mg167,00€50mg268,00€100mg401,00€200mg580,00€ML-211
CAS:ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the related LYPLA2 (IC50 = 30 nM)
Fórmula:C25H30N4O2Pureza:97.07%Cor e Forma:SolidPeso molecular:418.531-Naphthaleneacetic acid potassium salt
CAS:1-Naphthaleneacetic acid potassium salt (1-NAA Potassium Salt) is a synthetic phytogrowth hormone that promotes plant growth and a PLA2 inhibitor.Fórmula:C12H9O2·KPureza:97.68%Cor e Forma:Off-White To Beige PowderPeso molecular:224.3Difluprednate
CAS:Difluprednate (Myser)(Durezol) is a corticosteroid, approved for the treatment of post-operative ocular inflammation and pain.Fórmula:C27H34F2O7Pureza:99.23% - 99.86%Cor e Forma:SolidPeso molecular:508.55Cambinol
CAS:Cambinol is a SIRT1/2 inhibitor (IC50: 56/59 μM), non-competitive with NAD, weak on SIRT5, and prompts apoptosis in lymphoma cells.Fórmula:C21H16N2O2SPureza:98.02% - 99.83%Cor e Forma:SolidPeso molecular:360.43Ref: TM-T4019
1mg38,00€2mg50,00€1mL*10mM (DMSO)63,00€5mg80,00€10mg117,00€25mg207,00€50mg333,00€100mg495,00€500mg1.071,00€CAY10594
CAS:CAY10594, a PLD2 inhibitor, mitigates acetaminophen liver damage via the p-GSK-3β/JNK pathway.Fórmula:C26H28N4O2Pureza:98%Cor e Forma:SolidPeso molecular:428.53trans-Benzylideneacetone
CAS:trans-Benzylideneacetone (Acetocinnamone) is used in various synthetic preparations.Fórmula:C10H10OPureza:97.48%Cor e Forma:Light Yellow Low Melting Crystalline MassPeso molecular:146.19Aristolochic acid C
CAS:Aristolochic acid C is a derivative of Aristolochic acid which is a phospholipase A2 inhibitor.Fórmula:C16H9NO7Pureza:99.8%Cor e Forma:White PowderPeso molecular:327.25CAY10650
CAS:CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).Fórmula:C28H25NO6Pureza:97.33%Cor e Forma:SolidPeso molecular:471.5Ref: TM-TQ0105
1mg49,00€5mg114,00€1mL*10mM (DMSO)118,00€10mg172,00€25mg334,00€50mg467,00€100mg620,00€U-73122
CAS:U-73122 (U73122) , an effective PLC inhibitor, reduces agonist-induced Ca2+ increases in platelets and PMN.Fórmula:C29H40N2O3Pureza:97.50%Cor e Forma:Solid Off-WhitePeso molecular:464.64m-3M3FBS
CAS:m-3M3FBS is a phospholipase C (PLC) activator.Fórmula:C16H16F3NO2SPureza:99.66%Cor e Forma:SolidPeso molecular:343.36Melittin
CAS:Melittin: principal bee venom toxin, 26 amino acids, activates low-weight PLA2, not high-weight PLA2.Fórmula:C131H229N39O31Pureza:98.37% - 99.92%Cor e Forma:SolidPeso molecular:2846.46Neomycin sulfate
CAS:Neomycin sulfate (Framycin sulfate) is a broad-spectrum aminoglycoside antibiotic that blocks the synthesis of bacterial proteins in order to exertFórmula:C23H46N6O13·3H2SO4Pureza:99.4% - 99.88%Cor e Forma:Tan PowderPeso molecular:908.87VU0155056
CAS:VU0155056 is a dual PLD1/2 inhibitor with IC50 < 1 µM in cellular assays, inhibits breast cancer cell invasion.Fórmula:C25H26N4O2Pureza:98.6% - 99.15%Cor e Forma:SolidPeso molecular:414.5LCL521
CAS:LCL521 inhibits lysosomal acid sphingomyelinase (ASMase).LCL521 is an acid ceramidase (ACDase) inhibitor.Fórmula:C31H52N4O7Pureza:98%Cor e Forma:SolidPeso molecular:592.77Omeprazole Sodium
CAS:Omeprazole Sodium is a proton pump inhibitor(PPI) and suppresses gastric acid secretion.Fórmula:C17H18N3NaO3SPureza:99.84%Cor e Forma:Clear In WaterPeso molecular:367.42-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
CAS:2-Decenoylaminoethyl cyclohexylethyl sulfide prevents stress ulcers, stabilizes phospholipase A2 and prostaglandin E2.Fórmula:C20H37NOSPureza:98%Cor e Forma:SolidPeso molecular:339.58ML299
CAS:ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).Fórmula:C23H26BrFN4O2Pureza:98.23%Cor e Forma:SolidPeso molecular:489.38Ref: TM-T8968
100mgA consultar1mL*10mM (DMSO)A consultar500µg101,00€1mg152,00€5mg371,00€10mg558,00€25mg868,00€50mg1.153,00€Lp-PLA2-IN-3
CAS:Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.Fórmula:C20H13ClF3N3O3SPureza:99.84%Cor e Forma:SolidPeso molecular:467.85Ref: TM-T11874
1mg90,00€2mg132,00€5mg215,00€1mL*10mM (DMSO)220,00€10mg340,00€25mg565,00€50mg797,00€100mg1.063,00€500mg2.142,00€ASM-IN-1
CAS:ASM-IN-1: Oral acid sphingomyelinase inhibitor, IC50 = 1.5 µM; reduces lipid plaques, plasma ceramide, Ox-LDL.Fórmula:C16H12BrN3O4Pureza:98%Cor e Forma:SolidPeso molecular:390.19GK187
CAS:GK187 is a selective and potent Group VIA calcium-independent phospholipase A2 (GVIA iPLA2) inhibitor, used in the study of neurological disorders.Fórmula:C14H15F5O2Cor e Forma:SolidPeso molecular:310.26Ref: TM-T37221
1mg79,00€5mg172,00€1mL*10mM (DMSO)178,00€10mg268,00€25mg510,00€50mg802,00€100mg1.305,00€Halopemide
CAS:Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Fórmula:C21H22ClFN4O2Pureza:96.57%Cor e Forma:SolidPeso molecular:416.88Giripladib
CAS:Giripladib (PLA695/PLX-695) blocks radiation-boosted phosphorylation of ERK and Akt in endothelial cells.
