Receptor adrenérgico
Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.
Subcategorias de "Receptor adrenérgico"
Foram encontrados 645 produtos de "Receptor adrenérgico"
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Pronetalol
CAS:<p>Pronethalol ((±)-Pronethalol), a non-selective β-adrenergic antagonist, effectively inhibits Sox2 expression and offers protection against Digitalis-induced ventricular arrhythmias. Additionally, it can reverse such arrhythmias and limit the development of cerebral arteriovenous malformations (AVMs) [1] [2].</p>Fórmula:C15H19NOCor e Forma:SolidPeso molecular:229.32SDZ-NVI-085
CAS:<p>SDZ-NVI-085 is an α1 adrenergic receptor agonist and a competitive antagonist of 5-hydroxytryptamine.</p>Fórmula:C15H21NO2SCor e Forma:SolidPeso molecular:279.4Lidamidine
CAS:<p>Lidamidine (Lidamidinum) is an effective antidiarrheal agent that inhibits intestinal secretion, reduces intestinal transit, and inhibits smooth muscle</p>Fórmula:C11H16N4OPureza:99.98%Cor e Forma:SolidPeso molecular:220.27Ro-70-0004
CAS:<p>Ro-70-0004 is a selective antagonist of alpha1A-adrenoceptor.</p>Fórmula:C20H24F4N4O3Cor e Forma:SolidPeso molecular:444.42KUC-7322
CAS:<p>Ritobegron is used as a selective β3-adrenoceptor agonist and the prodrug of the active compound, KUC-7322.</p>Fórmula:C21H27NO5Cor e Forma:SolidPeso molecular:373.44Vemtoberant
CAS:<p>Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.</p>Fórmula:C29H37N3O8S2Cor e Forma:SolidPeso molecular:619.75Phentolamine Analogue 1
CAS:<p>Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.</p>Fórmula:C17H19N3OPureza:99.96%Cor e Forma:SolidPeso molecular:281.35Bufuralol
CAS:<p>Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.</p>Fórmula:C16H23NO2Pureza:98.26%Cor e Forma:SolidPeso molecular:261.36GW-597901
CAS:<p>GW-597901, an β2 adrenergic receptor agonist, is used potentially for the treatment of asthma and chronic obstructive.</p>Fórmula:C25H38N2O6SCor e Forma:SolidPeso molecular:494.64Domesticine, (-)-
CAS:<p>Domesticine, (-)- is an antagonist of alpha-1D-adrenoceptor.</p>Fórmula:C19H19NO4Pureza:98%Cor e Forma:SolidPeso molecular:325.360990CL
CAS:<p>0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMP</p>Fórmula:C21H21N5Pureza:98.58%Cor e Forma:SolidPeso molecular:343.42α1 adrenoceptor-MO-1
CAS:<p>α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.</p>Fórmula:C20H24ClN5OPureza:99.20% - 99.29%Cor e Forma:SolidPeso molecular:385.89OPC-28326
CAS:<p>OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.</p>Fórmula:C26H35N3O2Pureza:99.79%Cor e Forma:SolidPeso molecular:421.58CGP-20712
CAS:<p>CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.</p>Fórmula:C23H25F3N4O5Pureza:99.40% - 99.58%Cor e Forma:SolidPeso molecular:494.46(±)-Prenalterol
CAS:<p>(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.</p>Fórmula:C12H19NO3Pureza:99.73%Cor e Forma:SolidPeso molecular:225.28Talibegron hydrochloride
CAS:<p>Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.</p>Fórmula:C18H22ClNO4Pureza:99.82%Cor e Forma:SolidPeso molecular:351.83Deriglidole
CAS:<p>Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.</p>Fórmula:C16H21N3Pureza:97.31% - 98.23%Cor e Forma:SolidPeso molecular:255.36(±)-Penbutolol
CAS:<p>(±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic receptor antagonist. (±)-Penbutolol mitigates the tachycardia induced by exercise, reduces the increase in peak expiratory flow rate (PEFR) caused by physical activity, and decreases plasma renin activity (PRA) at rest. The peak plasma concentration of this compound is achieved one hour after oral administration, with a half-life of 4.5 hours, and it is metabolized into active metabolites in the body. This compound is utilized in research related to cardiovascular diseases.</p>Fórmula:C18H29NO2Cor e Forma:SolidPeso molecular:291.43TAAR1 agonist 3
CAS:<p>TAAR1 agonist 3 is a potent agonist of Trace Amine-Associated Receptor 1 (TAAR1) with a pEC50 value of 7.6. Additionally, it acts as a full agonist at the α2AR with a pEC50 of 6. TAAR1 agonist 3 is utilized in the research of neuropsychiatric disorders.</p>Fórmula:C10H13NOCor e Forma:SolidPeso molecular:163.22Teoprolol
CAS:<p>Teoprolol is a blocker of β-adrenergic receptor.</p>Fórmula:C23H30N6O4Pureza:98%Cor e Forma:SolidPeso molecular:454.52
