Protease serina
Os inibidores de serina protease são compostos que inibem as serina proteases, um grupo de enzimas caracterizado por um resíduo de serina no seu sítio ativo. Essas proteases estão envolvidas em vários processos fisiológicos, incluindo digestão, resposta imunológica, coagulação sanguínea e inflamação. Os inibidores de serina protease são importantes para o estudo de doenças onde essas enzimas estão desreguladas, como doenças cardiovasculares, câncer e condições inflamatórias. Na CymitQuimica, oferecemos inibidores de serina protease para apoiar sua pesquisa em enzimologia, mecanismos de doenças e intervenções terapêuticas.
Foram encontrados 50 produtos de "Protease serina"
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Chymotrypsinogen
CAS:<p>Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .</p>Cor e Forma:SolidPKR-IN-C51
CAS:<p>PKR-IN-C51 is ATP-competitive protein kinase R (PKR) inhibitor that inhibits intracellular PKR activation and autophosphorylation. Ser/Thr kinase.</p>Fórmula:C23H21N5Pureza:98.94%Cor e Forma:SolidPeso molecular:367.45Urokinase
CAS:<p>Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.</p>Cor e Forma:SolidGSK-690693
CAS:<p>GSK-690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM, also sensitive to the AGC kinase family: PKA, PrkX and PKC isozymes. Phase 1.</p>Fórmula:C21H27N7O3Pureza:98.07% - 99.77%Cor e Forma:SolidPeso molecular:425.482-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one
CAS:<p>2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one is an human neutrophil elastase inhibitor.</p>Fórmula:C14H7BrClNO2Pureza:97.36%Cor e Forma:SolidPeso molecular:336.57Cetraxate hydrochloride
CAS:<p>Cetraxate hydrochloride (DV10062) is an oral gastrointestinal medication. It has a cytoprotective effect.</p>Fórmula:C17H24ClNO4Pureza:99.75%Cor e Forma:SolidPeso molecular:341.83WNK463
CAS:<p>WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).</p>Fórmula:C21H24F3N7O2Pureza:>99.99% - ≥95%Cor e Forma:SolidPeso molecular:463.46WNK-IN-11
CAS:<p>WNK-IN-11 (Allosteric WNK Kinase Inhibitor) is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)</p>Fórmula:C21H21Cl2N5OSPureza:98.32%Cor e Forma:SolidPeso molecular:462.4Alvelestat
CAS:<p>Alvelestat (AZD9668) is an orally bioavailable, selective and reversible inhibitor of human neutrophil elastase (NE), with potential anti-inflammatory activity.</p>Fórmula:C25H22F3N5O4SPureza:98% - >99.99%Cor e Forma:SolidPeso molecular:545.53ML281
CAS:<p>ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.</p>Fórmula:C22H19N3O2SPureza:99.12% - 99.87%Cor e Forma:SolidPeso molecular:389.472,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
CAS:<p>2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urine</p>Fórmula:C13H16O3Pureza:99.53% - 99.81%Cor e Forma:SolidPeso molecular:220.26Ceritinib
CAS:<p>Ceritinib (LDK378) is an ALK inhibitor with selective, ATP-competitive, and oral activity. Ceritinib has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C28H36ClN5O3SPureza:98.52% - 99.77%Cor e Forma:SolidPeso molecular:558.14Lanadelumab
CAS:<p>Lanadelumab (SHP643), a humanized IgG1 antibody, inhibits plasma kallikrein and its interaction with HMWK, supporting hereditary angioedema research.</p>Pureza:95% - 95%Cor e Forma:LiquidGalegenimab
CAS:<p>Galegenimab (FHTR 2163; RG 6147; RO 7171009) is an HTRA1 antibody fragment for AMD research.</p>Pureza:95% - 95%Cor e Forma:LiquidMEGA-9
CAS:<p>MEGA-9 (Nonanoyl-N-Methylglucamide) solubilizes membrane protein and can be used as a nonionic detergent.</p>Fórmula:C16H33NO6Pureza:99.9%Cor e Forma:SolidPeso molecular:335.44BMS-363131
CAS:<p>BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.</p>Fórmula:C28H40N6O5Pureza:97.99%Cor e Forma:SolidPeso molecular:540.65p-Aminobenzamidine dihydrochloride
CAS:<p>4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase type</p>Fórmula:C7H11Cl2N3Pureza:99.00% - 99.56%Cor e Forma:SolidPeso molecular:208.088ZD8321
CAS:<p>ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).</p>Fórmula:C18H28F3N3O5Pureza:98%Cor e Forma:SolidPeso molecular:423.43ZD-0892
CAS:<p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>Fórmula:C24H32F3N3O5Pureza:95% - 99.53%Cor e Forma:SolidPeso molecular:499.52APC 366
CAS:<p>APC 366: Mast cell tryptase inhibitor, Ki 7.1 μM. Reduces EAR, LAR, BHR in allergic asthma (sheep model).</p>Fórmula:C22H28N6O4Pureza:99.8%Cor e Forma:SolidPeso molecular:440.5
