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CaMK

CaMK

Os inibidores da Proteína Quinase Dependente de Cálcio/Calmodulina (CaMK) são compostos especializados que inibem a atividade da CaMK, uma quinase crucial envolvida em uma variedade de processos celulares, particularmente no sistema nervoso. A CaMK é essencial para traduzir sinais de cálcio em várias respostas celulares, incluindo a plasticidade sináptica, a formação de memória e a expressão gênica. A desregulação da atividade da CaMK está associada a vários distúrbios neurológicos, tornando esses inibidores ferramentas valiosas para o estudo da sinalização sináptica, do aprendizado e da memória. Na CymitQuimica, oferecemos inibidores de CaMK de alta qualidade para apoiar sua pesquisa em plasticidade sináptica, função cognitiva e neurofarmacologia.

Foram encontrados 66 produtos para "CaMK".

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  • CAMKIV Protein, Human, Recombinant (GST)


    CAMKIV Protein, Human, Recombinant (GST) is expressed in Baculovirus insect cells with GST tag.
    Cor e Forma:Lyophilized Powder
    Peso molecular:79 kDa (predicted); 100 kDa (reducing conditions)

    Ref: TM-TMPY-04543

    5µg
    79,00€
    10µg
    110,00€
    20µg
    177,00€
    50µg
    413,00€
  • CALP2 acetate


    CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM.
    Fórmula:C68H104N14O13S
    Pureza:99.91%
    Cor e Forma:White Solid
    Peso molecular:1357.7

    Ref: TM-TP1909L1

    1mg
    55,00€
    5mg
    103,00€
    10mg
    168,00€
    25mg
    301,00€
    50mg
    424,00€
    100mg
    605,00€
  • Syntide 2 acetate


    Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).
    Fórmula:C70H126N20O20
    Pureza:99.87%
    Cor e Forma:Purple Liquid
    Peso molecular:1567.85

    Ref: TM-TP1403L

    1mg
    50,00€
    5mg
    159,00€
    10mg
    253,00€
    25mg
    414,00€
    50mg
    583,00€
    100mg
    783,00€
  • KN-92

    CAS:
    KN-92 is an inactive analog of the CaM kinase II inhibitor KN 93.
    Fórmula:C24H25ClN2O3S
    Cor e Forma:Solid
    Peso molecular:456.98

    Ref: TM-T4530L

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • GSK3i XIII

    CAS:
    GSK3i XIII (GSK3 inhibitor XIII) is a GSK-3 ATP-binding site inhibitor.
    Fórmula:C18H19N5
    Pureza:99.46%
    Cor e Forma:Solid
    Peso molecular:305.38

    Ref: TM-T24111

    1mg
    50,00€
    5mg
    101,00€
    1mL*10mM (DMSO)
    111,00€
    10mg
    150,00€
    25mg
    241,00€
    50mg
    353,00€
    100mg
    572,00€
  • KN-92 hydrochloride

    CAS:
    KN-92 hydrochloride is an inactive derivative of KN-93.
    Fórmula:C24H26Cl2N2O3S
    Pureza:99.68%
    Cor e Forma:White Solid
    Peso molecular:493.45

    Ref: TM-T8543

    1mg
    34,00€
    5mg
    99,00€
    1mL*10mM (DMSO)
    107,00€
    10mg
    167,00€
    25mg
    268,00€
    50mg
    409,00€
    100mg
    580,00€
  • IGS-1.76

    CAS:
    IGS-1.76 binds strongly to hNCS-1, modulates its Ric8a interaction, and inhibits the hNCS-1/Ric8a complex.
    Fórmula:C22H18N2OS
    Pureza:98.18% - 98.56%
    Cor e Forma:Solid
    Peso molecular:358.456

    Ref: TM-T8784

    2mg
    34,00€
    5mg
    50,00€
    1mL*10mM (DMSO)
    55,00€
    10mg
    79,00€
    25mg
    128,00€
    50mg
    173,00€
    100mg
    243,00€
  • Trifluoperazine

    CAS:
    Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
    Fórmula:C21H24F3N3S
    Pureza:98.3% - 99.98%
    Cor e Forma:Solid
    Peso molecular:407.496

    Ref: TM-T8389

    1mg
    42,00€
    2mg
    50,00€
    5mg
    77,00€
    10mg
    103,00€
    25mg
    182,00€
    50mg
    284,00€
    100mg
    430,00€
    200mg
    620,00€
  • NH125

    CAS:
    NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, >125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.
    Fórmula:C27H45IN2
    Pureza:98.60%
    Cor e Forma:Solid
    Peso molecular:524.56

    Ref: TM-T6605

    1mg
    38,00€
    2mg
    50,00€
    5mg
    84,00€
    1mL*10mM (DMSO)
    93,00€
    10mg
    113,00€
    25mg
    250,00€
    50mg
    430,00€
    100mg
    620,00€
  • KN-62

