
Receptor adrenérgico
Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.
Subcategorias de "Receptor adrenérgico"
Foram encontrados 721 produtos de "Receptor adrenérgico"
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(±)5(6)-EET
CAS:5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.Fórmula:C20H32O3Cor e Forma:SolidPeso molecular:320.4735-hydroxy Propranolol
CAS:5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.Fórmula:C16H21NO3Cor e Forma:SolidPeso molecular:275.348Prazobind
CAS:Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.Fórmula:C23H27N5O3Cor e Forma:SolidPeso molecular:421.501Mapenterol hydrochloride
CAS:Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.Fórmula:C14H21Cl2F3N2OPureza:98.11% - 99.98%Cor e Forma:SolidPeso molecular:361.23Carbazochrome salicylate
CAS:Carbazochrome salicylate can be used as a coagulant.Fórmula:C17H18N4NaO6Cor e Forma:White Crystalline PowderPeso molecular:397.343Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS:Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Fórmula:C25H26O13Cor e Forma:SolidPeso molecular:534.47(R)-(+)-Atenolol
CAS:<p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>Fórmula:C14H22N2O3Pureza:98.72%Cor e Forma:SolidPeso molecular:266.34Sibenadet hydrochloride
CAS:Sibenadet, a D2/beta2-agonist, is potential useful for the treatment of symptoms of chronic obstructive pulmonary disease.Fórmula:C22H29ClN2O5S2Cor e Forma:SolidPeso molecular:501.06AG-825
CAS:AG-825(Tyrphostin C15) is a selective and competitive ErbB2 inhibitor that inhibits tyrosine phosphorylation with an IC50 value of 0.35 μM.AG-825 (TyrphostinFórmula:C19H15N3O3S2Pureza:99.52%Cor e Forma:Yellow SolidPeso molecular:397.47α1A-AR Degrader 9c
CAS:α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.Fórmula:C38H43N11O11Pureza:98%Cor e Forma:SolidPeso molecular:829.82Nolomirole
CAS:Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.Fórmula:C19H27NO4Cor e Forma:SolidPeso molecular:333.42Besipirdine hydrochloride
CAS:<p>Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.</p>Fórmula:C16H18ClN3Pureza:98.45%Cor e Forma:SoildPeso molecular:287.79O-Desmethyl Mebeverine alcohol hydrochloride
CAS:O-Desmethyl Mebeverine alcohol HCl, a metabolite of Mebeverine, is a strong α1 inhibitor, relaxing the GI tract.Fórmula:C15H26ClNO2Cor e Forma:SolidPeso molecular:287.83Carazolol-d7
CAS:Carazolol-d7 is the deuterium-labeled isotope of Carazolol, commonly used in pharmacokinetic studies to investigate the metabolic pathways of Carazolol.Fórmula:C18H22N2O2Cor e Forma:SolidPeso molecular:305.42Terazosin dimer impurity dihydrochloride
CAS:Terazosin dimer impurity dihydrochloride is a chemical byproduct of the α1-antagonist Terazosin, derived from quinazoline.Fórmula:C24H30Cl2N8O4Cor e Forma:SolidPeso molecular:565.46Oxaprotiline hydrochloride
CAS:Oxaprotiline hydrochloride is an antidepressant.Fórmula:C20H24ClNOPureza:98%Cor e Forma:SolidPeso molecular:329.86Formoterol O-β-D-Glucuronide
CAS:Formoterol O-β-D-glucuronide is a metabolite of formoterol .Fórmula:C25H32N2O10Cor e Forma:SolidPeso molecular:520.535Quinazosin hydrochloride
CAS:Quinazosin hydrochloride is an antihypertensive agent.Fórmula:C17H25Cl2N5O2Cor e Forma:SolidPeso molecular:402.32Idazoxan
CAS:Idazoxan is an alpha2 receptor antagonist that also exhibits activity at imidazoline [I1] and [I2] receptors, playing a role in modulating dopamine release.Fórmula:C11H12N2O2Peso molecular:204.23

