
Receptor adrenérgico
Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.
Subcategorias de "Receptor adrenérgico"
Foram encontrados 709 produtos de "Receptor adrenérgico"
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Meluadrine tartrate
CAS:<p>Meluadrine tartrate is an endogenous metabolite.</p>Fórmula:C16H24ClNO8Pureza:98%Cor e Forma:SolidPeso molecular:393.82Besipirdine hydrochloride
CAS:<p>Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.</p>Fórmula:C16H18ClN3Pureza:98.45%Cor e Forma:SoildPeso molecular:287.79Oxaprotiline hydrochloride
CAS:Oxaprotiline hydrochloride is an antidepressant.Fórmula:C20H24ClNOPureza:98%Cor e Forma:SolidPeso molecular:329.86L-770644 dihydrochloride
CAS:L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.Fórmula:C30H38ClN7O4SCor e Forma:SolidPeso molecular:628.19O-Desmethyl Mebeverine alcohol
CAS:Mebeverine metabolite O-desmethyl alcohol inhibits α1 receptors, relaxing the gut.Fórmula:C15H25NO2Pureza:98%Cor e Forma:SolidPeso molecular:251.36Desglymidodrine
CAS:Desglymidodrine (ST 1059) is an α1-adrenoceptor agonist and vasoconstrictor, used in cardiovascular research and neurocardiogenic syncope studies.Fórmula:C10H15NO3Pureza:99.56%Cor e Forma:SolidPeso molecular:197.23Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.Fórmula:C22H30N2O7SPureza:97.05% - 98.53%Cor e Forma:SoildPeso molecular:466.55Carvedilol
CAS:<p>Carvedilol (SKF 105517) Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intrinsic sympathomimetic activity. The S enantiomer of carvedilol nonselectively binds to and blocks beta-adrenergic receptors, thereby exerting negative inotropic and chronotropic effects, and leading to a reduction in cardiac output. In addition, both enantiomers of carvedilol bind to and block alpha 1-adrenergic receptors, thereby causing vasodilation and reducing peripheral vascular resistance.</p>Fórmula:C24H26N2O4Pureza:99.73% - 99.97%Cor e Forma:Colourless Crystalline PowderPeso molecular:406.47AG-825
CAS:AG-825(Tyrphostin C15) is a selective and competitive ErbB2 inhibitor that inhibits tyrosine phosphorylation with an IC50 value of 0.35 μM.AG-825 (TyrphostinFórmula:C19H15N3O3S2Pureza:99.52%Cor e Forma:Yellow SolidPeso molecular:397.47Carbazochrome salicylate
CAS:Carbazochrome salicylate can be used as a coagulant.Fórmula:C17H18N4NaO6Cor e Forma:White Crystalline PowderPeso molecular:397.343Bromchlorbuterol hydrochloride
CAS:Bromchlorbuterol HCl, a potent β-agonist, is used to study lung diseases like asthma.Fórmula:C12H19BrCl2N2OCor e Forma:SolidPeso molecular:358.1Mabuterol free base
CAS:Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.Fórmula:C13H18ClF3N2OPureza:98%Cor e Forma:SolidPeso molecular:310.74Ivabradine-d3 hydrochloride
CAS:Ivabradine HCl: novel If blocker, IC50 2.9 μM, slows heart rate; D3 version is deuterium labeled.Fórmula:C27H37ClN2O5Pureza:98%Cor e Forma:SolidPeso molecular:508.07Propranolol hydrochloride
CAS:Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverseFórmula:C16H22ClNO2Pureza:99.94% - >99.99%Cor e Forma:White Or Almost White Powder White PowderPeso molecular:295.80Benzquinamide
CAS:<p>Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer</p>Fórmula:C22H32N2O5Pureza:94.86%Cor e Forma:SolidPeso molecular:404.5Corynanthine
CAS:Corynanthe is a plant alkaloid. Corynanthe also has an alpha-2-adrenergic blocking activity.Fórmula:C21H26N2O3Pureza:98%Cor e Forma:SolidPeso molecular:354.44Metaraminol
CAS:Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.Fórmula:C9H13NO2Cor e Forma:SolidPeso molecular:167.21SB-206606
CAS:<p>SB-206606 is a novel, highly specific radioactive ligand for the β3-adrenergic receptor.</p>Fórmula:C19H22ClNO4Cor e Forma:SolidPeso molecular:363.83Acrinor
CAS:Acrinor is a adrenergic beta receptor agonist.Fórmula:C35H46Cl2N10O8Pureza:98%Cor e Forma:SolidPeso molecular:805.72AA 497 HCl
CAS:AA 497, a beta-2 agonist, suppresses Ca spikes.Fórmula:C14H22ClNO3Cor e Forma:SolidPeso molecular:287.78