    CAS:
    KN-62 is a potent and specific Ca2+/calmodulin-dependent protein kinase II (CaMKII) inhibitor with Ki of 0.9 μM.
    Fórmula:C38H35N5O6S2
    Pureza:99.80% - >99.99%
    Cor e Forma:Solid
    Peso molecular:721.84

    Ref: TM-T2694

    1mg
    34,00€
    2mg
    49,00€
    5mg
    71,00€
    10mg
    105,00€
    1mL*10mM (DMSO)
    105,00€
    25mg
    207,00€
    50mg
    404,00€
    100mg
    592,00€
  • CaMKII-IN-1

    CAS:
    CaMKII-IN-1 is a potent and highly selective inhibitor of CaMKII (IC50 = 63 nM).
    Fórmula:C29H30ClN5O2S
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:548.1

    Ref: TM-T14860

    1mg
    50,00€
    2mg
    71,00€
    5mg
    113,00€
    1mL*10mM (DMSO)
    137,00€
    10mg
    166,00€
    25mg
    334,00€
    50mg
    520,00€
    100mg
    750,00€
  • lavendustin C

    CAS:
    lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.
    Fórmula:C14H13NO5
    Pureza:98.06%
    Cor e Forma:Solid
    Peso molecular:275.26

    Ref: TM-T4185

    1mg
    42,00€
    2mg
    55,00€
    1mL*10mM (DMSO)
    90,00€
    5mg
    93,00€
    10mg
    152,00€
    25mg
    330,00€
    50mg
    492,00€
    100mg
    707,00€
  • STO-609

    CAS:
    STO-609 inhibits CaM-KKα/KKβ (Ki: 80/15 ng/mL), is specific, cell-permeable, and targets Ca2+/calmodulin-dependent protein kinase kinase.
    Fórmula:C19H10N2O3
    Pureza:97.14% - 99.35%
    Cor e Forma:Solid
    Peso molecular:314.29

    Ref: TM-T3546

    1mg
    39,00€
    5mg
    84,00€
    1mL*10mM (DMSO)
    93,00€
    10mg
    120,00€
    25mg
    250,00€
    50mg
    400,00€
    100mg
    620,00€
    200mg
    873,00€
  • A-484954

    CAS:
    A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.
    Fórmula:C13H15N5O3
    Pureza:97.47% - 99.86%
    Cor e Forma:Solid
    Peso molecular:289.29

    Ref: TM-TQ0137

    1mg
    40,00€
    2mg
    52,00€
    5mg
    84,00€
    1mL*10mM (DMSO)
    93,00€
    10mg
    137,00€
    25mg
    289,00€
    50mg
    515,00€
    100mg
    733,00€
  • Autocamtide 2 TFA


    Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.
    Fórmula:C67H119F3N22O22
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:1641.79

    Ref: TM-TP1217L

    2mg
    42,00€
    5mg
    88,00€
    10mg
    122,00€
    25mg
    190,00€
    50mg
    261,00€
    100mg
    354,00€
  • KN-93

    CAS:
    KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase.
    Fórmula:C26H29ClN2O4S
    Pureza:99.56% - 99.95%
    Cor e Forma:White Solid
    Peso molecular:501.04

    Ref: TM-T2697

    1mg
    54,00€
    2mg
    74,00€
    5mg
    107,00€
    1mL*10mM (DMSO)
    120,00€
    10mg
    146,00€
    25mg
    289,00€
    50mg
    358,00€
    100mg
    523,00€
  • CaMKP Inhibitor

    CAS:
    CaMKP Inhibitor can inhibit CaMKP.
    Fórmula:C10H8NNaO7S2
    Pureza:99.91% - 99.98%
    Cor e Forma:Solid
    Peso molecular:341.28

    Ref: TM-T2159

    1mg
    34,00€
    5mg
    65,00€
    1mL*10mM (DMSO)
    73,00€
    10mg
    96,00€
    25mg
    182,00€
    50mg
    268,00€
    100mg
    369,00€
  • Stains-All

    CAS:
    Stains-All is a cationic dye of carbocyanine.
    Fórmula:C30H27BrN2S2
    Pureza:98.85% - 99.71%
    Cor e Forma:Black Solid
    Peso molecular:559.58

    Ref: TM-T16939

    100mg
    33,00€
    1mL*10mM (DMSO)
    33,00€
  • Autocamtide-2-related inhibitory peptide

    CAS:
    Autocamtide-2-related inhibitory peptide is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.
    Fórmula:C64H116N22O19
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1497.74

    Ref: TM-TP2310

    1mg
    58,00€
    5mg
    118,00€
    10mg
    172,00€
    25mg
    281,00€
    50mg
    396,00€
    100mg
    537,00€
    200mg
    712,00€
  • Autocamtide-2-related inhibitory peptide TFA salt


    Autocamtide-2-related inhibitory peptide TFA salt(CaM kinase II inhibitor TFA salt) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.
    Fórmula:C66H117F3N22O21
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1611.77

    Ref: TM-TP1216

    1mg
    73,00€
    5mg
    152,00€
    10mg
    215,00€
    25mg
    354,00€
    50mg
    522,00€
    100mg
    700,00€