Fórmula:C41H36ClF3N2O4SPureza:99.64%Cor e Forma:SolidPeso molecular:745.25VU0155069
CAS:VU0155069, a selective PLD1 inhibitor (IC50: 46 nM), halts cancer cell migration in transwell assays.Fórmula:C26H27ClN4O2Pureza:99.5%Cor e Forma:SolidPeso molecular:462.97VU0364739
CAS:VU0364739, a selective phospholipase D2 (PLD2) inhibitor with an IC50 of 22 nM, effectively reduces cancer cell proliferation [1].Fórmula:C26H27FN4O2Pureza:98%Cor e Forma:SolidPeso molecular:446.52Lp-PLA2-IN-13
CAS:Lp-PLA2-IN-13 (compound 15), a potent Lp-PLA2 inhibitor, holds potential for research in neurodegenerative-related diseases [1].Fórmula:C22H17F5N4O4Pureza:98%Cor e Forma:SolidPeso molecular:496.39Lp-PLA2-IN-2
CAS:Lp-PLA2-IN-2 is a selective and potent lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor, with an IC50 0f 120 nM for recombinant human Lp-PLA2.Fórmula:C19H23FN2O4SPureza:98%Cor e Forma:SolidPeso molecular:394.46Lp-PLA2-IN-14
CAS:Lp-PLA2-IN-14 (Compound 19), an inhibitor of rhLp-PLA2, exhibits a potent inhibitory effect with a pIC50 value of 8.4.Fórmula:C16H14F3N3O3Pureza:98%Cor e Forma:SolidPeso molecular:353.37,7-Dimethyl-(5Z,8Z)-eicosadienoic acid
CAS:7,7-Dimethyl-(5Z,8Z)-eicosadienoic acid (DEDA, 5 μM) significantly impacts the response to βA(25-35) stimulation. It reduces the formation of ROS.Fórmula:C22H40O2Cor e Forma:SolidPeso molecular:336.55Varespladib methyl
CAS:Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.Fórmula:C22H22N2O5Pureza:99.42% - 99.97%Cor e Forma:SolidPeso molecular:394.42Ref: TM-T17218
1mg93,00€2mg123,00€5mg200,00€1mL*10mM (DMSO)220,00€10mg319,00€25mg528,00€50mg730,00€100mg999,00€200mg1.333,00€Ecopladib
CAS:Ecopladib inhibits cPLA2α with IC50 of 0.15 μM (micelles) & 0.11 μM (rat blood).Fórmula:C39H33Cl3N2O5SPureza:95.15%Cor e Forma:SolidPeso molecular:748.11Ref: TM-T11149
1mL*10mM (DMSO)A consultar1mg315,00€5mg630,00€10mg850,00€25mg1.234,00€50mg1.693,00€100mg2.305,00€Rilapladib
CAS:Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activatingFórmula:C40H38F5N3O3SPureza:99.92%Cor e Forma:SolidPeso molecular:735.8Ref: TM-T16751
1mg87,00€5mg215,00€10mg349,00€1mL*10mM (DMSO)349,00€25mg537,00€50mg745,00€100mg1.108,00€200mg1.504,00€MAFP
CAS:MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase.Fórmula:C21H36FO2PCor e Forma:SolidPeso molecular:370.48GK420
CAS:GK420 (AVX420) is a potent inhibitor of cytoplasmic phospholipase A2α (cPLA2α), with an XI(50) value of 0.0016. It effectively inhibits the release of arachidonic acid, with an EC50 of 0.09 μM. GK420 plays a significant role in cancer research.Fórmula:C20H25NO5SCor e Forma:SolidPeso molecular:391.481Ro 23-9358
CAS:Ro 23-9358 is a potent inhibitor of secretory phospholipase A2, exhibiting anti-inflammatory properties.Fórmula:C30H51NO6Cor e Forma:SolidPeso molecular:521.729Lp-PLA2-IN-16
CAS:Lp-PLA2-IN-16 (Example 1) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential applications in Alzheimer's disease research [1].
Fórmula:C22H17F5N4O3Pureza:98%Cor e Forma:SolidPeso molecular:480.39Ref: TM-T79076
Produto descontinuadoLp-PLA2-IN-12
CAS:Lp-PLA2-IN-12 (compound 19), an Lp-PLA2 inhibitor, is utilized in researching neurodegenerative diseases including Alzheimer's disease (AD), glaucoma, age-
Fórmula:C24H23F2N5O3Pureza:98%Cor e Forma:SolidPeso molecular:467.47Ref: TM-T79010
Produto descontinuadoLp-PLA2-IN-15
CAS:Lp-PLA2-IN-15 (example 2) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential application in Alzheimer's disease research [1].
Fórmula:C22H17F5N4O3Pureza:98%Cor e Forma:SolidPeso molecular:480.39Ref: TM-T79075
Produto descontinuado
