
Receptor adrenérgico
Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.
Subcategorias de "Receptor adrenérgico"
Foram encontrados 645 produtos de "Receptor adrenérgico"
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(±)-N-Methylcoclaurine
CAS:<p>N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].</p>Fórmula:C18H21NO3Pureza:98%Cor e Forma:SolidPeso molecular:299.36Todralazine hydrochloride
CAS:<p>Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.</p>Fórmula:C11H13ClN4O2Pureza:99.91%Cor e Forma:SolidPeso molecular:268.7BMS-194449
CAS:<p>BMS-194449 is a full beta 3 agonist.</p>Fórmula:C24H24F4N2O6SCor e Forma:SolidPeso molecular:544.52Celiprolol hydrochloride
CAS:<p>Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.</p>Fórmula:C20H33N3O4·HClCor e Forma:White Crystalline SolidPeso molecular:415.96Bunazosin Hydrochloride
CAS:<p>Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.</p>Fórmula:C19H28ClN5O3Pureza:99.12%Cor e Forma:SolidPeso molecular:409.91BU-E 75
CAS:<p>BU-E 75 is an agonist of the histamine H2.</p>Fórmula:C21H24F2N6Cor e Forma:SolidPeso molecular:398.45β3-AR agonist 1
CAS:<p>β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/</p>Fórmula:C22H28N4O4SPureza:98%Cor e Forma:SolidPeso molecular:444.55L-796568 free base
CAS:<p>L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).</p>Fórmula:C31H27F3N4O3S2Cor e Forma:SolidPeso molecular:624.7RS100329 hydrochloride
CAS:<p>RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.</p>Fórmula:C20H26ClF3N4O3Pureza:99.95%Cor e Forma:SolidPeso molecular:462.89Bufuralol (hydrochloride)
CAS:<p>Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.</p>Fórmula:C16H24ClNO2Cor e Forma:SolidPeso molecular:297.82LK 204-545
CAS:<p>LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.</p>Fórmula:C25H32N4O6Cor e Forma:SolidPeso molecular:484.54NGD9002
CAS:<p>NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.</p>Fórmula:C20H31N5OPureza:98%Cor e Forma:SolidPeso molecular:357.49L-796568 dihydrochloride
CAS:<p>L-796568: potent β3 agonist (EC50 = 3.6 nM), >600-fold selectivity vs β1/β2, good oral bioavailability, long action.</p>Fórmula:C31H29Cl2F3N4O3S2Cor e Forma:SolidPeso molecular:697.62RS 17053 hydrochloride
CAS:<p>RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.</p>Fórmula:C24H30Cl2N2O2Pureza:99.27%Cor e Forma:SolidPeso molecular:449.41Ritodrine
CAS:<p>Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].</p>Fórmula:C17H21NO3Cor e Forma:SolidPeso molecular:287.35Binedaline
CAS:<p>Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.</p>Fórmula:C19H23N3Pureza:98%Cor e Forma:SolidPeso molecular:293.41Epinephrine HCl
CAS:<p>Epinephrine HCl is a hormone and neurotransmitter secreted by the adrenal medulla, agonist of α-adrenergic and β-adrenergic receptor.</p>Fórmula:C9H14ClNO3Pureza:99.48%Cor e Forma:SolidPeso molecular:219.67Dibenamine hydrochloride
CAS:<p>Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.</p>Fórmula:C16H19Cl2NPureza:96.43%Cor e Forma:Oily Liquid SolidPeso molecular:296.23AR-08
CAS:<p>AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.</p>Fórmula:C12H12N6Pureza:99.7%Cor e Forma:SolidPeso molecular:240.26Fiduxosin
CAS:<p>Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with Ki</p>Fórmula:C30H29N5O4SPureza:99.73%Cor e Forma:SolidPeso molecular:555.65
